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A straightforward approach to N -substituted-2 H -indazol-2-amines through reductive cyclization

Tetrahedron letters, 2017-04, Vol.58 (16), p.1633-1635

2017

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Development of High-Specificity Fluorescent Probes to Enable Cannabinoid Type 2 Receptor Studies in Living Cells

Journal of the American Chemical Society, 2020-10, Vol.142 (40), p.16953-16964

2020

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Revealing cytotoxic substructures in molecules using deep learning

Journal of computer-aided molecular design, 2020-07, Vol.34 (7), p.731-746

2020

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Isoform-selective targeting of PI3K: time to consider new opportunities?

Trends in pharmacological sciences (Regular ed.), 2023-09, Vol.44 (9), p.601-621

2023

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Detection of cannabinoid receptor type 2 in native cells and zebrafish with a highly potent, cell-permeable fluorescent probe

Chemical science (Cambridge), 2022-05, Vol.13 (19), p.5539-5545

2022

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Allosteric Inhibition of a Mammalian Lectin

Journal of the American Chemical Society, 2018-11, Vol.140 (44), p.14915-14925

2018

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DOTAM-Based, Targeted, Activatable Fluorescent Probes for the Highly Sensitive and Selective Detection of Cancer Cells

Bioconjugate chemistry, 2021-04, Vol.32 (4), p.702-712

2021

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Enhanced Properties of a Benzimidazole Benzylpyrazole Lysine Demethylase Inhibitor: Mechanism-of-Action, Binding Site Analysis, and Activity in Cellular Models of Prostate Cancer

Journal of medicinal chemistry, 2021-10, Vol.64 (19), p.14266-14282

2021

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Identification of High-Affinity P2Y12 Antagonists Based on a Phenylpyrazole Glutamic Acid Piperazine Backbone

Journal of medicinal chemistry, 2012-10, Vol.55 (20), p.8615-8629

2012

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Discovery of a Novel Series of Tankyrase Inhibitors by a Hybridization Approach

Journal of medicinal chemistry, 2017-12, Vol.60 (24), p.10013-10025

2017

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An Activatable Lanthanide Luminescent Probe for Time‐Gated Detection of Nitroreductase in Live Bacteria

Angewandte Chemie (International ed.), 2020-05, Vol.59 (22), p.8512-8516

International ed. in English, 2020

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Weizhouochrones: Gorgonian-Derived Symmetric Dimers and Their Structure Elucidation Using Anisotropic NMR Combined with DP4+ Probability and CASE-3D

Journal of natural products (Washington, D.C.), 2022-07, Vol.85 (7), p.1730-1737

2022

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A Palladium-Catalyzed Domino Reaction To Access 3‑Amino‑2H‑indazoles from Hydrazines and 2‑Halobenzonitriles

Organic letters, 2020-09, Vol.22 (18), p.7393-7396

2020

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An LPAR5-antagonist that reduces nociception and increases pruriception

Frontiers in pain research (Lausanne, Switzerland), 2022-07, Vol.3

2022

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A General One‐Pot Synthesis of 2H‐Indazoles Using an Organophosphorus–Silane System

Chemistry : a European journal, 2018-06, Vol.24 (36), p.9090-9100

2018

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Probing the Subpockets of Factor Xa Reveals Two Binding Modes for Inhibitors Based on a 2-Carboxyindole Scaffold: A Study Combining Structure-Activity Relationship and X-ray Crystallography

Journal of medicinal chemistry, 2005-07, Vol.48 (14), p.4511-4525

2005

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Preclinical Lead Optimization of a 1,2,4-Triazole Based Tankyrase Inhibitor

Journal of medicinal chemistry, 2020-07, Vol.63 (13), p.6834-6846

2020

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Development of a 1,2,4-Triazole-Based Lead Tankyrase Inhibitor: Part II

Journal of medicinal chemistry, 2021-12, Vol.64 (24), p.17936-17949

2021

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Structure-Based Design of Xanthine-Benzimidazole Derivatives as Novel and Potent Tryptophan Hydroxylase Inhibitors

Journal of medicinal chemistry, 2022-08, Vol.65 (16), p.11126-11149

2022

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Aβ Chronic Exposure Promotes an Activation State of Microglia through Endocannabinoid Signalling Imbalance

International journal of molecular sciences, 2023-04, Vol.24 (7), p.6684

2023

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CellFy: A Cell-Based Fragment Screen against C‑Type Lectins

ACS chemical biology, 2018-12, Vol.13 (12), p.3229-3235

2018

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NMR quality control of fragment libraries for screening

Journal of biomolecular NMR, 2020-11, Vol.74 (10-11), p.555-563

2020

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Identification of the Allosteric Binding Site for Thiazolopyrimidine on the C‑Type Lectin Langerin

ACS chemical biology, 2022-10, Vol.17 (10), p.2728-2733

2022

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From Pyrazolones to Azaindoles: Evolution of Active-Site SHP2 Inhibitors Based on Scaffold Hopping and Bioisosteric Replacement

Journal of medicinal chemistry, 2020-12, Vol.63 (23), p.14780-14804

2020

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A straightforward approach to N -substituted-2 H -indazol-2-amines through reductive cyclization

Development of High-Specificity Fluorescent Probes to Enable Cannabinoid Type 2 Receptor Studies in Living Cells

Revealing cytotoxic substructures in molecules using deep learning

Isoform-selective targeting of PI3K: time to consider new opportunities?

Detection of cannabinoid receptor type 2 in native cells and zebrafish with a highly potent, cell-permeable fluorescent probe

Allosteric Inhibition of a Mammalian Lectin

DOTAM-Based, Targeted, Activatable Fluorescent Probes for the Highly Sensitive and Selective Detection of Cancer Cells

Enhanced Properties of a Benzimidazole Benzylpyrazole Lysine Demethylase Inhibitor: Mechanism-of-Action, Binding Site Analysis, and Activity in Cellular Models of Prostate Cancer

Identification of High-Affinity P2Y12 Antagonists Based on a Phenylpyrazole Glutamic Acid Piperazine Backbone

Discovery of a Novel Series of Tankyrase Inhibitors by a Hybridization Approach

An Activatable Lanthanide Luminescent Probe for Time‐Gated Detection of Nitroreductase in Live Bacteria

Weizhouochrones: Gorgonian-Derived Symmetric Dimers and Their Structure Elucidation Using Anisotropic NMR Combined with DP4+ Probability and CASE-3D

A Palladium-Catalyzed Domino Reaction To Access 3‑Amino‑2H‑indazoles from Hydrazines and 2‑Halobenzonitriles

An LPAR5-antagonist that reduces nociception and increases pruriception

A General One‐Pot Synthesis of 2H‐Indazoles Using an Organophosphorus–Silane System

Probing the Subpockets of Factor Xa Reveals Two Binding Modes for Inhibitors Based on a 2-Carboxyindole Scaffold: A Study Combining Structure-Activity Relationship and X-ray Crystallography

Preclinical Lead Optimization of a 1,2,4-Triazole Based Tankyrase Inhibitor

Development of a 1,2,4-Triazole-Based Lead Tankyrase Inhibitor: Part II

Pentafluorosulfanyl (SF5) as a Superior 19F Magnetic Resonance Reporter Group: Signal Detection and Biological Activity of Teriflunomide Derivatives

Structure-Based Design of Xanthine-Benzimidazole Derivatives as Novel and Potent Tryptophan Hydroxylase Inhibitors

Aβ Chronic Exposure Promotes an Activation State of Microglia through Endocannabinoid Signalling Imbalance

CellFy: A Cell-Based Fragment Screen against C‑Type Lectins

NMR quality control of fragment libraries for screening

Identification of the Allosteric Binding Site for Thiazolopyrimidine on the C‑Type Lectin Langerin

From Pyrazolones to Azaindoles: Evolution of Active-Site SHP2 Inhibitors Based on Scaffold Hopping and Bioisosteric Replacement

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