UB Paderborn / Katalog / Suche / in CDI

Antibiotic-induced psychosis: A link to d -alanine?

Medical hypotheses, 2010-12, Vol.75 (6), p.676-677

Mehdi, Shujaath

2010

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Identification and neuroprotective properties of NA‐184, a calpain‐2 inhibitor

Pharmacology research & perspectives, 2024-04, Vol.12 (2), p.e1181-n/a

2024

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Cell-penetrating inhibitors of calpain

Trends in biochemical sciences (Amsterdam. Regular ed.), 1991, Vol.16 (4), p.150-153

Mehdi, Shujaath

1991

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Inhibition of Human Neutrophil Elastase. 4. Design, Synthesis, X-ray Crystallographic Analysis, and Structure−Activity Relationships for a Series of P2-Modified, Orally Active Peptidyl Pentafluoroethyl Ketones

Journal of medicinal chemistry, 1998-07, Vol.41 (14), p.2461-2480

1998

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Human kallikrein 6 inhibitors with a para-amidobenzylanmine P1 group identified through virtual screening

Bioorganic & medicinal chemistry letters, 2012-04, Vol.22 (7), p.2450-2455

2012

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Synthesis of peptidyl fluoromethyl ketones and peptidyl α-keto esters as inhibitors of porcine pancreatic elastase, human neutrophil elastase, and rat and human neutrophil cathepsin G

Journal of medicinal chemistry, 1990, Vol.33 (1), p.394-407

1990

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A Stereoselective method to (E)- and (Z)-fluorovinyl phosphonates Utilizing Palladium(0) coupling methodology

Tetrahedron letters, 1993-11, Vol.34 (45), p.7197-7200

1993

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Improved posthypoxic recovery with a membrane-permeable calpain inhibitor

European journal of pharmacology, 1991-12, Vol.209 (1), p.123-125

1991

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Inhibition of the proteolysis of rat erythrocyte membrane proteins by a synthetic inhibitor of calpain

Biochemical and biophysical research communications, 1988-12, Vol.157 (3), p.1117-1123

1988

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Dehydroquinate synthase: the role of divalent metal cations and of nicotinamide adenine dinucleotide in catalysis

Biochemistry (Easton), 1989-09, Vol.28 (19), p.7555-7560

1989

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Virtual Screening and X-ray Crystallography for Human Kallikrein 6 Inhibitors with an Amidinothiophene P1 Group

ACS medicinal chemistry letters, 2012-02, Vol.3 (2), p.159-164

2012

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Synthesis of a peptidyl 2,2-difluoro-3-aminopropionate

Bioorganic & medicinal chemistry letters, 1992-10, Vol.2 (10), p.1235-1238

1992

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The inhibition of human neutrophil elastase and cathepsin G by peptidyl 1,2-dicarbonyl derivatives

Biochemical and biophysical research communications, 1990-01, Vol.166 (2), p.595-600

1990

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COVALENT ENZYME INHIBITION IN DRUG DISCOVERY AND DEVELOPMENT

Enzyme Technologies, 2013, p.81-129

2013

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The Mechanism of Inhibition of S-Adenosyl-L-Homocysteine Hydrolase by Fluorine-Containing Adenosine Analogs

Journal of enzyme inhibition, 1990, Vol.4 (1), p.1-13

1990

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Synthetic and Naturally Occurring Protease Inhibitors Containing an Electrophilic Carbonyl Group

Bioorganic Chemistry, 1993-09, Vol.21 (3), p.249-259

Mehdi, S.

1993

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An assay for dihydroorotase using high-performance liquid chromatography with radioactivity detection

Analytical biochemistry, 1989, Vol.176 (1), p.105-108

1989

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Syntheses and configurational analyses of thymidine 4-nitrophenyl [17O,18O]phosphates and the stereochemical course of a reaction catalyzed by bovine pancreatic deoxyribonuclease I

Biochemistry (Easton), 1984-10, Vol.23 (21), p.4844-4852

1984

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Inhibition of Human Neutrophil Elastase. 4. Design, Synthesis, X-ray Crystallographic Analysis, and Structure−Activity Relationships for a Series of P 2 -Modified, Orally Active Peptidyl Pentafluoroethyl Ketones

Journal of medicinal chemistry, 1998-07, Vol.41 (14), p.2461-2480

1998

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Synthesis of peptidyl fluoromethyl ketones and peptidyl .alpha.-keto esters as inhibitors of porcine pancreatic elastase, human neutrophil elastase, and rat and human neutrophil cathepsin G

Journal of medicinal chemistry, 1990-01, Vol.33 (1), p.394-407

1990

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alpha.-Diketone and .alpha.-keto ester derivatives of N-protected amino acids and peptides as novel inhibitors of cysteine and serine proteinases

Journal of medicinal chemistry, 1990-01, Vol.33 (1), p.11-13

1990

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Molecular Design and Characterization of an α-Thrombin Inhibitor Containing a Novel P1 Moiety

Biochemistry (Easton), 1997-02, Vol.36 (5), p.1034-1040

1997

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Application of a conformationally restricted Phe-Leu dipeptide mimetic to the design of a combined inhibitor of angiotensin I-converting enzyme and neutral endopeptidase 24.11

Journal of medicinal chemistry, 1993-08, Vol.36 (16), p.2420-2423

1993

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An ultra-high throughput screening approach for an adenine transferase using fluorescence polarization

Journal of biomolecular screening, 2000-02, Vol.5 (1), p.31-37

2000

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Inhibition of Human Neutrophil Elastase with Peptidyl Electrophilic Ketones. 2. Orally Active PG-Val-Pro-Val Pentafluoroethyl Ketones

Journal of medicinal chemistry, 1994-12, Vol.37 (26), p.4538-4553

1994

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Antibiotic-induced psychosis: A link to d -alanine?

Identification and neuroprotective properties of NA‐184, a calpain‐2 inhibitor

Cell-penetrating inhibitors of calpain

Inhibition of Human Neutrophil Elastase. 4. Design, Synthesis, X-ray Crystallographic Analysis, and Structure−Activity Relationships for a Series of P2-Modified, Orally Active Peptidyl Pentafluoroethyl Ketones

Human kallikrein 6 inhibitors with a para-amidobenzylanmine P1 group identified through virtual screening

Synthesis of peptidyl fluoromethyl ketones and peptidyl α-keto esters as inhibitors of porcine pancreatic elastase, human neutrophil elastase, and rat and human neutrophil cathepsin G

A Stereoselective method to (E)- and (Z)-fluorovinyl phosphonates Utilizing Palladium(0) coupling methodology

Improved posthypoxic recovery with a membrane-permeable calpain inhibitor

Inhibition of the proteolysis of rat erythrocyte membrane proteins by a synthetic inhibitor of calpain

Dehydroquinate synthase: the role of divalent metal cations and of nicotinamide adenine dinucleotide in catalysis

Virtual Screening and X-ray Crystallography for Human Kallikrein 6 Inhibitors with an Amidinothiophene P1 Group

Synthesis of a peptidyl 2,2-difluoro-3-aminopropionate

The inhibition of human neutrophil elastase and cathepsin G by peptidyl 1,2-dicarbonyl derivatives

COVALENT ENZYME INHIBITION IN DRUG DISCOVERY AND DEVELOPMENT

The Mechanism of Inhibition of S-Adenosyl-L-Homocysteine Hydrolase by Fluorine-Containing Adenosine Analogs

Synthetic and Naturally Occurring Protease Inhibitors Containing an Electrophilic Carbonyl Group

An assay for dihydroorotase using high-performance liquid chromatography with radioactivity detection

Syntheses and configurational analyses of thymidine 4-nitrophenyl [17O,18O]phosphates and the stereochemical course of a reaction catalyzed by bovine pancreatic deoxyribonuclease I

Inhibition of Human Neutrophil Elastase. 4. Design, Synthesis, X-ray Crystallographic Analysis, and Structure−Activity Relationships for a Series of P 2 -Modified, Orally Active Peptidyl Pentafluoroethyl Ketones

Synthesis of peptidyl fluoromethyl ketones and peptidyl .alpha.-keto esters as inhibitors of porcine pancreatic elastase, human neutrophil elastase, and rat and human neutrophil cathepsin G

alpha.-Diketone and .alpha.-keto ester derivatives of N-protected amino acids and peptides as novel inhibitors of cysteine and serine proteinases

Molecular Design and Characterization of an α-Thrombin Inhibitor Containing a Novel P1 Moiety

Application of a conformationally restricted Phe-Leu dipeptide mimetic to the design of a combined inhibitor of angiotensin I-converting enzyme and neutral endopeptidase 24.11

An ultra-high throughput screening approach for an adenine transferase using fluorescence polarization

Inhibition of Human Neutrophil Elastase with Peptidyl Electrophilic Ketones. 2. Orally Active PG-Val-Pro-Val Pentafluoroethyl Ketones

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