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Novel N-Arylpyrazolo[3,2-c]-Based Ligands for the Glucocorticoid Receptor: Receptor Binding and in Vivo Activity

Journal of medicinal chemistry, 2004-05, Vol.47 (10), p.2441-2452

2004

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Allosteric Effects of Dexamethasone and RU486 on Glucocorticoid Receptor-DNA Interactions

The Journal of biological chemistry, 2002-01, Vol.277 (2), p.1538-1543

2002

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Novel ketal ligands for the glucocorticoid receptor: in vitro and in vivo activity

Bioorganic & medicinal chemistry letters, 2005-06, Vol.15 (11), p.2926-2931

2005

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Mechanism-Based Inhibition of Human Steroid 5α-Reductase by Finasteride: Enzyme-Catalyzed Formation of NADP−Dihydrofinasteride, a Potent Bisubstrate Analog Inhibitor

Journal of the American Chemical Society, 1996-03, Vol.118 (10), p.2359-2365

1996

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Steroid 5α-reductase inhibitors in androgen-dependent disorders

Current opinion in chemical biology, 1997-08, Vol.1 (2), p.254-259

1997

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Design and synthesis of novel antibacterial agents with inhibitory activity against DNA polymerase III

Bioorganic & medicinal chemistry letters, 2001-08, Vol.11 (16), p.2185-2188

2001

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Enzymatic preparation of high-specific-activity β- d-[6,6′- 3H]fructose-2,6-bisphosphate: Application to a sensitive assay for fructose-2,6-bisphosphatase

Analytical biochemistry, 2010-11, Vol.406 (2), p.97-104

2010

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Glucose-lowering in a db/db mouse model by dihydropyridine diacid glycogen phosphorylase inhibitors

Bioorganic & medicinal chemistry letters, 2003-10, Vol.13 (20), p.3405-3408

2003

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Novel Pyrazolo[3,4-d]pyrimidine-Based Inhibitors of Staphlococcus aureus DNA Polymerase III: Design, Synthesis, and Biological Evaluation

Journal of medicinal chemistry, 2003-05, Vol.46 (10), p.1824-1830

2003

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Activity of the Type 1 5α-Reductase Exhibits Regional Differences in Isolated Sebaceous Glands and Whole Skin

Journal of investigative dermatology, 1995-08, Vol.105 (2), p.209-214

1995

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4-Aza-3-oxo-5.alpha.-androst-1-ene-17.beta.-N-arylcarboxamides as Dual Inhibitors of Human Type 1 and Type 2 Steroid 5.alpha.-Reductases. Dramatic Effect of N-Aryl Substituents on Type 1 and Type 2 5.alpha.-Reductase Inhibitory Potency

Journal of medicinal chemistry, 1995-08, Vol.38 (17), p.3189-3192

1995

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Colorimetric Detection of Glutamine Synthetase-Catalyzed Transferase Activity in Glucocorticoid-Treated Skeletal Muscle Cells

Analytical biochemistry, 2001-02, Vol.289 (1), p.18-25

2001

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Discovery of betamethasone 17α-carbamates as dissociated glucocorticoid receptor modulators in the rat

Bioorganic & medicinal chemistry, 2008-08, Vol.16 (16), p.7535-7542

2008

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Novel heterocyclic glucocorticoids: in vitro profile and in vivo efficacy

Bioorganic & medicinal chemistry letters, 2005-04, Vol.15 (8), p.2163-2167

2005

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4-Aza-3-oxo-5α-androst-1-ene-17β-N-arylcarboxamides as Dual Inhibitors of Human Type 1 and Type 2 Steroid 5α-Reductases. Dramatic Effect of N-Aryl Substituents on Type 1 and Type 2 5α-Reductase Inhibitory Potency

Journal of medicinal chemistry, 1996-03, Vol.39 (5), p.1192-1192

1996

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Novel glucocorticoids containing a 6,5-bicyclic core fused to a pyrazole ring: Synthesis, in vitro profile, molecular modeling studies, and in vivo experiments

Bioorganic & medicinal chemistry letters, 2007-06, Vol.17 (12), p.3354-3361

2007

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A new class of glycogen phosphorylase inhibitors

Bioorganic & medicinal chemistry letters, 2003-11, Vol.13 (22), p.4125-4128

2003

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Novel 3,4-dihydroquinolin-2(1H)-one inhibitors of human glycogen phosphorylase a

Bioorganic & medicinal chemistry letters, 2003-12, Vol.13 (24), p.4385-4388

2003

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Skeletal muscle: a dual system to measure glucocorticoid-dependent transactivation and transrepression of gene regulation

The Journal of steroid biochemistry and molecular biology, 2004-02, Vol.88 (2), p.191-201

2004

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Discovery of betamethasone 17a-carbamates as dissociated glucocorticoid receptor modulators in the rat

Bioorganic & medicinal chemistry, 2008, Vol.16 (16), p.7535-7542

2008

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Selective glucocorticoid receptor nonsteroidal ligands completely antagonize the dexamethasone mediated induction of enzymes involved in gluconeogenesis and glutamine metabolism

The Journal of steroid biochemistry and molecular biology, 2004-12, Vol.92 (5), p.345-356

2004

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Modeling aided design of potent glycogen phosphorylase inhibitors

Journal of molecular graphics & modelling, 2005-04, Vol.23 (5), p.457-464

2005

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Identification and Selective Inhibition of an Isozyme of Steroid 5α- Reductase in Human Scalp

Proceedings of the National Academy of Sciences - PNAS, 1992-11, Vol.89 (22), p.10787-10791

1992

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Discovery of betamethasone 17alpha-carbamates as dissociated glucocorticoid receptor modulators in the rat

Bioorganic & medicinal chemistry, 2008-08, Vol.16 (16), p.7535-7542

2008

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4-Aza-3-oxo-5α-androst-1-ene-17β-N-aryl-carboxamides as dual inhibitors of human type 1 and type 2 steroid 5α-reductases. Dramatic effect of N-aryl substituents on type 1 and type 2 5α-reductase inhibitory potency

Journal of medicinal chemistry, 1995-08, Vol.38 (17), p.3189-3192

1995

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Novel N-Arylpyrazolo[3,2-c]-Based Ligands for the Glucocorticoid Receptor: Receptor Binding and in Vivo Activity

Allosteric Effects of Dexamethasone and RU486 on Glucocorticoid Receptor-DNA Interactions

Novel ketal ligands for the glucocorticoid receptor: in vitro and in vivo activity

Mechanism-Based Inhibition of Human Steroid 5α-Reductase by Finasteride: Enzyme-Catalyzed Formation of NADP−Dihydrofinasteride, a Potent Bisubstrate Analog Inhibitor

Steroid 5α-reductase inhibitors in androgen-dependent disorders

Design and synthesis of novel antibacterial agents with inhibitory activity against DNA polymerase III

Enzymatic preparation of high-specific-activity β- d-[6,6′- 3H]fructose-2,6-bisphosphate: Application to a sensitive assay for fructose-2,6-bisphosphatase

Glucose-lowering in a db/db mouse model by dihydropyridine diacid glycogen phosphorylase inhibitors

Novel Pyrazolo[3,4-d]pyrimidine-Based Inhibitors of Staphlococcus aureus DNA Polymerase III: Design, Synthesis, and Biological Evaluation

Activity of the Type 1 5α-Reductase Exhibits Regional Differences in Isolated Sebaceous Glands and Whole Skin

4-Aza-3-oxo-5.alpha.-androst-1-ene-17.beta.-N-arylcarboxamides as Dual Inhibitors of Human Type 1 and Type 2 Steroid 5.alpha.-Reductases. Dramatic Effect of N-Aryl Substituents on Type 1 and Type 2 5.alpha.-Reductase Inhibitory Potency

Colorimetric Detection of Glutamine Synthetase-Catalyzed Transferase Activity in Glucocorticoid-Treated Skeletal Muscle Cells

Discovery of betamethasone 17α-carbamates as dissociated glucocorticoid receptor modulators in the rat

Novel heterocyclic glucocorticoids: in vitro profile and in vivo efficacy

4-Aza-3-oxo-5α-androst-1-ene-17β-N-arylcarboxamides as Dual Inhibitors of Human Type 1 and Type 2 Steroid 5α-Reductases. Dramatic Effect of N-Aryl Substituents on Type 1 and Type 2 5α-Reductase Inhibitory Potency

Novel glucocorticoids containing a 6,5-bicyclic core fused to a pyrazole ring: Synthesis, in vitro profile, molecular modeling studies, and in vivo experiments

A new class of glycogen phosphorylase inhibitors

Novel 3,4-dihydroquinolin-2(1H)-one inhibitors of human glycogen phosphorylase a

Skeletal muscle: a dual system to measure glucocorticoid-dependent transactivation and transrepression of gene regulation

Discovery of betamethasone 17a-carbamates as dissociated glucocorticoid receptor modulators in the rat

Selective glucocorticoid receptor nonsteroidal ligands completely antagonize the dexamethasone mediated induction of enzymes involved in gluconeogenesis and glutamine metabolism

Modeling aided design of potent glycogen phosphorylase inhibitors

Identification and Selective Inhibition of an Isozyme of Steroid 5α- Reductase in Human Scalp

Discovery of betamethasone 17alpha-carbamates as dissociated glucocorticoid receptor modulators in the rat

4-Aza-3-oxo-5α-androst-1-ene-17β-N-aryl-carboxamides as dual inhibitors of human type 1 and type 2 steroid 5α-reductases. Dramatic effect of N-aryl substituents on type 1 and type 2 5α-reductase inhibitory potency

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