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Inhibition of Shikimate Kinase from Methicillin-Resistant Staphylococcus aureus by Benzimidazole Derivatives. Kinetic, Computational, Toxicological, and Biological Activity Studies

International journal of molecular sciences, 2024-05, Vol.25 (10), p.5077

2024

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In Silico Exploration of the Trypanothione Reductase (TryR) of L. mexicana

International journal of molecular sciences, 2023-11, Vol.24 (22), p.16046

2023

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Leishmania mexicana Trypanothione Reductase Inhibitors: Computational and Biological Studies

Molecules (Basel, Switzerland), 2019-09, Vol.24 (18), p.3216

2019

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Characterization of the Effect of N-(2-Methoxyphenyl)-1-methyl-1H-benzimidazol-2-amine, Compound 8, against Leishmania mexicana and Its In Vivo Leishmanicidal Activity

International journal of molecular sciences, 2024-01, Vol.25 (1), p.659

2024

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Computational Methods in Cooperation with Experimental Approaches to Design Protein Tyrosine Phosphatase 1B Inhibitors in Type 2 Diabetes Drug Design: A Review of the Achievements of This Century

Pharmaceuticals (Basel, Switzerland), 2022-07, Vol.15 (7), p.866

2022

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Structure‐based approaches for the design of benzimidazole‐2‐carbamate derivatives as tubulin polymerization inhibitors

Chemical biology & drug design, 2017-07, Vol.90 (1), p.40-51

2017

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Structure-Activity Relationship of N -Phenylthieno[2,3- b ]pyridine-2-carboxamide Derivatives Designed as Forkhead Box M1 Inhibitors: The Effect of Electron-Withdrawing and Donating Substituents on the Phenyl Ring

Pharmaceuticals (Basel, Switzerland), 2022-02, Vol.15 (3), p.283

2022

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Characterisation of the in vitro activity of a Nitazoxanide-N-methyl-1H-benzimidazole hybrid molecule against albendazole and nitazoxanide susceptible and resistant strains of Giardia intestinalis and its in vivo giardicidal activity

Memórias do Instituto Oswaldo Cruz, 2020-01, Vol.115, p.e190348

2020

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Alternative energy production pathways in Taenia crassiceps cysticerci in vitro exposed to a benzimidazole derivative (RCB20)

Parasitology, 2016-04, Vol.143 (4), p.488-493

2016

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JVG9, a benzimidazole derivative, alters the surface and cytoskeleton of Trypanosoma cruzi bloodstream trypomastigotes

Memórias do Instituto Oswaldo Cruz, 2014-09, Vol.109 (6), p.757-760

2014

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Novel triclabendazole prodrug: A highly water soluble alternative for the treatment of fasciolosis

Bioorganic & medicinal chemistry letters, 2017-02, Vol.27 (3), p.616-619

2017

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Praziquanamine enantiomers: Crystal structure, Hirshfeld surface analysis, and quantum chemical studies

Journal of molecular structure, 2023-07, Vol.1283, p.135343, Article 135343

2023

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Structure-Based Optimization of Carbendazim-Derived Tubulin Polymerization Inhibitors through Alchemical Free Energy Calculations

Journal of chemical information and modeling, 2023-11, Vol.63 (22), p.7228-7238

2023

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Fosfatriclaben, a prodrug of triclabendazole: Preparation, stability, and fasciolicidal activity of three new intramuscular formulations

Veterinary parasitology, 2024-04, Vol.327, p.110113-110113, Article 110113

2024

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Development and Pharmacokinetic Evaluation of Two Parenteral Formulations of Albendazole Using Prodrug and Cosolvent Approaches

AAPS PharmSciTech, 2023-07, Vol.24 (6), p.158-158, Article 158

2023

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Effectiveness of an experimental injectable prodrug formulation against Fasciola hepatica of different ages in experimentally infected sheep

Veterinary parasitology, 2021-10, Vol.298, p.109524-109524, Article 109524

2021

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Synthesis, antiprotozoal activity, and chemoinformatic analysis of 2-(methylthio)-1H-benzimidazole-5-carboxamide derivatives: Identification of new selective giardicidal and trichomonicidal compounds

European journal of medicinal chemistry, 2017-09, Vol.137, p.211-220

2017

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In silico hit optimization toward AKT inhibition: fragment-based approach, molecular docking and molecular dynamics study

Journal of biomolecular structure & dynamics, 2019-11, Vol.37 (16), p.4301-4311

2019

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5-Chloro-2-methylsulfanyl-6-(naphthalen-1-yloxy)-1H-benzimidazole methanol monosolvate

Acta crystallographica. Section E, Structure reports online, 2014-01, Vol.70 (1), p.o77-o77

2014

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Design, synthesis, kinetic, molecular dynamics, and hypoglycemic effect characterization of new and potential selective benzimidazole derivatives as Protein Tyrosine Phosphatase 1B inhibitors

Bioorganic & medicinal chemistry, 2021-10, Vol.48, p.116418-116418, Article 116418

2021

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Synthesis and trypanocidal activity of novel benzimidazole derivatives

Bioorganic & medicinal chemistry letters, 2016-09, Vol.26 (17), p.4377-4381

2016

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In search of AKT kinase inhibitors as anticancer agents: structure-based design, docking, and molecular dynamics studies of 2,4,6-trisubstituted pyridines

Journal of biomolecular structure & dynamics, 2018-02, Vol.36 (2), p.423-442

2018

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Efficiency comparison of experimental fosfatriclaben with three commercial fasciolicides in experimentally infected sheep

Parasitology research (1987), 2020-08, Vol.119 (8), p.2687-2693

2020

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Curcumin alters the cytoskeleton and microtubule organization on trophozoites of Giardia lamblia

Acta tropica, 2017-08, Vol.172, p.113-121

2017

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Synthesis and biological activity of 2-(trifluoromethyl)-1H-benzimidazole derivatives against some protozoa and Trichinella spiralis

European journal of medicinal chemistry, 2010-07, Vol.45 (7), p.3135-3141

2010

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Inhibition of Shikimate Kinase from Methicillin-Resistant Staphylococcus aureus by Benzimidazole Derivatives. Kinetic, Computational, Toxicological, and Biological Activity Studies

In Silico Exploration of the Trypanothione Reductase (TryR) of L. mexicana

Leishmania mexicana Trypanothione Reductase Inhibitors: Computational and Biological Studies

Characterization of the Effect of N-(2-Methoxyphenyl)-1-methyl-1H-benzimidazol-2-amine, Compound 8, against Leishmania mexicana and Its In Vivo Leishmanicidal Activity

Computational Methods in Cooperation with Experimental Approaches to Design Protein Tyrosine Phosphatase 1B Inhibitors in Type 2 Diabetes Drug Design: A Review of the Achievements of This Century

Structure‐based approaches for the design of benzimidazole‐2‐carbamate derivatives as tubulin polymerization inhibitors

Structure-Activity Relationship of N -Phenylthieno[2,3- b ]pyridine-2-carboxamide Derivatives Designed as Forkhead Box M1 Inhibitors: The Effect of Electron-Withdrawing and Donating Substituents on the Phenyl Ring

Characterisation of the in vitro activity of a Nitazoxanide-N-methyl-1H-benzimidazole hybrid molecule against albendazole and nitazoxanide susceptible and resistant strains of Giardia intestinalis and its in vivo giardicidal activity

Alternative energy production pathways in Taenia crassiceps cysticerci in vitro exposed to a benzimidazole derivative (RCB20)

JVG9, a benzimidazole derivative, alters the surface and cytoskeleton of Trypanosoma cruzi bloodstream trypomastigotes

Novel triclabendazole prodrug: A highly water soluble alternative for the treatment of fasciolosis

Praziquanamine enantiomers: Crystal structure, Hirshfeld surface analysis, and quantum chemical studies

Structure-Based Optimization of Carbendazim-Derived Tubulin Polymerization Inhibitors through Alchemical Free Energy Calculations

Fosfatriclaben, a prodrug of triclabendazole: Preparation, stability, and fasciolicidal activity of three new intramuscular formulations

Development and Pharmacokinetic Evaluation of Two Parenteral Formulations of Albendazole Using Prodrug and Cosolvent Approaches

Effectiveness of an experimental injectable prodrug formulation against Fasciola hepatica of different ages in experimentally infected sheep

Synthesis, antiprotozoal activity, and chemoinformatic analysis of 2-(methylthio)-1H-benzimidazole-5-carboxamide derivatives: Identification of new selective giardicidal and trichomonicidal compounds

In silico hit optimization toward AKT inhibition: fragment-based approach, molecular docking and molecular dynamics study

5-Chloro-2-methylsulfanyl-6-(naphthalen-1-yloxy)-1H-benzimidazole methanol monosolvate

Design, synthesis, kinetic, molecular dynamics, and hypoglycemic effect characterization of new and potential selective benzimidazole derivatives as Protein Tyrosine Phosphatase 1B inhibitors

Synthesis and trypanocidal activity of novel benzimidazole derivatives

In search of AKT kinase inhibitors as anticancer agents: structure-based design, docking, and molecular dynamics studies of 2,4,6-trisubstituted pyridines

Efficiency comparison of experimental fosfatriclaben with three commercial fasciolicides in experimentally infected sheep

Curcumin alters the cytoskeleton and microtubule organization on trophozoites of Giardia lamblia

Synthesis and biological activity of 2-(trifluoromethyl)-1H-benzimidazole derivatives against some protozoa and Trichinella spiralis

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