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New compound sets identified from high throughput phenotypic screening against three kinetoplastid parasites: an open resource

Scientific reports, 2015-03, Vol.5 (1), p.8771-8771, Article 8771

2015

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Hit-to-Lead Optimization of a Novel Class of Potent, Broad-Spectrum Trypanosomacides

Journal of medicinal chemistry, 2016-11, Vol.59 (21), p.9686-9720

2016

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Positive and Negative Allosteric Modulators of the Ca2+-sensing Receptor Interact within Overlapping but Not Identical Binding Sites in the Transmembrane Domain

The Journal of biological chemistry, 2004-04, Vol.279 (18), p.18990-18997

2004

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Novel chemical starting points for drug discovery in leishmaniasis and Chagas disease

International journal for parasitology -- drugs and drug resistance, 2019-08, Vol.10, p.58-68

2019

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Modeling and Mutagenesis of the Binding Site of Calhex 231, a Novel Negative Allosteric Modulator of the Extracellular Ca2+-sensing Receptor

The Journal of biological chemistry, 2003-12, Vol.278 (49), p.49487-49494

2003

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Novel Diarylthioether Compounds as Agents for the Treatment of Chagas Disease

Journal of medicinal chemistry, 2023-01, Vol.66 (2), p.1522-1542

2023

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Short-course combination treatment for experimental chronic Chagas disease

Science translational medicine, 2023-12, Vol.15 (726), p.eadg8105

2023

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A novel class of fast‐acting antimalarial agents: Substituted 15‐membered azalides

British journal of pharmacology, 2021-01, Vol.178 (2), p.363-377

2021

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Discovery of Potent N‑Ethylurea Pyrazole Derivatives as Dual Inhibitors of Trypanosoma brucei and Trypanosoma cruzi

ACS medicinal chemistry letters, 2020-03, Vol.11 (3), p.278-285

2020

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The Qi Site of Cytochrome b is a Promiscuous Drug Target in Trypanosoma cruzi and Leishmania donovani

ACS infectious diseases, 2020-03, Vol.6 (3), p.515-528

2020

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N -Benzoyl-N -[1-(1-naphthyl)ethyl]-trans-1,2-diaminocyclohexanes: Development of 4-Chlorophenylcarboxamide (Calhex 231) as a New Calcium Sensing Receptor Ligand Demonstrating Potent Calcilytic Activity

Journal of medicinal chemistry, 2006-08, Vol.49 (17), p.5119-5128

2006

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Rose Bengal analogs and vesicular glutamate transporters (VGLUTs)

Bioorganic & medicinal chemistry, 2010-09, Vol.18 (18), p.6922-6933

2010

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The Q i Site of Cytochrome b is a Promiscuous Drug Target in Trypanosoma cruzi and Leishmania donovani

ACS infectious diseases, 2020-03, Vol.6 (3), p.515-528

2020

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Indole Synthesis by Controlled Carbolithiation of o-Aminostyrenes

Journal of organic chemistry, 2004-11, Vol.69 (23), p.7836-7846

2004

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Molecular Tongs Containing Amino Acid Mimetic Fragments: New Inhibitors of Wild-Type and Mutated HIV-1 Protease Dimerization

Journal of medicinal chemistry, 2006-07, Vol.49 (15), p.4657-4664

2006

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Cyclopropyl Carboxamides: A New Oral Antimalarial Series Derived from the Tres Cantos Anti-Malarial Set (TCAMS)

ACS medicinal chemistry letters, 2011-11, Vol.2 (11), p.840-844

2011

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N(1)-Arylsulfonyl-N(2)-(1-(1-naphthyl)ethyl)-1,2-diaminocyclohexanes: a new class of calcilytic agents acting at the calcium-sensing receptor

Chembiochem : a European journal of chemical biology, 2004-08, Vol.5 (8), p.1131-1136

2004

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N 1 ‐Arylsulfonyl‐ N 2 ‐(1‐(1‐naphthyl)ethyl)‐1,2‐diaminocyclohexanes: A New Class of Calcilytic Agents Acting at the Calcium‐Sensing Receptor

Chembiochem : a European journal of chemical biology, 2004-08, Vol.5 (8), p.1131-1136

2004

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N1-benzoyl-N2-[1-(1-naphthyl)ethyl]-trans-1,2-diaminocyclohexanes : Development of 4-chlorophenylcarboxamide (Calhex 231) as a new calcium sensing receptor ligand demonstrating potent calcilytic activity

Journal of medicinal chemistry, 2006-08, Vol.49 (17), p.5119-5128

2006

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Molecular determinants of allosteric modulators of the calcium-sensing receptor

Journal of physiology, Paris, 2006-03, Vol.99 (2), p.2-3

2006

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N2-Benzyl- N1-(1-(1-naphthyl)ethyl)-3-phenylpropane-1,2-diamines and conformationally restrained indole analogues: development of calindol as a new calcimimetic acting at the calcium sensing receptor

Bioorganic & medicinal chemistry letters, 2004-06, Vol.14 (12), p.3345-3349

2004

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N1-Arylsulfonyl-N2-(1-(1-naphthyl)ethyl)-1,2-diaminocyclohexanes: A New Class of Calcilytic Agents Acting at the Calcium-Sensing Receptor

Chembiochem : a European journal of chemical biology, 2004-08, Vol.5 (8), p.1131-1136

2004

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N super(1)-Arylsulfonyl-N super(2)-(1-(1-naphthyl)ethyl)-1,2-diaminocyclohexanes: A New Class of Calcilytic Agents Acting at the Calcium-Sensing Receptor

Chembiochem : a European journal of chemical biology, 2004-01, Vol.5 (8), p.1131-1136

2004

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SUZUKI-MIYAURA CROSS-COUPLING: PREPARATION OF 2'-VINYLACETANILIDE

Organic syntheses, 2006, Vol.83, p.45

2006

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Indole Synthesis by Controlled Carbolithiation of o-Aminostyrenes

ChemInform, 2005-03, Vol.36 (12), p.no-no

2005

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New compound sets identified from high throughput phenotypic screening against three kinetoplastid parasites: an open resource

Hit-to-Lead Optimization of a Novel Class of Potent, Broad-Spectrum Trypanosomacides

Positive and Negative Allosteric Modulators of the Ca2+-sensing Receptor Interact within Overlapping but Not Identical Binding Sites in the Transmembrane Domain

Novel chemical starting points for drug discovery in leishmaniasis and Chagas disease

Modeling and Mutagenesis of the Binding Site of Calhex 231, a Novel Negative Allosteric Modulator of the Extracellular Ca2+-sensing Receptor

Novel Diarylthioether Compounds as Agents for the Treatment of Chagas Disease

Short-course combination treatment for experimental chronic Chagas disease

A novel class of fast‐acting antimalarial agents: Substituted 15‐membered azalides

Discovery of Potent N‑Ethylurea Pyrazole Derivatives as Dual Inhibitors of Trypanosoma brucei and Trypanosoma cruzi

The Qi Site of Cytochrome b is a Promiscuous Drug Target in Trypanosoma cruzi and Leishmania donovani

N -Benzoyl-N -[1-(1-naphthyl)ethyl]-trans-1,2-diaminocyclohexanes: Development of 4-Chlorophenylcarboxamide (Calhex 231) as a New Calcium Sensing Receptor Ligand Demonstrating Potent Calcilytic Activity

Rose Bengal analogs and vesicular glutamate transporters (VGLUTs)

The Q i Site of Cytochrome b is a Promiscuous Drug Target in Trypanosoma cruzi and Leishmania donovani

Indole Synthesis by Controlled Carbolithiation of o-Aminostyrenes

Molecular Tongs Containing Amino Acid Mimetic Fragments: New Inhibitors of Wild-Type and Mutated HIV-1 Protease Dimerization

Cyclopropyl Carboxamides: A New Oral Antimalarial Series Derived from the Tres Cantos Anti-Malarial Set (TCAMS)

N(1)-Arylsulfonyl-N(2)-(1-(1-naphthyl)ethyl)-1,2-diaminocyclohexanes: a new class of calcilytic agents acting at the calcium-sensing receptor

N 1 ‐Arylsulfonyl‐ N 2 ‐(1‐(1‐naphthyl)ethyl)‐1,2‐diaminocyclohexanes: A New Class of Calcilytic Agents Acting at the Calcium‐Sensing Receptor

N1-benzoyl-N2-[1-(1-naphthyl)ethyl]-trans-1,2-diaminocyclohexanes : Development of 4-chlorophenylcarboxamide (Calhex 231) as a new calcium sensing receptor ligand demonstrating potent calcilytic activity

Molecular determinants of allosteric modulators of the calcium-sensing receptor

N2-Benzyl- N1-(1-(1-naphthyl)ethyl)-3-phenylpropane-1,2-diamines and conformationally restrained indole analogues: development of calindol as a new calcimimetic acting at the calcium sensing receptor

N1-Arylsulfonyl-N2-(1-(1-naphthyl)ethyl)-1,2-diaminocyclohexanes: A New Class of Calcilytic Agents Acting at the Calcium-Sensing Receptor

N super(1)-Arylsulfonyl-N super(2)-(1-(1-naphthyl)ethyl)-1,2-diaminocyclohexanes: A New Class of Calcilytic Agents Acting at the Calcium-Sensing Receptor

SUZUKI-MIYAURA CROSS-COUPLING: PREPARATION OF 2'-VINYLACETANILIDE

Indole Synthesis by Controlled Carbolithiation of o-Aminostyrenes

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