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Principles of early drug discovery

British journal of pharmacology, 2011-03, Vol.162 (6), p.1239-1249

2011

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Thermodynamic analysis of ligands at cholecystokinin CCK2 receptors in rat cerebral cortex

British journal of pharmacology, 2007-08, Vol.151 (8), p.1352-1367

2007

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Retinoic acid receptor-α signalling antagonizes both intracellular and extracellular amyloid-β production and prevents neuronal cell death caused by amyloid-β

The European journal of neuroscience, 2010-10, Vol.32 (8), p.1246-1255

2010

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Unexpected relationship between plasma protein binding and the pharmacodynamics of 2‐NAP, a CCK1‐receptor antagonist

British journal of clinical pharmacology, 2007-05, Vol.63 (5), p.618-622

2007

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Thermodynamic analysis of ligands at cholecystokinin CCK 2 receptors in rat cerebral cortex

British journal of pharmacology, 2009-01, Vol.151 (8), p.1352-1367

2009

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Nonpeptide Cholecystokinin-2 Receptor Agonists

Journal of medicinal chemistry, 2001-04, Vol.44 (8), p.1125-1133

2001

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Development of Peptide 3D Structure Mimetics: Rational Design of Novel Peptoid Cholecystokinin Receptor Antagonists

Journal of medicinal chemistry, 2000-09, Vol.43 (19), p.3505-3517

2000

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Non-Peptide Cholecystokinin-B/Gastrin Receptor Antagonists Based on Bicyclic, Heteroaromatic Skeletons

Journal of medicinal chemistry, 1996-04, Vol.39 (9), p.1806-1815

1996

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Optimization of the in Vitro and in Vivo Properties of a Novel Series of 2,4,5-Trisubstituted Imidazoles as Potent Cholecystokinin-2 (CCK2) Antagonists

Journal of medicinal chemistry, 2005-11, Vol.48 (22), p.6803-6812

2005

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Improving the Affinity and Selectivity of a Nonpeptide Series of Cholecystokinin-B/Gastrin Receptor Antagonists Based on the Dibenzobicyclo[2.2.2]octane Skeleton

Journal of medicinal chemistry, 1995-10, Vol.38 (21), p.4294-4302

1995

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A recombinant, chimeric enzyme with a novel mechanism of action leading to greater potency and selectivity than tissue-type plasminogen activator

Circulation (New York, N.Y.), 1992-08, Vol.86 (2), p.548-552

1992

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2,7-Dioxo-2,3,4,5,6,7-hexahydro-1H-benzo[h][1,4]diazonine as a New Template for the Design of CCK2 Receptor Antagonists

Journal of medicinal chemistry, 2000-09, Vol.43 (19), p.3518-3529

2000

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From histamine to imidazolylalkyl-sulfonamides : The design of a novel series of histamine H3-RECEPTOR antagonists

Bioorganic & medicinal chemistry letters, 1999-07, Vol.9 (13), p.1825-1830

1999

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The use of active centre acylation to control the pharmacokinetic profile of a recombinant chimaeric plasminogen activator

Thrombosis and haemostasis, 1993, Vol.70 (6), p.984

1993

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Reagents for reversible coupling of proteins to the active centres of trypsin-like serine proteinases

Biochemical journal, 1987-12, Vol.248 (2), p.409-413

1987

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INCORPORATION OF CONFORMATIONALLY CONSTRAINED PHENYLALANINE DERIVATIVES TIC, SIC, HIC AND NIC INTO A CHOLECYSTOKININ-B/GASTRIN RECEPTOR ANTAGONIST

Bioorganic & medicinal chemistry letters, 1997-05, Vol.7 (10), p.1289-1292

1997

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Thermodynamic analysis of ligands at cholecystokinin CCK sub(2) receptors in rat cerebral cortex

British journal of pharmacology, 2007-08, Vol.151 (8), p.1352-1367

2007

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Retinoic acid receptor-a signalling antagonizes both intracellular and extracellular amyloid-b production and prevents neuronal cell death caused by amyloid-b

The European journal of neuroscience, 2010-10, Vol.32 (8), p.1246-1255

2010

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Thermodynamic analysis of ligands at cholecystokinin CCK2receptors in rat cerebral cortex

British journal of pharmacology, 2007, Vol.151 (8), p.1352-1367

2007

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The preparation and properties of novel reversible polymer-protein conjugates 2-ω-Methoxypolyethylene (5000) glycoxymethylene-3-methylmaleyl conjugates of plasminogen activators

FEBS letters, 1987-11, Vol.223 (2), p.361-365

1987

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The synthesis of a novel benzodiazocine via an intramolecular Staudinger/aza-Wittig cyclization

Tetrahedron letters, 1997-05, Vol.38 (20), p.3609-3610

1997

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A New Class of Non-peptidic Cholecystokinin-B/Gastrin Receptor Antagonists Based on Dibenzobicyclo[2.2.2]octane

Journal of medicinal chemistry, 1994-10, Vol.37 (22), p.3671-3673

1994

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Design, Synthesis, and Structure−Activity Relationships of Novel Non-Imidazole Histamine H3 Receptor Antagonists

Journal of medicinal chemistry, 2000-06, Vol.43 (12), p.2362-2370

2000

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Scaffold Hopping with Molecular Field Points: Identification of a Cholecystokinin-2 (CCK2) Receptor Pharmacophore and Its Use in the Design of a Prototypical Series of Pyrrole- and Imidazole-Based CCK2 Antagonists

Journal of medicinal chemistry, 2005-11, Vol.48 (22), p.6790-6802

2005

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Histamine H3 receptor antagonists

Expert opinion on therapeutic patents, 2000-07, Vol.10 (7), p.1045-1055

2000

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Principles of early drug discovery

Thermodynamic analysis of ligands at cholecystokinin CCK2 receptors in rat cerebral cortex

Retinoic acid receptor-α signalling antagonizes both intracellular and extracellular amyloid-β production and prevents neuronal cell death caused by amyloid-β

Unexpected relationship between plasma protein binding and the pharmacodynamics of 2‐NAP, a CCK1‐receptor antagonist

Thermodynamic analysis of ligands at cholecystokinin CCK 2 receptors in rat cerebral cortex

Nonpeptide Cholecystokinin-2 Receptor Agonists

Development of Peptide 3D Structure Mimetics: Rational Design of Novel Peptoid Cholecystokinin Receptor Antagonists

Non-Peptide Cholecystokinin-B/Gastrin Receptor Antagonists Based on Bicyclic, Heteroaromatic Skeletons

Optimization of the in Vitro and in Vivo Properties of a Novel Series of 2,4,5-Trisubstituted Imidazoles as Potent Cholecystokinin-2 (CCK2) Antagonists

Improving the Affinity and Selectivity of a Nonpeptide Series of Cholecystokinin-B/Gastrin Receptor Antagonists Based on the Dibenzobicyclo[2.2.2]octane Skeleton

A recombinant, chimeric enzyme with a novel mechanism of action leading to greater potency and selectivity than tissue-type plasminogen activator

2,7-Dioxo-2,3,4,5,6,7-hexahydro-1H-benzo[h][1,4]diazonine as a New Template for the Design of CCK2 Receptor Antagonists

From histamine to imidazolylalkyl-sulfonamides : The design of a novel series of histamine H3-RECEPTOR antagonists

The use of active centre acylation to control the pharmacokinetic profile of a recombinant chimaeric plasminogen activator

Reagents for reversible coupling of proteins to the active centres of trypsin-like serine proteinases

INCORPORATION OF CONFORMATIONALLY CONSTRAINED PHENYLALANINE DERIVATIVES TIC, SIC, HIC AND NIC INTO A CHOLECYSTOKININ-B/GASTRIN RECEPTOR ANTAGONIST

Thermodynamic analysis of ligands at cholecystokinin CCK sub(2) receptors in rat cerebral cortex

Retinoic acid receptor-a signalling antagonizes both intracellular and extracellular amyloid-b production and prevents neuronal cell death caused by amyloid-b

Thermodynamic analysis of ligands at cholecystokinin CCK2receptors in rat cerebral cortex

The preparation and properties of novel reversible polymer-protein conjugates 2-ω-Methoxypolyethylene (5000) glycoxymethylene-3-methylmaleyl conjugates of plasminogen activators

The synthesis of a novel benzodiazocine via an intramolecular Staudinger/aza-Wittig cyclization

A New Class of Non-peptidic Cholecystokinin-B/Gastrin Receptor Antagonists Based on Dibenzobicyclo[2.2.2]octane

Design, Synthesis, and Structure−Activity Relationships of Novel Non-Imidazole Histamine H3 Receptor Antagonists

Scaffold Hopping with Molecular Field Points: Identification of a Cholecystokinin-2 (CCK2) Receptor Pharmacophore and Its Use in the Design of a Prototypical Series of Pyrrole- and Imidazole-Based CCK2 Antagonists

Histamine H3 receptor antagonists

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