UB Paderborn / Katalog / Suche / in CDI

Chloroquine and its analogs: A new promise of an old drug for effective and safe cancer therapies

European journal of pharmacology, 2009-12, Vol.625 (1), p.220-233

2009

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An overview of quinazolines: Pharmacological significance and recent developments

European journal of medicinal chemistry, 2018-05, Vol.151, p.628-685

2018

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Examination of novel 4-aminoquinoline derivatives designed and synthesized by a hybrid pharmacophore approach to enhance their anticancer activities

Scientific reports, 2019-04, Vol.9 (1), p.6315, Article 6315

2019

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Hybrid pharmacophore design and synthesis of isatin–benzothiazole analogs for their anti-breast cancer activity

Bioorganic & medicinal chemistry, 2009-11, Vol.17 (21), p.7585-7592

2009

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Design and synthesis of anti-breast cancer agents from 4-piperazinylquinoline: A hybrid pharmacophore approach

Bioorganic & medicinal chemistry, 2010-02, Vol.18 (4), p.1563-1572

2010

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Synthesis and pharmacological evaluation of some 3-phenyl-2-substituted-3H-quinazolin-4-one as analgesic, anti-inflammatory agents

Bioorganic & medicinal chemistry, 2007-01, Vol.15 (1), p.235-241

2007

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Synthesis and Antimalarial Activity of Side Chain Modified 4-Aminoquinoline Derivatives

Journal of medicinal chemistry, 2007-01, Vol.50 (2), p.394-398

2007

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Pharmacophore modelling-based drug repurposing approaches for monkeypox therapeutics

Journal of biomolecular structure & dynamics, 2023-12, Vol.ahead-of-print (ahead-of-print), p.1-12

2023

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Investigating the Role of Loop C Hydrophilic Residue 'T244' in the Binding Site of ρ1 GABAC Receptors via Site Mutation and Partial Agonism

PloS one, 2016-05, Vol.11 (5), p.e0156618-e0156618

2016

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Computational Search for Potential COVID-19 Drugs from Ayurvedic Medicinal Plants to Identify Potential Inhibitors against SARS-CoV-2 Targets

Current computer-aided drug design, 2023-01, Vol.19 (1), p.51

2023

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Design and Synthesis of 3‐Substituted‐thiazolyl‐2‐iminothiazolidin‐4‐ones as a New Class of Anticonvulsants

Journal of heterocyclic chemistry, 2016-09, Vol.53 (5), p.1635-1639

2016

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The efficacy and selectivity of tumor cell killing by Akt inhibitors are substantially increased by chloroquine

Bioorganic & medicinal chemistry, 2008-09, Vol.16 (17), p.7888-7893

2008

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A 4-aminoquinoline derivative that markedly sensitizes tumor cell killing by Akt inhibitors with a minimum cytotoxicity to non-cancer cells

European journal of medicinal chemistry, 2010-02, Vol.45 (2), p.705-709

2010

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Design, synthesis and characterization of novel quinacrine analogs that preferentially kill cancer over non-cancer cells through the down-regulation of Bcl-2 and up-regulation of Bax and Bad

European journal of medicinal chemistry, 2017-09, Vol.137, p.156-166

2017

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3-(3-Ethylphenyl)-2-substituted hydrazino-3H-quinazolin-4-one Derivatives: New Class of Analgesic and Anti-Inflammatory Agents

Chemical biology & drug design, 2009-04, Vol.73 (4), p.471-479

2009

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Design and synthesis of novel quinacrine-[1,3]-thiazinan-4-one hybrids for their anti-breast cancer activity

European journal of medicinal chemistry, 2018-01, Vol.143, p.1028-1038

2018

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Synthesis of 2-mercapto-3-substituted-5,6-dimethylthieno[2,3- d ] pyrimidin-4(3 H )-ones as new analgesic, anti-inflammatory agents

Biomedicine & pharmacotherapy, 2007-06, Vol.61 (5), p.285-291

2007

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VR23: A Quinoline-Sulfonyl Hybrid Proteasome Inhibitor That Selectively Kills Cancer via Cyclin E-Mediated Centrosome Amplification

Cancer research (Chicago, Ill.), 2015-10, Vol.75 (19), p.4164-4175

2015

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Design and synthesis of new antimalarial agents from 4-aminoquinoline

Bioorganic & medicinal chemistry, 2005-03, Vol.13 (6), p.2157-2165

2005

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Anti-breast cancer activity of heteroaryl chalcone derivatives

Biomedicine & pharmacotherapy, 2012-04, Vol.66 (3), p.213-220

2012

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Design and synthesis of 3-(4-Ethylphenyl)-2-substituted amino-3H-quinazolin-4-ones as a novel class of analgesic and anti-inflammatory agents

Journal of enzyme inhibition and medicinal chemistry, 2008-01, Vol.23 (6), p.839-847

2008

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Design, Synthesis, and Structure–Activity Relationships of Novel N-Substituted-5-phenyl-[1,2,4]triazolo[1,5-c]quinazolin-2-amine for Their Anti-HIV and Antibacterial Activities

Russian journal of bioorganic chemistry, 2022-12, Vol.48 (6), p.1221-1229

2022

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Isolation, Functionalization, In Silico Investigation, and Synthesis of 1,8-Cineole Analog as Antitubercular Agent Targeting InhA

Russian journal of bioorganic chemistry, 2023-04, Vol.49 (2), p.390-402

2023

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The potential of quinoline derivatives for the treatment of Toxoplasma gondii infection

Experimental parasitology, 2014-10, Vol.145, p.135-144

2014

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Design, Synthesis, and Structure–Activity Relationships of Novel 1-(Substituted)-2-Methyl-3-(4-Oxo-2-Methylquinazolin-3(4H)-yl) Isothioureas for Their Anti-HIV and Antibacterial Activities

Russian journal of bioorganic chemistry, 2022, Vol.48 (3), p.548-556

2022

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Chloroquine and its analogs: A new promise of an old drug for effective and safe cancer therapies

An overview of quinazolines: Pharmacological significance and recent developments

Examination of novel 4-aminoquinoline derivatives designed and synthesized by a hybrid pharmacophore approach to enhance their anticancer activities

Hybrid pharmacophore design and synthesis of isatin–benzothiazole analogs for their anti-breast cancer activity

Design and synthesis of anti-breast cancer agents from 4-piperazinylquinoline: A hybrid pharmacophore approach

Synthesis and pharmacological evaluation of some 3-phenyl-2-substituted-3H-quinazolin-4-one as analgesic, anti-inflammatory agents

Synthesis and Antimalarial Activity of Side Chain Modified 4-Aminoquinoline Derivatives

Pharmacophore modelling-based drug repurposing approaches for monkeypox therapeutics

Investigating the Role of Loop C Hydrophilic Residue 'T244' in the Binding Site of ρ1 GABAC Receptors via Site Mutation and Partial Agonism

Computational Search for Potential COVID-19 Drugs from Ayurvedic Medicinal Plants to Identify Potential Inhibitors against SARS-CoV-2 Targets

Design and Synthesis of 3‐Substituted‐thiazolyl‐2‐iminothiazolidin‐4‐ones as a New Class of Anticonvulsants

The efficacy and selectivity of tumor cell killing by Akt inhibitors are substantially increased by chloroquine

A 4-aminoquinoline derivative that markedly sensitizes tumor cell killing by Akt inhibitors with a minimum cytotoxicity to non-cancer cells

Design, synthesis and characterization of novel quinacrine analogs that preferentially kill cancer over non-cancer cells through the down-regulation of Bcl-2 and up-regulation of Bax and Bad

3-(3-Ethylphenyl)-2-substituted hydrazino-3H-quinazolin-4-one Derivatives: New Class of Analgesic and Anti-Inflammatory Agents

Design and synthesis of novel quinacrine-[1,3]-thiazinan-4-one hybrids for their anti-breast cancer activity

Synthesis of 2-mercapto-3-substituted-5,6-dimethylthieno[2,3- d ] pyrimidin-4(3 H )-ones as new analgesic, anti-inflammatory agents

VR23: A Quinoline-Sulfonyl Hybrid Proteasome Inhibitor That Selectively Kills Cancer via Cyclin E-Mediated Centrosome Amplification

Design and synthesis of new antimalarial agents from 4-aminoquinoline

Anti-breast cancer activity of heteroaryl chalcone derivatives

Design and synthesis of 3-(4-Ethylphenyl)-2-substituted amino-3H-quinazolin-4-ones as a novel class of analgesic and anti-inflammatory agents

Design, Synthesis, and Structure–Activity Relationships of Novel N-Substituted-5-phenyl-[1,2,4]triazolo[1,5-c]quinazolin-2-amine for Their Anti-HIV and Antibacterial Activities

Isolation, Functionalization, In Silico Investigation, and Synthesis of 1,8-Cineole Analog as Antitubercular Agent Targeting InhA

The potential of quinoline derivatives for the treatment of Toxoplasma gondii infection

Design, Synthesis, and Structure–Activity Relationships of Novel 1-(Substituted)-2-Methyl-3-(4-Oxo-2-Methylquinazolin-3(4H)-yl) Isothioureas for Their Anti-HIV and Antibacterial Activities

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