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Discovery of Orally Bioavailable Cathepsin S Inhibitors for the Reversal of Neuropathic Pain

Journal of medicinal chemistry, 2008-09, Vol.51 (18), p.5502-5505

2008

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Thioamide Synthesis: Thioacyl-N-phthalimides as Thioacylating Agents

Journal of organic chemistry, 1997-06, Vol.62 (12), p.3808-3809

1997

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7-tert-Butyl-6-(4-chloro-phenyl)-2-thioxo-2,3-dihydro-1H-pyrido[2,3-d]pyrimidin-4-one, a classic polymodal inhibitor of transient receptor potential vanilloid type 1 with a reduced liability for hyperthermia, is analgesic and ameliorates visceral hypersensitivity

The Journal of pharmacology and experimental therapeutics, 2012-08, Vol.342 (2), p.389

2012

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Bradyzide, a potent non‐peptide B 2 bradykinin receptor antagonist with long‐lasting oral activity in animal models of inflammatory hyperalgesia

British journal of pharmacology, 2009-01, Vol.129 (1), p.77-86

2009

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Discovery of selective and nonpeptidic cathepsin S inhibitors

Bioorganic & medicinal chemistry, 2008-07, Vol.18 (14), p.3959-3962

2008

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Overcoming hERG issues for brain-penetrating cathepsin S inhibitors: 2-Cyanopyrimidines. Part 2

Bioorganic & medicinal chemistry, 2008-10, Vol.18 (19), p.5280-5284

2008

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4-Amino-2-cyanopyrimidines: Novel scaffold for nonpeptidic cathepsin S inhibitors

Bioorganic & medicinal chemistry letters, 2008-08, Vol.18 (16), p.4642-4646

2008

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Bradyzide, a potent non‐peptide B2 bradykinin receptor antagonist with long‐lasting oral activity in animal models of inflammatory hyperalgesia

British journal of pharmacology, 2000-01, Vol.129 (1), p.77-86

2000

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Sulfonamido-aryl ethers as bradykinin B1 receptor antagonists

Bioorganic & medicinal chemistry letters, 2009, Vol.19 (1), p.119-122

2009

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Nonpeptide Bradykinin B2 Receptor Antagonists: Conversion of Rodent-Selective Bradyzide Analogues into Potent, Orally-Active Human Bradykinin B2 Receptor Antagonists

Journal of medicinal chemistry, 2002-05, Vol.45 (11), p.2160-2172

2002

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Nonpeptide Bradykinin B 2 Receptor Antagonists: Conversion of Rodent-Selective Bradyzide Analogues into Potent, Orally-Active Human Bradykinin B 2 Receptor Antagonists

Journal of medicinal chemistry, 2002-05, Vol.45 (11), p.2160-2172

2002

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1-(2-Nitrophenyl)thiosemicarbazides: A Novel Class of Potent, Orally Active Non-Peptide Antagonist for the Bradykinin B 2 Receptor

Journal of medicinal chemistry, 2000-03, Vol.43 (5), p.769-771

2000

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N-Thioacylation of β-Amino Alcohols by N-(Thioacyl)phthalimides: A Facile Synthesis of α-Amino Acid Thiazolines

Tetrahedron letters, 1998, Vol.39 (1), p.127-130

1998

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1-(2-Nitrophenyl)thiosemicarbazides: A Novel Class of Potent, Orally Active Non-Peptide Antagonist for the Bradykinin B2 Receptor

Journal of medicinal chemistry, 2000-03, Vol.43 (5), p.769-771

2000

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The Synthesis of Peptides Related to Prothrombin

Prague, Czechoslovakia, August 29–September 3, 1982, 2019, Vol.17., p.273-276

2019

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Zur Synthese von Human-Big-Gastrin I und seinem 32-Leucin-Analogon 3. Mitteilung: Darstellung der allseits gesch tzten Gesamtsequenzen

Monatshefte für Chemie, 1979, Vol.110 (6), p.1407-1428

1979

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A Study of the Renin Inhibitor H142 in Man

Journal of hypertension, 1985-12, Vol.3 (6), p.653-658

1985

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The structure of a synthetic pepsin inhibitor complexed with endothiapepsin

European journal of biochemistry, 1987-11, Vol.169 (1), p.215-221

1987

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A Transition-state Analogue Inhibitor of Human Renin (H.261): Test in vitro and a Comparison with Captopril in the Anaesthetized Baboon

Journal of hypertension, 1985-02, Vol.3 (1), p.13-18

1985

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The Purification of a High-molecular-weight, Enzymatically Inactive Renin Precursor from Human Kidney

Journal of hypertension, 1984-06, Vol.2 (3), p.305-310

1984

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New Inhibitors of Human Renin Tested in vitro and in vivo in the Anaesthetized Baboon

Journal of hypertension, 1983-12, Vol.1 (4), p.399-403

1983

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Human renin inhibitors

Biochemical Society transactions, 1985-12, Vol.13 (6), p.1029

1985

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Clinical and Biochemical Effects of the Renin Inhibitor H142 in Humans

Journal of cardiovascular pharmacology, 1987, Vol.10 Suppl 7, p.69-74

1987

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Discovery of Orally Bioavailable Cathepsin S Inhibitors for the Reversal of Neuropathic Pain

Thioamide Synthesis: Thioacyl-N-phthalimides as Thioacylating Agents

7-tert-Butyl-6-(4-chloro-phenyl)-2-thioxo-2,3-dihydro-1H-pyrido[2,3-d]pyrimidin-4-one, a classic polymodal inhibitor of transient receptor potential vanilloid type 1 with a reduced liability for hyperthermia, is analgesic and ameliorates visceral hypersensitivity

Bradyzide, a potent non‐peptide B 2 bradykinin receptor antagonist with long‐lasting oral activity in animal models of inflammatory hyperalgesia

Identification and Biological Characterization of 6-Aryl-7-isopropylquinazolinones as Novel TRPV1 Antagonists that Are Effective in Models of Chronic Pain

Discovery of selective and nonpeptidic cathepsin S inhibitors

Overcoming hERG issues for brain-penetrating cathepsin S inhibitors: 2-Cyanopyrimidines. Part 2

4-Amino-2-cyanopyrimidines: Novel scaffold for nonpeptidic cathepsin S inhibitors

Bradyzide, a potent non‐peptide B2 bradykinin receptor antagonist with long‐lasting oral activity in animal models of inflammatory hyperalgesia

Sulfonamido-aryl ethers as bradykinin B1 receptor antagonists

Identification and biological characterization of 6-aryl-7-isopropylquinazolinones as novel TRPV1 antagonists that are effective in models of chronicpain

Nonpeptide Bradykinin B2 Receptor Antagonists: Conversion of Rodent-Selective Bradyzide Analogues into Potent, Orally-Active Human Bradykinin B2 Receptor Antagonists

Nonpeptide Bradykinin B 2 Receptor Antagonists: Conversion of Rodent-Selective Bradyzide Analogues into Potent, Orally-Active Human Bradykinin B 2 Receptor Antagonists

1-(2-Nitrophenyl)thiosemicarbazides: A Novel Class of Potent, Orally Active Non-Peptide Antagonist for the Bradykinin B 2 Receptor

N-Thioacylation of β-Amino Alcohols by N-(Thioacyl)phthalimides: A Facile Synthesis of α-Amino Acid Thiazolines

1-(2-Nitrophenyl)thiosemicarbazides: A Novel Class of Potent, Orally Active Non-Peptide Antagonist for the Bradykinin B2 Receptor

The Synthesis of Peptides Related to Prothrombin

Zur Synthese von Human-Big-Gastrin I und seinem 32-Leucin-Analogon 3. Mitteilung: Darstellung der allseits gesch tzten Gesamtsequenzen

A Study of the Renin Inhibitor H142 in Man

The structure of a synthetic pepsin inhibitor complexed with endothiapepsin

A Transition-state Analogue Inhibitor of Human Renin (H.261): Test in vitro and a Comparison with Captopril in the Anaesthetized Baboon

The Purification of a High-molecular-weight, Enzymatically Inactive Renin Precursor from Human Kidney

New Inhibitors of Human Renin Tested in vitro and in vivo in the Anaesthetized Baboon

Human renin inhibitors

Clinical and Biochemical Effects of the Renin Inhibitor H142 in Humans

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