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Facile One-Pot Synthesis of N-Difluoromethyl-2-pyridone Derivatives

Organic letters, 2006-08, Vol.8 (17), p.3805-3808

2006

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Identification of 2-[2-(4-tert-Butylphenyl)ethyl]-N-[4-(3-cyclopentylpropyl)-2-fluorophenyl]-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide as an Orally Active MGAT2 Inhibitor

Chemical and Pharmaceutical Bulletin, 2016/03/01, Vol.64(3), pp.228-238

2016

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Identification of 2-[2-(4-tert-butylphenyl)ethyl]-N-(4-fluorophenyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide (29) as an orally available MGAT2 inhibitor

Bioorganic & medicinal chemistry, 2015-09, Vol.23 (17), p.5922-5931

2015

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Synthesis, Structure−Activity Relationships, and Biological Profiles of a Quinazolinone Class of Histamine H3 Receptor Inverse Agonists

Journal of medicinal chemistry, 2008-08, Vol.51 (15), p.4780-4789

2008

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Morphological and habitat characteristics of settling and newly settled Roughscale Sole Clidoderma asperrimum collected in the coastal waters of northeastern Japan

Fisheries science, 2013-09, Vol.79 (5), p.767-777

2013

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neuropeptide Y Y5 antagonist selectively ameliorates body weight gain and associated parameters in diet-induced obese mice

Proceedings of the National Academy of Sciences - PNAS, 2006-05, Vol.103 (18), p.7154-7158

2006

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Synthesis and evaluation of a spiro-isobenzofuranone class of histamine H3 receptor inverse agonists

Bioorganic & medicinal chemistry letters, 2008-09, Vol.18 (18), p.5101-5106

2008

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5,5-Dimethyl-3-(5-methyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazol-4-yl)-1-phenyl-3-(trifluoromethyl)-3,5,6,7-tetrahydro-1H-indole-2,4-dione, a potent inhibitor for mammalian elongase of long-chain fatty acids family 6: examination of its potential utility as a pharmacological tool

The Journal of pharmacology and experimental therapeutics, 2009-07, Vol.330 (1), p.249

2009

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Discovery of substituted 2,4,4-triarylimidazoline derivatives as potent and selective neuropeptide Y Y5 receptor antagonists

Bioorganic & medicinal chemistry letters, 2009-03, Vol.19 (6), p.1670-1674

2009

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Synthesis, structure–activity relationships, and biological profiles of a dihydrobenzoxathiin class of histamine H3 receptor inverse agonists

Bioorganic & medicinal chemistry letters, 2009-08, Vol.19 (15), p.4232-4236

2009

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Total synthesis of octalactin A via ring-closing metathesis reaction

Tetrahedron letters, 2002-01, Vol.43 (2), p.181-184

2002

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Synthesis and evaluation of a novel 2-azabicyclo[2.2.2]octane class of long chain fatty acid elongase 6 (ELOVL6) inhibitors

Bioorganic & medicinal chemistry, 2009-08, Vol.17 (15), p.5639-5647

2009

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Development of novel 2-[4-(aminoalkoxy)phenyl]-4(3H)-quinazolinone derivatives as potent and selective histamine H3 receptor inverse agonists

Bioorganic & medicinal chemistry letters, 2008-12, Vol.18 (23), p.6041-6045

2008

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Identification and Characterization of a Selective Radioligand for ELOVL6

Journal of biochemistry (Tokyo), 2009-09, Vol.146 (3), p.429-437

2009

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Design and Synthesis of the Potent, Orally Available, Brain-Penetrable Arylpyrazole Class of Neuropeptide Y5 Receptor Antagonists

Journal of medicinal chemistry, 2003-02, Vol.46 (5), p.666-669

2003

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Modulation of neuropeptide Y receptors for the treatment of obesity

Expert opinion on therapeutic patents, 2009-10, Vol.19 (10), p.1401-1415

2009

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Development of a selective and potent radioactive ligand for histamine H3 receptors: A compound potentially useful for receptor occupancy studies

Bioorganic & medicinal chemistry letters, 2009-08, Vol.19 (15), p.4075-4078

2009

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Development of novel 2-[4-(aminoalkoxy)phenyl]-4 (3H)-quinazolinone derivatives as potent and selective histamine H3 receptor inverse agonists

Bioorganic & medicinal chemistry letters, 2008-12, Vol.18 (23), p.6041-6045

2008

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Synthesis and Evaluation of a Novel Indoledione Class of Long Chain Fatty Acid Elongase 6 (ELOVL6) Inhibitors

Journal of medicinal chemistry, 2009-05, Vol.52 (10), p.3142-3145

2009

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(9S)-9-(2-Hydroxy-4,4-dimethyl-6-oxo-1-cyclohexen-1-yl)-3,3-dimethyl-2,3,4,9-tetrahydro-1H-xanthen-1-one, a Selective and Orally Active Neuropeptide Y Y5 Receptor Antagonist

Journal of medicinal chemistry, 2008-08, Vol.51 (15), p.4765-4770

2008

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Synthesis, characterization, and monkey positron emission tomography (PET) studies of [18F]Y1-973, a PET tracer for the neuropeptide Y Y1 receptor

NeuroImage (Orlando, Fla.), 2011-02, Vol.54 (4), p.2635-2642

2011

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Synthesis and evaluation of a spiro-isobenzofuranone class of histamine H 3 receptor inverse agonists

Bioorganic & medicinal chemistry letters, 2008-09, Vol.18 (18), p.5101-5106

2008

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Discovery and characterization of a novel potent, selective and orally active inhibitor for mammalian ELOVL6

European journal of pharmacology, 2010-03, Vol.630 (1), p.34-41

2010

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Synthesis and Evaluation of Structurally Constrained Quinazolinone Derivatives as Potent and Selective Histamine H3 Receptor Inverse Agonists

Journal of medicinal chemistry, 2008-11, Vol.51 (21), p.6889-6901

2008

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Inverse agonist histamine H3 receptor PET tracers labelled with carbon-11 or fluorine-18

Synapse (New York, N.Y.), 2009-12, Vol.63 (12), p.1122-1132

2009

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Facile One-Pot Synthesis of N-Difluoromethyl-2-pyridone Derivatives

Identification of 2-[2-(4-tert-Butylphenyl)ethyl]-N-[4-(3-cyclopentylpropyl)-2-fluorophenyl]-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide as an Orally Active MGAT2 Inhibitor

Identification of 2-[2-(4-tert-butylphenyl)ethyl]-N-(4-fluorophenyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide (29) as an orally available MGAT2 inhibitor

Synthesis, Structure−Activity Relationships, and Biological Profiles of a Quinazolinone Class of Histamine H3 Receptor Inverse Agonists

Morphological and habitat characteristics of settling and newly settled Roughscale Sole Clidoderma asperrimum collected in the coastal waters of northeastern Japan

neuropeptide Y Y5 antagonist selectively ameliorates body weight gain and associated parameters in diet-induced obese mice

Synthesis and evaluation of a spiro-isobenzofuranone class of histamine H3 receptor inverse agonists

5,5-Dimethyl-3-(5-methyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazol-4-yl)-1-phenyl-3-(trifluoromethyl)-3,5,6,7-tetrahydro-1H-indole-2,4-dione, a potent inhibitor for mammalian elongase of long-chain fatty acids family 6: examination of its potential utility as a pharmacological tool

Discovery of substituted 2,4,4-triarylimidazoline derivatives as potent and selective neuropeptide Y Y5 receptor antagonists

Synthesis, structure–activity relationships, and biological profiles of a dihydrobenzoxathiin class of histamine H3 receptor inverse agonists

Total synthesis of octalactin A via ring-closing metathesis reaction

Synthesis and evaluation of a novel 2-azabicyclo[2.2.2]octane class of long chain fatty acid elongase 6 (ELOVL6) inhibitors

Development of novel 2-[4-(aminoalkoxy)phenyl]-4(3H)-quinazolinone derivatives as potent and selective histamine H3 receptor inverse agonists

Identification and Characterization of a Selective Radioligand for ELOVL6

Design and Synthesis of the Potent, Orally Available, Brain-Penetrable Arylpyrazole Class of Neuropeptide Y5 Receptor Antagonists

Modulation of neuropeptide Y receptors for the treatment of obesity

Development of a selective and potent radioactive ligand for histamine H3 receptors: A compound potentially useful for receptor occupancy studies

Development of novel 2-[4-(aminoalkoxy)phenyl]-4 (3H)-quinazolinone derivatives as potent and selective histamine H3 receptor inverse agonists

Synthesis and Evaluation of a Novel Indoledione Class of Long Chain Fatty Acid Elongase 6 (ELOVL6) Inhibitors

(9S)-9-(2-Hydroxy-4,4-dimethyl-6-oxo-1-cyclohexen-1-yl)-3,3-dimethyl-2,3,4,9-tetrahydro-1H-xanthen-1-one, a Selective and Orally Active Neuropeptide Y Y5 Receptor Antagonist

Synthesis, characterization, and monkey positron emission tomography (PET) studies of [18F]Y1-973, a PET tracer for the neuropeptide Y Y1 receptor

Synthesis and evaluation of a spiro-isobenzofuranone class of histamine H 3 receptor inverse agonists

Discovery and characterization of a novel potent, selective and orally active inhibitor for mammalian ELOVL6

Synthesis and Evaluation of Structurally Constrained Quinazolinone Derivatives as Potent and Selective Histamine H3 Receptor Inverse Agonists

Inverse agonist histamine H3 receptor PET tracers labelled with carbon-11 or fluorine-18

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