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The pharmacology of TUG-891, a potent and selective agonist of the free fatty acid receptor 4 (FFA4/GPR120), demonstrates both potential opportunity and possible challenges to therapeutic agonism

Molecular pharmacology, 2013-11, Vol.84 (5), p.710-725

2013

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Orexin-1 Receptor-Cannabinoid CB1 Receptor Heterodimerization Results in Both Ligand-dependent and -independent Coordinated Alterations of Receptor Localization and Function

The Journal of biological chemistry, 2006-12, Vol.281 (50), p.38812-38824

2006

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Spatial intensity distribution analysis quantifies the extent and regulation of homodimerization of the secretin receptor

Biochemical journal, 2017-05, Vol.474 (11), p.1879-1895

2017

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Roundabout 1 exists predominantly as a basal dimeric complex and this is unaffected by binding of the ligand Slit2

Biochemical journal, 2014-07, Vol.461 (1), p.61-73

2014

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A Molecular Basis for Selective Antagonist Destabilization of Dopamine D3 Receptor Quaternary Organization

Scientific reports, 2017-05, Vol.7 (1), p.1-17, Article 2134

2017

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The orexin OX1 receptor exists predominantly as a homodimer in the basal state: potential regulation of receptor organization by both agonist and antagonist ligands

Biochemical journal, 2011-10, Vol.439 (1), p.171-183

2011

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Ligand‐induced internalization of the orexin OX1 and cannabinoid CB1 receptors assessed via N‐terminal SNAP and CLIP‐tagging

British journal of pharmacology, 2011-03, Vol.162 (6), p.1439-1452

2011

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Spatial Intensity Distribution Analysis: Studies of G Protein-Coupled Receptor Oligomerisation

Trends in pharmacological sciences (Regular ed.), 2018-02, Vol.39 (2), p.175-186

2018

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Regulation of Oligomeric Organization of the Serotonin 5-Hydroxytryptamine 2C (5-HT2C) Receptor Observed by Spatial Intensity Distribution Analysis

The Journal of biological chemistry, 2015-05, Vol.290 (20), p.12844-12857

2015

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A general method to quantify ligand-driven oligomerization from fluorescence-based images

Nature methods, 2019-06, Vol.16 (6), p.493

2019

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Heteromultimerization of Cannabinoid CB1 Receptor and Orexin OX1 Receptor Generates a Unique Complex in Which Both Protomers Are Regulated by Orexin A

The Journal of biological chemistry, 2011-10, Vol.286 (43), p.37414-37428

2011

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Chemokine receptor CXCR4 oligomerization is disrupted selectively by the antagonist ligand IT1t

The Journal of biological chemistry, 2021-01, Vol.296, p.100139-100139, Article 100139

2021

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Dynamic Regulation of Quaternary Organization of the M1 Muscarinic Receptor by Subtype-selective Antagonist Drugs

The Journal of biological chemistry, 2016-06, Vol.291 (25), p.13132-13146

2016

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The M 1 muscarinic receptor is present in situ as a ligand-regulated mixture of monomers and oligomeric complexes

Proceedings of the National Academy of Sciences - PNAS, 2022-06, Vol.119 (24), p.e2201103119

2022

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The M1 muscarinic receptor is present in situ as a ligand-regulated mixture of monomers and oligomeric complexes

Proceedings of the National Academy of Sciences - PNAS, 2022-06, Vol.119 (24), p.1-e2201103119

2022

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Ligand‐induced internalization of the orexin OX 1 and cannabinoid CB 1 receptors assessed via N‐terminal SNAP and CLIP‐tagging

British journal of pharmacology, 2011-03, Vol.162 (6), p.1439-1452

2011

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Applications of fluorescence and bioluminescence resonance energy transfer to drug discovery at G protein coupled receptors

Analytical and bioanalytical chemistry, 2010-09, Vol.398 (1), p.167-180

2010

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Developing chemical genetic approaches to explore G protein-coupled receptor function: validation of the use of a receptor activated solely by synthetic ligand (RASSL)

Molecular pharmacology, 2011-12, Vol.80 (6), p.1033-1046

2011

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Novel Role for Proteinase-activated Receptor 2 (PAR2) in Membrane Trafficking of Proteinase-activated Receptor 4 (PAR4)

The Journal of biological chemistry, 2012-05, Vol.287 (20), p.16656-16669

2012

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Intramolecular Fluorescence Resonance Energy Transfer (FRET) Sensors of the Orexin OX1 and OX2 Receptors Identify Slow Kinetics of Agonist Activation

The Journal of biological chemistry, 2012-04, Vol.287 (18), p.14937-14949

2012

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Visualization of the activation of the histamine H3 receptor (H3R) using novel fluorescence resonance energy transfer biosensors and their potential application to the study of H3R pharmacology

The FEBS journal, 2018-06, Vol.285 (12), p.2319-2336

2018

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Agonist occupancy of a single monomeric element is sufficient to cause internalization of the dimeric β2-adrenoceptor

Cellular signalling, 2007-09, Vol.19 (9), p.1928-1938

2007

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The protein kinase C inhibitor, Ro-31-7459, is a potent activator of ERK and JNK MAP kinases in HUVECs and yet inhibits cyclic AMP-stimulated SOCS-3 gene induction through inactivation of the transcription factor c-Jun

Cellular signalling, 2012-08, Vol.24 (8), p.1690-1699

2012

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Ligand Regulation of the Quaternary Organization of Cell Surface M3 Muscarinic Acetylcholine Receptors Analyzed by Fluorescence Resonance Energy Transfer (FRET) Imaging and Homogeneous Time-resolved FRET

The Journal of biological chemistry, 2010-07, Vol.285 (30), p.23318-23330

2010

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Oligomeric structure of the α1b-adrenoceptor : Comparisons with rhodopsin

Vision research (Oxford), 2006-12, Vol.46 (27), p.4434-4441

2006

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The pharmacology of TUG-891, a potent and selective agonist of the free fatty acid receptor 4 (FFA4/GPR120), demonstrates both potential opportunity and possible challenges to therapeutic agonism

Orexin-1 Receptor-Cannabinoid CB1 Receptor Heterodimerization Results in Both Ligand-dependent and -independent Coordinated Alterations of Receptor Localization and Function

Spatial intensity distribution analysis quantifies the extent and regulation of homodimerization of the secretin receptor

Roundabout 1 exists predominantly as a basal dimeric complex and this is unaffected by binding of the ligand Slit2

A Molecular Basis for Selective Antagonist Destabilization of Dopamine D3 Receptor Quaternary Organization

The orexin OX1 receptor exists predominantly as a homodimer in the basal state: potential regulation of receptor organization by both agonist and antagonist ligands

Ligand‐induced internalization of the orexin OX1 and cannabinoid CB1 receptors assessed via N‐terminal SNAP and CLIP‐tagging

Spatial Intensity Distribution Analysis: Studies of G Protein-Coupled Receptor Oligomerisation

Regulation of Oligomeric Organization of the Serotonin 5-Hydroxytryptamine 2C (5-HT2C) Receptor Observed by Spatial Intensity Distribution Analysis

A general method to quantify ligand-driven oligomerization from fluorescence-based images

Heteromultimerization of Cannabinoid CB1 Receptor and Orexin OX1 Receptor Generates a Unique Complex in Which Both Protomers Are Regulated by Orexin A

Chemokine receptor CXCR4 oligomerization is disrupted selectively by the antagonist ligand IT1t

Dynamic Regulation of Quaternary Organization of the M1 Muscarinic Receptor by Subtype-selective Antagonist Drugs

The M 1 muscarinic receptor is present in situ as a ligand-regulated mixture of monomers and oligomeric complexes

The M1 muscarinic receptor is present in situ as a ligand-regulated mixture of monomers and oligomeric complexes

Ligand‐induced internalization of the orexin OX 1 and cannabinoid CB 1 receptors assessed via N‐terminal SNAP and CLIP‐tagging

Applications of fluorescence and bioluminescence resonance energy transfer to drug discovery at G protein coupled receptors

Developing chemical genetic approaches to explore G protein-coupled receptor function: validation of the use of a receptor activated solely by synthetic ligand (RASSL)

Novel Role for Proteinase-activated Receptor 2 (PAR2) in Membrane Trafficking of Proteinase-activated Receptor 4 (PAR4)

Intramolecular Fluorescence Resonance Energy Transfer (FRET) Sensors of the Orexin OX1 and OX2 Receptors Identify Slow Kinetics of Agonist Activation

Visualization of the activation of the histamine H3 receptor (H3R) using novel fluorescence resonance energy transfer biosensors and their potential application to the study of H3R pharmacology

Agonist occupancy of a single monomeric element is sufficient to cause internalization of the dimeric β2-adrenoceptor

The protein kinase C inhibitor, Ro-31-7459, is a potent activator of ERK and JNK MAP kinases in HUVECs and yet inhibits cyclic AMP-stimulated SOCS-3 gene induction through inactivation of the transcription factor c-Jun

Ligand Regulation of the Quaternary Organization of Cell Surface M3 Muscarinic Acetylcholine Receptors Analyzed by Fluorescence Resonance Energy Transfer (FRET) Imaging and Homogeneous Time-resolved FRET

Oligomeric structure of the α1b-adrenoceptor : Comparisons with rhodopsin

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