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Discovery of 7‑Methyl-5-(1-{[3-(trifluoromethyl)phenyl]acetyl}-2,3-dihydro‑1H‑indol-5-yl)‑7H‑pyrrolo[2,3‑d]pyrimidin-4-amine (GSK2606414), a Potent and Selective First-in-Class Inhibitor of Protein Kinase R (PKR)-like Endoplasmic Reticulum Kinase (PERK)

Journal of medicinal chemistry, 2012-08, Vol.55 (16), p.7193-7207

2012

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Discovery of GSK2656157: An Optimized PERK Inhibitor Selected for Preclinical Development

ACS medicinal chemistry letters, 2013-10, Vol.4 (10), p.964-968

2013

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Identification of Potent, Selective, Cell-Active Inhibitors of the Histone Lysine Methyltransferase EZH2

ACS medicinal chemistry letters, 2012-12, Vol.3 (12), p.1091-1096

2012

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Structure-Based Design of Potent and Selective 3-Phosphoinositide-Dependent Kinase-1 (PDK1) Inhibitors

Journal of medicinal chemistry, 2011-03, Vol.54 (6), p.1871-1895

2011

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Stereoselective cascade reactions that incorporate a 7-exo acyl radical cyclization

Organic letters, 2006-04, Vol.8 (9), p.1867-1870

2006

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Rapid synthesis of diversely functionalized 3,4,7-trisubstituted indoles

Tetrahedron letters, 2011-06, Vol.52 (26), p.3376-3378

2011

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Acylprolinamides: A new class of peptide deformylase inhibitors with in vivo antibacterial activity

Bioorganic & medicinal chemistry letters, 2012-06, Vol.22 (12), p.4028-4032

2012

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Discovery of a new series of Aurora inhibitors through truncation of GSK1070916

Bioorganic & medicinal chemistry letters, 2010-04, Vol.20 (8), p.2552-2555

2010

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Stereoselective Cascade Reactions that Incorporate a 7-e xo Acyl Radical Cyclization

Organic letters, 2006-04, Vol.8 (9), p.1867-1870

2006

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Abstract 2939: Discovery and synthesis of highly potent and selective small molecule inhibitors of the histone methyltransferase EZH2

Cancer research (Chicago, Ill.), 2012-04, Vol.72 (8_Supplement), p.2939-2939

2012

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ChemInform Abstract: Rapid Synthesis of Diversely Functionalized 3,4,7-Trisubstituted Indoles

ChemInform, 2011-10, Vol.42 (42), p.no-no

2011

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Stereoselective Cascade Reactions that Incorporate a 7-exo Acyl Radical Cyclization

ChemInform, 2006-08, Vol.37 (35), p.no-no

2006

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The Role of DNA Copy Number Variation in Schizophrenia

Biological psychiatry (1969), 2009-12, Vol.66 (11), p.1005-1012

2009

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Robust nanoscopy of a synaptic protein in living mice by organic-fluorophore labeling

Proceedings of the National Academy of Sciences - PNAS, 2018-08, Vol.115 (34), p.E8047-E8056

2018

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Supramolecular organization of NMDA receptors and the postsynaptic density

Current opinion in neurobiology, 2017-08, Vol.45, p.139-147

2017

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NMDA receptors are selectively partitioned into complexes and supercomplexes during synapse maturation

Nature communications, 2016-04, Vol.7 (1), p.11264-11264, Article 11264

2016

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Proteomic analysis of NMDA receptor-adhesion protein signaling complexes

Nature neuroscience, 2000-07, Vol.3 (7), p.661-669

2000

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Adipose Tissue Macrophages Promote Myelopoiesis and Monocytosis in Obesity

Cell metabolism, 2014-05, Vol.19 (5), p.821-835

2014

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Arc Requires PSD95 for Assembly into Postsynaptic Complexes Involved with Neural Dysfunction and Intelligence

Cell reports (Cambridge), 2017-10, Vol.21 (3), p.679-691

2017

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Hierarchical organization and genetically separable subfamilies of PSD95 postsynaptic supercomplexes

Journal of neurochemistry, 2017-08, Vol.142 (4), p.504-511

2017

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Molecular characterization and comparison of the components and multiprotein complexes in the postsynaptic proteome

Journal of neurochemistry, 2006-04, Vol.97 (s1), p.16-23

2006

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Neurobeachin Regulates Glutamate- and GABA-Receptor Targeting to Synapses via Distinct Pathways

Molecular neurobiology, 2016-05, Vol.53 (4), p.2112-2123

2016

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A systematic review of rodent pest research in Afro-Malagasy small-holder farming systems: Are we asking the right questions?

PloS one, 2017-03, Vol.12 (3), p.e0174554-e0174554

2017

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Understanding the relationship between geopolymer composition, microstructure and mechanical properties

Colloids and surfaces. A, Physicochemical and engineering aspects, 2005-11, Vol.269 (1), p.47-58

2005

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Discovery of 7‑Methyl-5-(1-{[3-(trifluoromethyl)phenyl]acetyl}-2,3-dihydro‑1H‑indol-5-yl)‑7H‑pyrrolo[2,3‑d]pyrimidin-4-amine (GSK2606414), a Potent and Selective First-in-Class Inhibitor of Protein Kinase R (PKR)-like Endoplasmic Reticulum Kinase (PERK)

Discovery of GSK2656157: An Optimized PERK Inhibitor Selected for Preclinical Development

Identification of Potent, Selective, Cell-Active Inhibitors of the Histone Lysine Methyltransferase EZH2

Structure-Based Design of Potent and Selective 3-Phosphoinositide-Dependent Kinase-1 (PDK1) Inhibitors

Stereoselective cascade reactions that incorporate a 7-exo acyl radical cyclization

Rapid synthesis of diversely functionalized 3,4,7-trisubstituted indoles

Acylprolinamides: A new class of peptide deformylase inhibitors with in vivo antibacterial activity

Discovery of a new series of Aurora inhibitors through truncation of GSK1070916

Stereoselective Cascade Reactions that Incorporate a 7-e xo Acyl Radical Cyclization

Abstract 2939: Discovery and synthesis of highly potent and selective small molecule inhibitors of the histone methyltransferase EZH2

Discovery of 7-Methyl-5-(1-{[3-(trifluoromethyl)phenyl]acetyl}-2,3-dihydro-1 H -indol-5-yl)-7 H -pyrrolo[2,3- d ]pyrimidin-4-amine (GSK2606414), a Potent and Selective First-in-Class Inhibitor of Protein Kinase R (PKR)-like Endoplasmic Reticulum Kinase (PERK)

ChemInform Abstract: Rapid Synthesis of Diversely Functionalized 3,4,7-Trisubstituted Indoles

Stereoselective Cascade Reactions that Incorporate a 7-exo Acyl Radical Cyclization

The Role of DNA Copy Number Variation in Schizophrenia

Robust nanoscopy of a synaptic protein in living mice by organic-fluorophore labeling

Supramolecular organization of NMDA receptors and the postsynaptic density

NMDA receptors are selectively partitioned into complexes and supercomplexes during synapse maturation

Proteomic analysis of NMDA receptor-adhesion protein signaling complexes

Adipose Tissue Macrophages Promote Myelopoiesis and Monocytosis in Obesity

Arc Requires PSD95 for Assembly into Postsynaptic Complexes Involved with Neural Dysfunction and Intelligence

Hierarchical organization and genetically separable subfamilies of PSD95 postsynaptic supercomplexes

Molecular characterization and comparison of the components and multiprotein complexes in the postsynaptic proteome

Neurobeachin Regulates Glutamate- and GABA-Receptor Targeting to Synapses via Distinct Pathways

A systematic review of rodent pest research in Afro-Malagasy small-holder farming systems: Are we asking the right questions?

Understanding the relationship between geopolymer composition, microstructure and mechanical properties

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