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Discovery, Structure−Activity Relationships, Pharmacokinetics, and Efficacy of Glucokinase Activator (2R)-3-Cyclopentyl-2-(4-methanesulfonylphenyl)-N-thiazol-2-yl-propionamide (RO0281675)

Journal of medicinal chemistry, 2010-05, Vol.53 (9), p.3618-3625

2010

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Discovery, Modeling, and Human Pharmacokinetics of N-(2-Acetyl-4,6-dimethylphenyl)-3-(3,4-dimethylisoxazol-5-ylsulfamoyl)thiophene-2-carboxamide (TBC3711), a Second Generation, ETA Selective, and Orally Bioavailable Endothelin Antagonist

Journal of medicinal chemistry, 2004-04, Vol.47 (8), p.1969-1986

2004

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Development of cell adhesion molecule antagonists as therapeutics for asthma and COPD

Pulmonary pharmacology & therapeutics, 2004-01, Vol.17 (1), p.1-10

2004

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Acyl Substitution at the Ortho Position of Anilides Enhances Oral Bioavailability of Thiophene Sulfonamides: TBC3214, an ETA Selective Endothelin Antagonist

Journal of medicinal chemistry, 2001-04, Vol.44 (8), p.1211-1216

2001

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Endothelin Antagonists: Substituted Mesitylcarboxamides with High Potency and Selectivity for ETA Receptors

Journal of medicinal chemistry, 1999-11, Vol.42 (22), p.4485-4499

1999

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Recently discovered sulfonamide-, acyl sulfonamide- and carboxylic acid-based endothelin antagonists

IDrugs : the investigational drugs journal, 2003-03, Vol.6 (3), p.232

2003

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Chapter 7. Antagonists of VILA-4

Annual Reports in Medicinal Chemistry, 2002, Vol.37, p.65-74

2002

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Versatile prostaglandin synthesis. Use of a carboxy-inversion reaction

Journal of organic chemistry, 1973-09, Vol.38 (19), p.3440-3442

1973

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Solution-Phase Parallel Synthesis of Substituted Benzimidazoles

Journal of combinatorial chemistry, 2002-07, Vol.4 (4), p.320-328

2002

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A 3D Structure Model of Integrin α4β1 Complex: I. Construction of a Homology Model of β1 and Ligand Binding Analysis

Biophysical journal, 2002-01, Vol.82 (1), p.447-457

2002

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A 3D structure model of integrin alpha 4 beta 1 complex: I. Construction of a homology model of beta 1 and ligand binding analysis

Biophysical journal, 2002-01, Vol.82 (1 Pt 1), p.447-457

2002

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Nonpeptide endothelin antagonists in clinical development

Drugs of today (Barcelona, Spain : 1998), 2001-07, Vol.37 (7), p.441-453

2001

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Discovery, modeling, and human pharmacokinetics of N-(2-acetyl-4,6-dimethylphenyl)-3-(3,4-dimethylisoxazol-5-ylsulfamoyl)-thiophene -2-carboxamide (TBC3711), a second generation, ETA selective, and orally bioavailable endothelin antagonists

Journal of medicinal chemistry, 2004, Vol.47 (8), p.1969-1986

2004

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Discovery, Modeling, and Human Pharmacokinetics of N -(2-Acetyl-4,6-dimethylphenyl)-3-(3,4-dimethylisoxazol-5-ylsulfamoyl)thiophene-2-carboxamide (TBC3711), a Second Generation, ET A Selective, and Orally Bioavailable Endothelin Antagonist

Journal of medicinal chemistry, 2004-04, Vol.47 (8), p.1969-1986

2004

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Endothelin antagonists: substituted mesitylcarboxamides with high potency and selectivity for ET(A) receptors

Journal of medicinal chemistry, 1999-11, Vol.42 (22), p.4485-4499

1999

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A 3D Structure Model of Integrin α4 β1 Complex: I. Construction of a Homology Model of β1 and Ligand Binding Analysis

Biophysical journal, 2002, Vol.82 (1), p.447-457

2002

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SELECTIVE ALKYLATION/ACYLATION OF DI- OR TRIANIONS: EXPEDITIOUS DERIVATIZATION OF ENDOTHELIN ANTAGONISTS[1]

Synthetic communications, 2002-01, Vol.32 (10), p.1615-1624

2002

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Application of electron spin resonance spectroscopy to problems of structure and conformation. XVI. Stereochemistry of the reaction of the 7-norbornenyl radical with tri-n-butyltin deuteride

Journal of the American Chemical Society, 1969-07, Vol.91 (14), p.3968-3969

1969

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Acyl Substitution at the Ortho Position of Anilides Enhances Oral Bioavailability of Thiophene Sulfonamides: TBC3214, an ET A Selective Endothelin Antagonist

Journal of medicinal chemistry, 2001-04, Vol.44 (8), p.1211-1216

2001

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New four-carbon-atom homologation involving the free-radical chain reaction of 1,3-butadiene monoxide with organoboranes. Synthesis of 4-alkyl-2-buten-1-ols from olefins via hydroboration

Journal of the American Chemical Society, 1971-06, Vol.93 (11), p.2792-2793

1971

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Semidiones. VI. Bicyclo[2.2.2]octane-2,3-semidione and derivatives

Journal of the American Chemical Society, 1967-12, Vol.89 (25), p.6629-6635

1967

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Aliphatic semidiones. XXV. Bicyclo[n.2.1]alkane-2,3-semidiones

Journal of the American Chemical Society, 1974-11, Vol.96 (23), p.7237-7248

1974

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Behavior of chloro alkenes in sulfur trioxide-sulfuric acid and in fluorosulfonic acid

Journal of organic chemistry, 1967-05, Vol.32 (5), p.1496-1498

1967

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Benzenepropanoic acids containing chromanone or naphthalenone moieties are potent and orally active leukotriene B4 antagonists

Bioorganic & medicinal chemistry letters, 1994-12, Vol.4 (24), p.2883-2888

1994

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Benzenepropanoic acids containing chromanone or naphthalenone moieties are potent and orally active leukotriene B 4 antagonists

Bioorganic & medicinal chemistry letters, 1994-12, Vol.4 (24), p.2883-2888

1994

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Discovery, Structure−Activity Relationships, Pharmacokinetics, and Efficacy of Glucokinase Activator (2R)-3-Cyclopentyl-2-(4-methanesulfonylphenyl)-N-thiazol-2-yl-propionamide (RO0281675)

Discovery, Modeling, and Human Pharmacokinetics of N-(2-Acetyl-4,6-dimethylphenyl)-3-(3,4-dimethylisoxazol-5-ylsulfamoyl)thiophene-2-carboxamide (TBC3711), a Second Generation, ETA Selective, and Orally Bioavailable Endothelin Antagonist

Development of cell adhesion molecule antagonists as therapeutics for asthma and COPD

Acyl Substitution at the Ortho Position of Anilides Enhances Oral Bioavailability of Thiophene Sulfonamides: TBC3214, an ETA Selective Endothelin Antagonist

Endothelin Antagonists: Substituted Mesitylcarboxamides with High Potency and Selectivity for ETA Receptors

Recently discovered sulfonamide-, acyl sulfonamide- and carboxylic acid-based endothelin antagonists

Chapter 7. Antagonists of VILA-4

Versatile prostaglandin synthesis. Use of a carboxy-inversion reaction

Solution-Phase Parallel Synthesis of Substituted Benzimidazoles

A 3D Structure Model of Integrin α4β1 Complex: I. Construction of a Homology Model of β1 and Ligand Binding Analysis

A 3D structure model of integrin alpha 4 beta 1 complex: I. Construction of a homology model of beta 1 and ligand binding analysis

Nonpeptide endothelin antagonists in clinical development

Discovery, modeling, and human pharmacokinetics of N-(2-acetyl-4,6-dimethylphenyl)-3-(3,4-dimethylisoxazol-5-ylsulfamoyl)-thiophene -2-carboxamide (TBC3711), a second generation, ETA selective, and orally bioavailable endothelin antagonists

Discovery, Modeling, and Human Pharmacokinetics of N -(2-Acetyl-4,6-dimethylphenyl)-3-(3,4-dimethylisoxazol-5-ylsulfamoyl)thiophene-2-carboxamide (TBC3711), a Second Generation, ET A Selective, and Orally Bioavailable Endothelin Antagonist

Endothelin antagonists: substituted mesitylcarboxamides with high potency and selectivity for ET(A) receptors

A 3D Structure Model of Integrin α4 β1 Complex: I. Construction of a Homology Model of β1 and Ligand Binding Analysis

SELECTIVE ALKYLATION/ACYLATION OF DI- OR TRIANIONS: EXPEDITIOUS DERIVATIZATION OF ENDOTHELIN ANTAGONISTS[1]

Application of electron spin resonance spectroscopy to problems of structure and conformation. XVI. Stereochemistry of the reaction of the 7-norbornenyl radical with tri-n-butyltin deuteride

Acyl Substitution at the Ortho Position of Anilides Enhances Oral Bioavailability of Thiophene Sulfonamides: TBC3214, an ET A Selective Endothelin Antagonist

New four-carbon-atom homologation involving the free-radical chain reaction of 1,3-butadiene monoxide with organoboranes. Synthesis of 4-alkyl-2-buten-1-ols from olefins via hydroboration

Semidiones. VI. Bicyclo[2.2.2]octane-2,3-semidione and derivatives

Aliphatic semidiones. XXV. Bicyclo[n.2.1]alkane-2,3-semidiones

Behavior of chloro alkenes in sulfur trioxide-sulfuric acid and in fluorosulfonic acid

Benzenepropanoic acids containing chromanone or naphthalenone moieties are potent and orally active leukotriene B4 antagonists

Benzenepropanoic acids containing chromanone or naphthalenone moieties are potent and orally active leukotriene B 4 antagonists

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