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Synthesis of Sulfonic Acid Derivatives by Oxidative Deprotection of Thiols Using tert-Butyl Hypochlorite

Organic letters, 2013-05, Vol.15 (9), p.2294-2297

2013

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Design, Synthesis, and In Vitro Biological Activities of a Bio-Oxidizable Prodrug to Deliver Both ChEs and DYRK1A Inhibitors for AD Therapy

Molecules (Basel, Switzerland), 2019-04, Vol.24 (7), p.1264

2019

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Donepezil-Based Central Acetylcholinesterase Inhibitors by Means of a “Bio-Oxidizable” Prodrug Strategy: Design, Synthesis, and in Vitro Biological Evaluation

Journal of medicinal chemistry, 2017-07, Vol.60 (13), p.5909-5926

2017

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Dihydroquinoline Carbamate DQS1-02 as a Prodrug of a Potent Acetylcholinesterase Inhibitor for Alzheimer’s Disease Therapy: Multigram-Scale Synthesis, Mechanism Investigations, in Vitro Safety Pharmacology, and Preliminary in Vivo Toxicology Profile

ACS omega, 2018-12, Vol.3 (12), p.18387-18397

2018

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Chemical Delivery System of MIBG to the Central Nervous System: Synthesis, 11C‑Radiosynthesis, and in Vivo Evaluation

ACS medicinal chemistry letters, 2019-03, Vol.10 (3), p.352-357

2019

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Selective Inhibition of Factor Inhibiting Hypoxia-Inducible Factor

Journal of the American Chemical Society, 2005-06, Vol.127 (21), p.7680-7681

2005

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Exploring the synthesis and metal complexation behavior of mono and bis substituted hexaazamacrocyclic cage derivatives

Inorganic chemistry communications, 2017-08, Vol.82, p.48-51

2017

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A technique to determine the thermal stability of uracil and uracil derivatives in a molecular beam

International journal of mass spectrometry, 2016-11, Vol.409, p.73-80

2016

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Palladium-Catalyzed Carbonylation of (Hetero)Aryl, Alkenyl and Allyl Halides by Means of N-Hydroxysuccinimidyl Formate as CO Surrogate

Journal of organic chemistry, 2015-07, Vol.80 (13), p.6537-6544

2015

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Straightforward Access to a New Class of Dual DYRK1A/CLK1 Inhibitors Possessing a Simple Dihydroquinoline Core

Molecules (Basel, Switzerland), 2023-01, Vol.28 (1), p.36

2023

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Access to Highly Enantioenriched Donepezil-like 1,4-Dihydropyridines as Promising Anti-Alzheimer Prodrug Candidates via Enantioselective Tsuji Allylation and Organocatalytic Aza-Ene-Type Domino Reactions

Journal of organic chemistry, 2018-09, Vol.83 (17), p.10231-10240

2018

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Rational design of central selective acetylcholinesterase inhibitors by means of a "bio-oxidisable prodrug" strategy

Organic & biomolecular chemistry, 2009-06, Vol.7 (12), p.2612-8

2009

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DMAP-Organocatalyzed O-Silyl-O-(or C-)-Benzoyl Interconversions by Means of Benzoyl Fluoride

Synlett, 2007-02, Vol.2007 (3), p.0381-0386

2007

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Novel donepezil-like N-benzylpyridinium salt derivatives as AChE inhibitors and their corresponding dihydropyridine “bio-oxidizable” prodrugs: Synthesis, biological evaluation and structure-activity relationship

European journal of medicinal chemistry, 2018-02, Vol.145, p.165-190

2018

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Modular Synthesis of Benzene-Centered Porphyrin Trimers and a Dendritic Porphyrin Hexamer

Journal of organic chemistry, 1998-08, Vol.63 (16), p.5568-5580

1998

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Rational design of carbamate-based dual binding site and central AChE inhibitors by a “biooxidisable” prodrug approach: Synthesis, in vitro evaluation and docking studies

European journal of medicinal chemistry, 2018-07, Vol.155, p.171-182

2018

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Amine Capture Strategy for Peptide Bond Formation by Means of Quinolinium Thioester Salts

Journal of the American Chemical Society, 2005-11, Vol.127 (45), p.15668-15669

2005

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Design, synthesis and preliminary biological evaluation of rivastigmine-INDY hybrids as multitarget ligands against Alzheimer's disease by targeting butyrylcholinesterase and DYRK1A/CLK1 kinases

RSC medicinal chemistry, 2024-03, Vol.15 (3), p.963-98

2024

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Delivering FLT to the Central Nervous System by Means of a Promising Targeting System: Synthesis, [11C]Radiosynthesis, and in Vivo Evaluation

ACS chemical neuroscience, 2017-11, Vol.8 (11), p.2457-2467

2017

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Dihydroquinoline Carbamate Derivatives as “Bio-oxidizable” Prodrugs for Brain Delivery of Acetylcholinesterase Inhibitors: [11C] Radiosynthesis and Biological Evaluation

ACS chemical neuroscience, 2015-05, Vol.6 (5), p.737-744

2015

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Investigations of Electronic Energy Transfer Dynamics in Multiporphyrin Arrays

The journal of physical chemistry. A, Molecules, spectroscopy, kinetics, environment, & general theory, 1999-07, Vol.103 (30), p.5858-5870

1999

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Access to Highly Enantioenriched Donepezil-like 1,4-Dihydropyridines as Promising Anti-Alzheimer Prodrug Candidates via Enantioselective Tsuji Allylation and Organocatalytic Aza-Ene-Type Domino Reactions

Journal of organic chemistry, 2018-07, Vol.83 (17), p.10231-10240

2018

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Chemical Delivery System of MIBG to the Central Nervous System: Synthesis, 11 C-Radiosynthesis, and in Vivo Evaluation

ACS medicinal chemistry letters, 2019-03, Vol.10 (3), p.352-357

2019

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New developments in redox chemical delivery systems by means of 1,4-dihydroquinoline-based targetor: Application to galantamine delivery to the brain

European journal of medicinal chemistry, 2014-06, Vol.81, p.218-226

2014

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The 1.5-A structure of Chryseobacterium meningosepticum zinc beta-lactamase in complex with the inhibitor, D-captopril

The Journal of biological chemistry, 2003-06, Vol.278 (26), p.23868-23873

2003

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Synthesis of Sulfonic Acid Derivatives by Oxidative Deprotection of Thiols Using tert-Butyl Hypochlorite

Design, Synthesis, and In Vitro Biological Activities of a Bio-Oxidizable Prodrug to Deliver Both ChEs and DYRK1A Inhibitors for AD Therapy

Donepezil-Based Central Acetylcholinesterase Inhibitors by Means of a “Bio-Oxidizable” Prodrug Strategy: Design, Synthesis, and in Vitro Biological Evaluation

Dihydroquinoline Carbamate DQS1-02 as a Prodrug of a Potent Acetylcholinesterase Inhibitor for Alzheimer’s Disease Therapy: Multigram-Scale Synthesis, Mechanism Investigations, in Vitro Safety Pharmacology, and Preliminary in Vivo Toxicology Profile

Chemical Delivery System of MIBG to the Central Nervous System: Synthesis, 11C‑Radiosynthesis, and in Vivo Evaluation

Selective Inhibition of Factor Inhibiting Hypoxia-Inducible Factor

Exploring the synthesis and metal complexation behavior of mono and bis substituted hexaazamacrocyclic cage derivatives

A technique to determine the thermal stability of uracil and uracil derivatives in a molecular beam

Palladium-Catalyzed Carbonylation of (Hetero)Aryl, Alkenyl and Allyl Halides by Means of N-Hydroxysuccinimidyl Formate as CO Surrogate

Straightforward Access to a New Class of Dual DYRK1A/CLK1 Inhibitors Possessing a Simple Dihydroquinoline Core

Access to Highly Enantioenriched Donepezil-like 1,4-Dihydropyridines as Promising Anti-Alzheimer Prodrug Candidates via Enantioselective Tsuji Allylation and Organocatalytic Aza-Ene-Type Domino Reactions

Rational design of central selective acetylcholinesterase inhibitors by means of a "bio-oxidisable prodrug" strategy

DMAP-Organocatalyzed O-Silyl-O-(or C-)-Benzoyl Interconversions by Means of Benzoyl Fluoride

Novel donepezil-like N-benzylpyridinium salt derivatives as AChE inhibitors and their corresponding dihydropyridine “bio-oxidizable” prodrugs: Synthesis, biological evaluation and structure-activity relationship

Modular Synthesis of Benzene-Centered Porphyrin Trimers and a Dendritic Porphyrin Hexamer

Rational design of carbamate-based dual binding site and central AChE inhibitors by a “biooxidisable” prodrug approach: Synthesis, in vitro evaluation and docking studies

Amine Capture Strategy for Peptide Bond Formation by Means of Quinolinium Thioester Salts

Design, synthesis and preliminary biological evaluation of rivastigmine-INDY hybrids as multitarget ligands against Alzheimer's disease by targeting butyrylcholinesterase and DYRK1A/CLK1 kinases

Delivering FLT to the Central Nervous System by Means of a Promising Targeting System: Synthesis, [11C]Radiosynthesis, and in Vivo Evaluation

Dihydroquinoline Carbamate Derivatives as “Bio-oxidizable” Prodrugs for Brain Delivery of Acetylcholinesterase Inhibitors: [11C] Radiosynthesis and Biological Evaluation

Investigations of Electronic Energy Transfer Dynamics in Multiporphyrin Arrays

Access to Highly Enantioenriched Donepezil-like 1,4-Dihydropyridines as Promising Anti-Alzheimer Prodrug Candidates via Enantioselective Tsuji Allylation and Organocatalytic Aza-Ene-Type Domino Reactions

Chemical Delivery System of MIBG to the Central Nervous System: Synthesis, 11 C-Radiosynthesis, and in Vivo Evaluation

New developments in redox chemical delivery systems by means of 1,4-dihydroquinoline-based targetor: Application to galantamine delivery to the brain

The 1.5-A structure of Chryseobacterium meningosepticum zinc beta-lactamase in complex with the inhibitor, D-captopril

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