UB Paderborn / Katalog / Suche / in CDI

Sortiert nach

Einfacher Volltextzugriff von (fast) überall

Installieren Sie die LibKey Nomad-Browsererweiterung und erhalten Sie von vielen Webseiten einfachen Zugriff auf lizenzierte Volltexte oder Open Access Publikationen. Mehr erfahren...

A sting in the tail： the N-terminal domain of the androgen receptor as a drug target

Asian journal of andrology, 2016-09, Vol.18 (5), p.687-694

2016

Volltextzugriff (PDF)

International Union of Basic and Clinical Pharmacology. LXXXVIII. G protein-coupled receptor list: recommendations for new pairings with cognate ligands

Pharmacological reviews, 2013-07, Vol.65 (3), p.967-986

2013

Volltextzugriff (PDF)

Development of a High-Throughput Screening Assay for Small-Molecule Inhibitors of Androgen Receptor Splice Variants

Assay and drug development technologies, 2022-04, Vol.20 (3), p.111-124

2022

Volltextzugriff (PDF)

Enhanced insulin signalling ameliorates C9orf72 hexanucleotide repeat expansion toxicity in Drosophila

eLife, 2021-03, Vol.10

2021

Volltextzugriff (PDF)

Structural Insights into Notum Covalent Inhibition

Journal of medicinal chemistry, 2021-08, Vol.64 (15), p.11354-11363

2021

Volltextzugriff (PDF)

Virtual Screening Directly Identifies New Fragment-Sized Inhibitors of Carboxylesterase Notum with Nanomolar Activity

Journal of medicinal chemistry, 2022-01, Vol.65 (1), p.562-578

2022

Volltextzugriff (PDF)

5‑Phenyl-1,3,4-oxadiazol-2(3H)‑ones Are Potent Inhibitors of Notum Carboxylesterase Activity Identified by the Optimization of a Crystallographic Fragment Screening Hit

Journal of medicinal chemistry, 2020-11, Vol.63 (21), p.12942-12956

2020

Volltextzugriff (PDF)

Design of a Potent, Selective, and Brain-Penetrant Inhibitor of Wnt-Deactivating Enzyme Notum by Optimization of a Crystallographic Fragment Hit

Journal of medicinal chemistry, 2022-05, Vol.65 (10), p.7212-7230

2022

Volltextzugriff (PDF)

Screening of a Custom-Designed Acid Fragment Library Identifies 1‑Phenylpyrroles and 1‑Phenylpyrrolidines as Inhibitors of Notum Carboxylesterase Activity

Journal of medicinal chemistry, 2020-09, Vol.63 (17), p.9464-9483

2020

Volltextzugriff (PDF)

Scaffold-hopping identifies furano[2,3-d]pyrimidine amides as potent Notum inhibitors

Bioorganic & medicinal chemistry letters, 2020-02, Vol.30 (3), p.126751, Article 126751

2020

Volltextzugriff (PDF)

Discovery of 2-phenoxyacetamides as inhibitors of the Wnt-depalmitoleating enzyme NOTUM from an X-ray fragment screen

MedChemComm, 2019-08, Vol.1 (8), p.1361-1369

2019

Volltextzugriff (PDF)

Discovery of 2-phenoxyacetamides as inhibitors of the Wnt-depalmitoleating enzyme NOTUM from an X-ray fragment screen† †This work was first presented at the following international conferences: E. Y. J. Biochemical Society Meeting. Acylation of intracellular and secreted proteins: mechanisms and functional outcomes; 10–12th September 2018; Brighton, UK. P. V. F. EFMC: XXVth International Symposium on Medicinal Chemistry; 2–6th September 2018; Ljubljana, Slovenia. ‡ ‡Electronic supplementary info

MedChemComm, 2019-04, Vol.10 (8), p.1361-1369

2019

Volltextzugriff (PDF)

Chemerin receptors in GtoPdb v.2023.1

IUPHAR/BPS Guide to Pharmacology CITE, 2023-04, Vol.2023 (1)

2023

Volltextzugriff (PDF)

The amino terminal domain of steroid hormone receptors as a novel drug target: identification of small molecule inhibitors

Monaghan, Amy Elizabeth

2016

Volltextzugriff (PDF)

Chemerin receptors in GtoPdb v.2021.3

IUPHAR/BPS Guide to Pharmacology CITE, 2021-09, Vol.2021 (3)

2021

Volltextzugriff (PDF)

Free fatty acid receptors in GtoPdb v.2023.1

IUPHAR/BPS Guide to Pharmacology CITE, 2023-04, Vol.2023 (1)

2023

Volltextzugriff (PDF)

Chemerin receptors (version 2019.4) in the IUPHAR/BPS Guide to Pharmacology Database

IUPHAR/BPS Guide to Pharmacology CITE, 2019-09, Vol.2019 (4)

2019

Volltextzugriff (PDF)

Class A Orphans in GtoPdb v.2023.1

IUPHAR/BPS Guide to Pharmacology CITE, 2023-04, Vol.2023 (1)

2023

Volltextzugriff (PDF)

Free fatty acid receptors (version 2019.4) in the IUPHAR/BPS Guide to Pharmacology Database

IUPHAR/BPS Guide to Pharmacology CITE, 2019-09, Vol.2019 (4)

2019

Volltextzugriff (PDF)

Chemokine receptors in GtoPdb v.2023.1

IUPHAR/BPS Guide to Pharmacology CITE, 2023-04, Vol.2023 (1)

2023

Volltextzugriff (PDF)

Class A Orphans in GtoPdb v.2022.3

IUPHAR/BPS Guide to Pharmacology CITE, 2022-10, Vol.2022 (3)

2022

Volltextzugriff (PDF)

The amino terminal domain of steroid hormone receptors as a novel drug target: Identification of small molecule inhibitors

Endocrine Abstracts, 2016-09

2016

Volltextzugriff (PDF)

Class A Orphans in GtoPdb v.2021.3

IUPHAR/BPS Guide to Pharmacology CITE, 2021-09, Vol.2021 (3)

2021

Volltextzugriff (PDF)

Class A Orphans (version 2020.5) in the IUPHAR/BPS Guide to Pharmacology Database

IUPHAR/BPS Guide to Pharmacology CITE, 2020-11, Vol.2020 (5)

2020

Volltextzugriff (PDF)

1 – 25 von 100

Suche als RSS-Feed

Suchergebnisse filtern

Filter anzeigen

Nur zeigen

Geprüft (Peer-Review)
(78)
Mit Volltextzugriff
(74)

Publikationsform

Sprache

Englisch
(100)
Japanisch
(7)

Erscheinungsjahr

n.n

Thema

15 weitere anzeigen...

Weniger anzeigen...

Kollektion

15 weitere anzeigen...

Weniger anzeigen...

Neu hinzugefügt

... seit 90 Tagen
(1)

Menü

Weitere Dienste

Einstellungen

A sting in the tail： the N-terminal domain of the androgen receptor as a drug target

International Union of Basic and Clinical Pharmacology. LXXXVIII. G protein-coupled receptor list: recommendations for new pairings with cognate ligands

Development of a High-Throughput Screening Assay for Small-Molecule Inhibitors of Androgen Receptor Splice Variants

Enhanced insulin signalling ameliorates C9orf72 hexanucleotide repeat expansion toxicity in Drosophila

Structural Insights into Notum Covalent Inhibition

Virtual Screening Directly Identifies New Fragment-Sized Inhibitors of Carboxylesterase Notum with Nanomolar Activity

5‑Phenyl-1,3,4-oxadiazol-2(3H)‑ones Are Potent Inhibitors of Notum Carboxylesterase Activity Identified by the Optimization of a Crystallographic Fragment Screening Hit

Design of a Potent, Selective, and Brain-Penetrant Inhibitor of Wnt-Deactivating Enzyme Notum by Optimization of a Crystallographic Fragment Hit

Screening of a Custom-Designed Acid Fragment Library Identifies 1‑Phenylpyrroles and 1‑Phenylpyrrolidines as Inhibitors of Notum Carboxylesterase Activity

Scaffold-hopping identifies furano[2,3-d]pyrimidine amides as potent Notum inhibitors

Discovery of 2-phenoxyacetamides as inhibitors of the Wnt-depalmitoleating enzyme NOTUM from an X-ray fragment screen

Chemerin receptors in GtoPdb v.2023.1

The amino terminal domain of steroid hormone receptors as a novel drug target: identification of small molecule inhibitors

Chemerin receptors in GtoPdb v.2021.3

Free fatty acid receptors in GtoPdb v.2023.1

Chemerin receptors (version 2019.4) in the IUPHAR/BPS Guide to Pharmacology Database

Class A Orphans in GtoPdb v.2023.1

Free fatty acid receptors (version 2019.4) in the IUPHAR/BPS Guide to Pharmacology Database

Chemokine receptors in GtoPdb v.2023.1

Class A Orphans in GtoPdb v.2022.3

The amino terminal domain of steroid hormone receptors as a novel drug target: Identification of small molecule inhibitors

Class A Orphans in GtoPdb v.2021.3

Class A Orphans (version 2020.5) in the IUPHAR/BPS Guide to Pharmacology Database

Chemokine receptors (version 2020.5) in the IUPHAR/BPS Guide to Pharmacology Database

Suchergebnisse filtern