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Synthesis of Novel GABA Uptake Inhibitors. 3. Diaryloxime and Diarylvinyl Ether Derivatives of Nipecotic Acid and Guvacine as Anticonvulsant Agents

Journal of medicinal chemistry, 1999-09, Vol.42 (18), p.3447-3462

1999

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Synthesis of Novel GABA Uptake Inhibitors. 4. Bioisosteric Transformation and Successive Optimization of Known GABA Uptake Inhibitors Leading to a Series of Potent Anticonvulsant Drug Candidates

Journal of medicinal chemistry, 1999-10, Vol.42 (21), p.4281-4291

1999

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Characterization of tiagabine (NO-328), a new potent and selective GABA uptake inhibitor

European journal of pharmacology, 1991-04, Vol.196 (3), p.257,IN1,261,IN3,263-260,IN2,262,IN4,266

1991

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NNC-711, a novel potent and selective γ-aminobutyric acid uptake inhibitor: pharmacological characterization

European journal of pharmacology, 1992-12, Vol.224 (2), p.189-198

1992

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The synthesis of new adenosine A3 selective ligands containing bioisosteric isoxazoles

Bioorganic & medicinal chemistry letters, 1998-07, Vol.8 (13), p.1767-1770

1998

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Contrasting effects of adenosine A1 and A2 receptor ligands in different chemoconvulsive rodent models

European journal of pharmacology, 1993-10, Vol.242 (3), p.221-228

1993

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N-Substituted Adenosines as Novel Neuroprotective A1 Agonists with Diminished Hypotensive Effects

Journal of medicinal chemistry, 1999-09, Vol.42 (18), p.3463-3477

1999

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N-substituted adenosines as novel neuroprotective A(1) agonists with diminished hypotensive effects

Journal of medicinal chemistry, 1999-09, Vol.42 (18), p.3463-3477

1999

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The synthesis of novel GABA uptake inhibitors. 1. Elucidation of the structure-activity studies leading to the choice of (R)-1-[4,4-bis(3-methyl-2-thienyl)-3-butenyl]-3-piperidinecarboxylic acid (Tiagabine) as an anticonvulsant drug candidate

Journal of medicinal chemistry, 1993-06, Vol.36 (12), p.1716-1725

1993

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KW-6002 (Kyowa Hakko Kogyo)

Current opinion in investigational drugs (London, England : 2000), 2001-05, Vol.2 (5), p.668

2001

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(R)‐N‐[4,4‐Bis(3‐Methyl‐2‐Thienyl)but‐3‐en‐1‐yl]Nipecotic Acid Binds with High Affinity to the Brain γ‐Aminobutyric Acid Uptake Carrier

Journal of neurochemistry, 1990-02, Vol.54 (2), p.639-647

1990

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Reliability and validity of high-frequency (8-20 kHz) thresholds obtained on a computer-based audiometer as compared to a documented laboratory system

Journal of the American Academy of Audiology, 1990-07, Vol.1 (3), p.162

1990

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In vivo labeling of the central GABA uptake carrier with 3H-tiagabine

Life sciences (1973), 1992, Vol.51 (24), p.1857-1868

1992

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Unexpected neuroprotection observed with the adenosine A2A receptor agonist CGS 21680

Drug development research, 1996-09, Vol.39 (1), p.108-114

1996

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Adenosine A1 and A3 selective N-alkoxypurines as novel cytokine modulators and neuroprotectants

Drug development research, 1998-11, Vol.45 (3-4), p.214-221

1998

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The synthesis and biochemical evaluation of new A1 selective adenosine receptor agonists containing 6-hydrazinopurine moieties

Bioorganic & medicinal chemistry letters, 1993-12, Vol.3 (12), p.2661-2666

1993

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14C-labelling of a novel antiischaemic adenosine A1 agonist at purine C-8

Journal of labelled compounds & radiopharmaceuticals, 1996-05, Vol.38 (5), p.497-507

1996

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Synthesis and antiviral properties of 5-(2-substituted vinyl)-6-aza-2'-deoxyuridines

Journal of medicinal chemistry, 1986-05, Vol.29 (5), p.809-816

1986

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Synthesis of [8-14C]-2,6-dichloro-9H-purine, a radiolabelled precursor for 14C-nucleosides

Journal of labelled compounds & radiopharmaceuticals, 1995-05, Vol.36 (5), p.457-464

1995

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ChemInform Abstract: The Chemistry of 2′-Deoxyribo-C-nucleosides

ChemInform, 1992-10, Vol.23 (40), p.no-no

KNUTSEN, L. J. S.

1992

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The synthesis of novel GABA uptake inhibitors. I: Elucidation of the structure-activity studies leading to the choice of (R)-1-[4,4-bis(3-methyl-2-thienyl)-3-butenyl]-3-piperidinecarboxylic acid (tiagabine) as an anticonvulsant drug candidate

Journal of medicinal chemistry, 1993, Vol.36 (12), p.1716-1725

1993

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The Chemistry of 2′-Deoxyribo-C-Nucleosides

Nucleosides & nucleotides, 1992-06, Vol.11 (5), p.961-983

Knutsen, Lars J. S.

1992

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(R)-N-[4,4-bis(3-methyl-2-thienyl)but-3-en-1-yl]nipecotic acids binds with high affinity to the brain γ-aminobutyric acid uptake carrier

Journal of neurochemistry, 1990, Vol.54 (2), p.639-647

1990

Volltextzugriff (PDF)

ChemInform Abstract: The Synthesis of New Adenosine A3 Selective Ligands Containing Bioisosteric Isoxazoles

ChemInform, 1998-11, Vol.29 (47), p.no-no

1998

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ChemInform Abstract: The Synthesis of New Adenosine A 3 Selective Ligands Containing Bioisosteric Isoxazoles

ChemInform, 1998-11, Vol.29 (47)

1998

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Synthesis of Novel GABA Uptake Inhibitors. 3. Diaryloxime and Diarylvinyl Ether Derivatives of Nipecotic Acid and Guvacine as Anticonvulsant Agents

Synthesis of Novel GABA Uptake Inhibitors. 4. Bioisosteric Transformation and Successive Optimization of Known GABA Uptake Inhibitors Leading to a Series of Potent Anticonvulsant Drug Candidates

Characterization of tiagabine (NO-328), a new potent and selective GABA uptake inhibitor

NNC-711, a novel potent and selective γ-aminobutyric acid uptake inhibitor: pharmacological characterization

The synthesis of new adenosine A3 selective ligands containing bioisosteric isoxazoles

Contrasting effects of adenosine A1 and A2 receptor ligands in different chemoconvulsive rodent models

N-Substituted Adenosines as Novel Neuroprotective A1 Agonists with Diminished Hypotensive Effects

N-substituted adenosines as novel neuroprotective A(1) agonists with diminished hypotensive effects

The synthesis of novel GABA uptake inhibitors. 1. Elucidation of the structure-activity studies leading to the choice of (R)-1-[4,4-bis(3-methyl-2-thienyl)-3-butenyl]-3-piperidinecarboxylic acid (Tiagabine) as an anticonvulsant drug candidate

KW-6002 (Kyowa Hakko Kogyo)

(R)‐N‐[4,4‐Bis(3‐Methyl‐2‐Thienyl)but‐3‐en‐1‐yl]Nipecotic Acid Binds with High Affinity to the Brain γ‐Aminobutyric Acid Uptake Carrier

Reliability and validity of high-frequency (8-20 kHz) thresholds obtained on a computer-based audiometer as compared to a documented laboratory system

In vivo labeling of the central GABA uptake carrier with 3H-tiagabine

Unexpected neuroprotection observed with the adenosine A2A receptor agonist CGS 21680

Adenosine A1 and A3 selective N-alkoxypurines as novel cytokine modulators and neuroprotectants

The synthesis and biochemical evaluation of new A1 selective adenosine receptor agonists containing 6-hydrazinopurine moieties

14C-labelling of a novel antiischaemic adenosine A1 agonist at purine C-8

Synthesis and antiviral properties of 5-(2-substituted vinyl)-6-aza-2'-deoxyuridines

Synthesis of [8-14C]-2,6-dichloro-9H-purine, a radiolabelled precursor for 14C-nucleosides

ChemInform Abstract: The Chemistry of 2′-Deoxyribo-C-nucleosides

The synthesis of novel GABA uptake inhibitors. I: Elucidation of the structure-activity studies leading to the choice of (R)-1-[4,4-bis(3-methyl-2-thienyl)-3-butenyl]-3-piperidinecarboxylic acid (tiagabine) as an anticonvulsant drug candidate

The Chemistry of 2′-Deoxyribo-C-Nucleosides

(R)-N-[4,4-bis(3-methyl-2-thienyl)but-3-en-1-yl]nipecotic acids binds with high affinity to the brain γ-aminobutyric acid uptake carrier

ChemInform Abstract: The Synthesis of New Adenosine A3 Selective Ligands Containing Bioisosteric Isoxazoles

ChemInform Abstract: The Synthesis of New Adenosine A 3 Selective Ligands Containing Bioisosteric Isoxazoles

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