UB Paderborn / Katalog / Suche / in CDI

1 – 25 von 38

Sortiert nach

Design and Optimization of Benzimidazole-Containing Transient Receptor Potential Melastatin 8 (TRPM8) Antagonists

Journal of medicinal chemistry, 2011-01, Vol.54 (1), p.233-247

2011

Volltextzugriff (PDF)

Discovery of novel benzo[b]thiophene tetrazoles as non-carboxylate GPR40 agonists

Bioorganic & medicinal chemistry letters, 2018-02, Vol.28 (3), p.429-436

2018

Volltextzugriff (PDF)

Discovery of a novel potent GPR40 full agonist

Bioorganic & medicinal chemistry letters, 2018-02, Vol.28 (4), p.720-726

2018

Volltextzugriff (PDF)

Discovery of a GPR40 Superagonist: The Impact of Aryl Propionic Acid α‑Fluorination

ACS medicinal chemistry letters, 2019-01, Vol.10 (1), p.16-21

2019

Volltextzugriff (PDF)

Synthesis and Characterization of Technetium-99m-Labeled Tropanes as Dopamine Transporter-Imaging Agents

Journal of medicinal chemistry, 1997-01, Vol.40 (1), p.9-17

1997

Volltextzugriff (PDF)

Discovery of novel potent imidazo[1,2-b]pyridazine PDE10a inhibitors

Bioorganic & medicinal chemistry letters, 2016-09, Vol.26 (17), p.4216-4222

2016

Volltextzugriff (PDF)

Discovery of vinylcycloalkyl-substituted benzimidazole TRPM8 antagonists effective in the treatment of cold allodynia

Bioorganic & medicinal chemistry letters, 2012-03, Vol.22 (5), p.1903-1907

2012

Volltextzugriff (PDF)

Synthesis and insecticidal activity of fluorinated 2-(2,6-dichloro-4-trifluoromethylphenyl)-2,4,5,6-tetrahydrocyclopentapyrazoles

Bioorganic & medicinal chemistry letters, 2006-03, Vol.16 (6), p.1702-1706

2006

Volltextzugriff (PDF)

Optimization of a Potent Class of Arylamide Colony-Stimulating Factor-1 Receptor Inhibitors Leading to Anti-inflammatory Clinical Candidate 4-Cyano-N-[2-(1-cyclohexen-1-yl)-4-[1-[(dimethylamino)acetyl]-4-piperidinyl]phenyl]-1H-imidazole-2-carboxamide (JNJ-28312141)

Journal of medicinal chemistry, 2011-11, Vol.54 (22), p.7860-7883

2011

Volltextzugriff (PDF)

5-amino-1-(2,6-dichloro-4-trifluoromethyl-phenyl)-3-[3H3]-methylsulfanyl-1H-pyrazole-4-carbonitrile (CTOM): synthesis and characterization of a novel and selective insect GABA receptor radioligand

Bioorganic & medicinal chemistry letters, 2003-11, Vol.13 (22), p.4035-4037

2003

Volltextzugriff (PDF)

Specificity of Diastereomers of [99mTc]TRODAT-1 as Dopamine Transporter Imaging Agents

Journal of medicinal chemistry, 1998-02, Vol.41 (4), p.428-436

1998

Volltextzugriff (PDF)

Enhancement of kinase selectivity in a potent class of arylamide FMS inhibitors

Bioorganic & medicinal chemistry letters, 2013-12, Vol.23 (23), p.6363-6369

2013

Volltextzugriff (PDF)

Discovery of novel FMS kinase inhibitors as anti-inflammatory agents

Bioorganic & medicinal chemistry, 2008-03, Vol.18 (5), p.1642-1648

2008

Volltextzugriff (PDF)

Structure-based optimization of a potent class of arylamide FMS inhibitors

Bioorganic & medicinal chemistry, 2008-06, Vol.18 (12), p.3632-3637

2008

Volltextzugriff (PDF)

Reducing ion channel activity in a series of 4-heterocyclic arylamide FMS inhibitors

Bioorganic & medicinal chemistry letters, 2010-07, Vol.20 (13), p.3925-3929

2010

Volltextzugriff (PDF)

Synthesis and GABA receptor potency of 3-thiomethyl-4-(hetero)aryl-5-amino-1-phenylpyrazoles

Bioorganic & medicinal chemistry letters, 2004-10, Vol.14 (19), p.4949-4953

2004

Volltextzugriff (PDF)

Pharmacological effects of dopaminergic drugs on in vivo binding of [99mTc]TRODAT-1 to the central dopamine transporters in rats

European journal of nuclear medicine, 1998-01, Vol.25 (1), p.31-39

1998

Volltextzugriff (PDF)

Simultaneous SPECT Studies of Pre- and Postsynaptic Dopamine Binding Sites in Baboons

The Journal of nuclear medicine (1978), 1999-04, Vol.40 (4), p.660-666

1999

Volltextzugriff (PDF)

Kinetic Modeling of [99mTc]TRODAT-1: A Dopamine Transporter Imaging Agent

The Journal of nuclear medicine (1978), 1999-01, Vol.40 (1), p.150-158

1999

Volltextzugriff (PDF)

Synthesis and Pharmacological Evaluation of Isoindolo[1,2-b]quinazolinone and Isoindolo[2,1-a]benzimidazole Derivatives Related to the Antitumor Agent Batracylin

Journal of medicinal chemistry, 1994-09, Vol.37 (20), p.3434-3439

1994

Volltextzugriff (PDF)

A general synthetic route to isobenzofurans bearing a functionalized C-1 substituent

Journal of organic chemistry, 1991-03, Vol.56 (5), p.1882-1888

1991

Volltextzugriff (PDF)

Imaging of dopamine transporters in humans with technetium-99m TRODAT-1

European Journal of Nuclear Medicine, 1996-11, Vol.23 (11), p.1527-1530

1996

Volltextzugriff (PDF)

An unusual doubly substituted product from the phase-transfer-catalyzed Heck reactions of o-bromobenzaldehydes with methyl acrylate

Journal of organic chemistry, 1992-04, Vol.57 (8), p.2422-2427

1992

Volltextzugriff (PDF)

1 – 25 von 38

Suche als RSS-Feed

Suchergebnisse filtern

Filter anzeigen

Nur zeigen

Geprüft (Peer-Review)
(34)
Mit Volltextzugriff
(37)

Publikationsform

Artikel
(37)
Dissertationen
(1)

Sprache

Englisch
(38)
Japanisch
(5)

Erscheinungsjahr

n.n

Thema

Science & Technology
(26)
Life Sciences & Biomedicine
(24)
Animals
(20)
Chemistry
(19)
Chemistry, Medicinal
(17)
Pharmacology & Pharmacy
(17)
Biological And Medical Sciences
(14)
Chemistry, Organic
(14)
Physical Sciences
(14)
Rats
(14)
Structure-Activity Relationship
(13)
Medical Sciences
(11)
Humans
(10)
Dopamine Plasma Membrane Transport Proteins
(8)
Membrane Transport Proteins
(8)
Mice
(8)
Models, Molecular
(8)
Molecular Structure
(8)
Rats, Sprague-Dawley
(8)
Brain - Metabolism
(7)

15 weitere anzeigen...

Weniger anzeigen...

Menü

Weitere Dienste

Einstellungen

JNJ-28312141, a novel orally active colony-stimulating factor-1 receptor/FMS-related receptor tyrosine kinase-3 receptor tyrosine kinase inhibitor with potential utility in solid tumors, bone metastases, and acute myeloid leukemia

Design and Optimization of Benzimidazole-Containing Transient Receptor Potential Melastatin 8 (TRPM8) Antagonists

Discovery of novel benzo[b]thiophene tetrazoles as non-carboxylate GPR40 agonists

Discovery of a novel potent GPR40 full agonist

Discovery of a GPR40 Superagonist: The Impact of Aryl Propionic Acid α‑Fluorination

Synthesis and Characterization of Technetium-99m-Labeled Tropanes as Dopamine Transporter-Imaging Agents

Discovery of novel potent imidazo[1,2-b]pyridazine PDE10a inhibitors

Discovery of vinylcycloalkyl-substituted benzimidazole TRPM8 antagonists effective in the treatment of cold allodynia

Synthesis and insecticidal activity of fluorinated 2-(2,6-dichloro-4-trifluoromethylphenyl)-2,4,5,6-tetrahydrocyclopentapyrazoles

Optimization of a Potent Class of Arylamide Colony-Stimulating Factor-1 Receptor Inhibitors Leading to Anti-inflammatory Clinical Candidate 4-Cyano-N-[2-(1-cyclohexen-1-yl)-4-[1-[(dimethylamino)acetyl]-4-piperidinyl]phenyl]-1H-imidazole-2-carboxamide (JNJ-28312141)

5-amino-1-(2,6-dichloro-4-trifluoromethyl-phenyl)-3-[3H3]-methylsulfanyl-1H-pyrazole-4-carbonitrile (CTOM): synthesis and characterization of a novel and selective insect GABA receptor radioligand

Specificity of Diastereomers of [99mTc]TRODAT-1 as Dopamine Transporter Imaging Agents

Enhancement of kinase selectivity in a potent class of arylamide FMS inhibitors

Discovery of novel FMS kinase inhibitors as anti-inflammatory agents

Structure-based optimization of a potent class of arylamide FMS inhibitors

Reducing ion channel activity in a series of 4-heterocyclic arylamide FMS inhibitors

Synthesis and GABA receptor potency of 3-thiomethyl-4-(hetero)aryl-5-amino-1-phenylpyrazoles

Pharmacological effects of dopaminergic drugs on in vivo binding of [99mTc]TRODAT-1 to the central dopamine transporters in rats

Simultaneous SPECT Studies of Pre- and Postsynaptic Dopamine Binding Sites in Baboons

Kinetic Modeling of [99mTc]TRODAT-1: A Dopamine Transporter Imaging Agent

Optimization of a Potent Class of Arylamide Colony-Stimulating Factor-1 Receptor Inhibitors Leading to Anti-inflammatory Clinical Candidate 4-Cyano- N -[2-(1-cyclohexen-1-yl)-4-[1-[(dimethylamino)acetyl]-4-piperidinyl]phenyl]-1 H -imidazole-2-carboxamide (JNJ-28312141)

Synthesis and Pharmacological Evaluation of Isoindolo[1,2-b]quinazolinone and Isoindolo[2,1-a]benzimidazole Derivatives Related to the Antitumor Agent Batracylin

A general synthetic route to isobenzofurans bearing a functionalized C-1 substituent

Imaging of dopamine transporters in humans with technetium-99m TRODAT-1

An unusual doubly substituted product from the phase-transfer-catalyzed Heck reactions of o-bromobenzaldehydes with methyl acrylate

Suchergebnisse filtern