UB Paderborn / Katalog / Suche / in CDI

Concise Synthesis, Preparative Resolution, Absolute Configuration Determination, and Applications of an Atropisomeric Biaryl Catalyst for Asymmetric Acylation

Journal of organic chemistry, 2003-09, Vol.68 (19), p.7379-7385

2003

Volltextzugriff (PDF)

Optimization of Novel Acyl Pyrrolidine Inhibitors of Hepatitis C Virus RNA-Dependent RNA Polymerase Leading to a Development Candidate

Journal of medicinal chemistry, 2007-03, Vol.50 (5), p.897-900

2007

Volltextzugriff (PDF)

New atropisomeric biaryl derivatives of 4-aminopyridine—identification of an improved nucleophilic catalyst for asymmetric acylation of sec-alcohols

Tetrahedron, 2004-05, Vol.60 (20), p.4513-4525

2004

Volltextzugriff (PDF)

Variable Sensitivity to Bacterial Methionyl-tRNA Synthetase Inhibitors Reveals Subpopulations of Streptococcus pneumoniae with Two Distinct Methionyl-tRNA Synthetase Genes

Antimicrobial Agents and Chemotherapy, 2003-06, Vol.47 (6), p.1784-1789

2003

Volltextzugriff (PDF)

Discovery of Novel Urea-Based Hepatitis C Protease Inhibitors with High Potency against Protease-Inhibitor-Resistant Mutants

Journal of medicinal chemistry, 2012-04, Vol.55 (7), p.3021-3026

2012

Volltextzugriff (PDF)

Synthesis and SAR of acyclic HCV NS3 protease inhibitors with novel P4-benzoxaborole moieties

Bioorganic & medicinal chemistry letters, 2011-04, Vol.21 (7), p.2048-2054

2011

Volltextzugriff (PDF)

Synthesis and biological evaluations of P4-benzoxaborole-substituted macrocyclic inhibitors of HCV NS3 protease

Bioorganic & medicinal chemistry letters, 2010-12, Vol.20 (24), p.7317-7322

2010

Volltextzugriff (PDF)

Synthesis and evaluation of novel α-amino cyclic boronates as inhibitors of HCV NS3 protease

Bioorganic & medicinal chemistry letters, 2010-06, Vol.20 (12), p.3550-3556

2010

Volltextzugriff (PDF)

Novel macrocyclic HCV NS3 protease inhibitors derived from α-amino cyclic boronates

Bioorganic & medicinal chemistry letters, 2010-10, Vol.20 (19), p.5695-5700

2010

Volltextzugriff (PDF)

Synthesis of new acylsulfamoyl benzoxaboroles as potent inhibitors of HCV NS3 protease

Bioorganic & medicinal chemistry letters, 2010-12, Vol.20 (24), p.7493-7497

2010

Volltextzugriff (PDF)

6-Alkylquinolone-3-carboxylic acid tethered to macrolides synthesis and antimicrobial profile

Bioorganic & medicinal chemistry, 2010-09, Vol.18 (17), p.6569-6577

2010

Volltextzugriff (PDF)

The antimicrobial natural product chuangxinmycin and Some synthetic analogues are potent and selective inhibitors of bacterial tryptophanyl tRNA synthetase

Bioorganic & medicinal chemistry letters, 2002-11, Vol.12 (21), p.3171-3174

2002

Volltextzugriff (PDF)

Synthesis and antiviral activity of novel HCV NS3 protease inhibitors with P4 capping groups

Bioorganic & medicinal chemistry letters, 2012-12, Vol.22 (24), p.7351-7356

2012

Volltextzugriff (PDF)

Nanomolar Inhibitors of Staphylococcus aureus Methionyl tRNA Synthetase with Potent Antibacterial Activity against Gram-Positive Pathogens

Journal of medicinal chemistry, 2002-05, Vol.45 (10), p.1959-1962

2002

Volltextzugriff (PDF)

Synthesis and Activity of Analogues of SB-219383: Novel Potent Inhibitors of Bacterial Tyrosyl tRNA Synthetase

The Journal of Antibiotics, 2000/11/25, Vol.53(11), pp.1282-1292

2000

Volltextzugriff (PDF)

The synthesis of 5-alkoxy and 5-amino substituted thiophenes

Tetrahedron letters, 2000-03, Vol.41 (10), p.1597-1600

2000

Volltextzugriff (PDF)

Definition of the heterocyclic pharmacophore of bacterial methionyl tRNA synthetase inhibitors: potent antibacterially active non-quinolone analogues

Bioorganic & medicinal chemistry letters, 2004-08, Vol.14 (15), p.3937-3941

2004

Volltextzugriff (PDF)

Inhibition of herpes proteases and antiviral activity of 2-substituted thieno[2,3-d]oxazinones

Bioorganic & medicinal chemistry letters, 1999-02, Vol.9 (3), p.443-448

1999

Volltextzugriff (PDF)

Discovery and optimisation of potent, selective, ethanolamine inhibitors of bacterial phenylalanyl tRNA synthetase

Bioorganic & medicinal chemistry letters, 2005-05, Vol.15 (9), p.2305-2309

2005

Volltextzugriff (PDF)

Optimisation of aryl substitution leading to potent methionyl tRNA synthetase inhibitors with excellent gram-Positive antibacterial activity

Bioorganic & medicinal chemistry letters, 2003-02, Vol.13 (4), p.665-668

2003

Volltextzugriff (PDF)

Inhibition of HSV-1 protease by benzoxazinones

Bioorganic & medicinal chemistry letters, 1996-10, Vol.6 (20), p.2463-2466

1996

Volltextzugriff (PDF)

Conformational restriction of methionyl tRNA synthetase inhibitors leading to analogues with potent inhibition and excellent gram-Positive antibacterial activity

Bioorganic & medicinal chemistry letters, 2003-04, Vol.13 (7), p.1265-1268

2003

Volltextzugriff (PDF)

Inhibitors of bacterial tyrosyl tRNA synthetase: synthesis of four stereoisomeric analogues of the natural product SB-219383

Bioorganic & medicinal chemistry letters, 2000-08, Vol.10 (16), p.1811-1814

2000

Volltextzugriff (PDF)

Synthetic analogues of SB-219383. Novel C-glycosyl peptides as inhibitors of tyrosyl tRNA synthetase

Bioorganic & medicinal chemistry letters, 2001-03, Vol.11 (5), p.711-714

2001

Volltextzugriff (PDF)

Potent synthetic inhibitors of tyrosyl tRNA synthetase derived from C-pyranosyl analogues of SB-219383

Bioorganic & medicinal chemistry letters, 2001-03, Vol.11 (5), p.715-718

2001

Volltextzugriff (PDF)

Menü

Weitere Dienste

Einstellungen

Concise Synthesis, Preparative Resolution, Absolute Configuration Determination, and Applications of an Atropisomeric Biaryl Catalyst for Asymmetric Acylation

Optimization of Novel Acyl Pyrrolidine Inhibitors of Hepatitis C Virus RNA-Dependent RNA Polymerase Leading to a Development Candidate

New atropisomeric biaryl derivatives of 4-aminopyridine—identification of an improved nucleophilic catalyst for asymmetric acylation of sec-alcohols

Variable Sensitivity to Bacterial Methionyl-tRNA Synthetase Inhibitors Reveals Subpopulations of Streptococcus pneumoniae with Two Distinct Methionyl-tRNA Synthetase Genes

Discovery of Novel Urea-Based Hepatitis C Protease Inhibitors with High Potency against Protease-Inhibitor-Resistant Mutants

Synthesis and SAR of acyclic HCV NS3 protease inhibitors with novel P4-benzoxaborole moieties

Synthesis and biological evaluations of P4-benzoxaborole-substituted macrocyclic inhibitors of HCV NS3 protease

Synthesis and evaluation of novel α-amino cyclic boronates as inhibitors of HCV NS3 protease

Novel macrocyclic HCV NS3 protease inhibitors derived from α-amino cyclic boronates

Synthesis of new acylsulfamoyl benzoxaboroles as potent inhibitors of HCV NS3 protease

6-Alkylquinolone-3-carboxylic acid tethered to macrolides synthesis and antimicrobial profile

The antimicrobial natural product chuangxinmycin and Some synthetic analogues are potent and selective inhibitors of bacterial tryptophanyl tRNA synthetase

Synthesis and antiviral activity of novel HCV NS3 protease inhibitors with P4 capping groups

Nanomolar Inhibitors of Staphylococcus aureus Methionyl tRNA Synthetase with Potent Antibacterial Activity against Gram-Positive Pathogens

Synthesis and Activity of Analogues of SB-219383: Novel Potent Inhibitors of Bacterial Tyrosyl tRNA Synthetase

The synthesis of 5-alkoxy and 5-amino substituted thiophenes

Definition of the heterocyclic pharmacophore of bacterial methionyl tRNA synthetase inhibitors: potent antibacterially active non-quinolone analogues

Inhibition of herpes proteases and antiviral activity of 2-substituted thieno[2,3-d]oxazinones

Discovery and optimisation of potent, selective, ethanolamine inhibitors of bacterial phenylalanyl tRNA synthetase

Optimisation of aryl substitution leading to potent methionyl tRNA synthetase inhibitors with excellent gram-Positive antibacterial activity

Inhibition of HSV-1 protease by benzoxazinones

Conformational restriction of methionyl tRNA synthetase inhibitors leading to analogues with potent inhibition and excellent gram-Positive antibacterial activity

Inhibitors of bacterial tyrosyl tRNA synthetase: synthesis of four stereoisomeric analogues of the natural product SB-219383

Synthetic analogues of SB-219383. Novel C-glycosyl peptides as inhibitors of tyrosyl tRNA synthetase

Potent synthetic inhibitors of tyrosyl tRNA synthetase derived from C-pyranosyl analogues of SB-219383

Suchergebnisse filtern