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Concentration and pH Dependent Aggregation of Hydrophobic Drug Molecules and Relevance to Oral Bioavailability

Journal of medicinal chemistry, 2005-03, Vol.48 (6), p.1974-1983

2005

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SYNOPSIS: SYNthesize and OPtimize System in Silico

Journal of medicinal chemistry, 2003-06, Vol.46 (13), p.2765-2773

2003

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Potent and selective inhibition of HIV-1 replication in vitro by a novel series of TIBO derivatives

Nature (London), 1990-02, Vol.343 (6257), p.470-474

1990

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Synthesis of Novel Diarylpyrimidine Analogues and Their Antiviral Activity against Human Immunodeficiency Virus Type 1

Journal of medicinal chemistry, 2005-03, Vol.48 (6), p.2072-2079

2005

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Design, Synthesis, and SAR of a Novel Pyrazinone Series with Non-Nucleoside HIV-1 Reverse Transcriptase Inhibitory Activity

Journal of medicinal chemistry, 2005-03, Vol.48 (6), p.1910-1918

2005

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Structure Based Activity Prediction of HIV-1 Reverse Transcriptase Inhibitors

Journal of medicinal chemistry, 2005-03, Vol.48 (6), p.2176-2183

2005

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Pre-incubation of cell-free HIV-1 group M isolates with non-nucleoside reverse transcriptase inhibitors blocks subsequent viral replication in co-cultures of dendritic cells and T cells

Antiviral therapy, 2005-01, Vol.10 (2), p.255-262

2005

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A NEW SERIES OF POTENT ANALGESICS

Journal of pharmacy and pharmacology, 2011-04, Vol.9 (1), p.381-400

2011

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Prediction of Binding Affinities for TIBO Inhibitors of HIV-1 Reverse Transcriptase Using Monte Carlo Simulations in a Linear Response Method

Journal of medicinal chemistry, 1998-12, Vol.41 (26), p.5272-5286

1998

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Synthesis and anti-HIV-1 activity of 4,5,6,7-tetrahydro-5-methylimidazo[4,5,1-jk][1,4]benzodiazepin-2(1H)-one (TIBO) derivatives. 2

Journal of medicinal chemistry, 1991-11, Vol.34 (11), p.3187-3197

1991

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Synthetic 1,4-disubstituted 1,4-dihydro-5H-tetrazol-5-one derivatives of fentanyl: Alfentanil (R 39209), a potent, extremely short-acting narcotic analgesic

Journal of medicinal chemistry, 1986-11, Vol.29 (11), p.2290-2297

1986

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New antihistaminic N-heterocyclic 4-piperidinamines. 3. Synthesis and antihistaminic activity of N-(4-piperidinyl)-3H-imidazo[4,5-b]pyridin-2-amines

Journal of medicinal chemistry, 1985-12, Vol.28 (12), p.1943-1947

1985

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New antihistaminic N-heterocyclic 4-piperidinamines. 2. Synthesis and antihistaminic activity of 1-[(4-fluorophenyl)methyl]-N-(4-piperidinyl)-1H-benzimidazol-2-amines

Journal of medicinal chemistry, 1985-12, Vol.28 (12), p.1934-1943

1985

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Is there a case for P-450 inhibitors in cancer treatment?

Journal of medicinal chemistry, 1989-10, Vol.32 (10), p.2231-2239

1989

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Functional role of 5-HT2 receptors in the regulation of sleep and wakefulness in the rat

Psychopharmacologia, 1989-04, Vol.97 (4), p.436-442

1989

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Evolution of anti-HIV drug candidates. Part 3: diarylpyrimidine (DAPY) analogues

Bioorganic & medicinal chemistry letters, 2001-09, Vol.11 (17), p.2235-2239

2001

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Pharmacology of Potent and Selective S2-Serotonergic Antagonists

Journal of cardiovascular pharmacology, 1985, Vol.7 Suppl 7, p.2-11

Janssen, Paul A. J

1985

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Potent and Highly Selective Human Immunodeficiency Virus Type 1 (HIV-1) Inhibition by a Series of α-Anilinophenylacetamide Derivatives Targeted at HIV-1 Reverse Transcriptase

Proceedings of the National Academy of Sciences - PNAS, 1993-03, Vol.90 (5), p.1711-1715

1993

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Evolution of anti-HIV drug candidates. Part 2 : Diaryltriazine (DATA) analogues

Bioorganic & medicinal chemistry letters, 2001-09, Vol.11 (17), p.2229-2234

2001

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Synthetic analgesics. Synthesis and pharmacology of the diastereoisomers of N-[3-methyl-1-(2-phenylethyl)-4-piperidyl]-N-phenylpropanamide and N-[3-methyl-1-(1-methyl-2-phenylethyl)-4-piperidyl]-N-phenylpropanamide

Journal of medicinal chemistry, 1974-10, Vol.17 (10), p.1047-1051

1974

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A pharmacophore docking algorithm and its application to the cross-docking of 18 HIV-NNRTI's in their binding pockets

Proteins, structure, function, and bioinformatics, 2004-02, Vol.54 (3), p.526-533

2004

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Mode of Action Studies: Basis for the Search of New Antifungal Drugs

Annals of the New York Academy of Sciences, 1988-12, Vol.544 (1), p.191-207

1988

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Evolution of anti-HIV drug candidates. Part 1: From α-Anilinophenylacetamide (α-APA) to imidoyl thiourea (ITU)

Bioorganic & medicinal chemistry letters, 2001-09, Vol.11 (17), p.2225-2228

2001

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In Search of a Novel Anti-HIV Drug: Multidisciplinary Coordination in the Discovery of 4-[[4-[[4-[(1E)-2-Cyanoethenyl]-2,6-dimethylphenyl]amino]-2- pyrimidinyl]amino]benzonitrile (R278474, Rilpivirine)

Concentration and pH Dependent Aggregation of Hydrophobic Drug Molecules and Relevance to Oral Bioavailability

SYNOPSIS: SYNthesize and OPtimize System in Silico

Roles of Conformational and Positional Adaptability in Structure-Based Design of TMC125-R165335 (Etravirine) and Related Non-nucleoside Reverse Transcriptase Inhibitors That Are Highly Potent and Effective against Wild-Type and Drug-Resistant HIV-1 Variants

Potent and selective inhibition of HIV-1 replication in vitro by a novel series of TIBO derivatives

Synthesis of Novel Diarylpyrimidine Analogues and Their Antiviral Activity against Human Immunodeficiency Virus Type 1

Design, Synthesis, and SAR of a Novel Pyrazinone Series with Non-Nucleoside HIV-1 Reverse Transcriptase Inhibitory Activity

Structure Based Activity Prediction of HIV-1 Reverse Transcriptase Inhibitors

Pre-incubation of cell-free HIV-1 group M isolates with non-nucleoside reverse transcriptase inhibitors blocks subsequent viral replication in co-cultures of dendritic cells and T cells

A NEW SERIES OF POTENT ANALGESICS

Prediction of Binding Affinities for TIBO Inhibitors of HIV-1 Reverse Transcriptase Using Monte Carlo Simulations in a Linear Response Method

Synthesis and anti-HIV-1 activity of 4,5,6,7-tetrahydro-5-methylimidazo[4,5,1-jk][1,4]benzodiazepin-2(1H)-one (TIBO) derivatives. 2

Synthetic 1,4-disubstituted 1,4-dihydro-5H-tetrazol-5-one derivatives of fentanyl: Alfentanil (R 39209), a potent, extremely short-acting narcotic analgesic

New antihistaminic N-heterocyclic 4-piperidinamines. 3. Synthesis and antihistaminic activity of N-(4-piperidinyl)-3H-imidazo[4,5-b]pyridin-2-amines

New antihistaminic N-heterocyclic 4-piperidinamines. 2. Synthesis and antihistaminic activity of 1-[(4-fluorophenyl)methyl]-N-(4-piperidinyl)-1H-benzimidazol-2-amines

Is there a case for P-450 inhibitors in cancer treatment?

Functional role of 5-HT2 receptors in the regulation of sleep and wakefulness in the rat

Evolution of anti-HIV drug candidates. Part 3: diarylpyrimidine (DAPY) analogues

Pharmacology of Potent and Selective S2-Serotonergic Antagonists

Potent and Highly Selective Human Immunodeficiency Virus Type 1 (HIV-1) Inhibition by a Series of α-Anilinophenylacetamide Derivatives Targeted at HIV-1 Reverse Transcriptase

Evolution of anti-HIV drug candidates. Part 2 : Diaryltriazine (DATA) analogues

Synthetic analgesics. Synthesis and pharmacology of the diastereoisomers of N-[3-methyl-1-(2-phenylethyl)-4-piperidyl]-N-phenylpropanamide and N-[3-methyl-1-(1-methyl-2-phenylethyl)-4-piperidyl]-N-phenylpropanamide

A pharmacophore docking algorithm and its application to the cross-docking of 18 HIV-NNRTI's in their binding pockets

Mode of Action Studies: Basis for the Search of New Antifungal Drugs

Evolution of anti-HIV drug candidates. Part 1: From α-Anilinophenylacetamide (α-APA) to imidoyl thiourea (ITU)

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