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Crystal structure of dihydrofolate reductase from the filarial nematode W. bancrofti in complex with NADPH and folate

PLoS neglected tropical diseases, 2023-04, Vol.17 (4), p.e0011303-e0011303

2023

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Expression, purification, and inhibition profile of dihydrofolate reductase from the filarial nematode Wuchereria bancrofti

PloS one, 2018-05, Vol.13 (5), p.e0197173-e0197173

2018

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Investigating the Roles of Active Site Residues in Mycobacterium tuberculosis Indole-3-glycerol Phosphate Synthase, a Potential Target for Antitubercular Agents

ACS bio & med chem au, 2023-10, Vol.3 (5), p.438-447

2023

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Indole Naphthyridinones as Inhibitors of Bacterial Enoyl-ACP Reductases FabI and FabK

Journal of medicinal chemistry, 2003-04, Vol.46 (9), p.1627-1635

2003

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Structure of the C-terminally truncated human ProMMP9, a gelatin-binding matrix metalloproteinase

Acta crystallographica. Section D, Biological crystallography., 2002-07, Vol.58 (7), p.1182-1192

2002

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Mutational analysis confirms the presence of distal inhibitor-selectivity determining residues in B. stearothermophilus dihydrofolate reductase

Archives of biochemistry and biophysics, 2020-10, Vol.692, p.108545-108545, Article 108545

2020

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First X-ray Cocrystal Structure of a Bacterial FabH Condensing Enzyme and a Small Molecule Inhibitor Achieved Using Rational Design and Homology Modeling

Journal of medicinal chemistry, 2003-01, Vol.46 (1), p.5-8

2003

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Unique fold and active site in cytomegalovirus protease

Nature (London), 1996-09, Vol.383 (6597), p.275-279

1996

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The structure of XIAP BIR2: understanding the selectivity of the BIR domains

Acta crystallographica. Section D, Biological crystallography., 2013-09, Vol.69 (9), p.1717-1725

2013

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Benzazepinones and Benzoxazepinones as Antagonists of Inhibitor of Apoptosis Proteins (IAPs) Selective for the Second Baculovirus IAP Repeat (BIR2) Domain

Journal of medicinal chemistry, 2013-10, Vol.56 (20), p.7772-7787

2013

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4-Aryl-1,2,3-triazole: A Novel Template for a Reversible Methionine Aminopeptidase 2 Inhibitor, Optimized To Inhibit Angiogenesis in Vivo

Journal of medicinal chemistry, 2005-09, Vol.48 (18), p.5644-5647

2005

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Optimization of Benzodiazepinones as Selective Inhibitors of the X‑Linked Inhibitor of Apoptosis Protein (XIAP) Second Baculovirus IAP Repeat (BIR2) Domain

Journal of medicinal chemistry, 2013-10, Vol.56 (20), p.7788-7803

2013

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Structure of apo acyl carrier protein and a proposal to engineer protein crystallization through metal ions

Acta crystallographica. Section D, Biological crystallography., 2004-09, Vol.60 (9), p.1545-1554

2004

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Highly Potent Inhibitors of Methionine Aminopeptidase-2 Based on a 1,2,4-Triazole Pharmacophore

Journal of medicinal chemistry, 2007-08, Vol.50 (16), p.3777-3785

2007

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Crystal structure and substrate specificity of the β‐ketoacyl‐acyl carrier protein synthase III (FabH) from Staphylococcus aureus

Protein science, 2005-08, Vol.14 (8), p.2087-2094

2005

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Crystal Structure of the IMP-1 Metallo β-Lactamase from Pseudomonas aeruginosa and Its Complex with a Mercaptocarboxylate Inhibitor: Binding Determinants of a Potent, Broad-Spectrum Inhibitor

Biochemistry (Easton), 2000-04, Vol.39 (15), p.4288-4298

2000

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Refined structures of β-ketoacyl-acyl carrier protein synthase III

Journal of molecular biology, 2001-03, Vol.307 (1), p.341-356

2001

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Design of thymidylate synthase inhibitors using protein crystal structures: the synthesis and biological evaluation of a novel class of 5-substituted quinazolinones

Journal of medicinal chemistry, 1993-03, Vol.36 (6), p.733-746

1993

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Crystal Structure of Varicella-Zoster Virus Protease

Proceedings of the National Academy of Sciences - PNAS, 1997-04, Vol.94 (7), p.2874-2879

1997

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Structure Activity Relationships of 5-, 6-, and 7-Methyl-Substituted Azepan-3-one Cathepsin K Inhibitors

Journal of medicinal chemistry, 2006-03, Vol.49 (5), p.1597-1612

2006

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Identification of an Adamantyl Azaquinolone JNK Selective Inhibitor

ACS medicinal chemistry letters, 2012-09, Vol.3 (9), p.764-768

2012

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Azepanone-Based Inhibitors of Human and Rat Cathepsin K

Journal of medicinal chemistry, 2001-04, Vol.44 (9), p.1380-1395

2001

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Identification of a Series of Tricyclic Natural Products as Potent Broad-Spectrum Inhibitors of Metallo-β-Lactamases

Antimicrobial Agents and Chemotherapy, 2002-06, Vol.46 (6), p.1880-1886

2002

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1,4-Disubstituted imidazoles are potential antibacterial agents functioning as inhibitors of enoyl acyl carrier protein reductase (FabI)

Bioorganic & medicinal chemistry letters, 2001-08, Vol.11 (16), p.2061-2065

2001

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Cyclic Ketone Inhibitors of the Cysteine Protease Cathepsin K

Journal of medicinal chemistry, 2001-03, Vol.44 (5), p.725-736

2001

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Crystal structure of dihydrofolate reductase from the filarial nematode W. bancrofti in complex with NADPH and folate

Expression, purification, and inhibition profile of dihydrofolate reductase from the filarial nematode Wuchereria bancrofti

Investigating the Roles of Active Site Residues in Mycobacterium tuberculosis Indole-3-glycerol Phosphate Synthase, a Potential Target for Antitubercular Agents

Indole Naphthyridinones as Inhibitors of Bacterial Enoyl-ACP Reductases FabI and FabK

Structure of the C-terminally truncated human ProMMP9, a gelatin-binding matrix metalloproteinase

Mutational analysis confirms the presence of distal inhibitor-selectivity determining residues in B. stearothermophilus dihydrofolate reductase

First X-ray Cocrystal Structure of a Bacterial FabH Condensing Enzyme and a Small Molecule Inhibitor Achieved Using Rational Design and Homology Modeling

Unique fold and active site in cytomegalovirus protease

The structure of XIAP BIR2: understanding the selectivity of the BIR domains

Benzazepinones and Benzoxazepinones as Antagonists of Inhibitor of Apoptosis Proteins (IAPs) Selective for the Second Baculovirus IAP Repeat (BIR2) Domain

4-Aryl-1,2,3-triazole: A Novel Template for a Reversible Methionine Aminopeptidase 2 Inhibitor, Optimized To Inhibit Angiogenesis in Vivo

Optimization of Benzodiazepinones as Selective Inhibitors of the X‑Linked Inhibitor of Apoptosis Protein (XIAP) Second Baculovirus IAP Repeat (BIR2) Domain

Structure of apo acyl carrier protein and a proposal to engineer protein crystallization through metal ions

Highly Potent Inhibitors of Methionine Aminopeptidase-2 Based on a 1,2,4-Triazole Pharmacophore

Crystal structure and substrate specificity of the β‐ketoacyl‐acyl carrier protein synthase III (FabH) from Staphylococcus aureus

Crystal Structure of the IMP-1 Metallo β-Lactamase from Pseudomonas aeruginosa and Its Complex with a Mercaptocarboxylate Inhibitor: Binding Determinants of a Potent, Broad-Spectrum Inhibitor

Refined structures of β-ketoacyl-acyl carrier protein synthase III

Design of thymidylate synthase inhibitors using protein crystal structures: the synthesis and biological evaluation of a novel class of 5-substituted quinazolinones

Crystal Structure of Varicella-Zoster Virus Protease

Structure Activity Relationships of 5-, 6-, and 7-Methyl-Substituted Azepan-3-one Cathepsin K Inhibitors

Identification of an Adamantyl Azaquinolone JNK Selective Inhibitor

Azepanone-Based Inhibitors of Human and Rat Cathepsin K

Identification of a Series of Tricyclic Natural Products as Potent Broad-Spectrum Inhibitors of Metallo-β-Lactamases

1,4-Disubstituted imidazoles are potential antibacterial agents functioning as inhibitors of enoyl acyl carrier protein reductase (FabI)

Cyclic Ketone Inhibitors of the Cysteine Protease Cathepsin K

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