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Cav1.3 L-type Ca2+ channel-activated CaMKII/ERK2 pathway in the ventral tegmental area is required for cocaine conditioned place preference

Neuropharmacology, 2023-02, Vol.224, p.109368-109368, Article 109368

2023

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Esmethadone-HCl (REL-1017): a promising rapid antidepressant

European archives of psychiatry and clinical neuroscience, 2023-10, Vol.273 (7), p.1463-1476

2023

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The novel uncompetitive NMDA receptor antagonist esmethadone (REL-1017) has no meaningful abuse potential in recreational drug users

Translational psychiatry, 2023-06, Vol.13 (1), p.192-12, Article 192

2023

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Esmethadone (REL-1017) and Other Uncompetitive NMDAR Channel Blockers May Improve Mood Disorders via Modulation of Synaptic Kinase-Mediated Signaling

International journal of molecular sciences, 2022-10, Vol.23 (20), p.12196

2022

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REL-1017 (Esmethadone) Increases Circulating BDNF Levels in Healthy Subjects of a Phase 1 Clinical Study

Frontiers in pharmacology, 2021-04, Vol.12, p.671859-671859

2021

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Drug–Drug Interaction Studies of Esmethadone (REL-1017) Involving CYP3A4- and CYP2D6-Mediated Metabolism

Drugs in R&D, 2024-03, Vol.24 (1), p.51-68

2024

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The N-Methyl-D-Aspartate Receptor Blocker REL-1017 (Esmethadone) Reduces Calcium Influx Induced by Glutamate, Quinolinic Acid, and Gentamicin

Pharmaceuticals (Basel, Switzerland), 2022-07, Vol.15 (7), p.882

2022

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Patient-Reported Outcomes and Opioid Use by Outpatient Cancer Patients

The journal of pain, 2018-03, Vol.19 (3), p.278-290

2018

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Pharmacological Comparative Characterization of REL-1017 (Esmethadone-HCl) and Other NMDAR Channel Blockers in Human Heterodimeric N-Methyl-D-Aspartate Receptors

Pharmaceuticals (Basel, Switzerland), 2022-08, Vol.15 (8), p.997

2022

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Activation of the Neuronal Extracellular Signal-Regulated Kinase 2 in the Spinal Cord Dorsal Horn Is Required for Complete Freund's Adjuvant-Induced Pain Hypersensitivity

The Journal of neuroscience, 2008-12, Vol.28 (52), p.14087-14096

2008

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siRNA-Mediated Knockdown of the NR1 Subunit Gene of the NMDA Receptor Attenuates Formalin-Induced Pain Behaviors in Adult Rats

The journal of pain, 2009-04, Vol.10 (4), p.380-390

2009

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Comment on “Novel Glutamatergic Modulators for the Treatment of Mood Disorders: Current Status

CNS drugs, 2022-02, Vol.36 (2), p.203-204

2022

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Does transdermal fentanyl work in patients with low BMI? Patient‐reported outcomes of pain and percent pain relief in cancer patients on transdermal fentanyl

Cancer medicine (Malden, MA), 2019-12, Vol.8 (18), p.7516-7522

2019

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REL-1017 (Esmethadone) as Adjunctive Treatment in Patients With Major Depressive Disorder: A Phase 2a Randomized Double-Blind Trial

The American journal of psychiatry, 2022-02, Vol.179 (2), p.122-131

2022

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Using Chronic Pain Outcomes Data to Improve Outcomes

Anesthesiology clinics, 2016-06, Vol.34 (2), p.395-408

2016

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Design and evaluation of small interfering RNAs that target expression of the N-methyl-D-aspartate receptor NR1 subunit gene in the spinal cord dorsal horn

The Journal of pharmacology and experimental therapeutics, 2007-09, Vol.322 (3), p.982

2007

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A Conditional Deletion of the NR1 Subunit of the NMDA Receptor in Adult Spinal Cord Dorsal Horn Reduces NMDA Currents and Injury-Induced Pain

The Journal of neuroscience, 2003-06, Vol.23 (12), p.5031-5040

2003

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Estradiol and progesterone differentially regulate formalin-induced nociception in ovariectomized female rats

Hormones and behavior, 2006-04, Vol.49 (4), p.441-449

2006

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Clinical Pharmacology of Opioids for Pain

The Clinical journal of pain, 2002-07, Vol.18 (4 Suppl), p.S3-S13

Inturrisi, Charles E

2002

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The d- and l- isomers of methadone bind to the non-competitive site on the N-methyl- d-aspartate (NMDA) receptor in rat forebrain and spinal cord

Neuroscience letters, 1997-02, Vol.223 (1), p.5-8

1997

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Understanding Opioid Actions, Pain and Analgesia: A Tribute to Dr. Gavril Pasternak

Cellular and molecular neurobiology, 2021-07, Vol.41 (5), p.827-834

2021

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An antisense oligonucleotide to the N-methyl-D-aspartate (NMDA) subunit NMDAR1 attenuates NMDA-induced nociception, hyperalgesia, and morphine tolerance

The Journal of pharmacology and experimental therapeutics, 2005-02, Vol.312 (2), p.834

2005

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Stabilization of the μ-Opioid Receptor by Truncated Single Transmembrane Splice Variants through a Chaperone-like Action

The Journal of biological chemistry, 2013-07, Vol.288 (29), p.21211-21227

2013

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Deletion of the glutamate receptor 5 subunit of kainate receptors affects the development of morphine tolerance

The Journal of pharmacology and experimental therapeutics, 2009-02, Vol.328 (2), p.579

2009

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Personalized Medicine and Opioid Analgesic Prescribing for Chronic Pain: Opportunities and Challenges

The journal of pain, 2013-02, Vol.14 (2), p.103-113

2013

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Cav1.3 L-type Ca2+ channel-activated CaMKII/ERK2 pathway in the ventral tegmental area is required for cocaine conditioned place preference

Esmethadone-HCl (REL-1017): a promising rapid antidepressant

The novel uncompetitive NMDA receptor antagonist esmethadone (REL-1017) has no meaningful abuse potential in recreational drug users

Esmethadone (REL-1017) and Other Uncompetitive NMDAR Channel Blockers May Improve Mood Disorders via Modulation of Synaptic Kinase-Mediated Signaling

REL-1017 (Esmethadone) Increases Circulating BDNF Levels in Healthy Subjects of a Phase 1 Clinical Study

Drug–Drug Interaction Studies of Esmethadone (REL-1017) Involving CYP3A4- and CYP2D6-Mediated Metabolism

The N-Methyl-D-Aspartate Receptor Blocker REL-1017 (Esmethadone) Reduces Calcium Influx Induced by Glutamate, Quinolinic Acid, and Gentamicin

Patient-Reported Outcomes and Opioid Use by Outpatient Cancer Patients

Pharmacological Comparative Characterization of REL-1017 (Esmethadone-HCl) and Other NMDAR Channel Blockers in Human Heterodimeric N-Methyl-D-Aspartate Receptors

Activation of the Neuronal Extracellular Signal-Regulated Kinase 2 in the Spinal Cord Dorsal Horn Is Required for Complete Freund's Adjuvant-Induced Pain Hypersensitivity

siRNA-Mediated Knockdown of the NR1 Subunit Gene of the NMDA Receptor Attenuates Formalin-Induced Pain Behaviors in Adult Rats

Comment on “Novel Glutamatergic Modulators for the Treatment of Mood Disorders: Current Status

Does transdermal fentanyl work in patients with low BMI? Patient‐reported outcomes of pain and percent pain relief in cancer patients on transdermal fentanyl

REL-1017 (Esmethadone) as Adjunctive Treatment in Patients With Major Depressive Disorder: A Phase 2a Randomized Double-Blind Trial

Using Chronic Pain Outcomes Data to Improve Outcomes

Design and evaluation of small interfering RNAs that target expression of the N-methyl-D-aspartate receptor NR1 subunit gene in the spinal cord dorsal horn

A Conditional Deletion of the NR1 Subunit of the NMDA Receptor in Adult Spinal Cord Dorsal Horn Reduces NMDA Currents and Injury-Induced Pain

Estradiol and progesterone differentially regulate formalin-induced nociception in ovariectomized female rats

Clinical Pharmacology of Opioids for Pain

The d- and l- isomers of methadone bind to the non-competitive site on the N-methyl- d-aspartate (NMDA) receptor in rat forebrain and spinal cord

Understanding Opioid Actions, Pain and Analgesia: A Tribute to Dr. Gavril Pasternak

An antisense oligonucleotide to the N-methyl-D-aspartate (NMDA) subunit NMDAR1 attenuates NMDA-induced nociception, hyperalgesia, and morphine tolerance

Stabilization of the μ-Opioid Receptor by Truncated Single Transmembrane Splice Variants through a Chaperone-like Action

Deletion of the glutamate receptor 5 subunit of kainate receptors affects the development of morphine tolerance

Personalized Medicine and Opioid Analgesic Prescribing for Chronic Pain: Opportunities and Challenges

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