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A Fragment-Derived Clinical Candidate for Antagonism of X-Linked and Cellular Inhibitor of Apoptosis Proteins: 1-(6-[(4-Fluorophenyl)methyl]-5-(hydroxymethyl)-3,3-dimethyl-1 H,2 H,3 H-pyrrolo[3,2- b]pyridin-1-yl)-2-[(2 R,5 R)-5-methyl-2-([(3R)-3-methylmorpholin-4-yl]methyl)piperazin-1-yl]ethan-1-one (ASTX660)

Journal of medicinal chemistry, 2018-08, Vol.61 (16), p.7314-7329

2018

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Fragment-Based Approach to the Development of an Orally Bioavailable Lactam Inhibitor of Lipoprotein-Associated Phospholipase A2 (Lp-PLA2)

Journal of medicinal chemistry, 2016-12, Vol.59 (23), p.10738-10749

2016

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Exploitation of a Novel Binding Pocket in Human Lipoprotein-Associated Phospholipase A2 (Lp-PLA2) Discovered through X‑ray Fragment Screening

Journal of medicinal chemistry, 2016-06, Vol.59 (11), p.5356-5367

2016

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Fragment-Based Discovery of Potent and Selective DDR1/2 Inhibitors

ACS medicinal chemistry letters, 2015-07, Vol.6 (7), p.798-803

2015

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Synthesis and evaluation of 3-amino-6-aryl-pyridazines as selective CB2 agonists for the treatment of inflammatory pain

Bioorganic & medicinal chemistry letters, 2010-01, Vol.20 (2), p.465-468

2010

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An unusual methylene aziridine refined in P21/c and the nonstandard setting P21/n

Acta crystallographica. Section C, Crystal structure communications, 2009-12, Vol.65 (12), p.o635-o638

2009

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2-Amino-5-aryl-pyridines as selective CB2 agonists: Synthesis and investigation of structure-activity relationships

Bioorganic & medicinal chemistry letters, 2009-12, Vol.19 (23), p.6578-6581

2009

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Identification of [4-[4-(methylsulfonyl)phenyl]-6-(trifluoromethyl)-2-pyrimidinyl] amines and ethers as potent and selective cyclooxygenase-2 inhibitors

Bioorganic & medicinal chemistry letters, 2009-08, Vol.19 (15), p.4504-4508

2009

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An unusual methylene aziridine refined in P2(1)/c and the nonstandard setting P2(1)/n

Acta crystallographica. Section C, Crystal structure communications, 2009-12, Vol.65 (Pt 12), p.o635-o638

2009

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[1,3]Oxazolo[3,2- b][1,2,4]triazoles: a versatile synthesis of a novel heterocycle

Tetrahedron letters, 2010-07, Vol.51 (30), p.3907-3909

2010

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The acid-mediated intramolecular 1,3-dipolar cycloaddition of derived 2-nitro-1,1-ethenediamines for the synthesis of novel fused bicyclic isoxazoles

Tetrahedron letters, 2010-06, Vol.51 (26), p.3388-3391

2010

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An unusual methylene aziridine refined in P 2 1 / c and the nonstandard setting P 2 1 / n

Acta crystallographica. Section C, Crystal structure communications, 2009-12, Vol.65 (12), p.o635-o638

2009

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Synthesis and evaluation of 3-amino-6-aryl-pyridazines as selective CB sub(2) agonists for the treatment of inflammatory pain

Bioorganic & medicinal chemistry letters, 2010-01, Vol.20 (2), p.465-468

2010

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Synthesis and evaluation of 3-amino-6-aryl-pyridazines as selective CB 2 agonists for the treatment of inflammatory pain

Bioorganic & medicinal chemistry letters, 2010, Vol.20 (2), p.465-468

2010

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ChemInform Abstract: The Acid-Mediated Intramolecular 1,3-Dipolar Cycloaddition of Derived 2-Nitro-1,1-ethenediamines for the Synthesis of Novel Fused Bicyclic Isoxazoles

ChemInform, 2010-10, Vol.41 (42), p.no-no

2010

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2-Amino-5-aryl-pyridines as selective CB 2 agonists: Synthesis and investigation of structure–activity relationships

Bioorganic & medicinal chemistry letters, 2009, Vol.19 (23), p.6578-6581

2009

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Identification of [4-[4-(methylsulfonyl)phenyl]-6-(trifluoromethyl)-2-pyrimi-dinyl] amines and ethers as potent and selective cyclooxygenase-2 inhibitors

Bioorganic & medicinal chemistry letters, 2009, Vol.19 (15), p.4504-4508

2009

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Synthesis and evaluation of 3-amino-6-aryl-pyridazines as selective CB(2) agonists for the treatment of inflammatory pain

Bioorganic & medicinal chemistry letters, 2010-01, Vol.20 (2), p.465-468

2010

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ChemInform Abstract: The Intramolecular Amination of Allenes

ChemInform, 2010-09, Vol.41 (36), p.no-no

2010

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ChemInform Abstract: [1,3]Oxazolo[3,2-b][1,2,4]triazoles: A Versatile Synthesis of a Novel Heterocycle

ChemInform, 2010-11, Vol.41 (46), p.no-no

2010

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Subsidence and carbon loss in drained tropical peatlands

Biogeosciences, 2012-03, Vol.9 (3), p.1053-1071

2012

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Genome-wide Comparative Analysis of Atopic Dermatitis and Psoriasis Gives Insight into Opposing Genetic Mechanisms

American journal of human genetics, 2015-01, Vol.96 (1), p.104-120

2015

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An Immunohistochemical Algorithm for Ovarian Carcinoma Typing

International journal of gynecological pathology, 2016-09, Vol.35 (5), p.430

2016

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DFTB+, a software package for efficient approximate density functional theory based atomistic simulations

The Journal of chemical physics, 2020-03, Vol.152 (12), p.124101-124101

2020

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Fragment-Based Approach to the Development of an Orally Bioavailable Lactam Inhibitor of Lipoprotein-Associated Phospholipase A2 (Lp-PLA2)

Exploitation of a Novel Binding Pocket in Human Lipoprotein-Associated Phospholipase A2 (Lp-PLA2) Discovered through X‑ray Fragment Screening

Fragment-Based Discovery of Potent and Selective DDR1/2 Inhibitors

Synthesis and evaluation of 3-amino-6-aryl-pyridazines as selective CB2 agonists for the treatment of inflammatory pain

An unusual methylene aziridine refined in P21/c and the nonstandard setting P21/n

2-Amino-5-aryl-pyridines as selective CB2 agonists: Synthesis and investigation of structure-activity relationships

Identification of [4-[4-(methylsulfonyl)phenyl]-6-(trifluoromethyl)-2-pyrimidinyl] amines and ethers as potent and selective cyclooxygenase-2 inhibitors

An unusual methylene aziridine refined in P2(1)/c and the nonstandard setting P2(1)/n

[1,3]Oxazolo[3,2- b][1,2,4]triazoles: a versatile synthesis of a novel heterocycle

The acid-mediated intramolecular 1,3-dipolar cycloaddition of derived 2-nitro-1,1-ethenediamines for the synthesis of novel fused bicyclic isoxazoles

An unusual methylene aziridine refined in P 2 1 / c and the nonstandard setting P 2 1 / n

Synthesis and evaluation of 3-amino-6-aryl-pyridazines as selective CB sub(2) agonists for the treatment of inflammatory pain

Synthesis and evaluation of 3-amino-6-aryl-pyridazines as selective CB 2 agonists for the treatment of inflammatory pain

ChemInform Abstract: The Acid-Mediated Intramolecular 1,3-Dipolar Cycloaddition of Derived 2-Nitro-1,1-ethenediamines for the Synthesis of Novel Fused Bicyclic Isoxazoles

2-Amino-5-aryl-pyridines as selective CB 2 agonists: Synthesis and investigation of structure–activity relationships

Identification of [4-[4-(methylsulfonyl)phenyl]-6-(trifluoromethyl)-2-pyrimi-dinyl] amines and ethers as potent and selective cyclooxygenase-2 inhibitors

Synthesis and evaluation of 3-amino-6-aryl-pyridazines as selective CB(2) agonists for the treatment of inflammatory pain

ChemInform Abstract: The Intramolecular Amination of Allenes

ChemInform Abstract: [1,3]Oxazolo[3,2-b][1,2,4]triazoles: A Versatile Synthesis of a Novel Heterocycle

Subsidence and carbon loss in drained tropical peatlands

Genome-wide Comparative Analysis of Atopic Dermatitis and Psoriasis Gives Insight into Opposing Genetic Mechanisms

An Immunohistochemical Algorithm for Ovarian Carcinoma Typing

DFTB+, a software package for efficient approximate density functional theory based atomistic simulations

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