UB Paderborn / Katalog / Suche / in CDI

1 – 25 von 43

Sortiert nach

Targeting the nicotinic alpha7 acetylcholine receptor to enhance cognition in disease

Biochemical pharmacology, 2011-10, Vol.82 (8), p.891-903

2011

Volltextzugriff (PDF)

Distribution of kainate receptor subunit mRNAs in human hippocampus, neocortex and cerebellum, and bilateral reduction of hippocampal GluR6 and KA2 transcripts in schizophrenia

Brain research, 1997-03, Vol.751 (2), p.217-231

1997

Volltextzugriff (PDF)

Determination of key amino acids implicated in the actions of allosteric modulation by 3,3′-difluorobenzaldazine on rat mGlu5 receptors

European journal of pharmacology, 2006-01, Vol.529 (1), p.95-104

2006

Volltextzugriff (PDF)

Discovery of the imidazo[1,5-α][1,2,4].triazolo[1,5-d][1,4]benzodiazepine scaffold as a novel, potent and selective GABAA α5 inverse agonist series

Bioorganic & medicinal chemistry letters, 2009-10, Vol.19 (19), p.5746-5752

2009

Volltextzugriff (PDF)

Fenobam: a clinically validated nonbenzodiazepine anxiolytic is a potent, selective, and noncompetitive mGlu5 receptor antagonist with inverse agonist activity

The Journal of pharmacology and experimental therapeutics, 2005-11, Vol.315 (2), p.711

2005

Volltextzugriff (PDF)

Influence of the 5-HT6 Receptor on Acetylcholine Release in the Cortex: Pharmacological Characterization of 4-(2-Bromo-6-pyrrolidin-1-ylpyridine-4-sulfonyl)phenylamine, a Potent and Selective 5-HT6 Receptor Antagonist

Journal of medicinal chemistry, 2003-03, Vol.46 (7), p.1273-1276

2003

Volltextzugriff (PDF)

Characterization of iodoacetate-mediated neurotoxicity in vitro using primary cultures of rat cerebellar granule cells

Free radical biology & medicine, 2000-01, Vol.28 (1), p.102-107

2000

Volltextzugriff (PDF)

Mutational Analysis and Molecular Modeling of the Binding Pocket of the Metabotropic Glutamate 5 Receptor Negative Modulator 2-Methyl-6-(phenylethynyl)-pyridine

Molecular pharmacology, 2003-10, Vol.64 (4), p.823-832

2003

Volltextzugriff (PDF)

Comparison of the binding pockets of two chemically unrelated allosteric antagonists of the mGlu5 receptor and identification of crucial residues involved in the inverse agonism of MPEP

Journal of neurochemistry, 2006-07, Vol.98 (2), p.601-615

2006

Volltextzugriff (PDF)

The effect of chronic haloperidol treatment on glutamate receptor subunit (GluR1, GluR2, KA1, KA2, NR1) mRNAs and glutamate binding protein mRNA in rat forebrain

Neuroscience letters, 1996-07, Vol.212 (3), p.163-166

1996

Volltextzugriff (PDF)

Agonist-induced functional desensitization of recombinant human 5-HT2 receptors expressed in CHO-K1 cells22Abbreviations: 5-HT, 5-hydroxytryptamine; CHO, Chinese hamster ovary; PI, phosphoinositide; FLIPR, fluorimetric imaging plate reader; mCPP, m-chlorophenylpiperazine; DOI, 2,5-dimethoxy-4-iodoamphetamine hydrobromide, GPCR, G-protein-coupled receptor; and PCR, polymerase chain reaction

Biochemical pharmacology, 2001-08, Vol.62 (4), p.431-438

2001

Volltextzugriff (PDF)

An Automated System for the Analysis of G Protein-Coupled Receptor Transmembrane Binding Pockets: Alignment, Receptor-Based Pharmacophores, and Their Application

Journal of chemical information and modeling, 2005-09, Vol.45 (5), p.1324-1336

2005

Volltextzugriff (PDF)

Antagonists of the human adenosine A2A receptor. Part 1 Discovery and synthesis of thieno[3,2-d]pyrimidine-4-methanone derivatives

Bioorganic & medicinal chemistry letters, 2008-05, Vol.18 (9), p.2916-2919

2008

Volltextzugriff (PDF)

G protein-coupled receptor transmembrane binding pockets and their applications in GPCR research and drug discovery: a survey

Current topics in medicinal chemistry, 2011-08, Vol.11 (15), p.1902

2011

Volltextzugriff (PDF)

Glutamate and Parkinson's disease

Molecular neurobiology, 1996-02, Vol.12 (1), p.73-94

1996

Volltextzugriff (PDF)

Anatomy and physiology of glutamate in the CNS

Neurology, 1994-11, Vol.44 (11 Suppl 8), p.S7

1994

Volltextzugriff (PDF)

Metabolite Identification via LC-SPE-NMR-MS of the In vitro Biooxidation Products of a Lead mGlu5 Allosteric Antagonist and Impact on the Improvement of Metabolic Stability in the Series

ChemMedChem, 2008-01, Vol.3 (1), p.136-144

2008

Volltextzugriff (PDF)

GluR1 Glutamate Receptor Subunit Is Regulated Differentially in the Primate Basal Ganglia Following Nigrostriatal Dopamine Denervation

Journal of neurochemistry, 2000-03, Vol.74 (3), p.1166-1174

2000

Volltextzugriff (PDF)

Regional Variations in the Pharmacology of NMDA Receptor Channel Blockers: Implications for Therapeutic Potential

Journal of neurochemistry, 1995-02, Vol.64 (2), p.614-623

1995

Volltextzugriff (PDF)

Inhibition of Succinate Dehydrogenase by Malonic Acid Produces an “Excitotoxic” Lesion in Rat Striatum

Journal of neurochemistry, 1993-09, Vol.61 (3), p.1151-1154

1993

Volltextzugriff (PDF)

Arylmethoxypyridines as novel, potent and orally active mGlu5 receptor antagonists

Bioorganic & medicinal chemistry letters, 2006-04, Vol.16 (7), p.1892-1897

2006

Volltextzugriff (PDF)

Discovery of the imidazo[1,5- a][1,2,4]-triazolo[1,5- d][1,4]benzodiazepine scaffold as a novel, potent and selective GABA A α5 inverse agonist series

Bioorganic & medicinal chemistry letters, 2009, Vol.19 (19), p.5746-5752

2009

Volltextzugriff (PDF)

Polysynaptic regulation of glutamate receptors and mitochondrial enzyme activities in the basal ganglia of rats with unilateral dopamine depletion

The Journal of neuroscience, 1994-11, Vol.14 (11), p.7192-7199

1994

Volltextzugriff (PDF)

3,5-Disubstituted-4-hydroxyphenyls Linked to 3-Hydroxy-2-methyl- 4(1H)-pyridinone: Potent Inhibitors of Lipid Peroxidation and Cell Toxicity

Journal of medicinal chemistry, 2000-07, Vol.43 (15), p.2779-2782

2000

Volltextzugriff (PDF)

Antagonists of the human adenosine A 2A receptor. Part 1: Discovery and synthesis of thieno[3,2- d]pyrimidine-4-methanone derivatives

Bioorganic & medicinal chemistry letters, 2008, Vol.18 (9), p.2916-2919

2008

Volltextzugriff (PDF)

1 – 25 von 43

Suche als RSS-Feed

Suchergebnisse filtern

Filter anzeigen

Nur zeigen

Geprüft (Peer-Review)
(41)
Mit Volltextzugriff
(40)

Publikationsform

Artikel
(43)

Sprache

Englisch
(43)
Japanisch
(9)

Erscheinungsjahr

n.n

Thema

Life Sciences & Biomedicine
(30)
Science & Technology
(30)
Animals
(27)
Biological And Medical Sciences
(24)
Rats
(19)
Humans
(15)
Medical Sciences
(14)
Neurosciences & Neurology
(14)
Pharmacology & Pharmacy
(14)
Neurosciences
(13)
Fundamental And Applied Biological Sciences. Psychology
(10)
Male
(10)
Pharmacology. Drug Treatments
(10)
Rats, Sprague-Dawley
(9)
Autoradiography
(8)
Binding Sites
(8)
Neuropharmacology
(8)
Central Nervous System
(7)
Neurology
(7)
Vertebrates: Nervous System And Sense Organs
(7)

15 weitere anzeigen...

Weniger anzeigen...

Menü

Weitere Dienste

Einstellungen

Targeting the nicotinic alpha7 acetylcholine receptor to enhance cognition in disease

Distribution of kainate receptor subunit mRNAs in human hippocampus, neocortex and cerebellum, and bilateral reduction of hippocampal GluR6 and KA2 transcripts in schizophrenia

Determination of key amino acids implicated in the actions of allosteric modulation by 3,3′-difluorobenzaldazine on rat mGlu5 receptors

Discovery of the imidazo[1,5-α][1,2,4].triazolo[1,5-d][1,4]benzodiazepine scaffold as a novel, potent and selective GABAA α5 inverse agonist series

Fenobam: a clinically validated nonbenzodiazepine anxiolytic is a potent, selective, and noncompetitive mGlu5 receptor antagonist with inverse agonist activity

Influence of the 5-HT6 Receptor on Acetylcholine Release in the Cortex: Pharmacological Characterization of 4-(2-Bromo-6-pyrrolidin-1-ylpyridine-4-sulfonyl)phenylamine, a Potent and Selective 5-HT6 Receptor Antagonist

Characterization of iodoacetate-mediated neurotoxicity in vitro using primary cultures of rat cerebellar granule cells

Mutational Analysis and Molecular Modeling of the Binding Pocket of the Metabotropic Glutamate 5 Receptor Negative Modulator 2-Methyl-6-(phenylethynyl)-pyridine

Comparison of the binding pockets of two chemically unrelated allosteric antagonists of the mGlu5 receptor and identification of crucial residues involved in the inverse agonism of MPEP

The effect of chronic haloperidol treatment on glutamate receptor subunit (GluR1, GluR2, KA1, KA2, NR1) mRNAs and glutamate binding protein mRNA in rat forebrain

An Automated System for the Analysis of G Protein-Coupled Receptor Transmembrane Binding Pockets: Alignment, Receptor-Based Pharmacophores, and Their Application

Antagonists of the human adenosine A2A receptor. Part 1 Discovery and synthesis of thieno[3,2-d]pyrimidine-4-methanone derivatives

G protein-coupled receptor transmembrane binding pockets and their applications in GPCR research and drug discovery: a survey

Glutamate and Parkinson's disease

Anatomy and physiology of glutamate in the CNS

Metabolite Identification via LC-SPE-NMR-MS of the In vitro Biooxidation Products of a Lead mGlu5 Allosteric Antagonist and Impact on the Improvement of Metabolic Stability in the Series

GluR1 Glutamate Receptor Subunit Is Regulated Differentially in the Primate Basal Ganglia Following Nigrostriatal Dopamine Denervation

Regional Variations in the Pharmacology of NMDA Receptor Channel Blockers: Implications for Therapeutic Potential

Inhibition of Succinate Dehydrogenase by Malonic Acid Produces an “Excitotoxic” Lesion in Rat Striatum

Arylmethoxypyridines as novel, potent and orally active mGlu5 receptor antagonists

Discovery of the imidazo[1,5- a][1,2,4]-triazolo[1,5- d][1,4]benzodiazepine scaffold as a novel, potent and selective GABA A α5 inverse agonist series

Polysynaptic regulation of glutamate receptors and mitochondrial enzyme activities in the basal ganglia of rats with unilateral dopamine depletion

3,5-Disubstituted-4-hydroxyphenyls Linked to 3-Hydroxy-2-methyl- 4(1H)-pyridinone: Potent Inhibitors of Lipid Peroxidation and Cell Toxicity

Antagonists of the human adenosine A 2A receptor. Part 1: Discovery and synthesis of thieno[3,2- d]pyrimidine-4-methanone derivatives

Suchergebnisse filtern