UB Paderborn / Katalog / Suche / in CDI

Nonclinical Evaluation of Antibacterial Oxazolidinones Contezolid and Contezolid Acefosamil with Low Serotonergic Neurotoxicity

Chemical research in toxicology, 2021-05, Vol.34 (5), p.1348-1354

2021

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New Potent Antibacterial Oxazolidinone (MRX-I) with an Improved Class Safety Profile

Journal of medicinal chemistry, 2014-06, Vol.57 (11), p.4487-4497

2014

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Preclinical toxicity evaluation of novel antibacterial contezolid acefosamil in rats and dogs

Journal of applied toxicology, 2024-05, Vol.44 (5), p.770-783

2024

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Pharmacokinetics and Disposition of Contezolid in Humans: Resolution of a Disproportionate Human Metabolite for Clinical Development

Antimicrobial agents and chemotherapy, 2021-10, Vol.65 (11), p.e0040921

2021

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Approaches to Combinatorial Synthesis of Heterocycles: A Solid-Phase Synthesis of 1,4-Dihydropyridines

Journal of organic chemistry, 1996-02, Vol.61 (3), p.924-928

1996

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Discovery of Antibacterial Contezolid Acefosamil: Innovative O‑Acyl Phosphoramidate Prodrug for IV and Oral Therapies

ACS medicinal chemistry letters, 2022-07, Vol.13 (7), p.1030-1035

2022

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Recent developments in the identification of novel oxazolidinone antibacterial agents

Bioorganic & medicinal chemistry, 2006-06, Vol.14 (12), p.4227-4240

2006

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Selection and characterisation of Staphylococcus aureus mutants with reduced susceptibility to the investigational oxazolidinone MRX-I

International journal of antimicrobial agents, 2014-05, Vol.43 (5), p.418-422

2014

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Synthesis of Aza-, Oxa-, and Thiabicyclo[3.1.0]hexane Heterocycles from a Common Synthetic Intermediate

Organic letters, 2005-06, Vol.7 (13), p.2627-2630

2005

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Novel antibacterial azetidine lincosamides

Bioorganic & medicinal chemistry, 2008-04, Vol.18 (8), p.2645-2648

2008

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Conformational Constraint in Oxazolidinone Antibacterials. Synthesis and Structure−Activity Studies of (Azabicyclo[3.1.0]hexylphenyl)oxazolidinones

Journal of medicinal chemistry, 2005-07, Vol.48 (15), p.5009-5024

2005

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Novel 6-position modified 1-thioalkyl-lincosamines

Tetrahedron letters, 2008-04, Vol.49 (18), p.2979-2981

2008

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Novel oxazolidinone–quinolone hybrid antimicrobials

Bioorganic & medicinal chemistry letters, 2003-12, Vol.13 (23), p.4213-4216

2003

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Synthesis and structure–activity studies of antibacterial oxazolidinones containing dihydrothiopyran or dihydrothiazine C-rings

Bioorganic & medicinal chemistry letters, 2006-07, Vol.16 (13), p.3475-3478

2006

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A distal methyl substituent attenuates mitochondrial protein synthesis inhibition in oxazolidinone antibacterials

Bioorganic & medicinal chemistry letters, 2007-09, Vol.17 (18), p.5036-5040

2007

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Approaches to combinatorial synthesis of heterocycles: Solid phase synthesis of pyridines and pyrido[2,3-d]pyrimidines

Tetrahedron letters, 1996-07, Vol.37 (27), p.4643-4646

1996

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Conformational constraint in oxazolidinone antibacterials. Part 2: Synthesis and structure–activity studies of oxa-, aza-, and thiabicyclo[3.1.0]hexylphenyl oxazolidinones

Bioorganic & medicinal chemistry letters, 2006-03, Vol.16 (5), p.1126-1129

2006

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New Antibacterial tetrahydro-4(2 H)-thiopyran and thiomorpholine S-oxide and S, S-dioxide phenyloxazolidinones

Bioorganic & medicinal chemistry letters, 2003-12, Vol.13 (23), p.4209-4212

2003

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A general and efficient solid phase synthesis of quinazoline-2,4-diones

Tetrahedron letters, 1997-03, Vol.38 (10), p.1729-1732

1997

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Solid-Phase Synthesis of β-Sultams

Journal of organic chemistry, 1997-11, Vol.62 (23), p.8177-8181

1997

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Combinatorial approaches to pharmacophoric heterocycles : A solid-phase synthesis of 3,1-benzoxazine-4-ones

Biotechnology and bioengineering, 1998-01, Vol.61 (1), p.13-16

GORDEEV, M. F

1998

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Lithium tetrafluoroborate-assisted reactions of N-(.alpha.-aminoalkyl)benzotriazoles with olefins and 1,3-dienes. New syntheses of 1,2,5,6-tetrahydropyridinium salts, 1,2,3,4-tetrahydroquinolines, and some related heterocyclic systems

Journal of organic chemistry, 1993-07, Vol.58 (15), p.4049-4053

1993

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A New and Safe Approach to (N-Vinylimino)phosphoranes

Journal of organic chemistry, 1994-05, Vol.59 (10), p.2740-2742

1994

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New synthetic routes to furans and dihydrofurans from 1-propargylbenzotriazole

Journal of organic chemistry, 1993-05, Vol.58 (11), p.3038-3041

1993

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Combinatorial chemistry of natural products: Solid phase synthesis of D- and L-cycloserine derivatives

Tetrahedron, 1998, Vol.54 (52), p.15879-15890

1998

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Nonclinical Evaluation of Antibacterial Oxazolidinones Contezolid and Contezolid Acefosamil with Low Serotonergic Neurotoxicity

New Potent Antibacterial Oxazolidinone (MRX-I) with an Improved Class Safety Profile

Preclinical toxicity evaluation of novel antibacterial contezolid acefosamil in rats and dogs

Pharmacokinetics and Disposition of Contezolid in Humans: Resolution of a Disproportionate Human Metabolite for Clinical Development

Approaches to Combinatorial Synthesis of Heterocycles: A Solid-Phase Synthesis of 1,4-Dihydropyridines

Discovery of Antibacterial Contezolid Acefosamil: Innovative O‑Acyl Phosphoramidate Prodrug for IV and Oral Therapies

Recent developments in the identification of novel oxazolidinone antibacterial agents

Selection and characterisation of Staphylococcus aureus mutants with reduced susceptibility to the investigational oxazolidinone MRX-I

Synthesis of Aza-, Oxa-, and Thiabicyclo[3.1.0]hexane Heterocycles from a Common Synthetic Intermediate

Novel antibacterial azetidine lincosamides

Conformational Constraint in Oxazolidinone Antibacterials. Synthesis and Structure−Activity Studies of (Azabicyclo[3.1.0]hexylphenyl)oxazolidinones

Novel 6-position modified 1-thioalkyl-lincosamines

Novel oxazolidinone–quinolone hybrid antimicrobials

Synthesis and structure–activity studies of antibacterial oxazolidinones containing dihydrothiopyran or dihydrothiazine C-rings

A distal methyl substituent attenuates mitochondrial protein synthesis inhibition in oxazolidinone antibacterials

Approaches to combinatorial synthesis of heterocycles: Solid phase synthesis of pyridines and pyrido[2,3-d]pyrimidines

Conformational constraint in oxazolidinone antibacterials. Part 2: Synthesis and structure–activity studies of oxa-, aza-, and thiabicyclo[3.1.0]hexylphenyl oxazolidinones

New Antibacterial tetrahydro-4(2 H)-thiopyran and thiomorpholine S-oxide and S, S-dioxide phenyloxazolidinones

A general and efficient solid phase synthesis of quinazoline-2,4-diones

Solid-Phase Synthesis of β-Sultams

Combinatorial approaches to pharmacophoric heterocycles : A solid-phase synthesis of 3,1-benzoxazine-4-ones

Lithium tetrafluoroborate-assisted reactions of N-(.alpha.-aminoalkyl)benzotriazoles with olefins and 1,3-dienes. New syntheses of 1,2,5,6-tetrahydropyridinium salts, 1,2,3,4-tetrahydroquinolines, and some related heterocyclic systems

A New and Safe Approach to (N-Vinylimino)phosphoranes

New synthetic routes to furans and dihydrofurans from 1-propargylbenzotriazole

Combinatorial chemistry of natural products: Solid phase synthesis of D- and L-cycloserine derivatives

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