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Discovery and Structure−Activity Relationships of Trisubstituted Pyrimidines/Pyridines as Novel Calcium-Sensing Receptor Antagonists

Journal of medicinal chemistry, 2009-02, Vol.52 (4), p.1204-1208

2009

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A Homogeneous Enzyme Fragment Complementation Cyclic AMP Screen for GPCR Agonists

SLAS discovery, 2002-12, Vol.7 (6), p.515-525

2002

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Muraglitazar, a Novel Dual (α/γ) Peroxisome Proliferator–Activated Receptor Activator, Improves Diabetes and Other Metabolic Abnormalities and Preserves β-Cell Function in db/db Mice

Diabetes (New York, N.Y.), 2006-01, Vol.55 (1), p.240-248

2006

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Discovery of Potent, Orally-Active, and Muscle-Selective Androgen Receptor Modulators Based on an N-Aryl-hydroxybicyclohydantoin Scaffold

Journal of medicinal chemistry, 2006-12, Vol.49 (26), p.7596-7599

2006

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Discovery of Potent and Muscle Selective Androgen Receptor Modulators through Scaffold Modifications

Journal of medicinal chemistry, 2007-06, Vol.50 (13), p.3015-3025

2007

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Characterization of Agonist-Induced Motilin Receptor Trafficking and Its Implications for Tachyphylaxis

Molecular pharmacology, 2006-01, Vol.69 (1), p.109-118

2006

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Cloning and Functional Expression of a cDNA Encoding a Human Type 2 Neuropeptide Y Receptor

The Journal of biological chemistry, 1995-09, Vol.270 (39), p.22661-22664

1995

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Acylation of Acylglycerols by Acyl Coenzyme A:Diacylglycerol Acyltransferase 1 (DGAT1)

The Journal of biological chemistry, 2008-10, Vol.283 (44), p.29802-29811

2008

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Characterization of a new class of selective nonsteroidal progesterone receptor agonists

Steroids, 2004-03, Vol.69 (3), p.201-217

2004

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Acylation of Acylglycerols by Acyl Coenzyme A:Diacylglycerol Acyltransferase 1 (DGAT1): FUNCTIONAL IMPORTANCE OF DGAT1 IN THE INTESTINAL FAT ABSORPTION

The Journal of biological chemistry, 2008-10, Vol.283 (44), p.29802-29811

2008

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Discovery of Clinical Candidate 2‑((2S,6S)‑2-Phenyl-6-hydroxyadamantan-2-yl)-1-(3′-hydroxyazetidin-1-yl)ethanone [BMS-816336], an Orally Active Novel Selective 11β-Hydroxysteroid Dehydrogenase Type 1 Inhibitor

Journal of medicinal chemistry, 2017-06, Vol.60 (12), p.4932-4948

2017

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Pharmacological and X-Ray Structural Characterization of a Novel Selective Androgen Receptor Modulator: Potent Hyperanabolic Stimulation of Skeletal Muscle with Hypostimulation of Prostate in Rats

Endocrinology (Philadelphia), 2007-01, Vol.148 (1), p.4-12

2007

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Discovery of pyridyl sulfonamide 11-beta-hydroxysteroid dehydrogenase type 1 (11β-HSD1) inhibitors for the treatment of metabolic disorders

Bioorganic & medicinal chemistry letters, 2014-11, Vol.24 (21), p.5045-5049

2014

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Synthesis and structure–activity relationship of 2-adamantylmethyl tetrazoles as potent and selective inhibitors of human 11β-hydroxysteroid dehydrogenase type 1 (11β-HSD1)

Bioorganic & medicinal chemistry letters, 2014-01, Vol.24 (2), p.654-660

2014

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Eleven Amino Acid Glucagon-like Peptide-1 Receptor Agonists with Antidiabetic Activity

Journal of medicinal chemistry, 2009-12, Vol.52 (23), p.7788-7799

2009

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Fluorescence Polarization Competition Immunoassay for Tyrosine Kinases

Methods (San Diego, Calif.), 2000-09, Vol.22 (1), p.61-70

Seethala, Ramakrishna

2000

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Generation of 3,8-substituted 1,2,4-triazolopyridines as potent inhibitors of human 11β-hydroxysteroid dehydrogenase type 1 (11β-HSD-1)

Bioorganic & medicinal chemistry letters, 2011-07, Vol.21 (14), p.4146-4149

2011

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Discovery of Clinical Candidate BMS-823778 as an Inhibitor of Human 11β-Hydroxysteroid Dehydrogenase Type 1 (11β-HSD-1)

ACS medicinal chemistry letters, 2018-12, Vol.9 (12), p.1170-1174

2018

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Synthesis and structure-activity relationship of 2-adamantylmethyl tetrazoles as potent and selective inhibitors of human 11I2-hydroxysteroid dehydrogenase type 1 (11I2-HSD1)

Bioorganic & medicinal chemistry letters, 2014-01, Vol.24 (2), p.654-660

2014

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A homogeneous scintillation proximity assay for acetyl coenzyme A carboxylase coupled to fatty acid synthase

Analytical biochemistry, 2006-11, Vol.358 (2), p.257-265

2006

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Identification of a potent and metabolically stable series of fluorinated diphenylpyridylethanamine-based cholesteryl ester transfer protein inhibitors

Bioorganic & medicinal chemistry letters, 2012-10, Vol.22 (20), p.6503-6508

2012

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Optimization of 1,2,4-Triazolopyridines as Inhibitors of Human 11β-Hydroxysteroid Dehydrogenase Type 1 (11β-HSD-1)

ACS medicinal chemistry letters, 2014-07, Vol.5 (7), p.803-808

2014

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A Fluorescence Polarization Competition Immunoassay for Tyrosine Kinases

Analytical biochemistry, 1998-01, Vol.255 (2), p.257-262

1998

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Synthesis and Characterization of 3-Arylquinazolinone and 3-Arylquinazolinethione Derivatives as Selective Estrogen Receptor Beta Modulators

Journal of medicinal chemistry, 2006-04, Vol.49 (8), p.2440-2455

2006

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Discovery and Structure−Activity Relationships of Trisubstituted Pyrimidines/Pyridines as Novel Calcium-Sensing Receptor Antagonists

A Homogeneous Enzyme Fragment Complementation Cyclic AMP Screen for GPCR Agonists

Muraglitazar, a Novel Dual (α/γ) Peroxisome Proliferator–Activated Receptor Activator, Improves Diabetes and Other Metabolic Abnormalities and Preserves β-Cell Function in db/db Mice

Discovery of Potent, Orally-Active, and Muscle-Selective Androgen Receptor Modulators Based on an N-Aryl-hydroxybicyclohydantoin Scaffold

Discovery of Potent and Muscle Selective Androgen Receptor Modulators through Scaffold Modifications

Characterization of Agonist-Induced Motilin Receptor Trafficking and Its Implications for Tachyphylaxis

Cloning and Functional Expression of a cDNA Encoding a Human Type 2 Neuropeptide Y Receptor

Acylation of Acylglycerols by Acyl Coenzyme A:Diacylglycerol Acyltransferase 1 (DGAT1)

Characterization of a new class of selective nonsteroidal progesterone receptor agonists

Acylation of Acylglycerols by Acyl Coenzyme A:Diacylglycerol Acyltransferase 1 (DGAT1): FUNCTIONAL IMPORTANCE OF DGAT1 IN THE INTESTINAL FAT ABSORPTION

Discovery of Clinical Candidate 2‑((2S,6S)‑2-Phenyl-6-hydroxyadamantan-2-yl)-1-(3′-hydroxyazetidin-1-yl)ethanone [BMS-816336], an Orally Active Novel Selective 11β-Hydroxysteroid Dehydrogenase Type 1 Inhibitor

Pharmacological and X-Ray Structural Characterization of a Novel Selective Androgen Receptor Modulator: Potent Hyperanabolic Stimulation of Skeletal Muscle with Hypostimulation of Prostate in Rats

Discovery of pyridyl sulfonamide 11-beta-hydroxysteroid dehydrogenase type 1 (11β-HSD1) inhibitors for the treatment of metabolic disorders

Synthesis and structure–activity relationship of 2-adamantylmethyl tetrazoles as potent and selective inhibitors of human 11β-hydroxysteroid dehydrogenase type 1 (11β-HSD1)

Eleven Amino Acid Glucagon-like Peptide-1 Receptor Agonists with Antidiabetic Activity

Fluorescence Polarization Competition Immunoassay for Tyrosine Kinases

Design and Synthesis of N-[(4-Methoxyphenoxy)carbonyl]-N-[[4-[2-(5- methyl-2-phenyl-4-oxazolyl)ethoxy]phenyl]methyl]glycine [Muraglitazar/BMS-298585], a Novel Peroxisome Proliferator-Activated Receptor α/γ Dual Agonist with Efficacious Glucose and Lipid-Lowering Activities

Generation of 3,8-substituted 1,2,4-triazolopyridines as potent inhibitors of human 11β-hydroxysteroid dehydrogenase type 1 (11β-HSD-1)

Discovery of Clinical Candidate BMS-823778 as an Inhibitor of Human 11β-Hydroxysteroid Dehydrogenase Type 1 (11β-HSD-1)

Synthesis and structure-activity relationship of 2-adamantylmethyl tetrazoles as potent and selective inhibitors of human 11I2-hydroxysteroid dehydrogenase type 1 (11I2-HSD1)

A homogeneous scintillation proximity assay for acetyl coenzyme A carboxylase coupled to fatty acid synthase

Identification of a potent and metabolically stable series of fluorinated diphenylpyridylethanamine-based cholesteryl ester transfer protein inhibitors

Optimization of 1,2,4-Triazolopyridines as Inhibitors of Human 11β-Hydroxysteroid Dehydrogenase Type 1 (11β-HSD-1)

A Fluorescence Polarization Competition Immunoassay for Tyrosine Kinases

Synthesis and Characterization of 3-Arylquinazolinone and 3-Arylquinazolinethione Derivatives as Selective Estrogen Receptor Beta Modulators

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