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The SMARCA2/4 ATPase Domain Surpasses the Bromodomain as a Drug Target in SWI/SNF-Mutant Cancers: Insights from cDNA Rescue and PFI-3 Inhibitor Studies

Cancer research (Chicago, Ill.), 2015-09, Vol.75 (18), p.3865-3878

2015

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Structure-Guided Design of IACS-9571, a Selective High-Affinity Dual TRIM24-BRPF1 Bromodomain Inhibitor

Journal of medicinal chemistry, 2016-02, Vol.59 (4), p.1440-1454

2016

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Discovery of IPN60090, a Clinical Stage Selective Glutaminase‑1 (GLS-1) Inhibitor with Excellent Pharmacokinetic and Physicochemical Properties

Journal of medicinal chemistry, 2020-11, Vol.63 (21), p.12957-12977

2020

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Development of small molecule inhibitors of BRPF1 and TRIM24 bromodomains

Drug discovery today. Technologies, 2016-03, Vol.19, p.65-71

Palmer, Wylie S.

2016

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Observed bromodomain flexibility reveals histone peptide- and small molecule ligand-compatible forms of ATAD2

Biochemical journal, 2015-03, Vol.466 (2), p.337-346

2015

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Discovery of Novel PI3-Kinase δ Specific Inhibitors for the Treatment of Rheumatoid Arthritis: Taming CYP3A4 Time-Dependent Inhibition

Journal of medicinal chemistry, 2012-06, Vol.55 (12), p.5887-5900

2012

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Development of novel cellular histone-binding and chromatin-displacement assays for bromodomain drug discovery

Epigenetics & chromatin, 2015-09, Vol.8 (1), p.37-37, Article 37

2015

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Development of amino-pyrimidine inhibitors of c-Jun N-terminal kinase (JNK): Kinase profiling guided optimization of a 1,2,3-benzotriazole lead

Bioorganic & medicinal chemistry letters, 2013-03, Vol.23 (5), p.1486-1492

2013

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Synthesis of Silirenes by Palladium-Catalyzed Transfer of Silylene from Siliranes to Alkynes

Organometallics, 1997-10, Vol.16 (22), p.4824-4827

1997

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Palladium-Catalyzed Reactions of Di-tert-butylsiliranes with Electron-Deficient Alkynes and Investigations of the Catalytic Cycle

Organometallics, 2001-08, Vol.20 (17), p.3691-3697

2001

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Stereospecific Palladium-Catalyzed Reactions of Siliranes with Alkynes

Organometallics, 1997-03, Vol.16 (6), p.1097-1099

1997

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Stereospecific and Regioselective Isocyanide Insertions into Siliranes and Reactions of the Resulting Iminosilacyclobutanes

Journal of organic chemistry, 1999-03, Vol.64 (6), p.1843-1848

1999

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Abstract 1023: Functional genomics reveals dependency on 6-phosphogluconate dehydrogenase in OXPHOS-deficient tumors

Cancer research (Chicago, Ill.), 2016-07, Vol.76 (14_Supplement), p.1023-1023

2016

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Observed bromodomain flexibility reveals histone peptide- and small molecule ligand-compatible forms of ATAD2A

Biochemical journal, 2015-03, Vol.466 (2), p.337-346

2015

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Abstract 3528: The SMARCA2/4 catalytic activity, but not the bromodomain, is a drug target in SWI/SNF mutant cancers

Cancer research (Chicago, Ill.), 2015-08, Vol.75 (15_Supplement), p.3528-3528

2015

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Development of indole/indazole-aminopyrimidines as inhibitors of c-Jun N-terminal kinase (JNK): Optimization for JNK potency and physicochemical properties

Bioorganic & medicinal chemistry letters, 2013-06, Vol.23 (12), p.3565-3569

2013

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N-Arylpiperazinyl-N‘-propylamino Derivatives of Heteroaryl Amides as Functional Uroselective α1-Adrenoceptor Antagonists

Journal of medicinal chemistry, 1997-08, Vol.40 (17), p.2674-2687

1997

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Stereo- and Regioselectivity of Reactions of Siliranes with Aldehydes and Related Substrates

Journal of organic chemistry, 1997-07, Vol.62 (14), p.4737-4745

1997

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Stereo- and Regiochemistry of Aldehyde Insertions into the C-Si Bonds of Siliranes

Journal of the American Chemical Society, 1995-10, Vol.117 (42), p.10575-10576

1995

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Joint Meeting on Medicinal Chemistry in Vienna

Angewandte Chemie (International ed.), 2005-08, Vol.44 (34), p.5364-5366

2005

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Fachtagung medizinische Chemie in Wien

Angewandte Chemie, 2005-08, Vol.117 (34), p.5498-5500

2005

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Fachtagung medizinische Chemie in Wien

Angewandte Chemie, 2005-08, Vol.117 (34), p.5498-5500

2005

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The chemistry of di-tert-butylsiliranes: Investigations of ring-opening, ring-expansion, and silylene transfer reactions to form various organosilanes

Palmer, Wylie Solang

1999

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On the utility of α-heteroatom substituted orthoesters in the Johnson Claisen rearrangement

Tetrahedron letters, 1994-07, Vol.35 (28), p.4951-4954

1994

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The SMARCA2/4 ATPase Domain Surpasses the Bromodomain as a Drug Target in SWI/SNF-Mutant Cancers: Insights from cDNA Rescue and PFI-3 Inhibitor Studies

Structure-Guided Design of IACS-9571, a Selective High-Affinity Dual TRIM24-BRPF1 Bromodomain Inhibitor

Discovery of IPN60090, a Clinical Stage Selective Glutaminase‑1 (GLS-1) Inhibitor with Excellent Pharmacokinetic and Physicochemical Properties

Functional Genomics Reveals Synthetic Lethality between Phosphogluconate Dehydrogenase and Oxidative Phosphorylation

Development of small molecule inhibitors of BRPF1 and TRIM24 bromodomains

Observed bromodomain flexibility reveals histone peptide- and small molecule ligand-compatible forms of ATAD2

Discovery of Novel PI3-Kinase δ Specific Inhibitors for the Treatment of Rheumatoid Arthritis: Taming CYP3A4 Time-Dependent Inhibition

Development of novel cellular histone-binding and chromatin-displacement assays for bromodomain drug discovery

Development of amino-pyrimidine inhibitors of c-Jun N-terminal kinase (JNK): Kinase profiling guided optimization of a 1,2,3-benzotriazole lead

Synthesis of Silirenes by Palladium-Catalyzed Transfer of Silylene from Siliranes to Alkynes

Palladium-Catalyzed Reactions of Di-tert-butylsiliranes with Electron-Deficient Alkynes and Investigations of the Catalytic Cycle

Stereospecific Palladium-Catalyzed Reactions of Siliranes with Alkynes

Stereospecific and Regioselective Isocyanide Insertions into Siliranes and Reactions of the Resulting Iminosilacyclobutanes

Abstract 1023: Functional genomics reveals dependency on 6-phosphogluconate dehydrogenase in OXPHOS-deficient tumors

Observed bromodomain flexibility reveals histone peptide- and small molecule ligand-compatible forms of ATAD2A

Abstract 3528: The SMARCA2/4 catalytic activity, but not the bromodomain, is a drug target in SWI/SNF mutant cancers

Development of indole/indazole-aminopyrimidines as inhibitors of c-Jun N-terminal kinase (JNK): Optimization for JNK potency and physicochemical properties

N-Arylpiperazinyl-N‘-propylamino Derivatives of Heteroaryl Amides as Functional Uroselective α1-Adrenoceptor Antagonists

Stereo- and Regioselectivity of Reactions of Siliranes with Aldehydes and Related Substrates

Stereo- and Regiochemistry of Aldehyde Insertions into the C-Si Bonds of Siliranes

Joint Meeting on Medicinal Chemistry in Vienna

Fachtagung medizinische Chemie in Wien

Fachtagung medizinische Chemie in Wien

The chemistry of di-tert-butylsiliranes: Investigations of ring-opening, ring-expansion, and silylene transfer reactions to form various organosilanes

On the utility of α-heteroatom substituted orthoesters in the Johnson Claisen rearrangement

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