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Series of Novel and Highly Potent Cyclic Peptide PCSK9 Inhibitors Derived from an mRNA Display Screen and Optimized via Structure-Based Design

Journal of medicinal chemistry, 2020-11, Vol.63 (22), p.13796-13824

2020

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Platensimycin and Platencin Congeners from Streptomyces platensis

Journal of natural products (Washington, D.C.), 2011-03, Vol.74 (3), p.329-340

2011

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A Series of Novel, Highly Potent, and Orally Bioavailable Next-Generation Tricyclic Peptide PCSK9 Inhibitors

Journal of medicinal chemistry, 2021-11, Vol.64 (22), p.16770-16800

2021

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A Family of Highly Selective Allosteric Modulators of the Metabotropic Glutamate Receptor Subtype 5

Molecular pharmacology, 2003-09, Vol.64 (3), p.731-740

2003

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A novel selective allosteric modulator potentiates the activity of native metabotropic glutamate receptor subtype 5 in rat forebrain

The Journal of pharmacology and experimental therapeutics, 2004-05, Vol.309 (2), p.568-577

2004

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Molecular Simulations Identify Binding Poses and Approximate Affinities of Stapled α‑Helical Peptides to MDM2 and MDMX

Journal of chemical theory and computation, 2017-02, Vol.13 (2), p.863-869

2017

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Synthesis and biological evaluation of platensimycin analogs

Bioorganic & medicinal chemistry letters, 2009-03, Vol.19 (6), p.1623-1627

2009

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Isolation, structure and biological activities of platencin A2–A4 from Streptomyces platensis

Bioorganic & medicinal chemistry, 2010-04, Vol.18 (7), p.2602-2610

2010

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Synthesis and evaluation of N-[(1 S,2 S)-3-(4-chlorophenyl)-2-(3-cyanophenyl)-1-methylpropyl]-2-methyl-2-aminopropanamide as human cannabinoid-1 receptor (CB1R) inverse agonists

Bioorganic & medicinal chemistry letters, 2009-09, Vol.19 (17), p.5195-5199

2009

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Discovery of benzamides as potent human β3 adrenergic receptor agonists

Bioorganic & medicinal chemistry letters, 2016-01, Vol.26 (1), p.55-59

2016

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Investigation of piperazine benzamides as human β3 adrenergic receptor agonists for the treatment of overactive bladder

Bioorganic & medicinal chemistry letters, 2017-02, Vol.27 (4), p.1094-1098

2017

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Investigation of piperazine benzamides as human β 3 adrenergic receptor agonists for the treatment of overactive bladder

Bioorganic & medicinal chemistry letters, 2017-02, Vol.27 (4), p.1094-1098

2017

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Nodulisporic Acids D−F: Structure, Biological Activities, and Biogenetic Relationships

Journal of natural products (Washington, D.C.), 2004-09, Vol.67 (9), p.1496-1506

2004

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Mini review on molecular modeling of P-glycoprotein (Pgp)

Current topics in medicinal chemistry, 2007-08, Vol.7 (15), p.1525-1529

2007

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Isolation, structure and biological activities of platencin A(2)-A(4) from Streptomyces platensis

Bioorganic & medicinal chemistry, 2010-04, Vol.18 (7), p.2602-2610

2010

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Challenges in the development of mGluR5 positive allosteric modulators: The discovery of CPPHA

Bioorganic & medicinal chemistry letters, 2007-03, Vol.17 (5), p.1386-1391

2007

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Potent Kv1.3 inhibitors from correolide—modification of the C18 position

Bioorganic & medicinal chemistry letters, 2005-01, Vol.15 (2), p.447-451

2005

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Orally Bioavailable Macrocyclic Peptide That Inhibits Binding of PCSK9 to the Low Density Lipoprotein Receptor

Circulation (New York, N.Y.), 2023-07, Vol.148 (2), p.144-158

2023

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A Gly/Ala switch contributes to high affinity binding of benzoxazinone-based non-peptide oxytocin receptor antagonists

FEBS letters, 2005-01, Vol.579 (2), p.349-356

2005

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Binding modes of dihydroquinoxalinones in a homology model of bradykinin receptor 1

Biochemical and biophysical research communications, 2005-05, Vol.331 (1), p.159-166

2005

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Identification of the Critical Residues of Bradykinin Receptor B1 for Interaction with the Kinins Guided by Site-Directed Mutagenesis and Molecular Modeling

Biochemistry (Easton), 2006-12, Vol.45 (48), p.14355-14361

2006

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Molecular Simulations Identify Binding Poses and Approximate Affinities of Stapled [alpha]-Helical Peptides to MDM2 and MDMX

Journal of chemical theory and computation, 2017-02, Vol.13 (2), p.863-869

2017

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A revised potential-energy surface for molecular mechanics studies of carbohydrates

Carbohydrate research, 1988-09, Vol.180 (2), p.207-221

1988

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Difference in mGluR5 Interaction between Positive Allosteric Modulators from Two Structural Classes

Annals of the New York Academy of Sciences, 2003-11, Vol.1003 (1), p.481-484

2003

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Establishment of P‐Glycoprotein Structure–Transport Relationships to Optimize CNS Exposure in Drug Discovery

Blood‐Brain Barrier in Drug Discovery, 2015, p.113-124

2015

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Series of Novel and Highly Potent Cyclic Peptide PCSK9 Inhibitors Derived from an mRNA Display Screen and Optimized via Structure-Based Design

Platensimycin and Platencin Congeners from Streptomyces platensis

A Series of Novel, Highly Potent, and Orally Bioavailable Next-Generation Tricyclic Peptide PCSK9 Inhibitors

A Family of Highly Selective Allosteric Modulators of the Metabotropic Glutamate Receptor Subtype 5

A novel selective allosteric modulator potentiates the activity of native metabotropic glutamate receptor subtype 5 in rat forebrain

Molecular Simulations Identify Binding Poses and Approximate Affinities of Stapled α‑Helical Peptides to MDM2 and MDMX

Synthesis and biological evaluation of platensimycin analogs

Isolation, structure and biological activities of platencin A2–A4 from Streptomyces platensis

Synthesis and evaluation of N-[(1 S,2 S)-3-(4-chlorophenyl)-2-(3-cyanophenyl)-1-methylpropyl]-2-methyl-2-aminopropanamide as human cannabinoid-1 receptor (CB1R) inverse agonists

Discovery of benzamides as potent human β3 adrenergic receptor agonists

Investigation of piperazine benzamides as human β3 adrenergic receptor agonists for the treatment of overactive bladder

Investigation of piperazine benzamides as human β 3 adrenergic receptor agonists for the treatment of overactive bladder

Nodulisporic Acids D−F: Structure, Biological Activities, and Biogenetic Relationships

Mini review on molecular modeling of P-glycoprotein (Pgp)

Isolation, structure and biological activities of platencin A(2)-A(4) from Streptomyces platensis

Challenges in the development of mGluR5 positive allosteric modulators: The discovery of CPPHA

Potent Kv1.3 inhibitors from correolide—modification of the C18 position

Orally Bioavailable Macrocyclic Peptide That Inhibits Binding of PCSK9 to the Low Density Lipoprotein Receptor

A Gly/Ala switch contributes to high affinity binding of benzoxazinone-based non-peptide oxytocin receptor antagonists

Binding modes of dihydroquinoxalinones in a homology model of bradykinin receptor 1

Identification of the Critical Residues of Bradykinin Receptor B1 for Interaction with the Kinins Guided by Site-Directed Mutagenesis and Molecular Modeling

Molecular Simulations Identify Binding Poses and Approximate Affinities of Stapled [alpha]-Helical Peptides to MDM2 and MDMX

A revised potential-energy surface for molecular mechanics studies of carbohydrates

Difference in mGluR5 Interaction between Positive Allosteric Modulators from Two Structural Classes

Establishment of P‐Glycoprotein Structure–Transport Relationships to Optimize CNS Exposure in Drug Discovery

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