UB Paderborn / Katalog / Suche / in CDI

Discovery of Imigliptin, a Novel Selective DPP‑4 Inhibitor for the Treatment of Type 2 Diabetes

ACS medicinal chemistry letters, 2014-08, Vol.5 (8), p.921-926

2014

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Human Immunodeficiency Virus Type 1 Mutants Resistant to Nonnucleoside Inhibitors of Reverse Transcriptase Arise in Tissue Culture

Proceedings of the National Academy of Sciences - PNAS, 1991-12, Vol.88 (24), p.11241-11245

1991

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Inhibition of HIV-1 Replication by a Nonnucleoside Reverse Transcriptase Inhibitor

Science (American Association for the Advancement of Science), 1990-12, Vol.250 (4986), p.1411-1413

1990

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Trifluoromethyl group as a pharmacophore: Effect of replacing a CF 3 group on binding and agonist activity of a glucocorticoid receptor ligand

Bioorganic & medicinal chemistry letters, 2005-11, Vol.15 (21), p.4761-4769

2005

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Trifluoromethyl group as a pharmacophore : Effect of replacing a CF3 group on binding and agonist activity of a glucocorticoid receptor ligand

Bioorganic & medicinal chemistry letters, 2005-11, Vol.15 (21), p.4761-4769

2005

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Identification of dissociated non-steroidal glucocorticoid receptor agonists

Bioorganic & medicinal chemistry letters, 2007-09, Vol.17 (18), p.5025-5031

2007

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Substituted 2H-isoquinolin-1-one as potent Rho-Kinase inhibitors. Part 1: Hit-to-lead account

Bioorganic & medicinal chemistry letters, 2010-06, Vol.20 (11), p.3235-3239

2010

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Hit to Lead Account of the Discovery of Bisbenzamide and Related Ureidobenzamide Inhibitors of Rho Kinase

Journal of medicinal chemistry, 2010-01, Vol.53 (2), p.759-777

2010

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Nevirapine resistance mutations of human immunodeficiency virus type 1 selected during therapy

Journal of Virology, 1994-03, Vol.68 (3), p.1660-1666

1994

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Chimeric Human Immunodeficiency Virus Type 1/Type 2 Reverse Transcriptases Display Reversed Sensitivity to Nonnucleoside Analog Inhibitors

Proceedings of the National Academy of Sciences - PNAS, 1991-11, Vol.88 (21), p.9878-9882

1991

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Nonnucleoside inhibitors of HIV-1 reverse transcriptase : nevirapine as prototype drug

AIDS research and human retroviruses, 1992-02, Vol.8 (2), p.145-152

1992

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Steady state kinetics and inhibition of HIV-1 reverse transcriptase by a non-nucleoside dipyridodiazepinone, BI-RG-587, using a heteropolymeric template

Nucleic acids research, 1991-06, Vol.19 (11), p.3035-3039

1991

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Prophylaxis against HIV-1 infection in chimpanzees by nevirapine, a nonnucleoside inhibitor of reverse transcriptase

Nature medicine, 1997-06, Vol.3 (6), p.665-670

1997

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Novel Nonnucleoside Inhibitors of HIV-1 Reverse Transcriptase. 7. 8-Arylethyldipyridodiazepinones as Potent Broad-Spectrum Inhibitors of Wild-Type and Mutant Enzymes

Journal of medicinal chemistry, 1998-07, Vol.41 (16), p.2960-2971

1998

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Novel Nonnucleoside Inhibitors of HIV-1 Reverse Transcriptase. 8. 8-Aryloxymethyl- and 8-Arylthiomethyldipyridodiazepinones

Journal of medicinal chemistry, 1998-07, Vol.41 (16), p.2972-2984

1998

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Amino acid substitutions in HIV-1 reverse transcriptase with corresponding residues from HIV-2. Effect on kinetic constants and inhibition by non-nucleoside analogs

The Journal of biological chemistry, 1993-08, Vol.268 (22), p.16571-16577

1993

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Expression of reverse transcriptase from feline immunodeficiency virus in Escherichia coli

Antimicrobial Agents and Chemotherapy, 1994-02, Vol.38 (2), p.388-391

1994

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Nucleotide Sequence 5′of the Chicken c-myc Coding Region: Localization of a Noncoding Exon That is Absent from myc Transcripts in Most Avian Leukosis Virus-Induced Lymphomas

Proceedings of the National Academy of Sciences - PNAS, 1984-08, Vol.81 (15), p.4697-4701

1984

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Expression of a proteolipid gene from a high-copy-number plasmid confers trifluoperazine resistance to Saccharomyces cerevisiae

Molecular and Cellular Biology, 1990-07, Vol.10 (7), p.3397-3404

1990

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Novel Non-Nucleoside Inhibitors of Human Immunodeficiency Virus Type 1 Reverse Transcriptase. 6. 2-Indol-3-yl- and 2-Azaindol-3-yl- dipyridodiazepinones

Journal of medicinal chemistry, 1997-07, Vol.40 (15), p.2430-2433

1997

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Novel Non-nucleoside Inhibitors of Human Immunodeficiency Virus Type 1 (HIV-1) Reverse Transcriptase. 4. 2-Substituted Dipyridodiazepinones as Potent Inhibitors of Both Wild-Type and Cysteine-181 HIV-1 Reverse Transcriptase Enzymes

Journal of medicinal chemistry, 1995-11, Vol.38 (24), p.4830-4838

1995

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A dominant trifluoperazine resistance gene from Saccharomyces cerevisiae has homology with F0F1 ATP synthase and confers calcium-sensitive growth

Molecular and Cellular Biology, 1988-08, Vol.8 (8), p.3094-3103

1988

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Human immunodeficiency virus type 1 mutants resistant to nonucleoside inhibitors of reverse transcriptase arise in tissue culture

Proceedings of the National Academy of Sciences - PNAS, 1991, Vol.88 (24), p.11241-11245

1991

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Novel non-nucleoside inhibitors of human immunodeficiency virus type 1 (HIV-1) reverse transcriptase. IV: 2-substituted dipyridodiazepinones as potent inhibitors of both wild-type and cysteine-181 HIV-1 reverse transcriptase enzymes

Journal of medicinal chemistry, 1995, Vol.38 (24), p.4830-4838

1995

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STRUCTURE, EXPRESSION, AND TRANSFORMING ACTIVITY OF THE AVIAN C-MYC AND V-MYC GENES (ONCOGENE, DNA SEQUENCE)

SHIH, CHENG-KON

1985

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Discovery of Imigliptin, a Novel Selective DPP‑4 Inhibitor for the Treatment of Type 2 Diabetes

Human Immunodeficiency Virus Type 1 Mutants Resistant to Nonnucleoside Inhibitors of Reverse Transcriptase Arise in Tissue Culture

Inhibition of HIV-1 Replication by a Nonnucleoside Reverse Transcriptase Inhibitor

Trifluoromethyl group as a pharmacophore: Effect of replacing a CF 3 group on binding and agonist activity of a glucocorticoid receptor ligand

Trifluoromethyl group as a pharmacophore : Effect of replacing a CF3 group on binding and agonist activity of a glucocorticoid receptor ligand

Identification of dissociated non-steroidal glucocorticoid receptor agonists

Substituted 2H-isoquinolin-1-one as potent Rho-Kinase inhibitors. Part 1: Hit-to-lead account

Hit to Lead Account of the Discovery of Bisbenzamide and Related Ureidobenzamide Inhibitors of Rho Kinase

Nevirapine resistance mutations of human immunodeficiency virus type 1 selected during therapy

Chimeric Human Immunodeficiency Virus Type 1/Type 2 Reverse Transcriptases Display Reversed Sensitivity to Nonnucleoside Analog Inhibitors

Nonnucleoside inhibitors of HIV-1 reverse transcriptase : nevirapine as prototype drug

Steady state kinetics and inhibition of HIV-1 reverse transcriptase by a non-nucleoside dipyridodiazepinone, BI-RG-587, using a heteropolymeric template

Prophylaxis against HIV-1 infection in chimpanzees by nevirapine, a nonnucleoside inhibitor of reverse transcriptase

Novel Nonnucleoside Inhibitors of HIV-1 Reverse Transcriptase. 7. 8-Arylethyldipyridodiazepinones as Potent Broad-Spectrum Inhibitors of Wild-Type and Mutant Enzymes

Novel Nonnucleoside Inhibitors of HIV-1 Reverse Transcriptase. 8. 8-Aryloxymethyl- and 8-Arylthiomethyldipyridodiazepinones

Amino acid substitutions in HIV-1 reverse transcriptase with corresponding residues from HIV-2. Effect on kinetic constants and inhibition by non-nucleoside analogs

Expression of reverse transcriptase from feline immunodeficiency virus in Escherichia coli

Nucleotide Sequence 5′of the Chicken c-myc Coding Region: Localization of a Noncoding Exon That is Absent from myc Transcripts in Most Avian Leukosis Virus-Induced Lymphomas

Expression of a proteolipid gene from a high-copy-number plasmid confers trifluoperazine resistance to Saccharomyces cerevisiae

Novel Non-Nucleoside Inhibitors of Human Immunodeficiency Virus Type 1 Reverse Transcriptase. 6. 2-Indol-3-yl- and 2-Azaindol-3-yl- dipyridodiazepinones

Novel Non-nucleoside Inhibitors of Human Immunodeficiency Virus Type 1 (HIV-1) Reverse Transcriptase. 4. 2-Substituted Dipyridodiazepinones as Potent Inhibitors of Both Wild-Type and Cysteine-181 HIV-1 Reverse Transcriptase Enzymes

A dominant trifluoperazine resistance gene from Saccharomyces cerevisiae has homology with F0F1 ATP synthase and confers calcium-sensitive growth

Human immunodeficiency virus type 1 mutants resistant to nonucleoside inhibitors of reverse transcriptase arise in tissue culture

Novel non-nucleoside inhibitors of human immunodeficiency virus type 1 (HIV-1) reverse transcriptase. IV: 2-substituted dipyridodiazepinones as potent inhibitors of both wild-type and cysteine-181 HIV-1 reverse transcriptase enzymes

STRUCTURE, EXPRESSION, AND TRANSFORMING ACTIVITY OF THE AVIAN C-MYC AND V-MYC GENES (ONCOGENE, DNA SEQUENCE)

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