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Redox Modification of Nuclear Actin by MICAL-2 Regulates SRF Signaling

Cell, 2014-01, Vol.156 (3), p.563-576

2014

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A Pan-ALDH1A Inhibitor Induces Necroptosis in Ovarian Cancer Stem-like Cells

Cell reports (Cambridge), 2019-03, Vol.26 (11), p.3061-3075.e6

2019

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Structure-Based Optimization of a Novel Class of Aldehyde Dehydrogenase 1A (ALDH1A) Subfamily-Selective Inhibitors as Potential Adjuncts to Ovarian Cancer Chemotherapy

Journal of medicinal chemistry, 2018-10, Vol.61 (19), p.8754-8773

2018

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Inhibition of Myocardin-Related Transcription Factor/Serum Response Factor Signaling Decreases Lung Fibrosis and Promotes Mesenchymal Cell Apoptosis

The American journal of pathology, 2015-04, Vol.185 (4), p.969-986

2015

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Structure-mechanism-based engineering of chemical regulators targeting distinct pathological factors in Alzheimer's disease

Nature communications, 2016-10, Vol.7 (1), p.13115-13, Article 13115

2016

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The development and use of small molecule inhibitors of glycosphingolipid metabolism for lysosomal storage diseases

Journal of lipid research, 2014-07, Vol.55 (7), p.1215-1225

2014

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Novel inhibitors of Staphylococcus aureus virulence gene expression and biofilm formation

PloS one, 2012-10, Vol.7 (10), p.e47255

2012

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Targeting the myofibroblast genetic switch: inhibitors of myocardin-related transcription factor/serum response factor-regulated gene transcription prevent fibrosis in a murine model of skin injury

The Journal of pharmacology and experimental therapeutics, 2014-06, Vol.349 (3), p.480

2014

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Physicochemical properties and formulation development of a novel compound inhibiting Staphylococcus aureus biofilm formation

PloS one, 2021-02, Vol.16 (2), p.e0246408-e0246408

2021

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Local delivery of novel MRTF/SRF inhibitors prevents scar tissue formation in a preclinical model of fibrosis

Scientific reports, 2017-03, Vol.7 (1), p.518-13, Article 518

2017

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Structure-Based Design, Synthesis, and Biological Evaluation of Highly Selective and Potent G Protein-Coupled Receptor Kinase 2 Inhibitors

Journal of medicinal chemistry, 2016-04, Vol.59 (8), p.3793-3807

2016

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Optimization of novel nipecotic bis(amide) inhibitors of the Rho/MKL1/SRF transcriptional pathway as potential anti-metastasis agents

Bioorganic & medicinal chemistry letters, 2013-07, Vol.23 (13), p.3826-3832

2013

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Structural Determinants Influencing the Potency and Selectivity of Indazole-Paroxetine Hybrid G Protein-Coupled Receptor Kinase 2 Inhibitors

Molecular pharmacology, 2017-12, Vol.92 (6), p.707-717

2017

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Utilizing a structure-based docking approach to develop potent G protein-coupled receptor kinase (GRK) 2 and 5 inhibitors

Bioorganic & medicinal chemistry letters, 2018-05, Vol.28 (9), p.1507-1515

2018

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Inhibitor of streptokinase gene expression improves survival after group A streptococcus infection in mice

Proceedings of the National Academy of Sciences - PNAS, 2012-02, Vol.109 (9), p.3469-3474

2012

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Structural and functional analysis of g protein-coupled receptor kinase inhibition by paroxetine and a rationally designed analog

Molecular pharmacology, 2014-02, Vol.85 (2), p.237-248

2014

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Pharmacological Inhibition of Myocardin-related Transcription Factor Pathway Blocks Lung Metastases of RhoC-Overexpressing Melanoma

Molecular cancer therapeutics, 2017-01, Vol.16 (1), p.193-204

2017

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In vitro and in vivo delivery of a sustained release nanocarrier-based formulation of an MRTF/SRF inhibitor in conjunctival fibrosis

Journal of nanobiotechnology, 2018-11, Vol.16 (1), p.97-11, Article 97

2018

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Optimization of Eliglustat-Based Glucosylceramide Synthase Inhibitors as Substrate Reduction Therapy for Gaucher Disease Type 3

ACS chemical neuroscience, 2020-10, Vol.11 (20), p.3464-3473

2020

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Optimization of Novel Indole-2-carboxamide Inhibitors of Neurotropic Alphavirus Replication

Journal of medicinal chemistry, 2013-11, Vol.56 (22), p.9222-9241

2013

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Prevention of bleomycin‐induced lung fibrosis via inhibition of the MRTF/SRF transcription pathway

Pharmacology research & perspectives, 2022-12, Vol.10 (6), p.e01028-n/a

2022

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Property-based design of a glucosylceramide synthase inhibitor that reduces glucosylceramide in the brain

Journal of lipid research, 2012-02, Vol.53 (2), p.282-291

2012

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Inhibitors of Mycobacterium tuberculosis DosRST signaling and persistence

Nature chemical biology, 2017-02, Vol.13 (2), p.218

2017

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Identification of Thieno[3,2-b]Pyrrole Derivatives as Novel Small Molecule Inhibitors of Neurotropic Alphaviruses

The Journal of infectious diseases, 2009-04, Vol.199 (7), p.950-957

2009

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Gedunin- and Khivorin-Derivatives Are Small-Molecule Partial Agonists for Adhesion G Protein-Coupled Receptors GPR56/ADGRG1 and GPR114/ADGRG5

Molecular pharmacology, 2018-05, Vol.93 (5), p.477-488

2018

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Redox Modification of Nuclear Actin by MICAL-2 Regulates SRF Signaling

A Pan-ALDH1A Inhibitor Induces Necroptosis in Ovarian Cancer Stem-like Cells

Structure-Based Optimization of a Novel Class of Aldehyde Dehydrogenase 1A (ALDH1A) Subfamily-Selective Inhibitors as Potential Adjuncts to Ovarian Cancer Chemotherapy

Inhibition of Myocardin-Related Transcription Factor/Serum Response Factor Signaling Decreases Lung Fibrosis and Promotes Mesenchymal Cell Apoptosis

Structure-mechanism-based engineering of chemical regulators targeting distinct pathological factors in Alzheimer's disease

The development and use of small molecule inhibitors of glycosphingolipid metabolism for lysosomal storage diseases

Novel inhibitors of Staphylococcus aureus virulence gene expression and biofilm formation

Targeting the myofibroblast genetic switch: inhibitors of myocardin-related transcription factor/serum response factor-regulated gene transcription prevent fibrosis in a murine model of skin injury

Physicochemical properties and formulation development of a novel compound inhibiting Staphylococcus aureus biofilm formation

Local delivery of novel MRTF/SRF inhibitors prevents scar tissue formation in a preclinical model of fibrosis

Structure-Based Design, Synthesis, and Biological Evaluation of Highly Selective and Potent G Protein-Coupled Receptor Kinase 2 Inhibitors

Optimization of novel nipecotic bis(amide) inhibitors of the Rho/MKL1/SRF transcriptional pathway as potential anti-metastasis agents

Structural Determinants Influencing the Potency and Selectivity of Indazole-Paroxetine Hybrid G Protein-Coupled Receptor Kinase 2 Inhibitors

Utilizing a structure-based docking approach to develop potent G protein-coupled receptor kinase (GRK) 2 and 5 inhibitors

Inhibitor of streptokinase gene expression improves survival after group A streptococcus infection in mice

Structural and functional analysis of g protein-coupled receptor kinase inhibition by paroxetine and a rationally designed analog

Pharmacological Inhibition of Myocardin-related Transcription Factor Pathway Blocks Lung Metastases of RhoC-Overexpressing Melanoma

In vitro and in vivo delivery of a sustained release nanocarrier-based formulation of an MRTF/SRF inhibitor in conjunctival fibrosis

Optimization of Eliglustat-Based Glucosylceramide Synthase Inhibitors as Substrate Reduction Therapy for Gaucher Disease Type 3

Optimization of Novel Indole-2-carboxamide Inhibitors of Neurotropic Alphavirus Replication

Prevention of bleomycin‐induced lung fibrosis via inhibition of the MRTF/SRF transcription pathway

Property-based design of a glucosylceramide synthase inhibitor that reduces glucosylceramide in the brain

Inhibitors of Mycobacterium tuberculosis DosRST signaling and persistence

Identification of Thieno[3,2-b]Pyrrole Derivatives as Novel Small Molecule Inhibitors of Neurotropic Alphaviruses

Gedunin- and Khivorin-Derivatives Are Small-Molecule Partial Agonists for Adhesion G Protein-Coupled Receptors GPR56/ADGRG1 and GPR114/ADGRG5

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