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Lessons from crystal structures of kainate receptors

Neuropharmacology, 2017-01, Vol.112 (Pt A), p.16-28

2017

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Binding of a negative allosteric modulator and competitive antagonist can occur simultaneously at the ionotropic glutamate receptor GluA2

The FEBS journal, 2021-02, Vol.288 (3), p.995-1007

2021

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7‑Phenoxy-Substituted 3,4-Dihydro‑2H‑1,2,4-benzothiadiazine 1,1-Dioxides as Positive Allosteric Modulators of α‑Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid (AMPA) Receptors with Nanomolar Potency

Journal of medicinal chemistry, 2018-01, Vol.61 (1), p.251-264

2018

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Exploring thienothiadiazine dioxides as isosteric analogues of benzo- and pyridothiadiazine dioxides in the search of new AMPA and kainate receptor positive allosteric modulators

European journal of medicinal chemistry, 2024-01, Vol.264, p.116036-116036, Article 116036

2024

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The Structure of a High-Affinity Kainate Receptor: GluK4 Ligand-Binding Domain Crystallized with Kainate

Structure (London), 2016-09, Vol.24 (9), p.1582-1589

2016

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Neuroplastin-55 binds to and signals through the fibroblast growth factor receptor

The FASEB journal, 2010-04, Vol.24 (4), p.1139-1150

2010

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Structural Characterization of the Stringent Response Related Exopolyphosphatase/Guanosine Pentaphosphate Phosphohydrolase Protein Family

Biochemistry (Easton), 2004-07, Vol.43 (28), p.8894-8900

2004

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Structural basis for positive allosteric modulation of AMPA and kainate receptors

The Journal of physiology, 2022-01, Vol.600 (2), p.181-200

2022

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Small Angle X-ray Studies Reveal That Aspergillus niger Glucoamylase Has a Defined Extended Conformation and Can Form Dimers in Solution

The Journal of biological chemistry, 2008-05, Vol.283 (21), p.14772-14780

2008

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Recovery from desensitization in GluA2 AMPA receptors is affected by a single mutation in the N-terminal domain interface

The Journal of biological chemistry, 2024-03, Vol.300 (3), p.105717-105717, Article 105717

2024

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Tyr702 Is an Important Determinant of Agonist Binding and Domain Closure of the Ligand-Binding Core of GluR2

Molecular pharmacology, 2005-03, Vol.67 (3), p.703-713

2005

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Enhancing Action of Positive Allosteric Modulators through the Design of Dimeric Compounds

Journal of medicinal chemistry, 2018-06, Vol.61 (12), p.5279-5291

2018

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Differences between the GluD1 and GluD2 receptors revealed by GluD1 X‐ray crystallography, binding studies and molecular dynamics

The FEBS journal, 2023-08, Vol.290 (15), p.3781-3801

2023

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The positive allosteric modulator BPAM344 and L‐glutamate introduce an active‐like structure of the ligand‐binding domain of GluK2

FEBS letters, 2024-04, Vol.598 (7), p.743-757

2024

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Lessons from more than 80 structures of the GluA2 ligand-binding domain in complex with agonists, antagonists and allosteric modulators

Neuropharmacology, 2011, Vol.60 (1), p.135-150

2011

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Identification and Structure-Function Study of Positive Allosteric Modulators of Kainate Receptors

Molecular pharmacology, 2017-06, Vol.91 (6), p.576-585

2017

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Partial Agonism and Antagonism of the Ionotropic Glutamate Receptor iGLuR5

The Journal of biological chemistry, 2007-08, Vol.282 (35), p.25726-25736

2007

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A pharmacological profile of the high-affinity GluK5 kainate receptor

European journal of pharmacology, 2016-10, Vol.788, p.315-320

2016

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The low binding affinity of D-serine at the ionotropic glutamate receptor GluD2 can be attributed to the hinge region

Scientific reports, 2017-04, Vol.7 (1), p.46145-46145, Article 46145

2017

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Development of Thiochroman Dioxide Analogues of Benzothiadiazine Dioxides as New Positive Allosteric Modulators of α‑Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid (AMPA) Receptors

ACS chemical neuroscience, 2021-07, Vol.12 (14), p.2679-2692

2021

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(S)‑2-Amino-3-(5-methyl-3-hydroxyisoxazol-4-yl)propanoic Acid (AMPA) and Kainate Receptor Ligands: Further Exploration of Bioisosteric Replacements and Structural and Biological Investigation

Journal of medicinal chemistry, 2018-03, Vol.61 (5), p.2124-2130

2018

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Crystal Structures of Potent Dimeric Positive Allosteric Modulators at the Ligand-Binding Domain of the GluA2 Receptor

ACS medicinal chemistry letters, 2019-03, Vol.10 (3), p.243-247

2019

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Intersubunit bridge formation governs agonist efficacy at nicotinic acetylcholine α4β2 receptors: unique role of halogen bonding revealed

The Journal of biological chemistry, 2012-02, Vol.287 (6), p.4248-4259

2012

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The ionotropic glutamate receptor GluA2 in complex with bicyclic pyrimidinedione-based compounds: when small compound modifications have distinct effects on binding interactions

ACS chemical neuroscience, 2020-06, Vol.11 (12), p.1791-1800

2020

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Lessons from crystal structures of kainate receptors

Binding of a negative allosteric modulator and competitive antagonist can occur simultaneously at the ionotropic glutamate receptor GluA2

7‑Phenoxy-Substituted 3,4-Dihydro‑2H‑1,2,4-benzothiadiazine 1,1-Dioxides as Positive Allosteric Modulators of α‑Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid (AMPA) Receptors with Nanomolar Potency

Exploring thienothiadiazine dioxides as isosteric analogues of benzo- and pyridothiadiazine dioxides in the search of new AMPA and kainate receptor positive allosteric modulators

The Structure of a High-Affinity Kainate Receptor: GluK4 Ligand-Binding Domain Crystallized with Kainate

Neuroplastin-55 binds to and signals through the fibroblast growth factor receptor

Structural Characterization of the Stringent Response Related Exopolyphosphatase/Guanosine Pentaphosphate Phosphohydrolase Protein Family

Structural basis for positive allosteric modulation of AMPA and kainate receptors

Small Angle X-ray Studies Reveal That Aspergillus niger Glucoamylase Has a Defined Extended Conformation and Can Form Dimers in Solution

Recovery from desensitization in GluA2 AMPA receptors is affected by a single mutation in the N-terminal domain interface

Tyr702 Is an Important Determinant of Agonist Binding and Domain Closure of the Ligand-Binding Core of GluR2

Enhancing Action of Positive Allosteric Modulators through the Design of Dimeric Compounds

Differences between the GluD1 and GluD2 receptors revealed by GluD1 X‐ray crystallography, binding studies and molecular dynamics

The positive allosteric modulator BPAM344 and L‐glutamate introduce an active‐like structure of the ligand‐binding domain of GluK2

Lessons from more than 80 structures of the GluA2 ligand-binding domain in complex with agonists, antagonists and allosteric modulators

Identification and Structure-Function Study of Positive Allosteric Modulators of Kainate Receptors

Partial Agonism and Antagonism of the Ionotropic Glutamate Receptor iGLuR5

A pharmacological profile of the high-affinity GluK5 kainate receptor

Invisible detergents for structure determination of membrane proteins by small‐angle neutron scattering

The low binding affinity of D-serine at the ionotropic glutamate receptor GluD2 can be attributed to the hinge region

Development of Thiochroman Dioxide Analogues of Benzothiadiazine Dioxides as New Positive Allosteric Modulators of α‑Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid (AMPA) Receptors

(S)‑2-Amino-3-(5-methyl-3-hydroxyisoxazol-4-yl)propanoic Acid (AMPA) and Kainate Receptor Ligands: Further Exploration of Bioisosteric Replacements and Structural and Biological Investigation

Crystal Structures of Potent Dimeric Positive Allosteric Modulators at the Ligand-Binding Domain of the GluA2 Receptor

Intersubunit bridge formation governs agonist efficacy at nicotinic acetylcholine α4β2 receptors: unique role of halogen bonding revealed

The ionotropic glutamate receptor GluA2 in complex with bicyclic pyrimidinedione-based compounds: when small compound modifications have distinct effects on binding interactions

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