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The Alpha Keto Amide Moiety as a Privileged Motif in Medicinal Chemistry: Current Insights and Emerging Opportunities

Journal of medicinal chemistry, 2021-04, Vol.64 (7), p.3508-3545

2021

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Indol-3-ylglyoxylamide as Privileged Scaffold in Medicinal Chemistry

Pharmaceuticals (Basel, Switzerland), 2023-07, Vol.16 (7), p.997

2023

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An update into the medicinal chemistry of translocator protein (TSPO) ligands

European journal of medicinal chemistry, 2021-01, Vol.209, p.112924-112924, Article 112924

2021

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Multiple Topoisomerase I (TopoI), Topoisomerase II (TopoII) and Tyrosyl-DNA Phosphodiesterase (TDP) inhibitors in the development of anticancer drugs

European journal of pharmaceutical sciences, 2021-01, Vol.156, p.105594, Article 105594

2021

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New antiproliferative agents derived from tricyclic 3,4‐dihydrobenzo[4,5]imidazo[1,2‐a][1,3,5]triazine scaffold: Synthesis and pharmacological effects

Archiv der Pharmazie (Weinheim), 2022-11, Vol.355 (11), p.e2200295-n/a

2022

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New antiproliferative agents derived from tricyclic 3,4‐dihydrobenzoimidazotriazine scaffold: Synthesis and pharmacological effects

Archiv der Pharmazie (Weinheim), 2022-11, Vol.355 (11)

2022

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Alkyl-substituted N-methylaryl-N′-aryl-4-aminobenzamides: A new series of small molecule inhibitors for Wip1 phosphatase

European journal of medicinal chemistry, 2022-12, Vol.243, p.114763-114763, Article 114763

2022

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Novel fluorescent triazinobenzimidazole derivatives as probes for labelling human A1 and A2B adenosine receptor subtypes

Bioorganic & medicinal chemistry, 2018-12, Vol.26 (22), p.5885-5895

2018

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Lead Optimization of 2‑Phenylindolylglyoxylyldipeptide Murine Double Minute (MDM)2/Translocator Protein (TSPO) Dual Inhibitors for the Treatment of Gliomas

Journal of medicinal chemistry, 2016-05, Vol.59 (10), p.4526-4538

2016

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Benzothiopyranoindole- and pyridothiopyranoindole-based antiproliferative agents targeting topoisomerases

European journal of medicinal chemistry, 2019-03, Vol.165, p.46-58

2019

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Prodrug Strategy Extends the Use of Anti-HIV Sulfanylbenzamides for Application In Vivo

ACS pharmacology & translational science, 2024-01, Vol.7 (1), p.259-273

2024

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The structure-activity profile of mercaptobenzamides’ anti-HIV activity suggests that thermodynamics of metabolism is more important than binding affinity to the target

European journal of medicinal chemistry, 2019-09, Vol.178, p.818-837

2019

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Residence Time, a New parameter to Predict Neurosteroidogenic Efficacy of Translocator Protein (TSPO) Ligands: the Case Study of N,N‐Dialkyl‐2‐arylindol‐3‐ylglyoxylamides

ChemMedChem, 2017-08, Vol.12 (16), p.1275-1278

2017

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Toward PET imaging of A2B adenosine receptors: a carbon-11 labeled triazinobenzimidazole tracer: Synthesis and imaging of a new A2B PET tracer

Nuclear medicine and biology, 2016-05, Vol.43 (5), p.309-317

2016

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Toward PET imaging of A2B adenosine receptors: a carbon-11 labeled triazinobenzimidazole tracer

Nuclear medicine and biology, 2016-05, Vol.43 (5), p.309-317

2016

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Towards PET imaging of A2B Adenosine Receptors: a carbon-11 labeled triazinobenzimidazole tracer

Nuclear medicine and biology, 2016

2016

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Novel fluorescent triazinobenzimidazole derivatives as probes for labelling human A 1 and A 2B adenosine receptor subtypes

Bioorganic & medicinal chemistry, 2018-12, Vol.26 (22), p.5885

2018

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Precise 3D modulation of electro-optical parameters during neurotransmitter uncaging experiments with neurons in vitro

Scientific reports, 2020-08, Vol.10 (1), p.13380-13380, Article 13380

2020

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Study of Biophysical Parameters in Rubi-Gaba Uncaging using Non-Linear Photoactivation and Electrophysiology in Cerebellar Granule Cells

Biophysical journal, 2019-02, Vol.116 (3), p.275a-275a

2019

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Neurounina-1, a novel compound that increases Na+/Ca2+ exchanger activity, effectively protects against stroke damage

Molecular pharmacology, 2013-01, Vol.83 (1), p.142

2013

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Neurounina-1, a Novel Compound That Increases Na + /Ca 2+ Exchanger Activity, Effectively Protects against Stroke Damage

Molecular pharmacology, 2013-01, Vol.83 (1), p.142-156

2013

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Trypanosoma cruzi: Molecular characterization of an RNA binding protein differentially expressed in the parasite life cycle

Experimental parasitology, 2007-09, Vol.117 (1), p.99-105

2007

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Different chloride electrochemical gradients across the plasma membrane in subcellular compartments of rat cerebellum granules

Neuroscience letters, 2005-06, Vol.381 (1), p.139-143

2005

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Three-dimensional optical behaviour of a confocal microscope with single illumination and detection pinhole through imaging of subresolution beads

Microscopy research and technique, 1999-04, Vol.45 (2), p.130-131

1999

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Changes in the endoplasmic reticulum structure of Paramecium primaurelia in relation to different cellular physiological states

Journal of photochemistry and photobiology. B, Biology, 2000-01, Vol.54 (1), p.35-42

2000

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The Alpha Keto Amide Moiety as a Privileged Motif in Medicinal Chemistry: Current Insights and Emerging Opportunities

Indol-3-ylglyoxylamide as Privileged Scaffold in Medicinal Chemistry

An update into the medicinal chemistry of translocator protein (TSPO) ligands

Multiple Topoisomerase I (TopoI), Topoisomerase II (TopoII) and Tyrosyl-DNA Phosphodiesterase (TDP) inhibitors in the development of anticancer drugs

New antiproliferative agents derived from tricyclic 3,4‐dihydrobenzo[4,5]imidazo[1,2‐a][1,3,5]triazine scaffold: Synthesis and pharmacological effects

New antiproliferative agents derived from tricyclic 3,4‐dihydrobenzoimidazotriazine scaffold: Synthesis and pharmacological effects

Alkyl-substituted N-methylaryl-N′-aryl-4-aminobenzamides: A new series of small molecule inhibitors for Wip1 phosphatase

Novel fluorescent triazinobenzimidazole derivatives as probes for labelling human A1 and A2B adenosine receptor subtypes

Lead Optimization of 2‑Phenylindolylglyoxylyldipeptide Murine Double Minute (MDM)2/Translocator Protein (TSPO) Dual Inhibitors for the Treatment of Gliomas

Benzothiopyranoindole- and pyridothiopyranoindole-based antiproliferative agents targeting topoisomerases

Prodrug Strategy Extends the Use of Anti-HIV Sulfanylbenzamides for Application In Vivo

The structure-activity profile of mercaptobenzamides’ anti-HIV activity suggests that thermodynamics of metabolism is more important than binding affinity to the target

Residence Time, a New parameter to Predict Neurosteroidogenic Efficacy of Translocator Protein (TSPO) Ligands: the Case Study of N,N‐Dialkyl‐2‐arylindol‐3‐ylglyoxylamides

Toward PET imaging of A2B adenosine receptors: a carbon-11 labeled triazinobenzimidazole tracer: Synthesis and imaging of a new A2B PET tracer

Toward PET imaging of A2B adenosine receptors: a carbon-11 labeled triazinobenzimidazole tracer

Towards PET imaging of A2B Adenosine Receptors: a carbon-11 labeled triazinobenzimidazole tracer

Novel fluorescent triazinobenzimidazole derivatives as probes for labelling human A 1 and A 2B adenosine receptor subtypes

Precise 3D modulation of electro-optical parameters during neurotransmitter uncaging experiments with neurons in vitro

Study of Biophysical Parameters in Rubi-Gaba Uncaging using Non-Linear Photoactivation and Electrophysiology in Cerebellar Granule Cells

Neurounina-1, a novel compound that increases Na+/Ca2+ exchanger activity, effectively protects against stroke damage

Neurounina-1, a Novel Compound That Increases Na + /Ca 2+ Exchanger Activity, Effectively Protects against Stroke Damage

Trypanosoma cruzi: Molecular characterization of an RNA binding protein differentially expressed in the parasite life cycle

Different chloride electrochemical gradients across the plasma membrane in subcellular compartments of rat cerebellum granules

Three-dimensional optical behaviour of a confocal microscope with single illumination and detection pinhole through imaging of subresolution beads

Changes in the endoplasmic reticulum structure of Paramecium primaurelia in relation to different cellular physiological states

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