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Voltage sensor interaction site for selective small molecule inhibitors of voltage-gated sodium channels

Proceedings of the National Academy of Sciences - PNAS, 2013-07, Vol.110 (29), p.E2724-E2732

2013

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A comprehensive approach to identifying repurposed drugs to treat SCN8A epilepsy

Epilepsia (Copenhagen), 2018-04, Vol.59 (4), p.802-813

2018

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A-803467, a potent and selective Nav1.8 sodium channel blocker, attenuates neuropathic and inflammatory pain in the rat

Proceedings of the National Academy of Sciences - PNAS, 2007-05, Vol.104 (20), p.8520-8525

2007

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Sodium channels and nociception: recent concepts and therapeutic opportunities

Current opinion in pharmacology, 2008-02, Vol.8 (1), p.50-56

2008

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A-887826 is a structurally novel, potent and voltage-dependent Na(v)1.8 sodium channel blocker that attenuates neuropathic tactile allodynia in rats

Neuropharmacology, 2010-09, Vol.59 (3), p.201-207

2010

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Discovery and biological evaluation of potent, selective, orally bioavailable, pyrazine-based blockers of the Na(v)1.8 sodium channel with efficacy in a model of neuropathic pain

Bioorganic & medicinal chemistry, 2010-11, Vol.18 (22), p.7816-7825

2010

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Discovery and biological evaluation of potent, selective, orally bioavailable, pyrazine-based blockers of the Nav1.8 sodium channel with efficacy in a model of neuropathic pain

Bioorganic & medicinal chemistry, 2010-11, Vol.18 (22), p.7816-7825

2010

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Subtype-selective Na(v)1.8 sodium channel blockers: identification of potent, orally active nicotinamide derivatives

Bioorganic & medicinal chemistry letters, 2010-11, Vol.20 (22), p.6812-6815

2010

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Block of Nav1.8 by Small Molecules

Channels (Austin, Tex.), 2007-05, Vol.1 (3), p.152-153

2007

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The Effect of κ-Opioid Receptor Agonists on Tetrodotoxin-Resistant Sodium Channels in Primary Sensory Neurons

Anesthesia and analgesia, 2009-08, Vol.109 (2), p.632-640

2009

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Ion channels: applications in ion channel drug discovery

Combinatorial chemistry & high throughput screening, 2009-01, Vol.12 (1), p.1

Krafte, Douglas S

2009

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Direct Activation of an Inwardly Rectifying Potassium Channel by Arachidonic Acid

Molecular pharmacology, 2001-05, Vol.59 (5), p.1061-1068

2001

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Tenidap, a novel anti-inflammatory agent, is an opener of the inwardly rectifying K + channel hKir2.3

European journal of pharmacology, 2002-01, Vol.435 (2), p.153-160

2002

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Decrease of inward rectification as a mechanism for arachidonic acid-induced potentiation of hKir2.3

European biophysics journal, 2002-12, Vol.31 (7), p.497-503

2002

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A comprehensive approach to identifying repurposed drugs to treat SCN 8A epilepsy

Epilepsia (Copenhagen), 2018-04, Vol.59 (4), p.802-813

2018

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Synthesis and Structure-Activity Relationships of 6-Heterocyclic-Substituted Purines as Inactivation Modifiers of Cardiac Sodium Channels

Journal of medicinal chemistry, 1995-07, Vol.38 (14), p.2582-2595

1995

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A-887826 is a structurally novel, potent and voltage-dependent Nav1.8 sodium channel blocker that attenuates neuropathic tactile allodynia in rats

Neuropharmacology, 2010-09, Vol.59 (3), p.201-207

2010

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Novel Inhibitors of Potassium Ion Channels on Human T Lymphocytes

Journal of medicinal chemistry, 1995-05, Vol.38 (11), p.1877-1883

1995

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Subtype-selective Na sub(v)1.8 sodium channel blockers: Identification of potent, orally active nicotinamide derivatives

Bioorganic & medicinal chemistry letters, 2010-11, Vol.20 (22), p.6812-6815

2010

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Voltage Dependence of Cardiac Delayed Rectifier Block by Methanesulfonamide Class III Antiarrhythmic Agents

Journal of cardiovascular pharmacology, 1994-01, Vol.23 (1), p.37-41

1994

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An interview with Douglas S. Krafte, Ph.D. Interview by Vicki P. Glaser

Assay and drug development technologies, 2006-02, Vol.4 (1), p.1

Krafte, Douglas S

2006

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Voltage sensor interaction site for selective small molecule inhibitors of voltage-gated sodium channels

Proceedings of the National Academy of Sciences - PNAS, 2013-07, Vol.110 (29), p.11675-11675

2013

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Identification of a Specific Radioligand for the Cardiac Rapidly Activating Delayed Rectifier K+ Channel

Circulation research, 1993-03, Vol.72 (3), p.707-714

1993

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Subtype-selective Nav1.8 sodium channel blockers: Identification of potent, orally active nicotinamide derivatives

Bioorganic & medicinal chemistry letters, 2010-11, Vol.20 (22), p.6812-6815

2010

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Voltage sensor interaction site for selective small molecule inhibitors of voltage-gated sodium channels

A comprehensive approach to identifying repurposed drugs to treat SCN8A epilepsy

A-803467, a potent and selective Nav1.8 sodium channel blocker, attenuates neuropathic and inflammatory pain in the rat

Sodium channels and nociception: recent concepts and therapeutic opportunities

A-887826 is a structurally novel, potent and voltage-dependent Na(v)1.8 sodium channel blocker that attenuates neuropathic tactile allodynia in rats

Discovery and Biological Evaluation of 5-Aryl-2-furfuramides, Potent and Selective Blockers of the Nav1.8 Sodium Channel with Efficacy in Models of Neuropathic and Inflammatory Pain

Discovery and biological evaluation of potent, selective, orally bioavailable, pyrazine-based blockers of the Na(v)1.8 sodium channel with efficacy in a model of neuropathic pain

Discovery and biological evaluation of potent, selective, orally bioavailable, pyrazine-based blockers of the Nav1.8 sodium channel with efficacy in a model of neuropathic pain

Subtype-selective Na(v)1.8 sodium channel blockers: identification of potent, orally active nicotinamide derivatives

Block of Nav1.8 by Small Molecules

The Effect of κ-Opioid Receptor Agonists on Tetrodotoxin-Resistant Sodium Channels in Primary Sensory Neurons

Ion channels: applications in ion channel drug discovery

Direct Activation of an Inwardly Rectifying Potassium Channel by Arachidonic Acid

Tenidap, a novel anti-inflammatory agent, is an opener of the inwardly rectifying K + channel hKir2.3

Decrease of inward rectification as a mechanism for arachidonic acid-induced potentiation of hKir2.3

A comprehensive approach to identifying repurposed drugs to treat SCN 8A epilepsy

Synthesis and Structure-Activity Relationships of 6-Heterocyclic-Substituted Purines as Inactivation Modifiers of Cardiac Sodium Channels

A-887826 is a structurally novel, potent and voltage-dependent Nav1.8 sodium channel blocker that attenuates neuropathic tactile allodynia in rats

Novel Inhibitors of Potassium Ion Channels on Human T Lymphocytes

Subtype-selective Na sub(v)1.8 sodium channel blockers: Identification of potent, orally active nicotinamide derivatives

Voltage Dependence of Cardiac Delayed Rectifier Block by Methanesulfonamide Class III Antiarrhythmic Agents

An interview with Douglas S. Krafte, Ph.D. Interview by Vicki P. Glaser

Voltage sensor interaction site for selective small molecule inhibitors of voltage-gated sodium channels

Identification of a Specific Radioligand for the Cardiac Rapidly Activating Delayed Rectifier K+ Channel

Subtype-selective Nav1.8 sodium channel blockers: Identification of potent, orally active nicotinamide derivatives

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