UB Paderborn / Katalog / Suche / in CDI

Sortiert nach

Einfacher Volltextzugriff von (fast) überall

Installieren Sie die LibKey Nomad-Browsererweiterung und erhalten Sie von vielen Webseiten einfachen Zugriff auf lizenzierte Volltexte oder Open Access Publikationen. Mehr erfahren...

Design and synthesis of morpholine derivatives. SAR for dual serotonin & noradrenaline reuptake inhibition

Bioorganic & medicinal chemistry, 2008-04, Vol.18 (8), p.2562-2566

2008

Volltextzugriff (PDF)

Discovery of PF-184563, a potent and selective V1a antagonist for the treatment of dysmenorrhoea. The influence of compound flexibility on microsomal stability

Bioorganic & medicinal chemistry letters, 2011-10, Vol.21 (19), p.5684-5687

2011

Volltextzugriff (PDF)

Novel 2-imidazoles as potent, selective and CNS penetrant α1A adrenoceptor partial agonists

Bioorganic & medicinal chemistry letters, 2008-12, Vol.18 (24), p.6437-6440

2008

Volltextzugriff (PDF)

Pyridyl-phenyl ether monoamine reuptake inhibitors: Impact of lipophilicity on dual SNRI pharmacology and off-target promiscuity

Bioorganic & medicinal chemistry, 2008-05, Vol.18 (9), p.2896-2899

2008

Volltextzugriff (PDF)

[4-(Phenoxy)pyridin-3-yl]methylamines: A new class of selective noradrenaline reuptake inhibitors

Bioorganic & medicinal chemistry, 2008-03, Vol.18 (6), p.1795-1798

2008

Volltextzugriff (PDF)

Potent and selective α1A adrenoceptor partial agonists—Novel imidazole frameworks

Bioorganic & medicinal chemistry letters, 2009-06, Vol.19 (11), p.3118-3121

2009

Volltextzugriff (PDF)

Pharmacological Properties of 2-(( R -5-Chloro-4-methoxymethylindan-1-yl)-1 H -imidazole (PF-3774076), a Novel and Selective α1 A -Adrenergic Partial Agonist, in in Vitro and in Vivo Models of Urethral Function

The Journal of pharmacology and experimental therapeutics, 2009-09, Vol.330 (3), p.892-901

2009

Volltextzugriff (PDF)

Design, synthesis and evaluation of N-[(3 S)-pyrrolidin-3-yl]benzamides as selective noradrenaline reuptake inhibitors: CNS penetration in a more polar template

Bioorganic & medicinal chemistry letters, 2009-08, Vol.19 (16), p.4579-4583

2009

Volltextzugriff (PDF)

Structure−Activity Relationships of 1,4-Dihydro-(1H,4H)-quinoxaline-2,3-diones as N-Methyl-d-aspartate (Glycine Site) Receptor Antagonists. 1. Heterocyclic Substituted 5-Alkyl Derivatives

Journal of medicinal chemistry, 2001-06, Vol.44 (12), p.1951-1962

2001

Volltextzugriff (PDF)

4-Piperidines and 3-pyrrolidines as dual serotonin and noradrenaline reuptake inhibitors: Design, synthesis and structure–activity relationships

Bioorganic & medicinal chemistry letters, 2009-05, Vol.19 (10), p.2829-2834

2009

Volltextzugriff (PDF)

Potent and selective alpha 1A adrenoceptor partial agonists-Novel imidazole frameworks

Bioorganic & medicinal chemistry letters, 2009-06, Vol.19 (11), p.3118-3121

2009

Volltextzugriff (PDF)

Novel 2-imidazoles as potent, selective and CNS penetrant alpha sub(1A) adrenoceptor partial agonists

Bioorganic & medicinal chemistry, 2008-12, Vol.18 (24), p.6437-6440

2008

Volltextzugriff (PDF)

Novel 2-imidazoles as potent and selective α1A adrenoceptor partial agonists

Bioorganic & medicinal chemistry letters, 2008-05, Vol.18 (9), p.2930-2934

2008

Volltextzugriff (PDF)

N-Benzyl- N-(tetrahydro-2 H-pyran-4-yl)pyrrolidin-3-amines as selective dual serotonin/noradrenaline reuptake inhibitors

Bioorganic & medicinal chemistry letters, 2007-04, Vol.17 (7), p.2022-2025

2007

Volltextzugriff (PDF)

Novel Selective Inhibitors of Neutral Endopeptidase for the Treatment of Female Sexual Arousal Disorder. Synthesis and Activity of Functionalized Glutaramides

Journal of medicinal chemistry, 2006-07, Vol.49 (14), p.4409-4424

2006

Volltextzugriff (PDF)

Novel 2-imidazoles as potent and selective alpha sub(1A) adrenoceptor partial agonists

Bioorganic & medicinal chemistry, 2008-05, Vol.18 (9), p.2920-2923

2008

Volltextzugriff (PDF)

Designing rapid onset selective serotonin re-uptake inhibitors. Part 3: Site-directed metabolism as a strategy to avoid active circulating metabolites: Structure–activity relationships of (thioalkyl)phenoxy benzylamines

Bioorganic & medicinal chemistry letters, 2008-10, Vol.18 (19), p.5303-5306

2008

Volltextzugriff (PDF)

N-(1,2-Diphenylethyl)piperazines: A new class of dual serotonin/noradrenaline reuptake inhibitor

Bioorganic & medicinal chemistry letters, 2006-08, Vol.16 (16), p.4345-4348

2006

Volltextzugriff (PDF)

N-[(3 S)-Pyrrolidin-3-yl]benzamides as novel dual serotonin and noradrenaline reuptake inhibitors: Impact of small structural modifications on P-gp recognition and CNS penetration

Bioorganic & medicinal chemistry letters, 2009-09, Vol.19 (17), p.5078-5081

2009

Volltextzugriff (PDF)

N-Benzyl- N-(pyrrolidin-3-yl)carboxamides as a new class of selective dual serotonin/noradrenaline reuptake inhibitors

Bioorganic & medicinal chemistry, 2008-08, Vol.18 (15), p.4308-4311

2008

Volltextzugriff (PDF)

Structure–activity relationships of N-substituted piperazine amine reuptake inhibitors

Bioorganic & medicinal chemistry letters, 2006-08, Vol.16 (16), p.4349-4353

2006

Volltextzugriff (PDF)

Novel 2-imidazoles as potent and selective α 1A adrenoceptor partial agonists

Bioorganic & medicinal chemistry letters, 2008, Vol.18 (9), p.2930-2934

2008

Volltextzugriff (PDF)

Novel 2-imidazoles as potent, selective and CNS penetrant α 1A adrenoceptor partial agonists

Bioorganic & medicinal chemistry letters, 2008, Vol.18 (24), p.6437-6440

2008

Volltextzugriff (PDF)

Designing rapid onset selective serotonin re-uptake inhibitors. 2: Structure–activity relationships of substituted (aryl)benzylamines

Bioorganic & medicinal chemistry, 2008-07, Vol.18 (14), p.4018-4021

2008

Volltextzugriff (PDF)

Derivatives of (3 S)- N-(biphenyl-2-ylmethyl)pyrrolidin-3-amine as selective noradrenaline reuptake inhibitors: Reducing P-gp mediated efflux by modulation of H-bond acceptor capacity

Bioorganic & medicinal chemistry, 2008-08, Vol.18 (15), p.4355-4359

2008

Volltextzugriff (PDF)

1 – 25 von 53

Suche als RSS-Feed

Suchergebnisse filtern

Filter anzeigen

Nur zeigen

Geprüft (Peer-Review)
(42)
Mit Volltextzugriff
(45)

Publikationsform

Sprache

Englisch
(53)

Erscheinungsjahr

n.n

Thema

Science & Technology
(27)
Chemistry
(22)
Humans
(22)
Life Sciences & Biomedicine
(22)
Physical Sciences
(22)
Biological And Medical Sciences
(21)
Chemistry, Medicinal
(21)
Medical Sciences
(21)
Pharmacology & Pharmacy
(21)
Pharmacology. Drug Treatments
(21)
Chemistry, Organic
(19)
Structure-Activity Relationship
(18)
Neuropharmacology
(16)
Animals
(15)
Neurotransmitters. Neurotransmission. Receptors
(13)
Drug Design
(12)
Serotonin Uptake Inhibitors - Chemistry
(11)
Serotonin Uptake Inhibitors - Pharmacology
(11)
Rats
(10)
Dogs
(9)

15 weitere anzeigen...

Weniger anzeigen...

Menü

Weitere Dienste

Einstellungen

Design and synthesis of morpholine derivatives. SAR for dual serotonin & noradrenaline reuptake inhibition

Discovery of PF-184563, a potent and selective V1a antagonist for the treatment of dysmenorrhoea. The influence of compound flexibility on microsomal stability

Novel 2-imidazoles as potent, selective and CNS penetrant α1A adrenoceptor partial agonists

Pyridyl-phenyl ether monoamine reuptake inhibitors: Impact of lipophilicity on dual SNRI pharmacology and off-target promiscuity

[4-(Phenoxy)pyridin-3-yl]methylamines: A new class of selective noradrenaline reuptake inhibitors

Potent and selective α1A adrenoceptor partial agonists—Novel imidazole frameworks

Pharmacological Properties of 2-(( R -5-Chloro-4-methoxymethylindan-1-yl)-1 H -imidazole (PF-3774076), a Novel and Selective α1 A -Adrenergic Partial Agonist, in in Vitro and in Vivo Models of Urethral Function

Design, synthesis and evaluation of N-[(3 S)-pyrrolidin-3-yl]benzamides as selective noradrenaline reuptake inhibitors: CNS penetration in a more polar template

Structure−Activity Relationships of 1,4-Dihydro-(1H,4H)-quinoxaline-2,3-diones as N-Methyl-d-aspartate (Glycine Site) Receptor Antagonists. 1. Heterocyclic Substituted 5-Alkyl Derivatives

4-Piperidines and 3-pyrrolidines as dual serotonin and noradrenaline reuptake inhibitors: Design, synthesis and structure–activity relationships

Potent and selective alpha 1A adrenoceptor partial agonists-Novel imidazole frameworks

Novel 2-imidazoles as potent, selective and CNS penetrant alpha sub(1A) adrenoceptor partial agonists

Novel 2-imidazoles as potent and selective α1A adrenoceptor partial agonists

N-Benzyl- N-(tetrahydro-2 H-pyran-4-yl)pyrrolidin-3-amines as selective dual serotonin/noradrenaline reuptake inhibitors

Novel Selective Inhibitors of Neutral Endopeptidase for the Treatment of Female Sexual Arousal Disorder. Synthesis and Activity of Functionalized Glutaramides

Novel 2-imidazoles as potent and selective alpha sub(1A) adrenoceptor partial agonists

Designing rapid onset selective serotonin re-uptake inhibitors. Part 3: Site-directed metabolism as a strategy to avoid active circulating metabolites: Structure–activity relationships of (thioalkyl)phenoxy benzylamines

N-(1,2-Diphenylethyl)piperazines: A new class of dual serotonin/noradrenaline reuptake inhibitor

N-[(3 S)-Pyrrolidin-3-yl]benzamides as novel dual serotonin and noradrenaline reuptake inhibitors: Impact of small structural modifications on P-gp recognition and CNS penetration

N-Benzyl- N-(pyrrolidin-3-yl)carboxamides as a new class of selective dual serotonin/noradrenaline reuptake inhibitors

Structure–activity relationships of N-substituted piperazine amine reuptake inhibitors

Novel 2-imidazoles as potent and selective α 1A adrenoceptor partial agonists

Novel 2-imidazoles as potent, selective and CNS penetrant α 1A adrenoceptor partial agonists

Designing rapid onset selective serotonin re-uptake inhibitors. 2: Structure–activity relationships of substituted (aryl)benzylamines

Derivatives of (3 S)- N-(biphenyl-2-ylmethyl)pyrrolidin-3-amine as selective noradrenaline reuptake inhibitors: Reducing P-gp mediated efflux by modulation of H-bond acceptor capacity

Suchergebnisse filtern