UB Paderborn / Katalog / Suche / in CDI

Sortiert nach

Einfacher Volltextzugriff von (fast) überall

Installieren Sie die LibKey Nomad-Browsererweiterung und erhalten Sie von vielen Webseiten einfachen Zugriff auf lizenzierte Volltexte oder Open Access Publikationen. Mehr erfahren...

Conformational Restriction of Flexible Ligands Guided by the Transferred NOE Experiment: Potent Macrocyclic Inhibitors of Farnesyltransferase

Journal of the American Chemical Society, 2001-03, Vol.123 (9), p.2107-2108

2001

Volltextzugriff (PDF)

Non-Peptide GPIIb/IIIa Inhibitors. 20. Centrally Constrained Thienothiophene α-Sulfonamides Are Potent, Long Acting in Vivo Inhibitors of Platelet Aggregation

Journal of medicinal chemistry, 1999-07, Vol.42 (13), p.2409-2421

1999

Volltextzugriff (PDF)

In vitro and in vivo evaluation of dihydropyrimidinone C-5 amides as potent and selective alpha(1A) receptor antagonists for the treatment of benign prostatic hyperplasia

Journal of medicinal chemistry, 2000-07, Vol.43 (14), p.2703-2718

2000

Volltextzugriff (PDF)

Design of nonpeptidal ligands for a peptide receptor: cholecystokinin antagonists

Journal of medicinal chemistry, 1987-07, Vol.30 (7), p.1229-1239

1987

Volltextzugriff (PDF)

Development of Orally Active Oxytocin Antagonists: Studies on 1-(1-{4-[1-(2-Methyl-1-oxidopyridin-3-ylmethyl)piperidin-4-yloxy]-2- methoxybenzoyl}piperidin-4-yl)-1,4-dihydrobenz[d][1,3]oxazin-2-one (L-372,662) and Related Pyridines

Journal of medicinal chemistry, 1998-06, Vol.41 (12), p.2146-2163

1998

Volltextzugriff (PDF)

In vivo and in vitro metabolism studies on a class III antiarrhythmic agent

Drug metabolism and disposition, 1993-05, Vol.21 (3), p.467

1993

Volltextzugriff (PDF)

A simple and inexpensive synthesis of 4-(aminomethyl)-L-phenylalanine

Journal of organic chemistry, 1993-08, Vol.58 (18), p.5015-5016

1993

Volltextzugriff (PDF)

Evaluation of amino acid-based linkers in potent macrocyclic inhibitors of farnesyl-protein transferase

Bioorganic & medicinal chemistry letters, 2001-07, Vol.11 (14), p.1817-1821

2001

Volltextzugriff (PDF)

Asymmetric Synthesis of α,α-Difluoro-β-amino Acid Derivatives from Enantiomerically Pure N-tert-Butylsulfinimines

Journal of organic chemistry, 2002-11, Vol.67 (23), p.8276-8279

2002

Volltextzugriff (PDF)

A series of 5-(5,6)-dihydrouracil substituted 8-hydroxy-[1,6]naphthyridine-7-carboxylic acid 4-fluorobenzylamide inhibitors of HIV-1 integrase and viral replication in cells

Bioorganic & medicinal chemistry letters, 2005-10, Vol.15 (20), p.4550-4554

2005

Volltextzugriff (PDF)

9-Hydroxyazafluorenes and Their Use in Thrombin Inhibitors

Journal of medicinal chemistry, 2005-04, Vol.48 (7), p.2282-2293

2005

Volltextzugriff (PDF)

Benzodiazepines as Potent and Selective Bradykinin B1 Antagonists

Journal of medicinal chemistry, 2003-05, Vol.46 (10), p.1803-1806

2003

Volltextzugriff (PDF)

L-156, 602, A C5a ANTAGONIST WITH A NOVEL CYCLIC HEXADEPSIPEPTIDE STRUCTURE FROM Streptomyces sp. MA6348: FERMENTATION, ISOLATION AND STRUCTURE DETERMINATION

The Journal of Antibiotics, 1991/02/25, Vol.44(2), pp.249-254

1991

Volltextzugriff (PDF)

Benzodiazepines as Potent and Selective Bradykinin B 1 Antagonists

Journal of medicinal chemistry, 2003-05, Vol.46 (10), p.1803-1806

2003

Volltextzugriff (PDF)

Total synthesis of nonpeptidal cholecystokinin antagonists from Aspergillus alliaceus

Journal of organic chemistry, 1987-04, Vol.52 (8), p.1644-1646

1987

Volltextzugriff (PDF)

Glucagon releasing activity of a cyclic peptide related to somatostatin

International Journal of Peptide and Protein Research, 1987-02, Vol.29 (2), p.244-249

1987

Volltextzugriff (PDF)

A Selective Protection of 2,3-Diaminopropionic Acid

Synthetic communications, 1993-03, Vol.23 (5), p.703-709

1993

Volltextzugriff (PDF)

A new amine resolution method and its application to 3-aminobenzodiazepines

Tetrahedron letters, 1987, Vol.28 (5), p.521-522

1987

Volltextzugriff (PDF)

Inhibition of acute nociceptive responses in rat spinal cord by a bradykinin B 1 receptor antagonist

European journal of pharmacology, 2005-12, Vol.527 (1), p.44-51

2005

Volltextzugriff (PDF)

Non-peptide alpha(v)beta(3) antagonists. Part 5: identification of potent RGD mimetics incorporating 2-aryl beta-amino acids as aspartic acid replacements

Bioorganic & medicinal chemistry letters, 2002-12, Vol.12 (23), p.3483

2002

Volltextzugriff (PDF)

Synthesis and antiviral activity of a series of HIV-1 protease inhibitors with functionality tethered to the P1 or P1' phenyl substituents : X-ray crystal structure assisted design

Journal of medicinal chemistry, 1992-05, Vol.35 (10), p.1685-1701

1992

Volltextzugriff (PDF)

Selective α1A adrenergic receptor antagonists based on 4-aryl-3,4-dihydropyridine-2-ones

Bioorganic & medicinal chemistry letters, 2000-08, Vol.10 (15), p.1625-1628

2000

Volltextzugriff (PDF)

Selective alpha1a adrenergic receptor antagonists based on 4-aryl-3,4-dihydropyridine-2-ones

Bioorganic & medicinal chemistry letters, 2000-08, Vol.10 (15), p.1625-1628

2000

Volltextzugriff (PDF)

1 – 25 von 58

Suche als RSS-Feed

Suchergebnisse filtern

Filter anzeigen

Nur zeigen

Geprüft (Peer-Review)
(45)
Mit Volltextzugriff
(46)

Publikationsform

Artikel
(58)

Sprache

Englisch
(58)

Erscheinungsjahr

n.n

Thema

15 weitere anzeigen...

Weniger anzeigen...

Menü

Weitere Dienste

Einstellungen

Conformational Restriction of Flexible Ligands Guided by the Transferred NOE Experiment: Potent Macrocyclic Inhibitors of Farnesyltransferase

Non-Peptide GPIIb/IIIa Inhibitors. 20. Centrally Constrained Thienothiophene α-Sulfonamides Are Potent, Long Acting in Vivo Inhibitors of Platelet Aggregation

In vitro and in vivo evaluation of dihydropyrimidinone C-5 amides as potent and selective alpha(1A) receptor antagonists for the treatment of benign prostatic hyperplasia

Design and Biological Activity of (S)-4-(5-{[1-(3-Chlorobenzyl)-2- oxopyrrolidin-3-ylamino]methyl}imidazol-1-ylmethyl)benzonitrile, a 3-Aminopyrrolidinone Farnesyltransferase Inhibitor with Excellent Cell Potency

Design of nonpeptidal ligands for a peptide receptor: cholecystokinin antagonists

Development of Orally Active Oxytocin Antagonists: Studies on 1-(1-{4-[1-(2-Methyl-1-oxidopyridin-3-ylmethyl)piperidin-4-yloxy]-2- methoxybenzoyl}piperidin-4-yl)-1,4-dihydrobenz[d][1,3]oxazin-2-one (L-372,662) and Related Pyridines

In vivo and in vitro metabolism studies on a class III antiarrhythmic agent

A simple and inexpensive synthesis of 4-(aminomethyl)-L-phenylalanine

Evaluation of amino acid-based linkers in potent macrocyclic inhibitors of farnesyl-protein transferase

Asymmetric Synthesis of α,α-Difluoro-β-amino Acid Derivatives from Enantiomerically Pure N-tert-Butylsulfinimines

A series of 5-(5,6)-dihydrouracil substituted 8-hydroxy-[1,6]naphthyridine-7-carboxylic acid 4-fluorobenzylamide inhibitors of HIV-1 integrase and viral replication in cells

3-Aminopyrrolidinone Farnesyltransferase Inhibitors: Design of Macrocyclic Compounds with Improved Pharmacokinetics and Excellent Cell Potency

9-Hydroxyazafluorenes and Their Use in Thrombin Inhibitors

Benzodiazepines as Potent and Selective Bradykinin B1 Antagonists

L-156, 602, A C5a ANTAGONIST WITH A NOVEL CYCLIC HEXADEPSIPEPTIDE STRUCTURE FROM Streptomyces sp. MA6348: FERMENTATION, ISOLATION AND STRUCTURE DETERMINATION

Benzodiazepines as Potent and Selective Bradykinin B 1 Antagonists

Total synthesis of nonpeptidal cholecystokinin antagonists from Aspergillus alliaceus

Glucagon releasing activity of a cyclic peptide related to somatostatin

A Selective Protection of 2,3-Diaminopropionic Acid

A new amine resolution method and its application to 3-aminobenzodiazepines

Inhibition of acute nociceptive responses in rat spinal cord by a bradykinin B 1 receptor antagonist

Non-peptide alpha(v)beta(3) antagonists. Part 5: identification of potent RGD mimetics incorporating 2-aryl beta-amino acids as aspartic acid replacements

Synthesis and antiviral activity of a series of HIV-1 protease inhibitors with functionality tethered to the P1 or P1' phenyl substituents : X-ray crystal structure assisted design

Selective α1A adrenergic receptor antagonists based on 4-aryl-3,4-dihydropyridine-2-ones

Selective alpha1a adrenergic receptor antagonists based on 4-aryl-3,4-dihydropyridine-2-ones

Suchergebnisse filtern