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Design, synthesis, and SAR of cis-1,2-diaminocyclohexane derivatives as potent factor Xa inhibitors. Part I: Exploration of 5–6 fused rings as alternative S1 moieties

Bioorganic & medicinal chemistry, 2009-12, Vol.17 (24), p.8206-8220

2009

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Design, synthesis, and SAR of cis-1,2-diaminocyclohexane derivatives as potent factor Xa inhibitors. Part II: Exploration of 6–6 fused rings as alternative S1 moieties

Bioorganic & medicinal chemistry, 2009-12, Vol.17 (24), p.8221-8233

2009

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Enantioselective Synthesis of Piperidine Diamine Derivatives as Novel fXa Inhibitors

Heterocycles, 2008-07, Vol.75 (7), p.1659

2008

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Design, synthesis, and biological activity of piperidine diamine derivatives as factor Xa inhibitor

Bioorganic & medicinal chemistry, 2008-01, Vol.18 (2), p.782-787

2008

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2-Aminomethylphenylamine as a novel scaffold for factor Xa inhibitor

Bioorganic & medicinal chemistry, 2011-03, Vol.19 (5), p.1623-1642

2011

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Lead optimization of 5-amino-6-(2,2-dimethyl-5-oxo-4-phenylpiperazin-1-yl)-4-hydroxyhexanamides to reduce a cardiac safety issue: Discovery of DS-8108b, an orally active renin inhibitor

Bioorganic & medicinal chemistry, 2013-06, Vol.21 (11), p.3175-3196

2013

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Synthesis and optimization of novel (3S,5R)-5-(2,2-dimethyl-5-oxo-4-phenylpiperazin-1-yl)piperidine-3-carboxamides as orally active renin inhibitors

Bioorganic & medicinal chemistry, 2013-09, Vol.21 (18), p.5907-5922

2013

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Orally active zwitterionic factor Xa inhibitors with long duration of action

Bioorganic & medicinal chemistry letters, 2011-12, Vol.21 (24), p.7337-7343

2011

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Synthesis and optimization of novel (3S,5R)-5-(2,2-dimethyl-5-oxo-4-phenylpiperazin-1-yl)piperidine-3- c arboxamides as orally active renin inhibitors

Bioorganic & medicinal chemistry, 2013-09, Vol.21 (18), p.5907-5922

2013

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Design and discovery of new (3S,5R)-5-[4-(2-chlorophenyl)-2,2-dimethyl-5-oxopiperazin-1-yl]piperidine-3-carboxamides as potent renin inhibitors

Bioorganic & medicinal chemistry letters, 2012-12, Vol.22 (24), p.7677-7682

2012

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Design, synthesis and SAR of novel ethylenediamine and phenylenediamine derivatives as factor Xa inhibitors

Bioorganic & medicinal chemistry letters, 2011-04, Vol.21 (7), p.2133-2140

2011

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Design and discovery of new (3S,5R)-5-[4-(2-chlorophenyl)-2,2-dimethyl-5-oxopiperazin-1-yl]pip e ridine-3-carboxamides as potent renin inhibitors

Bioorganic & medicinal chemistry letters, 2012-12, Vol.22 (24), p.7677-7682

2012

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Lead optimization of 5-amino-6-(2,2-dimethyl-5-oxo-4-phenylpiperazin-1-yl)-4-hydroxyhex a namides to reduce a cardiac safety issue: Discovery of DS-8108b, an orally active renin inhibitor

Bioorganic & medicinal chemistry, 2013-06, Vol.21 (11), p.3175-3196

2013

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A Facile Synthesis of 5,6-Dihydro-4H-pyrrolo[3,4-d]thiazole and Other Pyrrolidine-Fused Aromatic Ring Systems via One-Step Cyclization from Diols

Heterocycles, 2012, Vol.85 (7), p.1711

2012

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Design, synthesis, and biological activity of novel factor Xa inhibitors: Improving metabolic stability by S1 and S4 ligand modification

Bioorganic & medicinal chemistry, 2006-03, Vol.14 (5), p.1309-1330

2006

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Design, synthesis, and biological activity of non-basic compounds as factor Xa inhibitors: SAR study of S1 and aryl binding sites

Bioorganic & medicinal chemistry, 2005-06, Vol.13 (12), p.3927-3954

2005

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Stereochemical course of the hydrogen migration in the boron trifluoride etherate-catalyzed rearrangement of 1,1-disubstituted epoxides

Tetrahedron: asymmetry, 2000-05, Vol.11 (9), p.1859-1868

2000

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ChemInform Abstract: A Facile Synthesis of 5,6-Dihydro-4H-pyrrolo[3,4-d]thiazole and Other Pyrrolidine-Fused Aromatic Ring Systems via One-Step Cyclization from Diols

ChemInform, 2012-10, Vol.43 (44), p.no-no

2012

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ChemInform Abstract: Enantioselective Synthesis of Piperidine Diamine Derivatives as Novel fXa Inhibitors

ChemInform, 2008-11, Vol.39 (48), p.no-no

2008

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Microwave spectrum, barrier to internal rotation, and dipole moment of 1,2,3-pentatriene

The Journal of chemical physics, 1987-09, Vol.87 (5), p.2531-2535

1987

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A Case of Canine Systemic Nocardiosis

The Japanese Journal of Veterinary Science, 1986, Vol.48(3), pp.629-632

1986

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A case of canine systemic nocardiosis

Japanese journal of veterinary science, 1986-06, Vol.48 (3), p.629-632

1986

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ノカルジア症と診断された犬の全身性肉芽腫の1例

日本獸醫學雜誌(The Japanese Journal of Veterinary Science), 1986, Vol.48(3), pp.629-632

1986

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The sphingosine-1-phosphate transporter Spns2 expressed on endothelial cells regulates lymphocyte trafficking in mice

The Journal of clinical investigation, 2012-04, Vol.122 (4), p.1416-1426

2012

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Two-staged Correction for Pouter Pigeon Chest: A Less Invasive Procedure

Journal of Plastic and Reconstructive Surgery, 2023-01, Vol.2 (1), p.17-19, Article 2021-0030

2023

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Design, synthesis, and SAR of cis-1,2-diaminocyclohexane derivatives as potent factor Xa inhibitors. Part I: Exploration of 5–6 fused rings as alternative S1 moieties

Design, synthesis, and SAR of cis-1,2-diaminocyclohexane derivatives as potent factor Xa inhibitors. Part II: Exploration of 6–6 fused rings as alternative S1 moieties

Enantioselective Synthesis of Piperidine Diamine Derivatives as Novel fXa Inhibitors

Design, synthesis, and biological activity of piperidine diamine derivatives as factor Xa inhibitor

2-Aminomethylphenylamine as a novel scaffold for factor Xa inhibitor

Lead optimization of 5-amino-6-(2,2-dimethyl-5-oxo-4-phenylpiperazin-1-yl)-4-hydroxyhexanamides to reduce a cardiac safety issue: Discovery of DS-8108b, an orally active renin inhibitor

Synthesis and optimization of novel (3S,5R)-5-(2,2-dimethyl-5-oxo-4-phenylpiperazin-1-yl)piperidine-3-carboxamides as orally active renin inhibitors

Orally active zwitterionic factor Xa inhibitors with long duration of action

Synthesis and optimization of novel (3S,5R)-5-(2,2-dimethyl-5-oxo-4-phenylpiperazin-1-yl)piperidine-3- c arboxamides as orally active renin inhibitors

Design and discovery of new (3S,5R)-5-[4-(2-chlorophenyl)-2,2-dimethyl-5-oxopiperazin-1-yl]piperidine-3-carboxamides as potent renin inhibitors

Design, synthesis and SAR of novel ethylenediamine and phenylenediamine derivatives as factor Xa inhibitors

Design and discovery of new (3S,5R)-5-[4-(2-chlorophenyl)-2,2-dimethyl-5-oxopiperazin-1-yl]pip e ridine-3-carboxamides as potent renin inhibitors

Lead optimization of 5-amino-6-(2,2-dimethyl-5-oxo-4-phenylpiperazin-1-yl)-4-hydroxyhex a namides to reduce a cardiac safety issue: Discovery of DS-8108b, an orally active renin inhibitor

A Facile Synthesis of 5,6-Dihydro-4H-pyrrolo[3,4-d]thiazole and Other Pyrrolidine-Fused Aromatic Ring Systems via One-Step Cyclization from Diols

Design, synthesis, and biological activity of novel factor Xa inhibitors: Improving metabolic stability by S1 and S4 ligand modification

Design, synthesis, and biological activity of non-basic compounds as factor Xa inhibitors: SAR study of S1 and aryl binding sites

Stereochemical course of the hydrogen migration in the boron trifluoride etherate-catalyzed rearrangement of 1,1-disubstituted epoxides

ChemInform Abstract: A Facile Synthesis of 5,6-Dihydro-4H-pyrrolo[3,4-d]thiazole and Other Pyrrolidine-Fused Aromatic Ring Systems via One-Step Cyclization from Diols

ChemInform Abstract: Enantioselective Synthesis of Piperidine Diamine Derivatives as Novel fXa Inhibitors

Microwave spectrum, barrier to internal rotation, and dipole moment of 1,2,3-pentatriene

A Case of Canine Systemic Nocardiosis

A case of canine systemic nocardiosis

ノカルジア症と診断された犬の全身性肉芽腫の1例

The sphingosine-1-phosphate transporter Spns2 expressed on endothelial cells regulates lymphocyte trafficking in mice

Two-staged Correction for Pouter Pigeon Chest: A Less Invasive Procedure

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