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Metal-Free TEMPO-Promoted C(sp3)–H Amination To Afford Multisubstituted Benzimidazoles

Journal of organic chemistry, 2014-05, Vol.79 (10), p.4727-4734

2014

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Solvent/Oxidant-Switchable Synthesis of Multisubstituted Quinazolines and Benzimidazoles via Metal-Free Selective Oxidative Annulation of Arylamidines

Organic letters, 2014-06, Vol.16 (11), p.2822-2825

2014

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Convergent synthesis of tetrahydropyranyl side chain of verucopeptin, an antitumor antibiotic active against multidrug-resistant cancers

Chemical communications (Cambridge, England), 2022-12, Vol.58 (97), p.13447-1345

2022

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Bioorthogonal chemistry: Optimization and application updates during 2013–2017

Tetrahedron letters, 2018-06, Vol.59 (23), p.2214-2228

2018

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Metal-free hypervalent iodine-promoted tandem carbonyl migration and unactivated C(Ph)-C(Alkyl) bond cleavage for quinolone scaffold synthesis

Chemical communications (Cambridge, England), 2022-07, Vol.58 (6), p.834-8343

2022

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Transition metal-free one-pot synthesis of 2-substituted 3-carboxy-4-quinolone and chromone derivatives

Chemical communications (Cambridge, England), 2013-01, Vol.49 (46), p.5313-5315

2013

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Discovery of a novel 5-carbonyl-1H-imidazole-4-carboxamide class of inhibitors of the HIV-1 integrase–LEDGF/p75 interaction

Bioorganic & medicinal chemistry, 2013-10, Vol.21 (19), p.5963-5972

2013

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Targeting Inactive Enzyme Conformation: Aryl Diketoacid Derivatives as a New Class of PTP1B Inhibitors

Journal of the American Chemical Society, 2008-12, Vol.130 (50), p.17075-17084

2008

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On-Demand Activation of a Bioorthogonal Prodrug of SN-38 with Fast Reaction Kinetics and High Releasing Efficiency In Vivo

Journal of medicinal chemistry, 2022-01, Vol.65 (1), p.333-342

2022

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Recent advances in the discovery of protein tyrosine phosphatase SHP2 inhibitors

RSC medicinal chemistry, 2022-03, Vol.13 (3), p.246-257

2022

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GPR40 agonists for the treatment of type 2 diabetes mellitus: The biological characteristics and the chemical space

Bioorganic & medicinal chemistry letters, 2016-12, Vol.26 (23), p.5603-5612

2016

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Rational Design and Synthesis of Novel Dimeric Diketoacid-Containing Inhibitors of HIV-1 Integrase: Implication for Binding to Two Metal Ions on the Active Site of Integrase

Journal of medicinal chemistry, 2004-05, Vol.47 (10), p.2561-2573

2004

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Direct Synthesis of 2‑Aryl-4-quinolones via Transition-Metal-Free Intramolecular Oxidative C(sp3)–H/C(sp3)–H Coupling

Organic letters, 2015-03, Vol.17 (5), p.1268-1271

2015

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Targeting the Hedgehog pathway with novel Gli1 hydrophobic tagging degraders

Bioorganic chemistry, 2023-09, Vol.138, p.106649-106649, Article 106649

2023

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The chemical diversity and structure-based evolution of non-peptide CXCR4 antagonists with diverse therapeutic potential

European journal of medicinal chemistry, 2018-04, Vol.149, p.148-169

2018

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Design, Synthesis, and Pharmacological Evaluation of 2‑(2,5-Dimethyl-5,6,7,8-tetrahydroquinolin-8-yl)‑N‑aryl Propanamides as Novel Smoothened (Smo) Antagonists

Journal of medicinal chemistry, 2016-12, Vol.59 (24), p.11050-11068

2016

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Discovery of Novel 2-N-Aryl-Substituted Benzenesulfonamidoacetamides: Orally Bioavailable Tubulin Polymerization Inhibitors with Marked Antitumor Activities

ChemMedChem, 2012-04, Vol.7 (4), p.680-693

2012

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Discovery of orally effective and safe GPR40 agonists by incorporating a chiral, rigid and polar sulfoxide into β-position to the carboxylic acid

European journal of medicinal chemistry, 2023-05, Vol.251, p.115267-115267, Article 115267

2023

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Discovery of Potent and Orally Bioavailable GPR40 Full Agonists Bearing Thiophen-2-ylpropanoic Acid Scaffold

Journal of medicinal chemistry, 2017-04, Vol.60 (7), p.2697-2717

2017

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Discovery and synthesis of 6,7,8,9-tetrahydro-5H-pyrido[4,3-c]azepin-5-one-based novel chemotype CCR2 antagonists via scaffold hopping strategy

Bioorganic & medicinal chemistry, 2018-07, Vol.26 (12), p.3559-3572

2018

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Clinical observation on scalp acupuncture combined with rehabilitation training for hemiplegia after stroke

Journal of acupuncture and tuina science, 2013-08, Vol.11 (4), p.226-229

Qiu, Ya-long

2013

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A novel proteolysis-resistant cyclic helix B peptide ameliorates kidney ischemia reperfusion injury

Biochimica et biophysica acta. Molecular basis of disease, 2014-11, Vol.1842 (11), p.2306-2317

2014

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4-Quinolone-3-carboxylic acids as cell-permeable inhibitors of protein tyrosine phosphatase 1B

Bioorganic & medicinal chemistry, 2014-07, Vol.22 (14), p.3670-3683

2014

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Studies toward the total synthesis of cyclodidemniserinol trisulfate. Part I: 3,5,7-Trisubstituted 6,8-dioxabicyclo [3.2.1] octane core structure construction via a convergent and a linear stereoselective synthesis

Tetrahedron letters, 2009-08, Vol.50 (32), p.4587-4591

2009

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Design of Cell-Permeable Stapled Peptides as HIV‑1 Integrase Inhibitors

Journal of medicinal chemistry, 2013-07, Vol.56 (13), p.5601-5612

2013

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Metal-Free TEMPO-Promoted C(sp3)–H Amination To Afford Multisubstituted Benzimidazoles

Solvent/Oxidant-Switchable Synthesis of Multisubstituted Quinazolines and Benzimidazoles via Metal-Free Selective Oxidative Annulation of Arylamidines

Convergent synthesis of tetrahydropyranyl side chain of verucopeptin, an antitumor antibiotic active against multidrug-resistant cancers

Bioorthogonal chemistry: Optimization and application updates during 2013–2017

Metal-free hypervalent iodine-promoted tandem carbonyl migration and unactivated C(Ph)-C(Alkyl) bond cleavage for quinolone scaffold synthesis

Transition metal-free one-pot synthesis of 2-substituted 3-carboxy-4-quinolone and chromone derivatives

Discovery of a novel 5-carbonyl-1H-imidazole-4-carboxamide class of inhibitors of the HIV-1 integrase–LEDGF/p75 interaction

Targeting Inactive Enzyme Conformation: Aryl Diketoacid Derivatives as a New Class of PTP1B Inhibitors

On-Demand Activation of a Bioorthogonal Prodrug of SN-38 with Fast Reaction Kinetics and High Releasing Efficiency In Vivo

Recent advances in the discovery of protein tyrosine phosphatase SHP2 inhibitors

GPR40 agonists for the treatment of type 2 diabetes mellitus: The biological characteristics and the chemical space

Rational Design and Synthesis of Novel Dimeric Diketoacid-Containing Inhibitors of HIV-1 Integrase: Implication for Binding to Two Metal Ions on the Active Site of Integrase

Direct Synthesis of 2‑Aryl-4-quinolones via Transition-Metal-Free Intramolecular Oxidative C(sp3)–H/C(sp3)–H Coupling

Targeting the Hedgehog pathway with novel Gli1 hydrophobic tagging degraders

The chemical diversity and structure-based evolution of non-peptide CXCR4 antagonists with diverse therapeutic potential

Design, Synthesis, and Pharmacological Evaluation of 2‑(2,5-Dimethyl-5,6,7,8-tetrahydroquinolin-8-yl)‑N‑aryl Propanamides as Novel Smoothened (Smo) Antagonists

Discovery of Novel 2-N-Aryl-Substituted Benzenesulfonamidoacetamides: Orally Bioavailable Tubulin Polymerization Inhibitors with Marked Antitumor Activities

Discovery of orally effective and safe GPR40 agonists by incorporating a chiral, rigid and polar sulfoxide into β-position to the carboxylic acid

Discovery of Potent and Orally Bioavailable GPR40 Full Agonists Bearing Thiophen-2-ylpropanoic Acid Scaffold

Discovery and synthesis of 6,7,8,9-tetrahydro-5H-pyrido[4,3-c]azepin-5-one-based novel chemotype CCR2 antagonists via scaffold hopping strategy

Clinical observation on scalp acupuncture combined with rehabilitation training for hemiplegia after stroke

A novel proteolysis-resistant cyclic helix B peptide ameliorates kidney ischemia reperfusion injury

4-Quinolone-3-carboxylic acids as cell-permeable inhibitors of protein tyrosine phosphatase 1B

Studies toward the total synthesis of cyclodidemniserinol trisulfate. Part I: 3,5,7-Trisubstituted 6,8-dioxabicyclo [3.2.1] octane core structure construction via a convergent and a linear stereoselective synthesis

Design of Cell-Permeable Stapled Peptides as HIV‑1 Integrase Inhibitors

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