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Recent advances in acetylcholinesterase Inhibitors and Reactivators: an update on the patent literature (2012-2015)

Expert opinion on therapeutic patents, 2017-04, Vol.27 (4), p.455-476

2017

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Oxamniquine derivatives overcome Praziquantel treatment limitations for Schistosomiasis

PLoS pathogens, 2023-07, Vol.19 (7), p.e1011018-e1011018

2023

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Selective and membrane-permeable small molecule inhibitors of nicotinamide N-methyltransferase reverse high fat diet-induced obesity in mice

Biochemical pharmacology, 2018-01, Vol.147, p.141-152

2018

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Tamoxifen Derivatives Alter Retromer-Dependent Endosomal Tubulation and Sorting to Block Retrograde Trafficking of Shiga Toxins

Toxins, 2021-06, Vol.13 (6), p.424

2021

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Addressing the oxamniquine in vitro-in vivo paradox to facilitate a new generation of anti-schistosome treatments

International journal for parasitology -- drugs and drug resistance, 2023-04, Vol.21, p.65-73

2023

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An iterative process produces oxamniquine derivatives that kill the major species of schistosomes infecting humans

PLoS neglected tropical diseases, 2020-08, Vol.14 (8), p.e0008517

2020

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Inhibition of Ca2+ entry by capsazepine analog CIDD-99 prevents oral squamous carcinoma cell proliferation

Frontiers in physiology, 2022-09, Vol.13, p.969000-969000

2022

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Rational approach to drug discovery for human schistosomiasis

International journal for parasitology -- drugs and drug resistance, 2021-08, Vol.16, p.140-147

2021

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Corrigendum to “Rational approach to drug discovery for human schistosomiasis” [Int. J. Parasitol. Drugs Drug Resist. 16 (2021) 140–147]

International journal for parasitology -- drugs and drug resistance, 2022-04, Vol.18, p.103-103

2022

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Schistosome Sulfotransferases: Mode of Action, Expression and Localization

Pharmaceutics, 2022-07, Vol.14 (7), p.1416

2022

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Why does oxamniquine kill Schistosoma mansoni and not S. haematobium and S. japonicum?

International journal for parasitology -- drugs and drug resistance, 2020-08, Vol.13, p.8-15

2020

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Structure–Activity Relationship for Small Molecule Inhibitors of Nicotinamide N‑Methyltransferase

Journal of medicinal chemistry, 2017-06, Vol.60 (12), p.5015-5028

2017

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A modular PROTAC design for target destruction using a degradation signal based on a single amino acid

The Journal of biological chemistry, 2019-10, Vol.294 (41), p.15172-15175

2019

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Targeting Candida albicans filamentation for antifungal drug development

Virulence, 2017-02, Vol.8 (2), p.150-158

2017

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Asymmetric Synthesis of CIDD-0072424 via an Enantioselective Nitro-Mannich Reaction: A Central Nervous System Penetrant, Selective Small Molecule Inhibitor of Protein Kinase C Epsilon

Journal of organic chemistry, 2024-04, Vol.89 (7), p.5134-5141

2024

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Small molecule nicotinamide N-methyltransferase inhibitor activates senescent muscle stem cells and improves regenerative capacity of aged skeletal muscle

Biochemical pharmacology, 2019-05, Vol.163, p.481-492

2019

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Development of Anti-Virulence Approaches for Candidiasis via a Novel Series of Small-Molecule Inhibitors of Candida albicans Filamentation

mBio, 2017-12, Vol.8 (6)

2017

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Structure–Activity Relationships of New Natural Product-Based Diaryloxazoles with Selective Activity against Androgen Receptor-Positive Breast Cancer Cells

Journal of medicinal chemistry, 2017-11, Vol.60 (22), p.9275-9289

2017

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Preclinical Development of Brain Permeable ERβ Agonist for the Treatment of Glioblastoma

Molecular cancer therapeutics, 2023-11, Vol.22 (11), p.1248

2023

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Noncoupled Fluorescent Assay for Direct Real-Time Monitoring of Nicotinamide N‑Methyltransferase Activity

Biochemistry (Easton), 2017-02, Vol.56 (6), p.824-832

2017

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Synthesis and SAR of novel capsazepine analogs with significant anti-cancer effects in multiple cancer types

Bioorganic & medicinal chemistry, 2019-01, Vol.27 (1), p.208-215

2019

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Molecular basis for hycanthone drug action in schistosome parasites

Molecular and biochemical parasitology, 2020-03, Vol.236 (C), p.111257, Article 111257

2020

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Modulation of α1β3γ2 GABAA receptors expressed in X. laevis oocytes using a propofol photoswitch tethered to the transmembrane helix

Proceedings of the National Academy of Sciences - PNAS, 2021-02, Vol.118 (8)

2021

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Modulation of α1β3γ2 GABA A receptors expressed in X. laevis oocytes using a propofol photoswitch tethered to the transmembrane helix

Proceedings of the National Academy of Sciences - PNAS, 2021-02, Vol.118 (8)

2021

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Structural and enzymatic insights into species-specific resistance to schistosome parasite drug therapy

The Journal of biological chemistry, 2017-07, Vol.292 (27), p.11154-11164

2017

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Recent advances in acetylcholinesterase Inhibitors and Reactivators: an update on the patent literature (2012-2015)

Oxamniquine derivatives overcome Praziquantel treatment limitations for Schistosomiasis

Selective and membrane-permeable small molecule inhibitors of nicotinamide N-methyltransferase reverse high fat diet-induced obesity in mice

Tamoxifen Derivatives Alter Retromer-Dependent Endosomal Tubulation and Sorting to Block Retrograde Trafficking of Shiga Toxins

Addressing the oxamniquine in vitro-in vivo paradox to facilitate a new generation of anti-schistosome treatments

An iterative process produces oxamniquine derivatives that kill the major species of schistosomes infecting humans

Inhibition of Ca2+ entry by capsazepine analog CIDD-99 prevents oral squamous carcinoma cell proliferation

Rational approach to drug discovery for human schistosomiasis

Corrigendum to “Rational approach to drug discovery for human schistosomiasis” [Int. J. Parasitol. Drugs Drug Resist. 16 (2021) 140–147]

Schistosome Sulfotransferases: Mode of Action, Expression and Localization

Why does oxamniquine kill Schistosoma mansoni and not S. haematobium and S. japonicum?

Structure–Activity Relationship for Small Molecule Inhibitors of Nicotinamide N‑Methyltransferase

A modular PROTAC design for target destruction using a degradation signal based on a single amino acid

Targeting Candida albicans filamentation for antifungal drug development

Asymmetric Synthesis of CIDD-0072424 via an Enantioselective Nitro-Mannich Reaction: A Central Nervous System Penetrant, Selective Small Molecule Inhibitor of Protein Kinase C Epsilon

Small molecule nicotinamide N-methyltransferase inhibitor activates senescent muscle stem cells and improves regenerative capacity of aged skeletal muscle

Development of Anti-Virulence Approaches for Candidiasis via a Novel Series of Small-Molecule Inhibitors of Candida albicans Filamentation

Structure–Activity Relationships of New Natural Product-Based Diaryloxazoles with Selective Activity against Androgen Receptor-Positive Breast Cancer Cells

Preclinical Development of Brain Permeable ERβ Agonist for the Treatment of Glioblastoma

Noncoupled Fluorescent Assay for Direct Real-Time Monitoring of Nicotinamide N‑Methyltransferase Activity

Synthesis and SAR of novel capsazepine analogs with significant anti-cancer effects in multiple cancer types

Molecular basis for hycanthone drug action in schistosome parasites

Modulation of α1β3γ2 GABAA receptors expressed in X. laevis oocytes using a propofol photoswitch tethered to the transmembrane helix

Modulation of α1β3γ2 GABA A receptors expressed in X. laevis oocytes using a propofol photoswitch tethered to the transmembrane helix

Structural and enzymatic insights into species-specific resistance to schistosome parasite drug therapy

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