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Carrageenan-induced Paw Edema in Rat Elicits a Predominant Prostaglandin E2 (PGE2) Response in the Central Nervous System Associated with the Induction of Microsomal PGE2 Synthase-1

The Journal of biological chemistry, 2004-06, Vol.279 (23), p.24866-24872

2004

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The discovery of odanacatib (MK-0822), a selective inhibitor of cathepsin K

Bioorganic & medicinal chemistry, 2008-02, Vol.18 (3), p.923-928

2008

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MF63 [2-(6-chloro-1H-phenanthro[9,10-d]imidazol-2-yl)-isophthalonitrile], a selective microsomal prostaglandin E synthase-1 inhibitor, relieves pyresis and pain in preclinical models of inflammation

The Journal of pharmacology and experimental therapeutics, 2008-09, Vol.326 (3), p.754-763

2008

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Cyclooxygenase-2 promotes early atherosclerotic lesion formation in LDL receptor-deficient mice

Circulation (New York, N.Y.), 2002-04, Vol.105 (15), p.1816-1823

2002

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Prostacyclin antagonism reduces pain and inflammation in rodent models of hyperalgesia and chronic arthritis

The Journal of pharmacology and experimental therapeutics, 2006-12, Vol.319 (3), p.1043-1050

2006

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A High Level of Cyclooxygenase-2 Inhibitor Selectivity is Associated with a Reduced Interference of Platelet Cyclooxygenase-1 Inactivation by Aspirin

Proceedings of the National Academy of Sciences - PNAS, 2001-12, Vol.98 (25), p.14583-14588

2001

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Cloning, Expression, and Up-regulation of Inducible Rat Prostaglandin E Synthase during Lipopolysaccharide-induced Pyresis and Adjuvant-induced Arthritis

The Journal of biological chemistry, 2001-02, Vol.276 (6), p.4469-4475

2001

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Effect of Cathepsin K Inhibitor Basicity on in Vivo Off-Target Activities

Molecular pharmacology, 2008-01, Vol.73 (1), p.147-156

2008

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Inhibition of the Activation of Multiple Serine Proteases with a Cathepsin C Inhibitor Requires Sustained Exposure to Prevent Pro-enzyme Processing

The Journal of biological chemistry, 2007-07, Vol.282 (29), p.20836-20846

2007

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In Vivo Inhibition of Serine Protease Processing Requires a High Fractional Inhibition of Cathepsin C

Molecular pharmacology, 2008-06, Vol.73 (6), p.1857-1865

2008

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Down-regulation of Microsomal Prostaglandin E₂ Synthase-1 in Adipose Tissue by High-fat Feeding

Obesity (Silver Spring, Md.), 2007, Vol.15 (1), p.60-68

2007

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Cyclo-oxygenase-2 contributes to constitutive prostanoid production in rat kidney and brain

Biochemical journal, 2005-11, Vol.391 (Pt 3), p.561-566

2005

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Inhibitors of the inducible microsomal prostaglandin E2 synthase (mPGES-1) derived from MK-886

Bioorganic & medicinal chemistry letters, 2005-07, Vol.15 (14), p.3352-3355

2005

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Discovery of disubstituted phenanthrene imidazoles as potent, selective and orally active mPGES-1 inhibitors

Bioorganic & medicinal chemistry letters, 2009-10, Vol.19 (20), p.5837-5841

2009

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Deletion of Microsomal Prostaglandin E2 (PGE2) Synthase-1 Reduces Inducible and Basal PGE2 Production and Alters the Gastric Prostanoid Profile

The Journal of biological chemistry, 2004-05, Vol.279 (22), p.23229-23237

2004

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Substituted coumarins as potent 5-lipoxygenase inhibitors

Bioorganic & medicinal chemistry letters, 2006-05, Vol.16 (9), p.2528-2531

2006

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Action of Cyclooxygenase Inhibitors and a Leukotriene Biosynthesis Inhibitor on Cisplatin-Induced Acute and Delayed Emesis in the Ferret

Journal of Pharmacological Sciences, 2007, Vol.103(2), pp.189-200

2007

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Identification and Characterization of a Novel Microsomal Enzyme with Glutathione-dependent Transferase and Peroxidase Activities

The Journal of biological chemistry, 1997-09, Vol.272 (36), p.22934-22939

1997

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Down‐regulation of Microsomal Prostaglandin E 2 Synthase‐1 in Adipose Tissue by High‐fat Feeding

Obesity (Silver Spring, Md.), 2012-09, Vol.15 (1), p.60-68

2012

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Arginine 120 of Prostaglandin G/H Synthase-1 Is Required for the Inhibition by Nonsteroidal Anti-inflammatory Drugs Containing a Carboxylic Acid Moiety

The Journal of biological chemistry, 1995-12, Vol.270 (49), p.29372-29377

1995

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Effects of COX-2 inhibitors on aortic prostacyclin production in cholesterol-fed rabbits

Atherosclerosis, 2001-08, Vol.157 (2), p.393-402

2001

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Down-regulation of Microsomal Prostaglandin E Synthase-1 in Adipose Tissue by High-fat Feeding

Obesity (Silver Spring, Md.), 2007-01, Vol.15 (1), p.60-68

2007

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Purification and characterization of recombinant microsomal prostaglandin E synthase-1

Protein expression and purification, 2002-12, Vol.26 (3), p.489-495

2002

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Evaluation of loxoprofen and its alcohol metabolites for potency and selectivity of inhibition of cyclooxygenase-2

Bioorganic & medicinal chemistry letters, 2004-03, Vol.14 (5), p.1201-1203

2004

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Lysosomotropism of Basic Cathepsin K Inhibitors Contributes to Increased Cellular Potencies against Off-Target Cathepsins and Reduced Functional Selectivity

Journal of medicinal chemistry, 2005-12, Vol.48 (24), p.7535-7543

2005

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Carrageenan-induced Paw Edema in Rat Elicits a Predominant Prostaglandin E2 (PGE2) Response in the Central Nervous System Associated with the Induction of Microsomal PGE2 Synthase-1

The discovery of odanacatib (MK-0822), a selective inhibitor of cathepsin K

MF63 [2-(6-chloro-1H-phenanthro[9,10-d]imidazol-2-yl)-isophthalonitrile], a selective microsomal prostaglandin E synthase-1 inhibitor, relieves pyresis and pain in preclinical models of inflammation

Cyclooxygenase-2 promotes early atherosclerotic lesion formation in LDL receptor-deficient mice

Prostacyclin antagonism reduces pain and inflammation in rodent models of hyperalgesia and chronic arthritis

A High Level of Cyclooxygenase-2 Inhibitor Selectivity is Associated with a Reduced Interference of Platelet Cyclooxygenase-1 Inactivation by Aspirin

Cloning, Expression, and Up-regulation of Inducible Rat Prostaglandin E Synthase during Lipopolysaccharide-induced Pyresis and Adjuvant-induced Arthritis

Effect of Cathepsin K Inhibitor Basicity on in Vivo Off-Target Activities

Inhibition of the Activation of Multiple Serine Proteases with a Cathepsin C Inhibitor Requires Sustained Exposure to Prevent Pro-enzyme Processing

In Vivo Inhibition of Serine Protease Processing Requires a High Fractional Inhibition of Cathepsin C

Down-regulation of Microsomal Prostaglandin E₂ Synthase-1 in Adipose Tissue by High-fat Feeding

Cyclo-oxygenase-2 contributes to constitutive prostanoid production in rat kidney and brain

Inhibitors of the inducible microsomal prostaglandin E2 synthase (mPGES-1) derived from MK-886

Discovery of disubstituted phenanthrene imidazoles as potent, selective and orally active mPGES-1 inhibitors

Deletion of Microsomal Prostaglandin E2 (PGE2) Synthase-1 Reduces Inducible and Basal PGE2 Production and Alters the Gastric Prostanoid Profile

Substituted coumarins as potent 5-lipoxygenase inhibitors

Action of Cyclooxygenase Inhibitors and a Leukotriene Biosynthesis Inhibitor on Cisplatin-Induced Acute and Delayed Emesis in the Ferret

Identification and Characterization of a Novel Microsomal Enzyme with Glutathione-dependent Transferase and Peroxidase Activities

Down‐regulation of Microsomal Prostaglandin E 2 Synthase‐1 in Adipose Tissue by High‐fat Feeding

Arginine 120 of Prostaglandin G/H Synthase-1 Is Required for the Inhibition by Nonsteroidal Anti-inflammatory Drugs Containing a Carboxylic Acid Moiety

Effects of COX-2 inhibitors on aortic prostacyclin production in cholesterol-fed rabbits

Down-regulation of Microsomal Prostaglandin E Synthase-1 in Adipose Tissue by High-fat Feeding

Purification and characterization of recombinant microsomal prostaglandin E synthase-1

Evaluation of loxoprofen and its alcohol metabolites for potency and selectivity of inhibition of cyclooxygenase-2

Lysosomotropism of Basic Cathepsin K Inhibitors Contributes to Increased Cellular Potencies against Off-Target Cathepsins and Reduced Functional Selectivity

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