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BU08073 a buprenorphine analogue with partial agonist activity at μ‐receptors in vitro but long‐lasting opioid antagonist activity in vivo in mice

British journal of pharmacology, 2015-01, Vol.172 (2), p.668-680

2015

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Activities of mixed NOP and μ‐opioid receptor ligands

British journal of pharmacology, 2008-02, Vol.153 (3), p.609-619

2008

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Small-molecule agonists and antagonists of the opioid receptor-like receptor (ORL1, NOP): ligand-based analysis of structural factors influencing intrinsic activity at NOP

The AAPS journal, 2005-10, Vol.7 (2), p.E345-E352

2005

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A Novel Series of Piperidin-4-yl-1,3-Dihydroindol-2-ones as Agonist and Antagonist Ligands at the Nociceptin Receptor

Journal of medicinal chemistry, 2004-06, Vol.47 (12), p.2973-2976

2004

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Characterization of opiates, neuroleptics, and synthetic analogs at ORL1 and opioid receptors

European journal of pharmacology, 2001-09, Vol.428 (1), p.29-36

2001

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A bifunctional nociceptin and mu opioid receptor agonist is analgesic without opioid side effects in nonhuman primates

Science translational medicine, 2018-08, Vol.10 (456)

2018

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Structural Determinants of Opioid and NOP Receptor Activity in Derivatives of Buprenorphine

Journal of medicinal chemistry, 2011-10, Vol.54 (19), p.6531-6537

2011

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Nociceptin/Orphanin FQ Antagonists Ameliorate the Disease Pathogenesis During Inflammatory Bowel Disease

Clinical immunology (Orlando, Fla.), 2009-01, Vol.131, p.S120-S120

2009

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Design, Chemical Synthesis, and Biological Evaluation of Thiosaccharide Analogues of Morphine- and Codeine-6-Glucuronide

Journal of medicinal chemistry, 2004-11, Vol.47 (23), p.5809-5815

2004

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BU 08073 a buprenorphine analogue with partial agonist activity at μ‐receptors in vitro but long‐lasting opioid antagonist activity in vivo in mice

British journal of pharmacology, 2015-01, Vol.172 (2), p.668-680

2015

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A Novel and Selective Nociceptin Receptor (NOP) Agonist (1‐(1‐((cis)‐4‐isopropylcyclohexyl)piperidin‐4‐yl)‐1H‐indol‐2‐yl)methanol (AT‐312) Decreases Acquisition of Ethanol‐Induced Conditioned Place Preference in Mice

Alcoholism, clinical and experimental research, 2018-02, Vol.42 (2), p.461-471

2018

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Designing bifunctional NOP receptor–mu opioid receptor ligands from NOP receptor-selective scaffolds. Part I

Bioorganic & medicinal chemistry letters, 2013-06, Vol.23 (11), p.3308-3313

2013

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Designing bifunctional NOP receptor–mu opioid receptor ligands from NOP-receptor selective scaffolds. Part II

Bioorganic & medicinal chemistry, 2014-04, Vol.22 (8), p.2508-2516

2014

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Anti‐Parkinsonian and anti‐dyskinetic profiles of two novel potent and selective nociceptin/orphanin FQ receptor agonists

British journal of pharmacology, 2018-03, Vol.175 (5), p.782-796

2018

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Ovarian sex steroid-dependent plasticity of nociceptin/orphanin FQ and opioid modulation of spinal dynorphin release

The Journal of pharmacology and experimental therapeutics, 2001-09, Vol.298 (3), p.1213

2001

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Regulation of transcription of the human prepronociceptin gene by Sp1

Gene, 2002-05, Vol.290 (1), p.45-52

2002

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Comparison of the antinociceptive and antirewarding profiles of novel bifunctional nociceptin receptor/mu-opioid receptor ligands: implications for therapeutic applications

The Journal of pharmacology and experimental therapeutics, 2009-12, Vol.331 (3), p.954-964

2009

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Characterization of the δ-opioid receptor found in SH-SY5Y neuroblastoma cells

European journal of pharmacology, 1997-04, Vol.323 (2), p.261-267

1997

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Structure-activity studies on high affinity NOP-active hexapeptides

The journal of peptide research, 2004-09, Vol.64 (3), p.87-94

2004

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N-terminal modifications leading to peptide ORL1 partial agonists and antagonists

The journal of peptide research, 2003-11, Vol.62 (5), p.191-198

2003

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Discovery of the First Small-Molecule Opioid Pan Antagonist with Nanomolar Affinity at Mu, Delta, Kappa, and Nociceptin Opioid Receptors

ACS chemical neuroscience, 2015-04, Vol.6 (4), p.646-657

2015

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Molecular determinants of benzodiazepine receptor affinities and anticonvulsant activities

Molecular pharmacology, 1989-10, Vol.36 (4), p.589-600

1989

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Activity of new NOP receptor ligands in a rat peripheral mononeuropathy model: Potentiation of morphine anti-allodynic activity by NOP receptor antagonists

European journal of pharmacology, 2009-05, Vol.610 (1), p.49-54

2009

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Structure-activity studies of morphiceptin analogs: receptor binding and molecular determinants of mu-affinity and selectivity

Molecular pharmacology, 1986-06, Vol.29 (6), p.546-553

1986

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Activities of mixed NOP and [mu]-opioid receptor ligands

British journal of pharmacology, 2008-02, Vol.153 (3), p.609

2008

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BU08073 a buprenorphine analogue with partial agonist activity at μ‐receptors in vitro but long‐lasting opioid antagonist activity in vivo in mice

Activities of mixed NOP and μ‐opioid receptor ligands

Small-molecule agonists and antagonists of the opioid receptor-like receptor (ORL1, NOP): ligand-based analysis of structural factors influencing intrinsic activity at NOP

A Novel Series of Piperidin-4-yl-1,3-Dihydroindol-2-ones as Agonist and Antagonist Ligands at the Nociceptin Receptor

Characterization of opiates, neuroleptics, and synthetic analogs at ORL1 and opioid receptors

A bifunctional nociceptin and mu opioid receptor agonist is analgesic without opioid side effects in nonhuman primates

Structural Determinants of Opioid and NOP Receptor Activity in Derivatives of Buprenorphine

Nociceptin/Orphanin FQ Antagonists Ameliorate the Disease Pathogenesis During Inflammatory Bowel Disease

Design, Chemical Synthesis, and Biological Evaluation of Thiosaccharide Analogues of Morphine- and Codeine-6-Glucuronide

BU 08073 a buprenorphine analogue with partial agonist activity at μ‐receptors in vitro but long‐lasting opioid antagonist activity in vivo in mice

A Novel and Selective Nociceptin Receptor (NOP) Agonist (1‐(1‐((cis)‐4‐isopropylcyclohexyl)piperidin‐4‐yl)‐1H‐indol‐2‐yl)methanol (AT‐312) Decreases Acquisition of Ethanol‐Induced Conditioned Place Preference in Mice

Designing bifunctional NOP receptor–mu opioid receptor ligands from NOP receptor-selective scaffolds. Part I

Designing bifunctional NOP receptor–mu opioid receptor ligands from NOP-receptor selective scaffolds. Part II

Anti‐Parkinsonian and anti‐dyskinetic profiles of two novel potent and selective nociceptin/orphanin FQ receptor agonists

Ovarian sex steroid-dependent plasticity of nociceptin/orphanin FQ and opioid modulation of spinal dynorphin release

Regulation of transcription of the human prepronociceptin gene by Sp1

Comparison of the antinociceptive and antirewarding profiles of novel bifunctional nociceptin receptor/mu-opioid receptor ligands: implications for therapeutic applications

Characterization of the δ-opioid receptor found in SH-SY5Y neuroblastoma cells

Structure-activity studies on high affinity NOP-active hexapeptides

N-terminal modifications leading to peptide ORL1 partial agonists and antagonists

Discovery of the First Small-Molecule Opioid Pan Antagonist with Nanomolar Affinity at Mu, Delta, Kappa, and Nociceptin Opioid Receptors

Molecular determinants of benzodiazepine receptor affinities and anticonvulsant activities

Activity of new NOP receptor ligands in a rat peripheral mononeuropathy model: Potentiation of morphine anti-allodynic activity by NOP receptor antagonists

Structure-activity studies of morphiceptin analogs: receptor binding and molecular determinants of mu-affinity and selectivity

Activities of mixed NOP and [mu]-opioid receptor ligands

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