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Pharmacological inhibition of RORγt suppresses the Th17 pathway and alleviates arthritis in vivo

PloS one, 2017-11, Vol.12 (11), p.e0188391-e0188391

2017

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Antagonizing Retinoic Acid-Related-Orphan Receptor Gamma Activity Blocks the T Helper 17/Interleukin-17 Pathway Leading to Attenuated Pro-inflammatory Human Keratinocyte and Skin Responses

Frontiers in immunology, 2019-03, Vol.10, p.577-577

2019

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Linkers and Cleavage Strategies in Solid-Phase Organic Synthesis and Combinatorial Chemistry

Chemical reviews, 2000-06, Vol.100 (6), p.2091-2158

2000

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Design and Synthesis of Selurampanel, a Novel Orally Active and Competitive AMPA Receptor Antagonist

ChemMedChem, 2017-02, Vol.12 (3), p.197-201

2017

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Fear-reducing effects of intra-amygdala neuropeptide Y infusion in animal models of conditioned fear: an NPY Y1 receptor independent effect

Psychopharmacologia, 2009-10, Vol.206 (2), p.291-301

2009

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Retinoic-acid-orphan-receptor-C inhibition suppresses Th17 cells and induces thymic aberrations

JCI insight, 2017-03, Vol.2 (5), p.e91127-e91127

2017

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Design and Synthesis of Selective and Potent Orally Active S1P5 Agonists

ChemMedChem, 2010-10, Vol.5 (10), p.1693-1696

2010

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Concise Synthesis of 1H-Pyrazin-2-ones and 2-Aminopyrazines

Synlett, 2004-09, Vol.2004 (11), p.2031-2033

2004

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Key aspects of the Novartis compound collection enhancement project for the compilation of a comprehensive chemogenomics drug discovery screening collection

Current topics in medicinal chemistry, 2005-01, Vol.5 (4), p.397

2005

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Structural States of RORγt: X‐ray Elucidation of Molecular Mechanisms and Binding Interactions for Natural and Synthetic Compounds

ChemMedChem, 2017-07, Vol.12 (13), p.1014-1021

2017

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Development of Selective, Orally Active GPR4 Antagonists with Modulatory Effects on Nociception, Inflammation, and Angiogenesis

Journal of medicinal chemistry, 2017-05, Vol.60 (9), p.3672-3683

2017

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Optimizing a Weakly Binding Fragment into a Potent RORγt Inverse Agonist with Efficacy in an in Vivo Inflammation Model

Journal of medicinal chemistry, 2018-08, Vol.61 (15), p.6724-6735

2018

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Synthesis and Biological Evaluation of New Triazolo- and Imidazolopyridine RORγt Inverse Agonists

ChemMedChem, 2016-12, Vol.11 (24), p.2640-2648

2016

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Pharmacological inhibition of ROR[gamma]t suppresses the Th17 pathway and alleviates arthritis in vivo.(Research Article)(retinoic acid receptor-related orphan receptor gamma t)

PloS one, 2017-11, Vol.12 (11), p.e0188391

2017

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Linkers and Cleavage Strategies in Solid-Phase Organic Synthesis and Combinatorial Chemistry. (Chem. Rev. 2000, 100, 2091. Published on the Web May 6, 2000)

Chemical reviews, 2000-10, Vol.100 (10), p.3859-3859

2000

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Structural States of ROR[gamma]t: X-ray Elucidation of Molecular Mechanisms and Binding Interactions for Natural and Synthetic Compounds

ChemMedChem, 2017-07, Vol.12 (13), p.1014

2017

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AMPA receptor antagonists: potential therapeutic applications

Recent patents on CNS drug discovery, 2006-11, Vol.1 (3), p.247

2006

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Piperidyl amides as novel, potent and orally active mGlu5 receptor antagonists with anxiolytic-like activity

Bioorganic & medicinal chemistry letters, 2010, Vol.20 (1), p.184-188

2010

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Discovery of 1H-pyrrolo[2,3-c]pyridine-7-carboxamides as novel, allosteric mGluR5 antagonists

Bioorganic & medicinal chemistry letters, 2012-10, Vol.22 (20), p.6454-6459

2012

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Cover Picture: Design and Synthesis of Selurampanel, a Novel Orally Active and Competitive AMPA Receptor Antagonist (ChemMedChem 3/2017)

ChemMedChem, 2017-02, Vol.12 (3), p.196-196

2017

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Synthesis and Biological Evaluation of New Triazolo- and Imidazolopyridine ROR[gamma]t Inverse Agonists

ChemMedChem, 2016-12, Vol.11 (24), p.2640-2648

2016

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Quinazolinedione sulfonamides: A novel class of competitive AMPA receptor antagonists with oral activity

Bioorganic & medicinal chemistry letters, 2011-06, Vol.21 (11), p.3358-3361

2011

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BZM055, an Iodinated Radiotracer Candidate for PET and SPECT Imaging of Myelin and FTY720 Brain Distribution

ChemMedChem, 2011-04, Vol.6 (4), p.667-677

2011

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Synthesis of Functionalized Deuterioallylic Compounds

Journal of organic chemistry, 1999-05, Vol.64 (10), p.3563-3566

1999

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Fluorescence Lifetime-Based Competitive Binding Assays for Measuring the Binding Potency of Protease Inhibitors In Vitro

Journal of biomolecular screening, 2014-07, Vol.19 (6), p.870-877

2014

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Pharmacological inhibition of RORγt suppresses the Th17 pathway and alleviates arthritis in vivo

Antagonizing Retinoic Acid-Related-Orphan Receptor Gamma Activity Blocks the T Helper 17/Interleukin-17 Pathway Leading to Attenuated Pro-inflammatory Human Keratinocyte and Skin Responses

Linkers and Cleavage Strategies in Solid-Phase Organic Synthesis and Combinatorial Chemistry

Design and Synthesis of Selurampanel, a Novel Orally Active and Competitive AMPA Receptor Antagonist

Fear-reducing effects of intra-amygdala neuropeptide Y infusion in animal models of conditioned fear: an NPY Y1 receptor independent effect

Retinoic-acid-orphan-receptor-C inhibition suppresses Th17 cells and induces thymic aberrations

Design and Synthesis of Selective and Potent Orally Active S1P5 Agonists

Concise Synthesis of 1H-Pyrazin-2-ones and 2-Aminopyrazines

Key aspects of the Novartis compound collection enhancement project for the compilation of a comprehensive chemogenomics drug discovery screening collection

Structural States of RORγt: X‐ray Elucidation of Molecular Mechanisms and Binding Interactions for Natural and Synthetic Compounds

Development of Selective, Orally Active GPR4 Antagonists with Modulatory Effects on Nociception, Inflammation, and Angiogenesis

Optimizing a Weakly Binding Fragment into a Potent RORγt Inverse Agonist with Efficacy in an in Vivo Inflammation Model

Synthesis and Biological Evaluation of New Triazolo- and Imidazolopyridine RORγt Inverse Agonists

Pharmacological inhibition of ROR[gamma]t suppresses the Th17 pathway and alleviates arthritis in vivo.(Research Article)(retinoic acid receptor-related orphan receptor gamma t)

Linkers and Cleavage Strategies in Solid-Phase Organic Synthesis and Combinatorial Chemistry. (Chem. Rev. 2000, 100, 2091. Published on the Web May 6, 2000)

Structural States of ROR[gamma]t: X-ray Elucidation of Molecular Mechanisms and Binding Interactions for Natural and Synthetic Compounds

AMPA receptor antagonists: potential therapeutic applications

Piperidyl amides as novel, potent and orally active mGlu5 receptor antagonists with anxiolytic-like activity

Discovery of 1H-pyrrolo[2,3-c]pyridine-7-carboxamides as novel, allosteric mGluR5 antagonists

Cover Picture: Design and Synthesis of Selurampanel, a Novel Orally Active and Competitive AMPA Receptor Antagonist (ChemMedChem 3/2017)

Synthesis and Biological Evaluation of New Triazolo- and Imidazolopyridine ROR[gamma]t Inverse Agonists

Quinazolinedione sulfonamides: A novel class of competitive AMPA receptor antagonists with oral activity

BZM055, an Iodinated Radiotracer Candidate for PET and SPECT Imaging of Myelin and FTY720 Brain Distribution

Synthesis of Functionalized Deuterioallylic Compounds

Fluorescence Lifetime-Based Competitive Binding Assays for Measuring the Binding Potency of Protease Inhibitors In Vitro

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