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CCR2B receptor antagonists: conversion of a weak HTS hit to a potent lead compound

Bioorganic & medicinal chemistry letters, 2000-08, Vol.10 (16), p.1803-1806

2000

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3-Anilino-4-arylmaleimides: potent and selective inhibitors of glycogen synthase kinase-3 (GSK-3)

Bioorganic & medicinal chemistry letters, 2001-03, Vol.11 (5), p.635-639

2001

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ATP-Citrate Lyase as a Target for Hypolipidemic Intervention. 2. Synthesis and Evaluation of (3R,5S)-ω-Substituted-3-carboxy-3,5-dihydroxyalkanoic Acids and Their γ-Lactone Prodrugs as Inhibitors of the Enzyme in Vitro and in Vivo

Journal of medicinal chemistry, 1998-09, Vol.41 (19), p.3582-3595

1998

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The inhibition of human cytomegalovirus (hCMV) protease by hydroxylamine derivatives

Bioorganic & medicinal chemistry letters, 1999-11, Vol.9 (21), p.3137-3142

1999

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Conformationally Restricted Indolopiperidine Derivatives as Potent CCR2B Receptor Antagonists

Bioorganic & medicinal chemistry letters, 2001-08, Vol.11 (16), p.2177-2180

2001

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Lipoprotein-associated phospholipase A2, platelet-activating factor acetylhydrolase, generates two bioactive products during the oxidation of low-density lipoprotein: use of a novel inhibitor

Biochemical journal, 1999-03, Vol.338 ( Pt 2) (2), p.479-487

1999

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Structures of histamine H1-receptor antagonists derived from the cimetidine group of histamine H2-receptor antagonists

Acta crystallographica. Section B, Structural science, 1994-04, Vol.50 (2), p.221-243

1994

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Solid-phase synthesis of cyclic alkoxyketones, inhibitors of the cysteine protease cathepsin K

Bioorganic & medicinal chemistry letters, 2001-01, Vol.11 (2), p.195-198

2001

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Photoaffinity Labeling of the Lumenal K+ Site of the Gastric (H+ + K+)-ATPase

The Journal of biological chemistry, 1989-04, Vol.264 (10), p.5552-5558

1989

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2-[[(4-Amino-2-pyridyl)methyl]sulfinyl]benzimidazole H+/K+-ATPase inhibitors. The relationship between pyridine basicity, stability, and activity

Journal of medicinal chemistry, 1989-08, Vol.32 (8), p.1970-1977

1989

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Diastereoselective synthesis, activity and chiral stability of cyclic alkoxyketone inhibitors of cathepsin K

Bioorganic & medicinal chemistry letters, 2001-01, Vol.11 (2), p.199-202

2001

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Studies on the mechanism of action of omeprazole

Biochemical pharmacology, 1985-08, Vol.34 (16), p.2967-2973

1985

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2-(alkylthio)pyrimidin-4-ones as novel, reversible inhibitors of lipoprotein-associated phospholipase A2

Bioorganic & medicinal chemistry letters, 2000-02, Vol.10 (4), p.395-398

2000

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Design of an Affinity Matrix for Purification of the Histamine H1 Receptor from Guinea Pig Cerebellum

Journal of neurochemistry, 1992-01, Vol.58 (1), p.350-356

1992

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Characterisation of the effects of anthranilic and (indanyloxy) acetic acid derivatives on chloride transport in membrane vesicles

Biochimica et biophysica acta, 1991-08, Vol.1067 (1), p.51-63

1991

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Reversible Inhibitors of the Gastric (H+/K+)-ATPase. 5. Substituted 2,4-Diaminoquinazolines and Thienopyrimidines

Journal of medicinal chemistry, 1995-07, Vol.38 (14), p.2763-2773

1995

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5-Aryl-pyrazolo[3,4- b]pyridines: potent inhibitors of glycogen synthase kinase-3 (GSK-3)

Bioorganic & medicinal chemistry letters, 2003-05, Vol.13 (9), p.1577-1580

2003

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[125I] Iodobolpyramine, a highly sensitive probe for histamine H1-receptors in guinea-pig brain

European journal of pharmacology, 1986-01, Vol.120 (2), p.151-160

1986

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Reversible inhibitors of the gastric (H+/K+)-ATPase. 3. 3-Substituted-4-(phenylamino)quinolines

Journal of medicinal chemistry, 1992-09, Vol.35 (18), p.3413-3422

1992

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SK&F 96067 is a reversible, lumenally acting inhibitor of the gastric (H + + K +)-ATPase

Biochemical pharmacology, 1991-06, Vol.42 (1), p.123-130

1991

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1-(Arylpiperazinylamidoalkyl)-pyrimidones: orally active inhibitors of lipoprotein-associated phospholipase A(2)

Bioorganic & medicinal chemistry letters, 2001-07, Vol.11 (14), p.1925

2001

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Properties of the reversible, K +-competitive inhibitor of the gastric (H +/K +)-ATPase, SK&F 97574. I. In vitro activity

Biochemical pharmacology, 1995-11, Vol.50 (10), p.1543-1549

1995

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Histamine receptors on leukocytes: the binding of histamine serum albumin conjugates is non-specific

International archives of allergy and applied immunology, 1985, Vol.76 (1), p.9

1985

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Reversible Inhibitors of the Gastric (H+/K+)-ATPase. 4. Identification of an Inhibitor with an Intermediate Duration of Action

Journal of medicinal chemistry, 1995-07, Vol.38 (14), p.2748-2762

1995

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Reversible inhibitors of the gastric (H+/K+)-ATPase. 2. 1-Arylpyrrolo[3,2-c]quinolines: effect of the 4-substituent

Journal of medicinal chemistry, 1992-05, Vol.35 (10), p.1845-1852

1992

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CCR2B receptor antagonists: conversion of a weak HTS hit to a potent lead compound

3-Anilino-4-arylmaleimides: potent and selective inhibitors of glycogen synthase kinase-3 (GSK-3)

ATP-Citrate Lyase as a Target for Hypolipidemic Intervention. 2. Synthesis and Evaluation of (3R,5S)-ω-Substituted-3-carboxy-3,5-dihydroxyalkanoic Acids and Their γ-Lactone Prodrugs as Inhibitors of the Enzyme in Vitro and in Vivo

The inhibition of human cytomegalovirus (hCMV) protease by hydroxylamine derivatives

Conformationally Restricted Indolopiperidine Derivatives as Potent CCR2B Receptor Antagonists

Lipoprotein-associated phospholipase A2, platelet-activating factor acetylhydrolase, generates two bioactive products during the oxidation of low-density lipoprotein: use of a novel inhibitor

Structures of histamine H1-receptor antagonists derived from the cimetidine group of histamine H2-receptor antagonists

Solid-phase synthesis of cyclic alkoxyketones, inhibitors of the cysteine protease cathepsin K

Photoaffinity Labeling of the Lumenal K+ Site of the Gastric (H+ + K+)-ATPase

2-[[(4-Amino-2-pyridyl)methyl]sulfinyl]benzimidazole H+/K+-ATPase inhibitors. The relationship between pyridine basicity, stability, and activity

Diastereoselective synthesis, activity and chiral stability of cyclic alkoxyketone inhibitors of cathepsin K

Studies on the mechanism of action of omeprazole

2-(alkylthio)pyrimidin-4-ones as novel, reversible inhibitors of lipoprotein-associated phospholipase A2

Design of an Affinity Matrix for Purification of the Histamine H1 Receptor from Guinea Pig Cerebellum

Characterisation of the effects of anthranilic and (indanyloxy) acetic acid derivatives on chloride transport in membrane vesicles

Reversible Inhibitors of the Gastric (H+/K+)-ATPase. 5. Substituted 2,4-Diaminoquinazolines and Thienopyrimidines

5-Aryl-pyrazolo[3,4- b]pyridines: potent inhibitors of glycogen synthase kinase-3 (GSK-3)

[125I] Iodobolpyramine, a highly sensitive probe for histamine H1-receptors in guinea-pig brain

Reversible inhibitors of the gastric (H+/K+)-ATPase. 3. 3-Substituted-4-(phenylamino)quinolines

SK&F 96067 is a reversible, lumenally acting inhibitor of the gastric (H + + K +)-ATPase

1-(Arylpiperazinylamidoalkyl)-pyrimidones: orally active inhibitors of lipoprotein-associated phospholipase A(2)

Properties of the reversible, K +-competitive inhibitor of the gastric (H +/K +)-ATPase, SK&F 97574. I. In vitro activity

Histamine receptors on leukocytes: the binding of histamine serum albumin conjugates is non-specific

Reversible Inhibitors of the Gastric (H+/K+)-ATPase. 4. Identification of an Inhibitor with an Intermediate Duration of Action

Reversible inhibitors of the gastric (H+/K+)-ATPase. 2. 1-Arylpyrrolo[3,2-c]quinolines: effect of the 4-substituent

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