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Hydrolytic instability of the important orexin 1 receptor antagonist SB-334867: Possible confounding effects on in vivo and in vitro studies

Bioorganic & medicinal chemistry letters, 2012-11, Vol.22 (21), p.6661-6664

2012

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Emergence and properties of spice and bath salts: A medicinal chemistry perspective

Life sciences (1973), 2014-02, Vol.97 (1), p.9-19

2014

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Structure of the human κ-opioid receptor in complex with JDTic

Nature (London), 2012-03, Vol.485 (7398), p.327-332

2012

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Designer drugs: a medicinal chemistry perspective

Annals of the New York Academy of Sciences, 2012-02, Vol.1248 (1), p.18-38

2012

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Structure–activity correlations for β-phenethylamines at human trace amine receptor 1

Bioorganic & medicinal chemistry, 2008-08, Vol.16 (15), p.7415-7423

2008

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Designer drugs: a medicinal chemistry perspective (II)

Annals of the New York Academy of Sciences, 2021-04, Vol.1489 (1), p.48-77

2021

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Quantitative Signaling and Structure-Activity Analyses Demonstrate Functional Selectivity at the Nociceptin/Orphanin FQ Opioid Receptor

Molecular pharmacology, 2015-09, Vol.88 (3), p.502-511

2015

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Potent and Selective Tetrahydroisoquinoline Kappa Opioid Receptor Antagonists of Lead Compound (3R)‑7-Hydroxy‑N‑[(1S)‑2-methyl-1-(piperidin-1-ylmethyl)propyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide (PDTic)

Journal of medicinal chemistry, 2018-09, Vol.61 (17), p.7525-7545

2018

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Bupropion and Bupropion Analogs as Treatments for CNS Disorders

Advances in Pharmacology, 2014, Vol.69, p.177-216

2014

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Potent and Selective Tetrahydroisoquinoline Kappa Opioid Receptor Antagonists of Lead Compound (3R)‑N‑[1R)‑1-(Cyclohexylmethyl)-2-methylpropyl]-7-hydroxy-1,2,3,4-tetrahydroisoquinoline-3-carboxamide (CDTic

Journal of medicinal chemistry, 2018-09, Vol.61 (17), p.7546-7559

2018

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Isolation of Hemiketal and Hydroxy Ketone Tautomers of Synthetic Intermediates Each Affording 18-Hydroxycortisol-1,6,7-d3

ACS omega, 2023-08, Vol.8 (31), p.28185-28195

2023

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Design, Synthesis, and Biological Evaluation of Structurally Rigid Analogues of 4‑(3-Hydroxyphenyl)piperidine Opioid Receptor Antagonists

Journal of organic chemistry, 2016-11, Vol.81 (21), p.10383-10391

2016

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Design, Synthesis, and Biological Evaluation of (3R)‑1,2,3,4-Tetrahydro-7-hydroxy‑N‑[(1S)‑1-[[(3R,4R)‑4-(3-hydroxyphenyl)-3,4-dimethyl-1-piperidinyl]methyl]-2-methylpropyl]-3-isoquinolinecarboxamide (JDTic) Analogues: In Vitro Pharmacology and ADME Profile

Journal of medicinal chemistry, 2014-09, Vol.57 (17), p.7367-7381

2014

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Synthesis, Nicotinic Acetylcholine Receptor Binding, and Antinociceptive Properties of 2′-Fluoro-3′-(substituted pyridinyl)-7-deschloroepibatidine Analogues

Journal of medicinal chemistry, 2014-02, Vol.57 (3), p.836-848

2014

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Isolation of Hemiketal and Hydroxy Ketone Tautomers of Synthetic Intermediates Each Affording 18-Hydroxycortisol-1,6,7‑d 3

ACS omega, 2023-08, Vol.8 (31), p.28185-28195

2023

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Synthesis and Nicotinic Acetylcholine Receptor in Vitro and in Vivo Pharmacological Properties of 2′-Fluoro-3′-(substituted phenyl)deschloroepibatidine Analogues of 2′-Fluoro-3′-(4-nitrophenyl)deschloroepibatidine

Journal of medicinal chemistry, 2012-07, Vol.55 (14), p.6512-6522

2012

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Synthesis and physicochemical characterization of the one-carbon carrier 10-formyltetrahydrofolate; a reference standard for metabolomics

Metabolomics, 2017-10, Vol.13 (10), p.1, Article 117

2017

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Design, synthesis, and pharmacological evaluation of JDTic analogs to examine the significance of the 3- and 4-methyl substituents

Bioorganic & medicinal chemistry, 2015-10, Vol.23 (19), p.6379-6388

2015

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Conformational characteristics of the interaction of SR141716A with the CB1 cannabinoid receptor as determined through the use of conformationally constrained analogs

The AAPS journal, 2006-10, Vol.8 (4), p.E665-E671

2006

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Design, synthesis, and pharmacological evaluation of JDTic analogs to examine the significance of replacement of the 3-hydroxyphenyl group with pyridine or thiophene bioisosteres

Bioorganic & medicinal chemistry, 2016-08, Vol.24 (16), p.3842-3848

2016

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Synthesis and Characterization of the Selective, Reversible PKC β Inhibitor (9 S)-9-[(Dimethylamino)methyl]-6,7,10,11-tetrahydro-9 H,18 H-5,21:12,17-dimethenodibenzo[ e,k]pyrrolo[3,4- h][1,4,13]oxadiazacyclohexadecine-18,20(19 H)-dione, Ruboxistaurin (LY333531)

ACS chemical neuroscience, 2019-01, Vol.10 (1), p.246-251

2019

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Synthesis and Characterization of in Vitro and in Vivo Profiles of Hydroxybupropion Analogues: Aids to Smoking Cessation

Journal of medicinal chemistry, 2010-06, Vol.53 (12), p.4731-4748

2010

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Synthesis and Biological Evaluation of Bupropion Analogues as Potential Pharmacotherapies for Smoking Cessation

Journal of medicinal chemistry, 2010-03, Vol.53 (5), p.2204-2214

2010

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Discovery of N‑{4-[(3-Hydroxyphenyl)-3-methylpiperazin-1-yl]methyl-2-methylpropyl}-4-phenoxybenzamide Analogues as Selective Kappa Opioid Receptor Antagonists

Journal of medicinal chemistry, 2013-06, Vol.56 (11), p.4551-4567

2013

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Simple Tetrahydroisoquinolines Are Potent and Selective Kappa Opioid Receptor Antagonists

ACS medicinal chemistry letters, 2017-07, Vol.8 (7), p.742-745

2017

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Hydrolytic instability of the important orexin 1 receptor antagonist SB-334867: Possible confounding effects on in vivo and in vitro studies

Emergence and properties of spice and bath salts: A medicinal chemistry perspective

Structure of the human κ-opioid receptor in complex with JDTic

Designer drugs: a medicinal chemistry perspective

Structure–activity correlations for β-phenethylamines at human trace amine receptor 1

Designer drugs: a medicinal chemistry perspective (II)

Quantitative Signaling and Structure-Activity Analyses Demonstrate Functional Selectivity at the Nociceptin/Orphanin FQ Opioid Receptor

Potent and Selective Tetrahydroisoquinoline Kappa Opioid Receptor Antagonists of Lead Compound (3R)‑7-Hydroxy‑N‑[(1S)‑2-methyl-1-(piperidin-1-ylmethyl)propyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide (PDTic)

Bupropion and Bupropion Analogs as Treatments for CNS Disorders

Potent and Selective Tetrahydroisoquinoline Kappa Opioid Receptor Antagonists of Lead Compound (3R)‑N‑[1R)‑1-(Cyclohexylmethyl)-2-methylpropyl]-7-hydroxy-1,2,3,4-tetrahydroisoquinoline-3-carboxamide (CDTic

Isolation of Hemiketal and Hydroxy Ketone Tautomers of Synthetic Intermediates Each Affording 18-Hydroxycortisol-1,6,7-d3

Design, Synthesis, and Biological Evaluation of Structurally Rigid Analogues of 4‑(3-Hydroxyphenyl)piperidine Opioid Receptor Antagonists

Design, Synthesis, and Biological Evaluation of (3R)‑1,2,3,4-Tetrahydro-7-hydroxy‑N‑[(1S)‑1-[[(3R,4R)‑4-(3-hydroxyphenyl)-3,4-dimethyl-1-piperidinyl]methyl]-2-methylpropyl]-3-isoquinolinecarboxamide (JDTic) Analogues: In Vitro Pharmacology and ADME Profile

Synthesis, Nicotinic Acetylcholine Receptor Binding, and Antinociceptive Properties of 2′-Fluoro-3′-(substituted pyridinyl)-7-deschloroepibatidine Analogues

Isolation of Hemiketal and Hydroxy Ketone Tautomers of Synthetic Intermediates Each Affording 18-Hydroxycortisol-1,6,7‑d 3

Synthesis and Nicotinic Acetylcholine Receptor in Vitro and in Vivo Pharmacological Properties of 2′-Fluoro-3′-(substituted phenyl)deschloroepibatidine Analogues of 2′-Fluoro-3′-(4-nitrophenyl)deschloroepibatidine

Synthesis and physicochemical characterization of the one-carbon carrier 10-formyltetrahydrofolate; a reference standard for metabolomics

Design, synthesis, and pharmacological evaluation of JDTic analogs to examine the significance of the 3- and 4-methyl substituents

Conformational characteristics of the interaction of SR141716A with the CB1 cannabinoid receptor as determined through the use of conformationally constrained analogs

Design, synthesis, and pharmacological evaluation of JDTic analogs to examine the significance of replacement of the 3-hydroxyphenyl group with pyridine or thiophene bioisosteres

Synthesis and Characterization of the Selective, Reversible PKC β Inhibitor (9 S)-9-[(Dimethylamino)methyl]-6,7,10,11-tetrahydro-9 H,18 H-5,21:12,17-dimethenodibenzo[ e,k]pyrrolo[3,4- h][1,4,13]oxadiazacyclohexadecine-18,20(19 H)-dione, Ruboxistaurin (LY333531)

Synthesis and Characterization of in Vitro and in Vivo Profiles of Hydroxybupropion Analogues: Aids to Smoking Cessation

Synthesis and Biological Evaluation of Bupropion Analogues as Potential Pharmacotherapies for Smoking Cessation

Discovery of N‑{4-[(3-Hydroxyphenyl)-3-methylpiperazin-1-yl]methyl-2-methylpropyl}-4-phenoxybenzamide Analogues as Selective Kappa Opioid Receptor Antagonists

Simple Tetrahydroisoquinolines Are Potent and Selective Kappa Opioid Receptor Antagonists

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