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Quaternary Diamines as Mass Spectrometry Cleavable Crosslinkers for Protein Interactions

Journal of the American Society for Mass Spectrometry, 2012-02, Vol.23 (2), p.201-212

2012

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Progress in the Synthesis of Canthine Alkaloids and Ring-Truncated Congeners

Journal of natural products (Washington, D.C.), 2013-03, Vol.76 (3), p.455-467

Showalter, H. D. Hollis

2013

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Enediol mimics as inhibitors of the d-arabinose 5-phosphate isomerase (KdsD) from Francisella tularensis

Bioorganic & medicinal chemistry letters, 2011-05, Vol.21 (9), p.2679-2682

2011

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Stereoselective Synthesis of (S)-3-(Methylamino)-3-((R)-pyrrolidin-3-yl)propanenitrile

Journal of organic chemistry, 2012-05, Vol.77 (10), p.4732-4739

2012

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X‑ray Crystal Structures of the Escherichia coli RNA Polymerase in Complex with Benzoxazinorifamycins

Journal of medicinal chemistry, 2013-06, Vol.56 (11), p.4758-4763

2013

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3-Aminoquinazolinediones as a New Class of Antibacterial Agents Demonstrating Excellent Antibacterial Activity Against Wild-Type and Multidrug Resistant Organisms

Journal of medicinal chemistry, 2006-11, Vol.49 (22), p.6435-6438

2006

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Protein cross-linking as a novel mechanism of action of a ubiquitin-activating enzyme inhibitor with anti-tumor activity

Biochemical pharmacology, 2011-08, Vol.82 (4), p.341-349

2011

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Property-based design of a glucosylceramide synthase inhibitor that reduces glucosylceramide in the brain

Journal of lipid research, 2012-02, Vol.53 (2), p.282-291

2012

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Design, synthesis and prostate cancer cell-based studies of analogs of the Rho/MKL1 transcriptional pathway inhibitor, CCG-1423

Bioorganic & medicinal chemistry letters, 2010-01, Vol.20 (2), p.665-672

2010

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Investigation of 3-aryl-pyrimido[5,4-e][1,2,4]triazine-5,7-diones as small molecule antagonists of β-catenin/TCF transcription

Bioorganic & medicinal chemistry letters, 2013-11, Vol.23 (21), p.5814-5820

2013

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A novel synthesis of 3-(substituted)pyrimido[4,5- c]pyridazine-5,7(1 H,6 H)-diones

Tetrahedron letters, 2010-03, Vol.51 (9), p.1326-1328

2010

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Rifamycins – Obstacles and opportunities

Tuberculosis (Edinburgh, Scotland), 2010-03, Vol.90 (2), p.94-118

2010

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Synthesis and structure–activity relationships of novel substituted 8-amino, 8-thio, and 1,8-pyrazole congeners of antitubercular rifamycin S and rifampin

Bioorganic & medicinal chemistry letters, 2011-10, Vol.21 (20), p.6094-6099

2011

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Tyrosine Kinase Inhibitors. 19. 6-Alkynamides of 4-Anilinoquinazolines and 4-Anilinopyrido[3,4-d]pyrimidines as Irreversible Inhibitors of the erbB Family of Tyrosine Kinase Receptors

Journal of medicinal chemistry, 2006-02, Vol.49 (4), p.1475-1485

2006

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3‑Substituted‑N‑(4-Hydroxynaphthalen-1-yl)arylsulfonamides as a Novel Class of Selective Mcl‑1 Inhibitors: Structure-Based Design, Synthesis, SAR, and Biological Evaluation

Journal of medicinal chemistry, 2014-05, Vol.57 (10), p.4111-4133

2014

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Synthesis and Structure−Activity Relationships of Soluble 7-Substituted 3-(3,5-Dimethoxyphenyl)-1,6-naphthyridin-2-amines and Related Ureas as Dual Inhibitors of the Fibroblast Growth Factor Receptor-1 and Vascular Endothelial Growth Factor Receptor-2 Tyrosine Kinases

Journal of medicinal chemistry, 2005-07, Vol.48 (14), p.4628-4653

2005

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An improved synthesis of a fluorophosphonate-polyethylene glycol-biotin probe and its use against competitive substrates

Beilstein journal of organic chemistry, 2013-01, Vol.9 (1), p.89-96

2013

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Synthesis and antibacterial activity of the C-7 side chain of 3-aminoquinazolinediones

Bioorganic & medicinal chemistry letters, 2008-09, Vol.18 (18), p.5087-5090

2008

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Tyrosine Kinase Inhibitors. 18. 6-Substituted 4-Anilinoquinazolines and 4-Anilinopyrido[3,4-d]pyrimidines as Soluble, Irreversible Inhibitors of the Epidermal Growth Factor Receptor

Journal of medicinal chemistry, 2001-02, Vol.44 (3), p.429-440

2001

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A roadmap for drug discovery and its translation to small molecule agents in clinical development for tuberculosis treatment

Tuberculosis (Edinburgh, Scotland), 2008-08, Vol.88, p.S3-S17

2008

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Synthesis and structure–activity relationships of 2-amino-3-carboxy-4-phenylthiophenes as novel atypical protein kinase C inhibitors

Bioorganic & medicinal chemistry letters, 2013-05, Vol.23 (10), p.3034-3038

2013

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Structure-Based Design of Novel Benzoxazinorifamycins with Potent Binding Affinity to Wild-Type and Rifampin-Resistant Mutant Mycobacterium tuberculosis RNA Polymerases

Journal of medicinal chemistry, 2012-04, Vol.55 (8), p.3814-3826

2012

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Tyrosine Kinase Inhibitors. 17. Irreversible Inhibitors of the Epidermal Growth Factor Receptor: 4-(Phenylamino)quinazoline- and 4-(Phenylamino)pyrido[3,2-d]pyrimidine-6-acrylamides Bearing Additional Solubilizing Functions

Journal of medicinal chemistry, 2000-04, Vol.43 (7), p.1380-1397

2000

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Tyrosine Kinase Inhibitors. 14. Structure−Activity Relationships for Methyl- amino-Substituted Derivatives of 4-[(3-Bromophenyl)amino]-6-(methylamino)- pyrido[3,4-d]pyrimidine (PD 158780), a Potent and Specific Inhibitor of the Tyrosine Kinase Activity of Receptors for the EGF Family of Growth Factors

Journal of medicinal chemistry, 1998-02, Vol.41 (5), p.742-751

1998

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Investigating the prevalence of queuine in Escherichia coli RNA via incorporation of the tritium-labeled precursor, preQ(1)

Biochemical and biophysical research communications, 2012-08, Vol.425 (1), p.83-88

2012

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Quaternary Diamines as Mass Spectrometry Cleavable Crosslinkers for Protein Interactions

Progress in the Synthesis of Canthine Alkaloids and Ring-Truncated Congeners

Enediol mimics as inhibitors of the d-arabinose 5-phosphate isomerase (KdsD) from Francisella tularensis

Stereoselective Synthesis of (S)-3-(Methylamino)-3-((R)-pyrrolidin-3-yl)propanenitrile

X‑ray Crystal Structures of the Escherichia coli RNA Polymerase in Complex with Benzoxazinorifamycins

3-Aminoquinazolinediones as a New Class of Antibacterial Agents Demonstrating Excellent Antibacterial Activity Against Wild-Type and Multidrug Resistant Organisms

Protein cross-linking as a novel mechanism of action of a ubiquitin-activating enzyme inhibitor with anti-tumor activity

Property-based design of a glucosylceramide synthase inhibitor that reduces glucosylceramide in the brain

Design, synthesis and prostate cancer cell-based studies of analogs of the Rho/MKL1 transcriptional pathway inhibitor, CCG-1423

Investigation of 3-aryl-pyrimido[5,4-e][1,2,4]triazine-5,7-diones as small molecule antagonists of β-catenin/TCF transcription

A novel synthesis of 3-(substituted)pyrimido[4,5- c]pyridazine-5,7(1 H,6 H)-diones

Rifamycins – Obstacles and opportunities

Synthesis and structure–activity relationships of novel substituted 8-amino, 8-thio, and 1,8-pyrazole congeners of antitubercular rifamycin S and rifampin

Tyrosine Kinase Inhibitors. 19. 6-Alkynamides of 4-Anilinoquinazolines and 4-Anilinopyrido[3,4-d]pyrimidines as Irreversible Inhibitors of the erbB Family of Tyrosine Kinase Receptors

3‑Substituted‑N‑(4-Hydroxynaphthalen-1-yl)arylsulfonamides as a Novel Class of Selective Mcl‑1 Inhibitors: Structure-Based Design, Synthesis, SAR, and Biological Evaluation

Synthesis and Structure−Activity Relationships of Soluble 7-Substituted 3-(3,5-Dimethoxyphenyl)-1,6-naphthyridin-2-amines and Related Ureas as Dual Inhibitors of the Fibroblast Growth Factor Receptor-1 and Vascular Endothelial Growth Factor Receptor-2 Tyrosine Kinases

An improved synthesis of a fluorophosphonate-polyethylene glycol-biotin probe and its use against competitive substrates

Synthesis and antibacterial activity of the C-7 side chain of 3-aminoquinazolinediones

Tyrosine Kinase Inhibitors. 18. 6-Substituted 4-Anilinoquinazolines and 4-Anilinopyrido[3,4-d]pyrimidines as Soluble, Irreversible Inhibitors of the Epidermal Growth Factor Receptor

A roadmap for drug discovery and its translation to small molecule agents in clinical development for tuberculosis treatment

Synthesis and structure–activity relationships of 2-amino-3-carboxy-4-phenylthiophenes as novel atypical protein kinase C inhibitors

Structure-Based Design of Novel Benzoxazinorifamycins with Potent Binding Affinity to Wild-Type and Rifampin-Resistant Mutant Mycobacterium tuberculosis RNA Polymerases

Tyrosine Kinase Inhibitors. 17. Irreversible Inhibitors of the Epidermal Growth Factor Receptor: 4-(Phenylamino)quinazoline- and 4-(Phenylamino)pyrido[3,2-d]pyrimidine-6-acrylamides Bearing Additional Solubilizing Functions

Investigating the prevalence of queuine in Escherichia coli RNA via incorporation of the tritium-labeled precursor, preQ(1)

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