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Prodrugs of Phosphates and Phosphonates

Journal of medicinal chemistry, 2008-04, Vol.51 (8), p.2328-2345

2008

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Discovery of Cyclic Boronic Acid QPX7728, an Ultrabroad-Spectrum Inhibitor of Serine and Metallo-β-lactamases

Journal of medicinal chemistry, 2020-07, Vol.63 (14), p.7491-7507

2020

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Cu-Catalyzed Decarboxylative Borylation

ACS catalysis, 2018-10, Vol.8 (10), p.9537-9542

2018

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A synthetic lipopeptide targeting top-priority multidrug-resistant Gram-negative pathogens

Nature communications, 2022-03, Vol.13 (1), p.1625-15, Article 1625

2022

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Discovery of a Cyclic Boronic Acid β‑Lactamase Inhibitor (RPX7009) with Utility vs Class A Serine Carbapenemases

Journal of medicinal chemistry, 2015-05, Vol.58 (9), p.3682-3692

2015

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Selection of QPX7831, an Orally Bioavailable Prodrug of Boronic Acid β‑Lactamase Inhibitor QPX7728

Journal of medicinal chemistry, 2021-12, Vol.64 (23), p.17523-17529

2021

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QPX7728, An Ultra-Broad-Spectrum B-Lactamase Inhibitor for Intravenous and Oral Therapy: Overview of Biochemical and Microbiological Characteristics

Frontiers in microbiology, 2021-07, Vol.12, p.697180-697180

2021

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Methodology for Monobactam Diversification: Syntheses and Studies of 4‑Thiomethyl Substituted β‑Lactams with Activity against Gram-Negative Bacteria, Including Carbapenemase Producing Acinetobacter baumannii

Journal of medicinal chemistry, 2017-11, Vol.60 (21), p.8933-8944

2017

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Broad-spectrum cyclic boronate β-lactamase inhibitors featuring an intramolecular prodrug for oral bioavailability

Bioorganic & medicinal chemistry, 2022-05, Vol.62, p.116722-116722, Article 116722

2022

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Scalable Synthesis of β‑Lactamase Inhibitor QPX7728 by Sequential Nickel-Catalyzed Boron Insertion into a Benzofuran Substrate and Enantioselective Cyclopropanation of the Resulting Vinylboronate

Organic process research & development, 2022-03, Vol.26 (3), p.925-935

2022

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Development of a Continuous Flow Process for a Matteson Reaction: From Lab Scale to Full-Scale Production of a Pharmaceutical Intermediate

Organic process research & development, 2019-05, Vol.23 (5), p.1069-1077

2019

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Scalable On-Demand Production of Purified Diazomethane Suitable for Sensitive Catalytic Reactions

Organic process research & development, 2021-03, Vol.25 (3), p.522-528

2021

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Antiviral Efficacy upon Administration of a HepDirect Prodrug of 2′-C-Methylcytidine to Hepatitis C Virus-Infected Chimpanzees

Antimicrobial Agents and Chemotherapy, 2011-08, Vol.55 (8), p.3854-3860

2011

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A Potent and Selective AMPK Activator That Inhibits de Novo Lipogenesis

ACS medicinal chemistry letters, 2010-12, Vol.1 (9), p.478-482

2010

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Synthesis and Biological Evaluation of a Series of Liver-Selective Phosphonic Acid Thyroid Hormone Receptor Agonists and Their Prodrugs

Journal of medicinal chemistry, 2008-11, Vol.51 (22), p.7075-7093

2008

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Liver-Targeted Prodrugs of 2‘-C-Methyladenosine for Therapy of Hepatitis C Virus Infection

Journal of medicinal chemistry, 2007-08, Vol.50 (16), p.3891-3896

2007

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Inhibitors of Efflux Pumps in Pseudomonas aeruginosa Potentiate the Activity of the Fluoroquinolone Antibacterial Levofloxacin

Journal of medicinal chemistry, 1999-12, Vol.42 (24), p.4928-4931

1999

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Quantitative Structure−Activity Relationships among Macrolide Antibacterial Agents: In Vitro and in Vivo Potency against Pasteurella multocida

Journal of medicinal chemistry, 1997-04, Vol.40 (9), p.1340-1346

1997

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Zinc finger protein 33B demonstrates sex interaction with atopy-related markers in childhood asthma

The European respiratory journal, 2023-01, Vol.61 (1), p.2200479

2023

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Stereochemical Elucidation and Total Synthesis of Dihydropacidamycin D, a Semisynthetic Pacidamycin

Journal of the American Chemical Society, 2001-02, Vol.123 (5), p.870-874

2001

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Synthetic dihydropacidamycin antibiotics: A modified spectrum of activity for the pacidamycin class

Bioorganic & medicinal chemistry letters, 2003-10, Vol.13 (19), p.3305-3309

2003

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Prodrugs of Cephalosporin RWJ-333441 (MC-04,546) with Improved Aqueous Solubility

Antimicrobial Agents and Chemotherapy, 2003-06, Vol.47 (6), p.2043-2046

2003

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Synthesis of base-modified dihydropacidamycins

Bioorganic & medicinal chemistry letters, 2002-04, Vol.12 (7), p.1121-1123

2002

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Discovery of RWJ-54428 (MC-02, 479), a New Cephalosporin Active Against Resistant Gram-positive Bacteria

The Journal of Antibiotics, 2000/11/25, Vol.53(11), pp.1272-1281

2000

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A tour of recent patent applications addressing antibacterial resistance

Expert opinion on therapeutic patents, 2002-08, Vol.12 (8), p.1159-1172

2002

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Prodrugs of Phosphates and Phosphonates

Discovery of Cyclic Boronic Acid QPX7728, an Ultrabroad-Spectrum Inhibitor of Serine and Metallo-β-lactamases

Cu-Catalyzed Decarboxylative Borylation

A synthetic lipopeptide targeting top-priority multidrug-resistant Gram-negative pathogens

Discovery of a Cyclic Boronic Acid β‑Lactamase Inhibitor (RPX7009) with Utility vs Class A Serine Carbapenemases

Selection of QPX7831, an Orally Bioavailable Prodrug of Boronic Acid β‑Lactamase Inhibitor QPX7728

QPX7728, An Ultra-Broad-Spectrum B-Lactamase Inhibitor for Intravenous and Oral Therapy: Overview of Biochemical and Microbiological Characteristics

Methodology for Monobactam Diversification: Syntheses and Studies of 4‑Thiomethyl Substituted β‑Lactams with Activity against Gram-Negative Bacteria, Including Carbapenemase Producing Acinetobacter baumannii

Broad-spectrum cyclic boronate β-lactamase inhibitors featuring an intramolecular prodrug for oral bioavailability

Scalable Synthesis of β‑Lactamase Inhibitor QPX7728 by Sequential Nickel-Catalyzed Boron Insertion into a Benzofuran Substrate and Enantioselective Cyclopropanation of the Resulting Vinylboronate

Development of a Continuous Flow Process for a Matteson Reaction: From Lab Scale to Full-Scale Production of a Pharmaceutical Intermediate

Scalable On-Demand Production of Purified Diazomethane Suitable for Sensitive Catalytic Reactions

Antiviral Efficacy upon Administration of a HepDirect Prodrug of 2′-C-Methylcytidine to Hepatitis C Virus-Infected Chimpanzees

A Potent and Selective AMPK Activator That Inhibits de Novo Lipogenesis

Synthesis and Biological Evaluation of a Series of Liver-Selective Phosphonic Acid Thyroid Hormone Receptor Agonists and Their Prodrugs

Liver-Targeted Prodrugs of 2‘-C-Methyladenosine for Therapy of Hepatitis C Virus Infection

Inhibitors of Efflux Pumps in Pseudomonas aeruginosa Potentiate the Activity of the Fluoroquinolone Antibacterial Levofloxacin

Quantitative Structure−Activity Relationships among Macrolide Antibacterial Agents: In Vitro and in Vivo Potency against Pasteurella multocida

Zinc finger protein 33B demonstrates sex interaction with atopy-related markers in childhood asthma

Stereochemical Elucidation and Total Synthesis of Dihydropacidamycin D, a Semisynthetic Pacidamycin

Synthetic dihydropacidamycin antibiotics: A modified spectrum of activity for the pacidamycin class

Prodrugs of Cephalosporin RWJ-333441 (MC-04,546) with Improved Aqueous Solubility

Synthesis of base-modified dihydropacidamycins

Discovery of RWJ-54428 (MC-02, 479), a New Cephalosporin Active Against Resistant Gram-positive Bacteria

A tour of recent patent applications addressing antibacterial resistance

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