UB Paderborn / Katalog / Suche / in CDI

Sortiert nach

Einfacher Volltextzugriff von (fast) überall

Installieren Sie die LibKey Nomad-Browsererweiterung und erhalten Sie von vielen Webseiten einfachen Zugriff auf lizenzierte Volltexte oder Open Access Publikationen. Mehr erfahren...

Analgesic Properties of Opioid/NK1 Multitarget Ligands with Distinct in Vitro Profiles in Naive and Chronic Constriction Injury Mice

ACS chemical neuroscience, 2017-10, Vol.8 (10), p.2315-2324

2017

Volltextzugriff (PDF)

Synthesis and biological evaluation of compact, conformationally constrained bifunctional opioid agonist – Neurokinin-1 antagonist peptidomimetics

European journal of medicinal chemistry, 2015-03, Vol.92, p.64-77

2015

Volltextzugriff (PDF)

‘Carba’-carfentanil (trans isomer): A μ opioid receptor (MOR) partial agonist with a distinct binding mode

Bioorganic & medicinal chemistry, 2014-09, Vol.22 (17), p.4581-4586

2014

Volltextzugriff (PDF)

Variation of the Net Charge, Lipophilicity, and Side Chain Flexibility in Dmt1‑DALDA: Effect on Opioid Activity and Biodistribution

Journal of medicinal chemistry, 2012-11, Vol.55 (22), p.9549-9561

2012

Volltextzugriff (PDF)

Variation of the net charge, lipophilicity, and side chain flexibility in Dmt(1)-DALDA: Effect on Opioid Activity and Biodistribution

Journal of medicinal chemistry, 2012-11, Vol.55 (22), p.9549

2012

Volltextzugriff (PDF)

Design of Novel Neurokinin 1 Receptor Antagonists Based on Conformationally Constrained Aromatic Amino Acids and Discovery of a Potent Chimeric Opioid Agonist-Neurokinin 1 Receptor Antagonist

Journal of medicinal chemistry, 2011-04, Vol.54 (7), p.2467-2476

2011

Volltextzugriff (PDF)

"Carba"-analogues of fentanyl are opioid receptor agonists

Journal of medicinal chemistry, 2010-04, Vol.53 (7), p.2875-2881

2010

Volltextzugriff (PDF)

Dicarba Analogues of the Cyclic Enkephalin Peptides H-Tyr-c[d-Cys-Gly-Phe-d(or l)-Cys]NH2 Retain High Opioid Activity

Journal of medicinal chemistry, 2007-03, Vol.50 (6), p.1414-1417

2007

Volltextzugriff (PDF)

Novel TIPP (H-Tyr-Tic-Phe-Phe-OH) analogues displaying a wide range of efficacies at the δ opioid receptor. Discovery of two highly potent and selective δ opioid agonists

Bioorganic & medicinal chemistry letters, 2012-03, Vol.22 (5), p.1899-1902

2012

Volltextzugriff (PDF)

Agonist vs Antagonist Behavior of δ Opioid Peptides Containing Novel Phenylalanine Analogues in Place of Tyr

Journal of medicinal chemistry, 2009-11, Vol.52 (21), p.6941-6945

2009

Volltextzugriff (PDF)

Synthesis and Characterization of Potent and Selective μ-Opioid Receptor Antagonists, [Dmt, d-2-Nal4]endomorphin-1 (Antanal-1) and [Dmt1, d-2-Nal4]endomorphin-2 (Antanal-2)

Journal of medicinal chemistry, 2007-02, Vol.50 (3), p.512-520

2007

Volltextzugriff (PDF)

Bifunctional μ/δ Opioid Peptides: Variation of the Type and Length of the Linker Connecting the Two Components

Chemical biology & drug design, 2012-02, Vol.79 (2), p.186-193

2012

Volltextzugriff (PDF)

Pseudoproline-Containing Analogues of Morphiceptin and Endomorphin-2: Evidence for a Cis Tyr−Pro Amide Bond in the Bioactive Conformation

Journal of medicinal chemistry, 2001-11, Vol.44 (23), p.3896-3903

2001

Volltextzugriff (PDF)

Variation of the Net Charge, Lipophilicity, and Side Chain Flexibility in Dmt 1 -DALDA: Effect on Opioid Activity and Biodistribution

Journal of medicinal chemistry, 2012-11, Vol.55 (22), p.9549-9561

2012

Volltextzugriff (PDF)

Blood−Brain Barrier Penetration by Two Dermorphin Tetrapeptide Analogues: Role of Lipophilicity vs Structural Flexibility

Journal of medicinal chemistry, 2008-04, Vol.51 (8), p.2571-2574

2008

Volltextzugriff (PDF)

Agonist vs Antagonist Behavior of δ Opioid Peptides Containing Novel Phenylalanine Analogues in Place of Tyr 1

Journal of medicinal chemistry, 2009-11, Vol.52 (21), p.6941-6945

2009

Volltextzugriff (PDF)

The Opioid μ Agonist/δ Antagonist DIPP-NH2[Ψ] Produces a Potent Analgesic Effect, No Physical Dependence, and Less Tolerance than Morphine in Rats

Journal of medicinal chemistry, 1999-09, Vol.42 (18), p.3520-3526

1999

Volltextzugriff (PDF)

Synthesis and in vitro opioid activity profiles of DALDA analogues

European journal of medicinal chemistry, 2000-10, Vol.35 (10), p.895-901

2000

Volltextzugriff (PDF)

Cyclic Opioid Peptide Agonists and Antagonists Obtained Via Ring-Closing Metathesis

Chemical biology & drug design, 2009-10, Vol.74 (4), p.329-334

2009

Volltextzugriff (PDF)

Structural Modifications of the N-terminal Tetrapeptide Segment of [D-Ala 2]Deltorphin I: Effects on Opioid Receptor Affinities and Activities In Vitro and on Antinociceptive Potency

Peptides (New York, N.Y. : 1980), 1997, Vol.18 (10), p.1615-1621

1997

Volltextzugriff (PDF)

[2‘,6‘-Dimethyltyrosine]Dynorphin A(1−11)-NH2 Analogues Lacking an N-Terminal Amino Group: Potent and Selective κ Opioid Antagonists

Journal of medicinal chemistry, 2001-09, Vol.44 (19), p.3048-3053

2001

Volltextzugriff (PDF)

“Carba”-Analogues of Fentanyl are Opioid Receptor Agonists ‡ Dedicated to the memory of Ralph F. Hirschmann

Journal of medicinal chemistry, 2010-04, Vol.53 (7), p.2875-2881

2010

Volltextzugriff (PDF)

N-Methylated Cyclic Enkephalin Analogues Retain High Opioid Receptor Binding Affinity

Chemical biology & drug design, 2010-02, Vol.75 (2), p.182-188

2010

Volltextzugriff (PDF)

Agonist vs Antagonist Behavior of δ Opioid Peptides Containing Novel Phenylalanine Analogues in Place of Tyr1

Journal of medicinal chemistry, 2009-11, Vol.52 (21), p.6941-6945

2009

Volltextzugriff (PDF)

Dicarba analogues of the cyclic enkephalin peptides H-Tyr-c[D-Cys-Gly-Phe-D(or L)-Cys]NH(2) retain high opioid activity

Journal of medicinal chemistry, 2007-03, Vol.50 (6), p.1414-1417

2007

Volltextzugriff (PDF)

1 – 25 von 113

Suche als RSS-Feed

Suchergebnisse filtern

Filter anzeigen

Nur zeigen

Geprüft (Peer-Review)
(108)
Mit Volltextzugriff
(105)

Publikationsform

Sprache

Englisch
(113)
Japanisch
(8)

Erscheinungsjahr

n.n

Thema

15 weitere anzeigen...

Weniger anzeigen...

Neu hinzugefügt

... seit 7 Tagen
(1)

Menü

Weitere Dienste

Einstellungen

Analgesic Properties of Opioid/NK1 Multitarget Ligands with Distinct in Vitro Profiles in Naive and Chronic Constriction Injury Mice

Synthesis and biological evaluation of compact, conformationally constrained bifunctional opioid agonist – Neurokinin-1 antagonist peptidomimetics

‘Carba’-carfentanil (trans isomer): A μ opioid receptor (MOR) partial agonist with a distinct binding mode

Variation of the Net Charge, Lipophilicity, and Side Chain Flexibility in Dmt1‑DALDA: Effect on Opioid Activity and Biodistribution

Variation of the net charge, lipophilicity, and side chain flexibility in Dmt(1)-DALDA: Effect on Opioid Activity and Biodistribution

Design of Novel Neurokinin 1 Receptor Antagonists Based on Conformationally Constrained Aromatic Amino Acids and Discovery of a Potent Chimeric Opioid Agonist-Neurokinin 1 Receptor Antagonist

"Carba"-analogues of fentanyl are opioid receptor agonists

Dicarba Analogues of the Cyclic Enkephalin Peptides H-Tyr-c[d-Cys-Gly-Phe-d(or l)-Cys]NH2 Retain High Opioid Activity

Novel TIPP (H-Tyr-Tic-Phe-Phe-OH) analogues displaying a wide range of efficacies at the δ opioid receptor. Discovery of two highly potent and selective δ opioid agonists

Agonist vs Antagonist Behavior of δ Opioid Peptides Containing Novel Phenylalanine Analogues in Place of Tyr

Synthesis and Characterization of Potent and Selective μ-Opioid Receptor Antagonists, [Dmt, d-2-Nal4]endomorphin-1 (Antanal-1) and [Dmt1, d-2-Nal4]endomorphin-2 (Antanal-2)

Bifunctional μ/δ Opioid Peptides: Variation of the Type and Length of the Linker Connecting the Two Components

Pseudoproline-Containing Analogues of Morphiceptin and Endomorphin-2: Evidence for a Cis Tyr−Pro Amide Bond in the Bioactive Conformation

Variation of the Net Charge, Lipophilicity, and Side Chain Flexibility in Dmt 1 -DALDA: Effect on Opioid Activity and Biodistribution

Blood−Brain Barrier Penetration by Two Dermorphin Tetrapeptide Analogues: Role of Lipophilicity vs Structural Flexibility

Agonist vs Antagonist Behavior of δ Opioid Peptides Containing Novel Phenylalanine Analogues in Place of Tyr 1

The Opioid μ Agonist/δ Antagonist DIPP-NH2[Ψ] Produces a Potent Analgesic Effect, No Physical Dependence, and Less Tolerance than Morphine in Rats

Synthesis and in vitro opioid activity profiles of DALDA analogues

Cyclic Opioid Peptide Agonists and Antagonists Obtained Via Ring-Closing Metathesis

Structural Modifications of the N-terminal Tetrapeptide Segment of [D-Ala 2]Deltorphin I: Effects on Opioid Receptor Affinities and Activities In Vitro and on Antinociceptive Potency

[2‘,6‘-Dimethyltyrosine]Dynorphin A(1−11)-NH2 Analogues Lacking an N-Terminal Amino Group: Potent and Selective κ Opioid Antagonists

“Carba”-Analogues of Fentanyl are Opioid Receptor Agonists ‡ Dedicated to the memory of Ralph F. Hirschmann

N-Methylated Cyclic Enkephalin Analogues Retain High Opioid Receptor Binding Affinity

Agonist vs Antagonist Behavior of δ Opioid Peptides Containing Novel Phenylalanine Analogues in Place of Tyr1

Dicarba analogues of the cyclic enkephalin peptides H-Tyr-c[D-Cys-Gly-Phe-D(or L)-Cys]NH(2) retain high opioid activity

Suchergebnisse filtern