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AZD1152, a Selective Inhibitor of Aurora B Kinase, Inhibits Human Tumor Xenograft Growth by Inducing Apoptosis

Clinical cancer research, 2007-06, Vol.13 (12), p.3682-3688

2007

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Discovery, Synthesis, and in Vivo Activity of a New Class of Pyrazoloquinazolines as Selective Inhibitors of Aurora B Kinase

Journal of medicinal chemistry, 2007-05, Vol.50 (9), p.2213-2224

2007

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SAR and inhibitor complex structure determination of a novel class of potent and specific Aurora kinase inhibitors

Bioorganic & medicinal chemistry letters, 2006-03, Vol.16 (5), p.1320-1323

2006

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Small-molecule androgen receptor downregulators as an approach to treatment of advanced prostate cancer

Bioorganic & medicinal chemistry letters, 2011-09, Vol.21 (18), p.5442-5445

2011

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Discovery of Novel and Potent Thiazoloquinazolines as Selective Aurora A and B Kinase Inhibitors

Journal of medicinal chemistry, 2006-02, Vol.49 (3), p.955-970

2006

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Synthesis and SAR of 1-acetanilide-4-aminopyrazole-substituted quinazolines: Selective inhibitors of Aurora B kinase with potent anti-tumor activity

Bioorganic & medicinal chemistry, 2008-03, Vol.18 (6), p.1904-1909

2008

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Progress in the development of selective inhibitors of aurora kinases

Current topics in medicinal chemistry, 2005-08, Vol.5 (8), p.807-821

2005

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Structure–activity relationship of a series of non peptidic RGD integrin antagonists targeting α5β1: Part 1

Bioorganic & medicinal chemistry letters, 2012-06, Vol.22 (12), p.4111-4116

2012

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Structure–activity relationship of a series of non peptidic RGD integrin antagonists targeting α5β1: Part 2

Bioorganic & medicinal chemistry letters, 2012-06, Vol.22 (12), p.4117-4121

2012

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Total Syntheses of (−)-Papuamine and (−)-Haliclonadiamine

Journal of organic chemistry, 1996-01, Vol.61 (2), p.700-709

1996

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Bifunctional chiral auxiliaries 5: The synthesis of 1,3-diacylimidazolidine-2-thiones and 1,3-diacylimidazolidin-2-ones from 1,2-diamines

Tetrahedron, 1993, Vol.49 (20), p.4419-4438

1993

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New Non-Peptide Endothelin-A Receptor Antagonists: Synthesis, Biological Properties, and Structure−Activity Relationships of 5-(Dimethylamino)-N-pyridyl-, -N-pyrimidinyl-, -N-pyridazinyl-, and -N-pyrazinyl-1-naphthalenesulfonamides

Journal of medicinal chemistry, 1997-03, Vol.40 (6), p.996-1004

1997

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Two New Syntheses of a 4-Aminopyrazole: Condensation of an N-Substituted Vinamidinium Salt with a Functionalized Hydrazine

Synthesis (Stuttgart), 2007-06, Vol.2007 (11), p.1697-1701

2007

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Bifunctional chiral auxiliaries 6: Alkylations of enolates derived from 1,3-diacylimidazolidine- 2-thiones and 1,3-diacylimidazolidin-2-ones

Tetrahedron: asymmetry, 1994-04, Vol.5 (4), p.585-606

1994

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Synthetic studies on CP-225,917 and CP-263,114: concise synthesis of the bicyclic core using an intramolecular Mukaiyama aldol reactionElectronic supplementary information (ESI) available: crystal data for 13a. See http://www.rsc.org/suppdata/p1/b2/b202752f

Perkin 1 : an international journal of organic and bio-organic chemistry, 2002-05 (11), p.1344-1350

2002

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Structureaactivity relationship of a series of non peptidic RGD integrin antagonists targeting I-5I21: Part 2

Bioorganic & medicinal chemistry letters, 2012-06, Vol.22 (12), p.4117-4121

2012

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Structureaactivity relationship of a series of non peptidic RGD integrin antagonists targeting I-5I21: Part 1

Bioorganic & medicinal chemistry letters, 2012-06, Vol.22 (12), p.4111-4116

2012

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N-methyl-2-[4-(2-methylpropyl)phenyl]-3-(3-methoxy-5-methylpyrazin-2-ylsulfamoyl)benzamide ; One of a class of novel benzenesulphonamides which are orally-active, ETA-Selective endothelin antagonists

Bioorganic & medicinal chemistry letters, 1997-06, Vol.7 (11), p.1399-1402

1997

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Discovery of AZD1152: A Selective Inhibitor of Aurora‐B Kinase with Potent Antitumor Activity

Kinase Inhibitor Drugs, 2009, p.309-332

2009

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Synthesis of the Bicyclo[4.4.1]decenone Core of CP-225,917 and CP-263,114

Synlett, 1998-05, Vol.1998 (5), p.552-553

1998

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Approaches to the γ-lactone unit of CP-225,917 and CP-263,114

Tetrahedron letters, 2002-08, Vol.43 (34), p.6027-6030

2002

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SARr and inhibitor complex structure determination of a novel class of potent and specific Aurora kinase inhibitors

Bioorganic & medicinal chemistry letters, 2006, Vol.16 (5), p.1320-1323

2006

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Bifunctional chiral auxiliaries 7: Aldol reactions of enolates derived from 1,3-diacyl-imidazolidine-2-thiones and 1,3-diacylimidazolidin-2-ones

Tetrahedron, 1994, Vol.50 (22), p.6621-6642

1994

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Asymmetric synthesis of (1R,8S)- and (1S,8S)-1-hydroxypyrrolizidin-3-ones via the aldol reaction between N-boc-(S)-prolinal and chiral acetate enolate equivalents derived from (S)- and (R)-[(η 5-C 5H 5)Fe(CO)(PPh 3)COCH 3]

Tetrahedron: asymmetry, 1992, Vol.3 (1), p.123-136

1992

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Bifunctional chiral auxiliaries 2: the synthesis of 1,3-diacylimidazolidin-2-ones from 1,2-diamines

Tetrahedron letters, 1991, Vol.32 (36), p.4791-4794

1991

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AZD1152, a Selective Inhibitor of Aurora B Kinase, Inhibits Human Tumor Xenograft Growth by Inducing Apoptosis

Discovery, Synthesis, and in Vivo Activity of a New Class of Pyrazoloquinazolines as Selective Inhibitors of Aurora B Kinase

SAR and inhibitor complex structure determination of a novel class of potent and specific Aurora kinase inhibitors

Small-molecule androgen receptor downregulators as an approach to treatment of advanced prostate cancer

Discovery of Novel and Potent Thiazoloquinazolines as Selective Aurora A and B Kinase Inhibitors

Synthesis and SAR of 1-acetanilide-4-aminopyrazole-substituted quinazolines: Selective inhibitors of Aurora B kinase with potent anti-tumor activity

Progress in the development of selective inhibitors of aurora kinases

Structure–activity relationship of a series of non peptidic RGD integrin antagonists targeting α5β1: Part 1

Structure–activity relationship of a series of non peptidic RGD integrin antagonists targeting α5β1: Part 2

Total Syntheses of (−)-Papuamine and (−)-Haliclonadiamine

Bifunctional chiral auxiliaries 5: The synthesis of 1,3-diacylimidazolidine-2-thiones and 1,3-diacylimidazolidin-2-ones from 1,2-diamines

New Non-Peptide Endothelin-A Receptor Antagonists: Synthesis, Biological Properties, and Structure−Activity Relationships of 5-(Dimethylamino)-N-pyridyl-, -N-pyrimidinyl-, -N-pyridazinyl-, and -N-pyrazinyl-1-naphthalenesulfonamides

Two New Syntheses of a 4-Aminopyrazole: Condensation of an N-Substituted Vinamidinium Salt with a Functionalized Hydrazine

Bifunctional chiral auxiliaries 6: Alkylations of enolates derived from 1,3-diacylimidazolidine- 2-thiones and 1,3-diacylimidazolidin-2-ones

Synthetic studies on CP-225,917 and CP-263,114: concise synthesis of the bicyclic core using an intramolecular Mukaiyama aldol reactionElectronic supplementary information (ESI) available: crystal data for 13a. See http://www.rsc.org/suppdata/p1/b2/b202752f

Structureaactivity relationship of a series of non peptidic RGD integrin antagonists targeting I-5I21: Part 2

Structureaactivity relationship of a series of non peptidic RGD integrin antagonists targeting I-5I21: Part 1

N-methyl-2-[4-(2-methylpropyl)phenyl]-3-(3-methoxy-5-methylpyrazin-2-ylsulfamoyl)benzamide ; One of a class of novel benzenesulphonamides which are orally-active, ETA-Selective endothelin antagonists

Discovery of AZD1152: A Selective Inhibitor of Aurora‐B Kinase with Potent Antitumor Activity

Synthesis of the Bicyclo[4.4.1]decenone Core of CP-225,917 and CP-263,114

Approaches to the γ-lactone unit of CP-225,917 and CP-263,114

SARr and inhibitor complex structure determination of a novel class of potent and specific Aurora kinase inhibitors

Bifunctional chiral auxiliaries 7: Aldol reactions of enolates derived from 1,3-diacyl-imidazolidine-2-thiones and 1,3-diacylimidazolidin-2-ones

Asymmetric synthesis of (1R,8S)- and (1S,8S)-1-hydroxypyrrolizidin-3-ones via the aldol reaction between N-boc-(S)-prolinal and chiral acetate enolate equivalents derived from (S)- and (R)-[(η 5-C 5H 5)Fe(CO)(PPh 3)COCH 3]

Bifunctional chiral auxiliaries 2: the synthesis of 1,3-diacylimidazolidin-2-ones from 1,2-diamines

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