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Novel Peptidyl Phosphorus Derivatives as Inhibitors of Human Calpain I

Journal of medicinal chemistry, 1998-09, Vol.41 (20), p.3912-3916

1998

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Neurotrophic 3,9-Bis[(alkylthio)methyl]- and -Bis(alkoxymethyl)-K-252a Derivatives

Journal of medicinal chemistry, 1997-06, Vol.40 (12), p.1863-1869

1997

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d-Amino Acid Containing, High-Affinity Inhibitors of Recombinant Human Calpain I

Journal of medicinal chemistry, 1998-07, Vol.41 (15), p.2663-2666

1998

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Synthesis and Biological Activity of a Series of Potent Fluoromethyl Ketone Inhibitors of Recombinant Human Calpain I

Journal of medicinal chemistry, 1997-11, Vol.40 (23), p.3820-3828

1997

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Antipicornavirus activity of tetrazole analogs related to disoxaril

Journal of medicinal chemistry, 1993-10, Vol.36 (22), p.3240-3250

1993

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Knowledge-Based, Central Nervous System (CNS) Lead Selection and Lead Optimization for CNS Drug Discovery

ACS chemical neuroscience, 2012-01, Vol.3 (1), p.50-68

2012

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Prodrug esters of the indolocarbazole CEP-751 (KT-6587)

Bioorganic & medicinal chemistry letters, 1998-07, Vol.8 (14), p.1873-1876

1998

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Knowledge-based chemoinformatic approaches to drug discovery

Drug discovery today, 2006-12, Vol.11 (23), p.1107-1114

2006

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WIN 63480, a hydrophilic TCP-site ligand, has reduced agonist-independent NMDA ion channel access compared to MK-801 and phencyclidine

Neuropharmacology, 1995-12, Vol.34 (12), p.1597-1606

1995

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P2-ACHIRAL, P'-extended α-ketoamide inhibitors of calpain I

Bioorganic & medicinal chemistry letters, 1999-08, Vol.9 (16), p.2371-2374

1999

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Synthesis and Mixed Lineage Kinase Activity of Pyrrolocarbazole and Isoindolone Analogs of (+)K-252a

Journal of medicinal chemistry, 2007-02, Vol.50 (3), p.433-441

2007

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Novel Benzo[b]quinolizinium Cations as Uncompetitive N-Methyl-D-aspartic Acid (NMDA) Antagonists: The Relationship between log D and Agonist Independent (Closed) NMDA Channel Block

Journal of medicinal chemistry, 1995-09, Vol.38 (18), p.3586-3592

1995

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Identification, Synthesis, and Characterization of a Unique Class of N-Methyl-D-aspartate Antagonists. The 6,11-Ethanobenzo[b]quinolizinium Cation

Journal of medicinal chemistry, 1994-12, Vol.37 (26), p.4438-4448

1994

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Antiandrogenic steroidal sulfonyl heterocycles. Utility of electrostatic complementarity in defining bioisosteric sulfonyl heterocycles

Journal of medicinal chemistry, 1992-05, Vol.35 (10), p.1663-1670

1992

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Synthesis and structure-activity studies of some disubstituted phenylisoxazoles against human picornavirus

Journal of medicinal chemistry, 1989-02, Vol.32 (2), p.450-455

1989

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Calpain inhibitors based on the quiescent affinity label concept: high rates of calpain inactivation with leaving groups derived from N-hydroxy peptide coupling reagents

Bioorganic & medicinal chemistry letters, 2000-10, Vol.10 (20), p.2315-2319

2000

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An Evaluation of the Antirhinoviral Activity of Acylfuran Replacements for 3-Methylisoxazoles. Are 2-Acetylfurans Bioisosteres for 3-Methylisoxazoles?

Journal of medicinal chemistry, 1994-11, Vol.37 (24), p.4177-4184

1994

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Synthesis and Evaluation of 6,11-Ethanohexahydrobenzo[b]quinolizidines: A New Class of Noncompetitive N-Methyl-D-aspartate Antagonists

Journal of medicinal chemistry, 1995-06, Vol.38 (13), p.2483-2489

1995

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Novel NMDA Antagonists: Replacement of the Pyridinium Ring of 6,11-Ethanobenzo[b]quinolizinium Cations with Heteroisoquinolinium Cations

Journal of medicinal chemistry, 1995-05, Vol.38 (10), p.1826-1830

1995

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Discovery of 6,11-Ethano-12,12-diaryl-6,11-dihydrobenzo[b]quinolizinium Cations, a Novel Class of N-Methyl-D-aspartate Antagonists

Journal of medicinal chemistry, 1995-01, Vol.38 (1), p.21-27

1995

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Antiandrogenic steroidal sulfonylpyrazoles

Journal of medicinal chemistry, 1990-08, Vol.33 (8), p.2094-2100

1990

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Structure-guided identification of novel VEGFR-2 kinase inhibitors via solution phase parallel synthesis

Bioorganic & medicinal chemistry letters, 2006-04, Vol.16 (8), p.2158-2162

2006

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Antipicornavirus Compounds: Use of Rational Drug Design and Molecular Modelling

Antiviral Chemistry and Chemotherapy, 1993-02, Vol.4 (1), p.1-10

1993

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Structure-activity studies of 5-[[4-(4,5-dihydro-2-oxazolyl)phenoxy]alkyl]-3-methylisoxazoles: inhibitors of picornavirus uncoating

Journal of medicinal chemistry, 1987-02, Vol.30 (2), p.383-388

1987

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1,2-Benzothiazine 1,1-dioxide α-ketoamide analogues as potent calpain I inhibitors

Bioorganic & medicinal chemistry letters, 2004-02, Vol.14 (4), p.1035-1038

2004

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Novel Peptidyl Phosphorus Derivatives as Inhibitors of Human Calpain I

Neurotrophic 3,9-Bis[(alkylthio)methyl]- and -Bis(alkoxymethyl)-K-252a Derivatives

d-Amino Acid Containing, High-Affinity Inhibitors of Recombinant Human Calpain I

Synthesis and Biological Activity of a Series of Potent Fluoromethyl Ketone Inhibitors of Recombinant Human Calpain I

Antipicornavirus activity of tetrazole analogs related to disoxaril

Knowledge-Based, Central Nervous System (CNS) Lead Selection and Lead Optimization for CNS Drug Discovery

Prodrug esters of the indolocarbazole CEP-751 (KT-6587)

Knowledge-based chemoinformatic approaches to drug discovery

WIN 63480, a hydrophilic TCP-site ligand, has reduced agonist-independent NMDA ion channel access compared to MK-801 and phencyclidine

P2-ACHIRAL, P'-extended α-ketoamide inhibitors of calpain I

Synthesis and Mixed Lineage Kinase Activity of Pyrrolocarbazole and Isoindolone Analogs of (+)K-252a

Novel Benzo[b]quinolizinium Cations as Uncompetitive N-Methyl-D-aspartic Acid (NMDA) Antagonists: The Relationship between log D and Agonist Independent (Closed) NMDA Channel Block

Identification, Synthesis, and Characterization of a Unique Class of N-Methyl-D-aspartate Antagonists. The 6,11-Ethanobenzo[b]quinolizinium Cation

Antiandrogenic steroidal sulfonyl heterocycles. Utility of electrostatic complementarity in defining bioisosteric sulfonyl heterocycles

Synthesis and structure-activity studies of some disubstituted phenylisoxazoles against human picornavirus

Calpain inhibitors based on the quiescent affinity label concept: high rates of calpain inactivation with leaving groups derived from N-hydroxy peptide coupling reagents

An Evaluation of the Antirhinoviral Activity of Acylfuran Replacements for 3-Methylisoxazoles. Are 2-Acetylfurans Bioisosteres for 3-Methylisoxazoles?

Synthesis and Evaluation of 6,11-Ethanohexahydrobenzo[b]quinolizidines: A New Class of Noncompetitive N-Methyl-D-aspartate Antagonists

Novel NMDA Antagonists: Replacement of the Pyridinium Ring of 6,11-Ethanobenzo[b]quinolizinium Cations with Heteroisoquinolinium Cations

Discovery of 6,11-Ethano-12,12-diaryl-6,11-dihydrobenzo[b]quinolizinium Cations, a Novel Class of N-Methyl-D-aspartate Antagonists

Antiandrogenic steroidal sulfonylpyrazoles

Structure-guided identification of novel VEGFR-2 kinase inhibitors via solution phase parallel synthesis

Antipicornavirus Compounds: Use of Rational Drug Design and Molecular Modelling

Structure-activity studies of 5-[[4-(4,5-dihydro-2-oxazolyl)phenoxy]alkyl]-3-methylisoxazoles: inhibitors of picornavirus uncoating

1,2-Benzothiazine 1,1-dioxide α-ketoamide analogues as potent calpain I inhibitors

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