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Discovery and Preclinical Profile of Saxagliptin (BMS-477118): A Highly Potent, Long-Acting, Orally Active Dipeptidyl Peptidase IV Inhibitor for the Treatment of Type 2 Diabetes

Journal of medicinal chemistry, 2005-07, Vol.48 (15), p.5025-5037

2005

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A Novel Series of Highly Potent Benzimidazole-Based Microsomal Triglyceride Transfer Protein Inhibitors

Journal of medicinal chemistry, 2001-03, Vol.44 (6), p.851-856

2001

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Synthesis, SAR, and atropisomerism of imidazolopyrimidine DPP4 inhibitors

Bioorganic & medicinal chemistry letters, 2010-11, Vol.20 (21), p.6273-6276

2010

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Synthesis of Novel Potent Dipeptidyl Peptidase IV Inhibitors with Enhanced Chemical Stability: Interplay between the N-Terminal Amino Acid Alkyl Side Chain and the Cyclopropyl Group of α-Aminoacyl-l-cis-4,5-methanoprolinenitrile-Based Inhibitors

Journal of medicinal chemistry, 2004-05, Vol.47 (10), p.2587-2598

2004

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N-Aryl-oxazolidin-2-imine Muscle Selective Androgen Receptor Modulators Enhance Potency through Pharmacophore Reorientation

Journal of medicinal chemistry, 2009-05, Vol.52 (9), p.2794-2798

2009

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Potent non-nitrile dipeptidic dipeptidyl peptidase IV inhibitors

Bioorganic & medicinal chemistry, 2007-12, Vol.17 (23), p.6476-6480

2007

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Pyridine amides as potent and selective inhibitors of 11β-hydroxysteroid dehydrogenase type 1

Bioorganic & medicinal chemistry, 2008-06, Vol.18 (11), p.3168-3172

2008

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Dual Metalloprotease Inhibitors: Mercaptoacetyl-Based Fused Heterocyclic Dipeptide Mimetics as Inhibitors of Angiotensin-Converting Enzyme and Neutral Endopeptidase

Journal of medicinal chemistry, 1997-05, Vol.40 (11), p.1570-1577

1997

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Diprolyl nitriles as potent dipeptidyl peptidase IV inhibitors

Bioorganic & medicinal chemistry letters, 2005-09, Vol.15 (18), p.3992-3995

2005

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Vasopeptidase Inhibitors: Incorporation of Geminal and Spirocyclic Substituted Azepinones in Mercaptoacyl Dipeptides

Journal of medicinal chemistry, 1999-01, Vol.42 (2), p.305-311

1999

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Dual Metalloprotease Inhibitors. 6. Incorporation of Bicyclic and Substituted Monocyclic Azepinones as Dipeptide Surrogates in Angiotensin-Converting Enzyme/Neutral Endopeptidase Inhibitors

Journal of medicinal chemistry, 1996-01, Vol.39 (2), p.494-502

1996

Volltextzugriff (PDF)

Peptidomimetic Synthesis: A Novel, Highly Stereoselective Route to Substituted Freidinger Lactams

Journal of the American Chemical Society, 1994-03, Vol.116 (6), p.2348-2355

1994

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An MTP Inhibitor that Normalizes Atherogenic Lipoprotein Levels in WHHL Rabbits

Science (American Association for the Advancement of Science), 1998-10, Vol.282 (5389), p.751-754

1998

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Phosphorus-containing inhibitors of HMG-CoA reductase. I. 4-[(2-Arylethyl)hydroxyphosphinyl]-3-hydroxybutanoic acids: a new class of cell selective inhibitors of cholesterol biosynthesis

Journal of medicinal chemistry, 1990-11, Vol.33 (11), p.2952-2956

1990

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N-formyl hydroxylamine containing dipeptides : Generation of a new class of vasopeptidase inhibitors

Bioorganic & medicinal chemistry letters, 2000-02, Vol.10 (3), p.257-260

2000

Volltextzugriff (PDF)

1-Acyltriazoles as antiinflammatory agents

Journal of medicinal chemistry, 1982-03, Vol.25 (3), p.331-333

1982

Volltextzugriff (PDF)

Pyridine amides as potent and selective inhibitors of 11beta-hydroxysteroid dehydrogenase type 1

Bioorganic & medicinal chemistry letters, 2008-06, Vol.18 (11), p.3168

2008

Volltextzugriff (PDF)

Dual metalloprotease inhibitors. I. constrained peptidomimetics of mercaptoacyl dipeptides

Bioorganic & medicinal chemistry letters, 1994-08, Vol.4 (15), p.1789-1794

1994

Volltextzugriff (PDF)

Phosphorus-containing inhibitors of HMG-CoA reductase. 1. 4-[(2-arylethyl)hydroxyphosphinyl]-3-hydroxy-butanoic acids: a new class of cell-selective inhibitors of cholesterol biosynthesis

Journal of medicinal chemistry, 1990-11, Vol.33 (11), p.2952-2956

1990

Volltextzugriff (PDF)

Dual metalloprotease inhibitors. II. Effect of substitution and stereochemistry on benzazepinone based mercaptoacetyls

Bioorganic & medicinal chemistry letters, 1994-08, Vol.4 (15), p.1795-1800

1994

Volltextzugriff (PDF)

Dual metalloprotease inhibitors. III. utilization of bicyclic and monocyclic diazepinone based mercaptoacetyls

Bioorganic & medicinal chemistry letters, 1994-08, Vol.4 (16), p.2055-2060

1994

Volltextzugriff (PDF)

Selective inhibition of urokinase by substituted phenylguanidines: quantitative structure-activity relationship analyses

Journal of medicinal chemistry, 1990-11, Vol.33 (11), p.2956-2961

1990

Volltextzugriff (PDF)

ChemInform Abstract: N-Formyl Hydroxylamine Containing Dipeptides: Generation of a New Class of Vasopeptidase Inhibitors

ChemInform, 2000-05, Vol.31 (21), p.no-no

2000

Volltextzugriff (PDF)

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Discovery and Preclinical Profile of Saxagliptin (BMS-477118): A Highly Potent, Long-Acting, Orally Active Dipeptidyl Peptidase IV Inhibitor for the Treatment of Type 2 Diabetes

A Novel Series of Highly Potent Benzimidazole-Based Microsomal Triglyceride Transfer Protein Inhibitors

Synthesis, SAR, and atropisomerism of imidazolopyrimidine DPP4 inhibitors

Synthesis of Novel Potent Dipeptidyl Peptidase IV Inhibitors with Enhanced Chemical Stability: Interplay between the N-Terminal Amino Acid Alkyl Side Chain and the Cyclopropyl Group of α-Aminoacyl-l-cis-4,5-methanoprolinenitrile-Based Inhibitors

N-Aryl-oxazolidin-2-imine Muscle Selective Androgen Receptor Modulators Enhance Potency through Pharmacophore Reorientation

Potent non-nitrile dipeptidic dipeptidyl peptidase IV inhibitors

Pyridine amides as potent and selective inhibitors of 11β-hydroxysteroid dehydrogenase type 1

Dual Metalloprotease Inhibitors: Mercaptoacetyl-Based Fused Heterocyclic Dipeptide Mimetics as Inhibitors of Angiotensin-Converting Enzyme and Neutral Endopeptidase

Diprolyl nitriles as potent dipeptidyl peptidase IV inhibitors

Vasopeptidase Inhibitors: Incorporation of Geminal and Spirocyclic Substituted Azepinones in Mercaptoacyl Dipeptides

Dual Metalloprotease Inhibitors. 6. Incorporation of Bicyclic and Substituted Monocyclic Azepinones as Dipeptide Surrogates in Angiotensin-Converting Enzyme/Neutral Endopeptidase Inhibitors

Peptidomimetic Synthesis: A Novel, Highly Stereoselective Route to Substituted Freidinger Lactams

An MTP Inhibitor that Normalizes Atherogenic Lipoprotein Levels in WHHL Rabbits

Phosphorus-containing inhibitors of HMG-CoA reductase. I. 4-[(2-Arylethyl)hydroxyphosphinyl]-3-hydroxybutanoic acids: a new class of cell selective inhibitors of cholesterol biosynthesis

N-formyl hydroxylamine containing dipeptides : Generation of a new class of vasopeptidase inhibitors

1-Acyltriazoles as antiinflammatory agents

Pyridine amides as potent and selective inhibitors of 11beta-hydroxysteroid dehydrogenase type 1

Dual metalloprotease inhibitors. I. constrained peptidomimetics of mercaptoacyl dipeptides

Phosphorus-containing inhibitors of HMG-CoA reductase. 1. 4-[(2-arylethyl)hydroxyphosphinyl]-3-hydroxy-butanoic acids: a new class of cell-selective inhibitors of cholesterol biosynthesis

Dual metalloprotease inhibitors. II. Effect of substitution and stereochemistry on benzazepinone based mercaptoacetyls

Dual metalloprotease inhibitors. III. utilization of bicyclic and monocyclic diazepinone based mercaptoacetyls

Selective inhibition of urokinase by substituted phenylguanidines: quantitative structure-activity relationship analyses

ChemInform Abstract: N-Formyl Hydroxylamine Containing Dipeptides: Generation of a New Class of Vasopeptidase Inhibitors

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