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JNJ-28312141, a novel orally active colony-stimulating factor-1 receptor/FMS-related receptor tyrosine kinase-3 receptor tyrosine kinase inhibitor with potential utility in solid tumors, bone metastases, and acute myeloid leukemia

Molecular cancer therapeutics, 2009-11, Vol.8 (11), p.3151-3161

2009

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Design and Optimization of Benzimidazole-Containing Transient Receptor Potential Melastatin 8 (TRPM8) Antagonists

Journal of medicinal chemistry, 2011-01, Vol.54 (1), p.233-247

2011

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Discovery of novel potent imidazo[1,2-b]pyridazine PDE10a inhibitors

Bioorganic & medicinal chemistry letters, 2016-09, Vol.26 (17), p.4216-4222

2016

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Enhancement of kinase selectivity in a potent class of arylamide FMS inhibitors

Bioorganic & medicinal chemistry letters, 2013-12, Vol.23 (23), p.6363-6369

2013

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Optimization of a Potent Class of Arylamide Colony-Stimulating Factor-1 Receptor Inhibitors Leading to Anti-inflammatory Clinical Candidate 4-Cyano-N-[2-(1-cyclohexen-1-yl)-4-[1-[(dimethylamino)acetyl]-4-piperidinyl]phenyl]-1H-imidazole-2-carboxamide (JNJ-28312141)

Journal of medicinal chemistry, 2011-11, Vol.54 (22), p.7860-7883

2011

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Synthesis and evaluation of novel 3,4,6-substituted 2-quinolones as FMS kinase inhibitors

Bioorganic & medicinal chemistry, 2008-03, Vol.18 (6), p.2097-2102

2008

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Discovery of novel FMS kinase inhibitors as anti-inflammatory agents

Bioorganic & medicinal chemistry, 2008-03, Vol.18 (5), p.1642-1648

2008

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Structure-based optimization of a potent class of arylamide FMS inhibitors

Bioorganic & medicinal chemistry, 2008-06, Vol.18 (12), p.3632-3637

2008

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Synthesis of thiophene-2-carboxamidines containing 2-aminothiazoles and their biological evaluation as urokinase inhibitors

Bioorganic & medicinal chemistry letters, 2001-04, Vol.11 (7), p.915-918

2001

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Reducing ion channel activity in a series of 4-heterocyclic arylamide FMS inhibitors

Bioorganic & medicinal chemistry letters, 2010-07, Vol.20 (13), p.3925-3929

2010

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A novel series of potent and selective small molecule inhibitors of the complement component C1s

Bioorganic & medicinal chemistry letters, 2004-06, Vol.14 (12), p.3043-3047

2004

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Design and Synthesis of 4,5-Disubstituted-thiophene-2-amidines as Potent Urokinase Inhibitors

Bioorganic & medicinal chemistry letters, 2002-02, Vol.12 (3), p.491-495

2002

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Structural Analysis of Thrombin Complexed with Potent Inhibitors Incorporating a Phenyl Group as a Peptide Mimetic and Aminopyridines as Guanidine Substitutes

Journal of medicinal chemistry, 1998-06, Vol.41 (12), p.2068-2075

1998

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Structure-activity and crystallographic analysis of a new class of non-amide-based thrombin inhibitor

Bioorganic & medicinal chemistry letters, 2000-01, Vol.10 (1), p.79-82

2000

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1,3,5-Trialkyl-2,4,6-triiodobenzenes: Novel X-ray Contrast Agents for Gastrointestinal Imaging

Journal of medicinal chemistry, 2000-05, Vol.43 (10), p.1940-1948

2000

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Cyano-Substituted 2-Carboxyimidazoles: Synthesis of 4-Cyano-1-{[2-(trimethylsilyl)ethoxy]methyl}-1 H -imidazole-2-carboxylate Potassium Salt

Synthesis (Stuttgart), 2008-11, Vol.2008 (21), p.3377-3379

2008

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In vitro evaluation and crystallographic analysis of a new class of selective, non-amide-based thrombin inhibitors

Bioorganic & medicinal chemistry letters, 1998-07, Vol.8 (13), p.1595-1600

1998

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Synthesis of thiophene-2-carboxamidines containing 2-amino-thiazoles and their biological evaluation as urokinase inhibitors

Bioorganic & medicinal chemistry letters, 2001-04, Vol.11 (7), p.915-918

2001

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Stereoselective synthesis of (.+-.)-cyanocycline

Journal of the American Chemical Society, 1986-04, Vol.108 (9), p.2478-2479

1986

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Amidinohydrazones as guanidine bioisosteres : Application to a new class of potent, selective and orally bioavailable, non-amide-based small-molecule thrombin inhibitors

Bioorganic & medicinal chemistry letters, 2000-01, Vol.10 (1), p.1-4

2000

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Structure-Based design, synthesis and sAR of a novel series of thiopheneamidine urokinase plasminogen activator inhibitors

Bioorganic & medicinal chemistry letters, 2001-06, Vol.11 (11), p.1379-1382

2001

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Gas Problems Since Phillips

Texas law review, 1956-01, Vol.35, p.647

Illig, Carl

1956

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CONSUMER CREDIT: MESHING TRUTH-IN-LENDING WITH THE TEXAS CODE

Texas bar journal, 1970-02, Vol.33 (2), p.87

Illig, Carl

1970

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Offshore Lands and Paramount Rights

University of Pittsburgh law review, 1952-01, Vol.14, p.10

Illig, Carl

1952

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JNJ-28312141, a novel orally active colony-stimulating factor-1 receptor/FMS-related receptor tyrosine kinase-3 receptor tyrosine kinase inhibitor with potential utility in solid tumors, bone metastases, and acute myeloid leukemia

Design and Optimization of Benzimidazole-Containing Transient Receptor Potential Melastatin 8 (TRPM8) Antagonists

Discovery of novel potent imidazo[1,2-b]pyridazine PDE10a inhibitors

Enhancement of kinase selectivity in a potent class of arylamide FMS inhibitors

Optimization of a Potent Class of Arylamide Colony-Stimulating Factor-1 Receptor Inhibitors Leading to Anti-inflammatory Clinical Candidate 4-Cyano-N-[2-(1-cyclohexen-1-yl)-4-[1-[(dimethylamino)acetyl]-4-piperidinyl]phenyl]-1H-imidazole-2-carboxamide (JNJ-28312141)

Synthesis and evaluation of novel 3,4,6-substituted 2-quinolones as FMS kinase inhibitors

Discovery of novel FMS kinase inhibitors as anti-inflammatory agents

Structure-based optimization of a potent class of arylamide FMS inhibitors

Synthesis of thiophene-2-carboxamidines containing 2-aminothiazoles and their biological evaluation as urokinase inhibitors

Reducing ion channel activity in a series of 4-heterocyclic arylamide FMS inhibitors

A novel series of potent and selective small molecule inhibitors of the complement component C1s

Design and Synthesis of 4,5-Disubstituted-thiophene-2-amidines as Potent Urokinase Inhibitors

Structural Analysis of Thrombin Complexed with Potent Inhibitors Incorporating a Phenyl Group as a Peptide Mimetic and Aminopyridines as Guanidine Substitutes

Optimization of a Potent Class of Arylamide Colony-Stimulating Factor-1 Receptor Inhibitors Leading to Anti-inflammatory Clinical Candidate 4-Cyano- N -[2-(1-cyclohexen-1-yl)-4-[1-[(dimethylamino)acetyl]-4-piperidinyl]phenyl]-1 H -imidazole-2-carboxamide (JNJ-28312141)

Structure-activity and crystallographic analysis of a new class of non-amide-based thrombin inhibitor

1,3,5-Trialkyl-2,4,6-triiodobenzenes: Novel X-ray Contrast Agents for Gastrointestinal Imaging

Cyano-Substituted 2-Carboxyimidazoles: Synthesis of 4-Cyano-1-{[2-(trimethylsilyl)ethoxy]methyl}-1 H -imidazole-2-carboxylate Potassium Salt

In vitro evaluation and crystallographic analysis of a new class of selective, non-amide-based thrombin inhibitors

Synthesis of thiophene-2-carboxamidines containing 2-amino-thiazoles and their biological evaluation as urokinase inhibitors

Stereoselective synthesis of (.+-.)-cyanocycline

Amidinohydrazones as guanidine bioisosteres : Application to a new class of potent, selective and orally bioavailable, non-amide-based small-molecule thrombin inhibitors

Structure-Based design, synthesis and sAR of a novel series of thiopheneamidine urokinase plasminogen activator inhibitors

Gas Problems Since Phillips

CONSUMER CREDIT: MESHING TRUTH-IN-LENDING WITH THE TEXAS CODE

Offshore Lands and Paramount Rights

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