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7-Azabicycloheptane Carboxylic Acid: A Proline Replacement in a Boroarginine Thrombin Inhibitor

Organic letters, 1999-12, Vol.1 (12), p.1875-1877

1999

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Determining appropriate substrate conversion for enzymatic assays in high-throughput screening

Journal of biomolecular screening, 2003-12, Vol.8 (6), p.694-700

2003

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Streamlined System for Purifying and Quantifying a Diverse Library of Compounds and the Effect of Compound Concentration Measurements on the Accurate Interpretation of Biological Assay Results

Analytical chemistry (Washington), 2004-12, Vol.76 (24), p.7278-7287

2004

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Rational Design of Potent, Bioavailable, Nonpeptide Cyclic Ureas as HIV Protease Inhibitors

Science (American Association for the Advancement of Science), 1994-01, Vol.263 (5145), p.380-384

1994

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Photobleaching-based flow measurement in a commercial capillary electrophoresis chip instrument

Electrophoresis, 2008-03, Vol.29 (6), p.1253-1263

2008

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Cyclic HIV Protease Inhibitors: Synthesis, Conformational Analysis, P2/P2‘ Structure−Activity Relationship, and Molecular Recognition of Cyclic Ureas

Journal of medicinal chemistry, 1996-08, Vol.39 (18), p.3514-3525

1996

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A molecular mechanics/grid method for evaluation of ligand-receptor interactions

Journal of computational chemistry, 1995-04, Vol.16 (4), p.454-464

1995

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Solvation studies of DMP323 and A76928 bound to HIV protease: Analysis of water sites using grand canonical Monte Carlo simulations

Protein science, 1998-03, Vol.7 (3), p.573-579

1998

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A Chemogenomic Approach to Discovering Target-Selective Drugs

Chemical biology & drug design, 2006-01, Vol.67 (1), p.85-86

2006

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Corticotropin-Releasing Hormone Receptor Antagonists: Framework Design and Synthesis Guided by Ligand Conformational Studies

Journal of medicinal chemistry, 1999-03, Vol.42 (5), p.819-832

1999

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Molecular Basis of HIV-1 Protease Drug Resistance: Structural Analysis of Mutant Proteases Complexed with Cyclic Urea Inhibitors

Biochemistry (Easton), 1997-02, Vol.36 (7), p.1573-1580

1997

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NMR and X-ray Evidence That the HIV Protease Catalytic Aspartyl Groups Are Protonated in the Complex Formed by the Protease and a Non-Peptide Cyclic Urea-Based Inhibitor

Journal of the American Chemical Society, 1994-11, Vol.116 (23), p.10791-10792

1994

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Assay development and high-throughput screening of caspases in microfluidic format

Combinatorial chemistry & high throughput screening, 2003-06, Vol.6 (4), p.303

2003

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Nonpeptide Cyclic Cyanoguanidines as HIV-1 Protease Inhibitors: Synthesis, Structure−Activity Relationships, and X-ray Crystal Structure Studies

Journal of medicinal chemistry, 1998-04, Vol.41 (9), p.1446-1455

1998

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Molecular Recognition of Cyclic Urea HIV-1 Protease Inhibitors

The Journal of biological chemistry, 1998-05, Vol.273 (20), p.12325-12331

1998

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Mapping Hydration Water Molecules in the HIV-1 Protease/DMP323 Complex in Solution by NMR Spectroscopy

Biochemistry (Easton), 1996-10, Vol.35 (39), p.12694-12704

1996

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Thermodynamic linkage between the binding of protons and inhibitors to HIV-1 protease

Protein science, 1999-01, Vol.8 (1), p.180-195

1999

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Crystal structure of scytalone dehydratase--a disease determinant of the rice pathogen, Magnaporthe grisea

Structure (London), 1994-10, Vol.2 (10), p.937-944

1994

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Transformations of Resin-Bound Pyridinium Ylides: I. A Stereoselective Synthesis of 2,2,3-Trisubstituted Cyclopropanecarboxylates

Tetrahedron letters, 1997-11, Vol.38 (46), p.7951-7954

1997

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Fitting an inhibitor into the active site of thermolysin: A molecular dynamics case study

Proteins, structure, function, and bioinformatics, 1996-02, Vol.24 (2), p.227-237

1996

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Discovery of highly selective inhibitors of p38alpha

Current topics in medicinal chemistry, 2005, Vol.5 (10), p.941

2005

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Calculated and Experimental Low-Energy Conformations of Cyclic Urea HIV Protease Inhibitors

Journal of the American Chemical Society, 1998-05, Vol.120 (19), p.4570-4581

1998

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A diazine heterocycle replaces a six-membered hydrogen-bonded array in the active site of scytalone dehydratase

Bioorganic & medicinal chemistry letters, 1993-08, Vol.3 (8), p.1605-1608

1993

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2,3-Dihydro-2,5-dihydroxy-4H-benzopyran-4-one: A Nonphysiological Substrate for Fungal Melanin Biosynthetic Enzymes

Analytical biochemistry, 1998-02, Vol.256 (1), p.1-6

1998

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7-Azabicycloheptane Carboxylic Acid: A Proline Replacement in a Boroarginine Thrombin Inhibitor

Determining appropriate substrate conversion for enzymatic assays in high-throughput screening

Streamlined System for Purifying and Quantifying a Diverse Library of Compounds and the Effect of Compound Concentration Measurements on the Accurate Interpretation of Biological Assay Results

Rational Design of Potent, Bioavailable, Nonpeptide Cyclic Ureas as HIV Protease Inhibitors

Photobleaching-based flow measurement in a commercial capillary electrophoresis chip instrument

Cyclic HIV Protease Inhibitors: Synthesis, Conformational Analysis, P2/P2‘ Structure−Activity Relationship, and Molecular Recognition of Cyclic Ureas

A molecular mechanics/grid method for evaluation of ligand-receptor interactions

Solvation studies of DMP323 and A76928 bound to HIV protease: Analysis of water sites using grand canonical Monte Carlo simulations

A Chemogenomic Approach to Discovering Target-Selective Drugs

Corticotropin-Releasing Hormone Receptor Antagonists: Framework Design and Synthesis Guided by Ligand Conformational Studies

Molecular Basis of HIV-1 Protease Drug Resistance: Structural Analysis of Mutant Proteases Complexed with Cyclic Urea Inhibitors

NMR and X-ray Evidence That the HIV Protease Catalytic Aspartyl Groups Are Protonated in the Complex Formed by the Protease and a Non-Peptide Cyclic Urea-Based Inhibitor

Assay development and high-throughput screening of caspases in microfluidic format

Nonpeptide Cyclic Cyanoguanidines as HIV-1 Protease Inhibitors: Synthesis, Structure−Activity Relationships, and X-ray Crystal Structure Studies

Molecular Recognition of Cyclic Urea HIV-1 Protease Inhibitors

Mapping Hydration Water Molecules in the HIV-1 Protease/DMP323 Complex in Solution by NMR Spectroscopy

Thermodynamic linkage between the binding of protons and inhibitors to HIV-1 protease

Crystal structure of scytalone dehydratase--a disease determinant of the rice pathogen, Magnaporthe grisea

Transformations of Resin-Bound Pyridinium Ylides: I. A Stereoselective Synthesis of 2,2,3-Trisubstituted Cyclopropanecarboxylates

Synthesis, Corticotropin-Releasing Factor Receptor Binding Affinity, and Pharmacokinetic Properties of Triazolo-, Imidazo-, and Pyrrolopyrimidines and -pyridines

Fitting an inhibitor into the active site of thermolysin: A molecular dynamics case study

Discovery of highly selective inhibitors of p38alpha

Calculated and Experimental Low-Energy Conformations of Cyclic Urea HIV Protease Inhibitors

A diazine heterocycle replaces a six-membered hydrogen-bonded array in the active site of scytalone dehydratase

2,3-Dihydro-2,5-dihydroxy-4H-benzopyran-4-one: A Nonphysiological Substrate for Fungal Melanin Biosynthetic Enzymes

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