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Development of a Potent Nurr1 Agonist Tool for In Vivo Applications

Journal of medicinal chemistry, 2023-05, Vol.66 (9), p.6391-6402

2023

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Structure-Guided Design of Nurr1 Agonists Derived from the Natural Ligand Dihydroxyindole

Journal of medicinal chemistry, 2023-10, Vol.66 (19), p.13556-13567

2023

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Structural Fusion of Natural and Synthetic Ligand Features Boosts RXR Agonist Potency

Journal of medicinal chemistry, 2023-12, Vol.66 (24), p.16762-16771

2023

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Development of New Photoswitchable Azobenzene Based γ‑Aminobutyric Acid (GABA) Uptake Inhibitors with Distinctly Enhanced Potency upon Photoactivation

Journal of medicinal chemistry, 2018-07, Vol.61 (14), p.6211-6235

2018

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First Photoswitchable Neurotransmitter Transporter Inhibitor: Light-Induced Control of γ‑Aminobutyric Acid Transporter 1 (GAT1) Activity in Mouse Brain

Journal of medicinal chemistry, 2014-08, Vol.57 (15), p.6809-6821

2014

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Synthesis and biological evaluation of fluorescent GAT-ligands based on meso-substituted BODIPY dyes

Medicinal chemistry research, 2020-02, Vol.29 (2), p.301-327

2020

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Asymmetric synthesis of all four stereoisomers of 1-amino-3-hydroxy-cyclopentane-1-carboxylic acid

Tetrahedron, 2015-01, Vol.71 (4), p.686-693

2015

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Novel, highly potent and in vivo active inhibitor of GABA transporter subtype 1 with anticonvulsant, anxiolytic, antidepressant and antinociceptive properties

Neuropharmacology, 2017-02, Vol.113 (Pt A), p.331-342

2017

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Synthesis and biological evaluation of 4-hydroxy-4-(4-methoxyphenyl)-substituted proline and pyrrolidin-2-ylacetic acid derivatives as GABA uptake inhibitors

Bioorganic & medicinal chemistry, 2013-01, Vol.21 (2), p.470-484

2013

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Development of Highly Potent GAT1 Inhibitors: Synthesis of Nipecotic Acid Derivatives by Suzuki-Miyaura Cross-Coupling Reactions

ChemMedChem, 2016-03, Vol.11 (5), p.519-538

2016

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Different Binding Modes of Small and Large Binders of GAT1

ChemMedChem, 2016-03, Vol.11 (5), p.509-518

2016

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Azetidine derivatives as novel γ-aminobutyric acid uptake inhibitors: Synthesis, biological evaluation, and structure–activity relationship

European journal of medicinal chemistry, 2010-06, Vol.45 (6), p.2453-2466

2010

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Development of an (S)-1-{2-[Tris(4-methoxyphenyl)methoxy]ethyl}piperidine-3-carboxylic acid [(S)-SNAP-5114] Carba Analogue Inhibitor for Murine γ-Aminobutyric Acid Transporter Type 4

ChemMedChem, 2012-07, Vol.7 (7), p.1245-1255

2012

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Development of imidazole alkanoic acids as mGAT3 selective GABA uptake inhibitors

European journal of medicinal chemistry, 2011-05, Vol.46 (5), p.1483-1498

2011

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Development of an (S)-1-{2-[Tris(4-methoxyphenyl)methoxy]ethyl}piperidine-3-carboxylic acid [(S)-SNAP-5114] Carba Analogue Inhibitor for Murine [gamma]-Aminobutyric Acid Transporter Type4

ChemMedChem, 2012-07, Vol.7 (7), p.1245

2012

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Asymmetric Synthesis of Pyrido[1,2-c]pyrimidinones

Zeitschrift für Naturforschung. B, A journal of chemical sciences, 2009-06, Vol.64 (6), p.653-661

2009

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Asymmetric Synthesis with 6-tert-Butyl-5-methoxy-6-methyl-3,6-dihydro-2H-1,4-oxazin-2-one as a New Chiral Glycine Equivalent: Preparation of Enantiomerically Pure α-Tertiary and α-Quaternary α-Amino Acids

European journal of organic chemistry, 2003-04, Vol.2003 (7), p.1244-1263

2003

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Generation of chiral N-acylpyridinium ions by means of silyl triflates and their diastereoselective trapping reactions: formation of N-acyldihydropyridines and N-acyldihydropyridones

Tetrahedron, 2002-08, Vol.58 (33), p.6757-6770

2002

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Synthesis and resolution of racemic eliprodil and evaluation of the enantiomers of eliprodil as NMDA receptor antagonists

Bioorganic & medicinal chemistry letters, 2000-06, Vol.10 (12), p.1377-1380

2000

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Asymmetric Synthesis with 6‐ tert ‐Butyl‐5‐methoxy‐6‐methyl‐3,6‐dihydro‐2 H ‐1,4‐oxazin‐2‐one as a New Chiral Glycine Equivalent: Preparation of Enantiomerically Pure α‐Tertiary and α‐Quaternary α‐Amino Acids

European journal of organic chemistry, 2003-03, Vol.2003 (7), p.1244-1263

2003

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Empagliflozin reduces Ca/calmodulin‐dependent kinase II activity in isolated ventricular cardiomyocytes

ESC Heart Failure, 2018-08, Vol.5 (4), p.642-648

2018

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Activation of protein phosphatase 1 by a selective phosphatase disrupting peptide reduces sarcoplasmic reticulum Ca2+ leak in human heart failure

European journal of heart failure, 2018-12, Vol.20 (12), p.1673-1685

2018

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Activation of protein phosphatase 1 by a selective phosphatase disrupting peptide reduces sarcoplasmic reticulum Ca 2+ leak in human heart failure

European journal of heart failure, 2018-12, Vol.20 (12), p.1673-1685

2018

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Sex-dependent alterations of Ca2+ cycling in human cardiac hypertrophy and heart failure

Europace (London, England), 2016-09, Vol.18 (9), p.1440-1448

2016

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Antimicrobial activities and matrix-assisted laser desorption/ionization mass spectrometry of Bacillus isolates from the marine sponge Aplysina aerophoba

Marine biotechnology (New York, N.Y.), 2003-09, Vol.5 (5), p.424-434

2003

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Development of a Potent Nurr1 Agonist Tool for In Vivo Applications

Structure-Guided Design of Nurr1 Agonists Derived from the Natural Ligand Dihydroxyindole

Structural Fusion of Natural and Synthetic Ligand Features Boosts RXR Agonist Potency

Development of New Photoswitchable Azobenzene Based γ‑Aminobutyric Acid (GABA) Uptake Inhibitors with Distinctly Enhanced Potency upon Photoactivation

First Photoswitchable Neurotransmitter Transporter Inhibitor: Light-Induced Control of γ‑Aminobutyric Acid Transporter 1 (GAT1) Activity in Mouse Brain

Synthesis and biological evaluation of fluorescent GAT-ligands based on meso-substituted BODIPY dyes

Asymmetric synthesis of all four stereoisomers of 1-amino-3-hydroxy-cyclopentane-1-carboxylic acid

Novel, highly potent and in vivo active inhibitor of GABA transporter subtype 1 with anticonvulsant, anxiolytic, antidepressant and antinociceptive properties

Synthesis and biological evaluation of 4-hydroxy-4-(4-methoxyphenyl)-substituted proline and pyrrolidin-2-ylacetic acid derivatives as GABA uptake inhibitors

Development of Highly Potent GAT1 Inhibitors: Synthesis of Nipecotic Acid Derivatives by Suzuki-Miyaura Cross-Coupling Reactions

Different Binding Modes of Small and Large Binders of GAT1

Azetidine derivatives as novel γ-aminobutyric acid uptake inhibitors: Synthesis, biological evaluation, and structure–activity relationship

Development of an (S)-1-{2-[Tris(4-methoxyphenyl)methoxy]ethyl}piperidine-3-carboxylic acid [(S)-SNAP-5114] Carba Analogue Inhibitor for Murine γ-Aminobutyric Acid Transporter Type 4

Development of imidazole alkanoic acids as mGAT3 selective GABA uptake inhibitors

Development of an (S)-1-{2-[Tris(4-methoxyphenyl)methoxy]ethyl}piperidine-3-carboxylic acid [(S)-SNAP-5114] Carba Analogue Inhibitor for Murine [gamma]-Aminobutyric Acid Transporter Type4

Asymmetric Synthesis of Pyrido[1,2-c]pyrimidinones

Asymmetric Synthesis with 6-tert-Butyl-5-methoxy-6-methyl-3,6-dihydro-2H-1,4-oxazin-2-one as a New Chiral Glycine Equivalent: Preparation of Enantiomerically Pure α-Tertiary and α-Quaternary α-Amino Acids

Generation of chiral N-acylpyridinium ions by means of silyl triflates and their diastereoselective trapping reactions: formation of N-acyldihydropyridines and N-acyldihydropyridones

Synthesis and resolution of racemic eliprodil and evaluation of the enantiomers of eliprodil as NMDA receptor antagonists

Asymmetric Synthesis with 6‐ tert ‐Butyl‐5‐methoxy‐6‐methyl‐3,6‐dihydro‐2 H ‐1,4‐oxazin‐2‐one as a New Chiral Glycine Equivalent: Preparation of Enantiomerically Pure α‐Tertiary and α‐Quaternary α‐Amino Acids

Empagliflozin reduces Ca/calmodulin‐dependent kinase II activity in isolated ventricular cardiomyocytes

Activation of protein phosphatase 1 by a selective phosphatase disrupting peptide reduces sarcoplasmic reticulum Ca2+ leak in human heart failure

Activation of protein phosphatase 1 by a selective phosphatase disrupting peptide reduces sarcoplasmic reticulum Ca 2+ leak in human heart failure

Sex-dependent alterations of Ca2+ cycling in human cardiac hypertrophy and heart failure

Antimicrobial activities and matrix-assisted laser desorption/ionization mass spectrometry of Bacillus isolates from the marine sponge Aplysina aerophoba

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